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Found 602 with Last Name = 'qin' and Initial = 'q'
TargetAurora kinase A(Homo sapiens (Human))
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50004205(MK-045 | MK-0457 | TOZASERTIB | US9249124, VX680 |...)
Affinity DataKi:  0.650nMAssay Description:Inhibition of Aurora A (unknown origin)More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAurora kinase B(Homo sapiens (Human))
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50004205(MK-045 | MK-0457 | TOZASERTIB | US9249124, VX680 |...)
Affinity DataKi:  3.40nMAssay Description:Inhibition of Aurora B (unknown origin)More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAurora kinase C(Homo sapiens (Human))
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50004205(MK-045 | MK-0457 | TOZASERTIB | US9249124, VX680 |...)
Affinity DataKi:  4.60nMAssay Description:Inhibition of Aurora C (unknown origin)More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSerine/threonine-protein kinase PLK4(Homo sapiens (Human))
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50004205(MK-045 | MK-0457 | TOZASERTIB | US9249124, VX680 |...)
Affinity DataKi:  7.70nMAssay Description:Inhibition of PLK4 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSerine/threonine-protein kinase PLK4(Homo sapiens (Human))
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50591934(CHEMBL5209160)
Affinity DataIC50:  0.100nMAssay Description:Inhibition of recombinant human PLK4 incubated for 60 mins by Lanthascreen Eu kinase binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetRetinol-binding protein 4(Homo sapiens (Human))
Albany Molecular Research

Curated by ChEMBL
LigandPNGBDBM50026260(CHEMBL3359024)
Affinity DataIC50:  0.121nMAssay Description:Antagonist activity at maltose binding protein-tagged RBP4 (unknown origin) expressed in Escherichia coli assessed as inhibition of retinol-induced p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinol-binding protein 4(Homo sapiens (Human))
Albany Molecular Research

Curated by ChEMBL
LigandPNGBDBM50019040(CHEMBL1230001)
Affinity DataIC50:  0.155nMAssay Description:Antagonist activity at maltose binding protein-tagged RBP4 (unknown origin) expressed in Escherichia coli assessed as inhibition of retinol-induced p...More data for this Ligand-Target Pair
TargetRetinol-binding protein 4(Homo sapiens (Human))
Albany Molecular Research

Curated by ChEMBL
LigandPNGBDBM50026258(CHEMBL3359022)
Affinity DataIC50:  0.179nMAssay Description:Antagonist activity at maltose binding protein-tagged RBP4 (unknown origin) expressed in Escherichia coli assessed as inhibition of retinol-induced p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PLK4(Homo sapiens (Human))
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50591949(CHEMBL5185001)
Affinity DataIC50:  0.200nMAssay Description:Inhibition of recombinant human PLK4 incubated for 60 mins by Lanthascreen Eu kinase binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetNT-3 growth factor receptor(Homo sapiens (Human))TBA
LigandPNGBDBM136597(US10005783, 14 | US10047097, 14 | US10774085, Exam...)
Affinity DataIC50:  0.200nMAssay Description:Inhibition of TRKC (unknown origin) using TK as substrate in presence of ATP incubated for 40 mins by HTRF KinEASE assayMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetRetinol-binding protein 4(Homo sapiens (Human))
Albany Molecular Research

Curated by ChEMBL
LigandPNGBDBM50026259(CHEMBL3359023)
Affinity DataIC50:  0.235nMAssay Description:Antagonist activity at maltose binding protein-tagged RBP4 (unknown origin) expressed in Escherichia coli assessed as inhibition of retinol-induced p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinol-binding protein 4(Homo sapiens (Human))
Albany Molecular Research

Curated by ChEMBL
LigandPNGBDBM50026255(CHEMBL3359017)
Affinity DataIC50:  0.285nMAssay Description:Antagonist activity at maltose binding protein-tagged RBP4 (unknown origin) expressed in Escherichia coli assessed as inhibition of retinol-induced p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinol-binding protein 4(Homo sapiens (Human))
Albany Molecular Research

Curated by ChEMBL
LigandPNGBDBM50026253(CHEMBL3359014)
Affinity DataIC50:  0.294nMAssay Description:Antagonist activity at maltose binding protein-tagged RBP4 (unknown origin) expressed in Escherichia coli assessed as inhibition of retinol-induced p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PLK4(Homo sapiens (Human))
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50591932(CHEMBL5171469)
Affinity DataIC50:  0.300nMAssay Description:Inhibition of recombinant human PLK4 incubated for 60 mins by Lanthascreen Eu kinase binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetRetinol-binding protein 4(Homo sapiens (Human))
Albany Molecular Research

Curated by ChEMBL
LigandPNGBDBM50026256(CHEMBL3359019)
Affinity DataIC50:  0.340nMAssay Description:Antagonist activity at maltose binding protein-tagged RBP4 (unknown origin) expressed in Escherichia coli assessed as inhibition of retinol-induced p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinol-binding protein 4(Homo sapiens (Human))
Albany Molecular Research

Curated by ChEMBL
LigandPNGBDBM50026254(CHEMBL3359015)
Affinity DataIC50:  0.481nMAssay Description:Antagonist activity at maltose binding protein-tagged RBP4 (unknown origin) expressed in Escherichia coli assessed as inhibition of retinol-induced p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinol-binding protein 4(Homo sapiens (Human))
Albany Molecular Research

Curated by ChEMBL
LigandPNGBDBM50026251(CHEMBL3359005)
Affinity DataIC50:  0.554nMAssay Description:Antagonist activity at maltose binding protein-tagged RBP4 (unknown origin) expressed in Escherichia coli assessed as inhibition of retinol-induced p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PLK4(Homo sapiens (Human))
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50591954(CHEMBL5183346)
Affinity DataIC50:  0.700nMAssay Description:Inhibition of recombinant human PLK4 incubated for 60 mins by Lanthascreen Eu kinase binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetSerine/threonine-protein kinase PLK4(Homo sapiens (Human))
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50591948(CHEMBL5188129)
Affinity DataIC50:  0.700nMAssay Description:Inhibition of recombinant human PLK4 incubated for 60 mins by Lanthascreen Eu kinase binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetSerine/threonine-protein kinase PLK4(Homo sapiens (Human))
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50591926(CHEMBL5171233)
Affinity DataIC50:  0.700nMAssay Description:Inhibition of recombinant human PLK4 incubated for 60 mins by Lanthascreen Eu kinase binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetSerine/threonine-protein kinase PLK4(Homo sapiens (Human))
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50591931(CHEMBL5200865)
Affinity DataIC50:  0.800nMAssay Description:Inhibition of recombinant human PLK4 incubated for 60 mins by Lanthascreen Eu kinase binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetRetinol-binding protein 4(Homo sapiens (Human))
Albany Molecular Research

Curated by ChEMBL
LigandPNGBDBM50026244(CHEMBL3359028)
Affinity DataIC50:  0.829nMAssay Description:Antagonist activity at maltose binding protein-tagged RBP4 (unknown origin) expressed in Escherichia coli assessed as inhibition of retinol-induced p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PLK4(Homo sapiens (Human))
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50591925(CHEMBL5185324)
Affinity DataIC50:  1nMAssay Description:Inhibition of recombinant human PLK4 incubated for 60 mins by Lanthascreen Eu kinase binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetNT-3 growth factor receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50577766(CHEMBL4856292)
Affinity DataIC50:  1nMAssay Description:Inhibition of N-terminal GST-tagged human TRKC (456 to 825 residues) expressed in Sf21 using TK as substrate in presence of ATP measured after 40 min...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHigh affinity nerve growth factor receptor(Homo sapiens (Human))
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM158154(US10081622, Compound 11 | US10370379, Entrectinib ...)
Affinity DataIC50:  1nMAssay Description:Inhibition of TRKA (unknown origin) by radiometric assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase PLK4(Homo sapiens (Human))
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50591953(CHEMBL5194020)
Affinity DataIC50:  1.10nMAssay Description:Inhibition of recombinant human PLK4 incubated for 60 mins by Lanthascreen Eu kinase binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetSerine/threonine-protein kinase PLK4(Homo sapiens (Human))
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50437841(CHEMBL2407900)
Affinity DataIC50:  1.60nMAssay Description:Inhibition of PLK4 (unknown origin) by Lanthascreen Eu Kinase binding assayMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetRetinol-binding protein 4(Homo sapiens (Human))
Albany Molecular Research

Curated by ChEMBL
LigandPNGBDBM50026257(CHEMBL3359020)
Affinity DataIC50:  1.60nMAssay Description:Antagonist activity at maltose binding protein-tagged RBP4 (unknown origin) expressed in Escherichia coli assessed as inhibition of retinol-induced p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PLK4(Homo sapiens (Human))
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50591955(CHEMBL5191641)
Affinity DataIC50:  1.80nMAssay Description:Inhibition of recombinant human PLK4 incubated for 60 mins by Lanthascreen Eu kinase binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetNT-3 growth factor receptor(Homo sapiens (Human))TBA
LigandPNGBDBM136597(US10005783, 14 | US10047097, 14 | US10774085, Exam...)
Affinity DataIC50:  2.5nMAssay Description:Inhibition of TRKC (unknown origin) incubated for 40 mins in presence of ATP by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetNT-3 growth factor receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50598103(CHEMBL5174615)
Affinity DataIC50:  2.5nMAssay Description:Inhibition of N-terminal human TRKC (456 to 825 residues) expressed in baculovirus expression system using TK as substrate measured after 40 mins in ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetRetinol-binding protein 4(Homo sapiens (Human))
Albany Molecular Research

Curated by ChEMBL
LigandPNGBDBM50026250(CHEMBL3358470)
Affinity DataIC50:  2.70nMAssay Description:Antagonist activity at maltose binding protein-tagged RBP4 (unknown origin) expressed in Escherichia coli assessed as inhibition of retinol-induced p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PLK4(Homo sapiens (Human))
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50591939(CHEMBL5185225)
Affinity DataIC50:  2.70nMAssay Description:Inhibition of PLK4 (unknown origin) by Lanthascreen Eu Kinase binding assayMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetNT-3 growth factor receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50577766(CHEMBL4856292)
Affinity DataIC50:  2.70nMAssay Description:Inhibition of N-terminal human TRKC (456 to 825 residues) expressed in baculovirus expression system using TK as substrate measured after 40 mins in ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetSerine/threonine-protein kinase PLK4(Homo sapiens (Human))
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50591950(CHEMBL5176789)
Affinity DataIC50:  2.70nMAssay Description:Inhibition of recombinant human PLK4 incubated for 60 mins by Lanthascreen Eu kinase binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetBDNF/NT-3 growth factors receptor(Homo sapiens (Human))
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50577766(CHEMBL4856292)
Affinity DataIC50:  2.90nMAssay Description:Inhibition of N-terminal human TRKB (456 to 822 residues) expressed in baculovirus expression system using TK as substrate measured after 40 mins in ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetSerine/threonine-protein kinase PLK4(Homo sapiens (Human))
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50591939(CHEMBL5185225)
Affinity DataIC50:  3nMAssay Description:Inhibition of recombinant human PLK4 incubated for 60 mins by Lanthascreen Eu kinase binding assayMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetBDNF/NT-3 growth factors receptor(Homo sapiens (Human))
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM158154(US10081622, Compound 11 | US10370379, Entrectinib ...)
Affinity DataIC50:  3nMAssay Description:Inhibition of TRKB (unknown origin) by radiometric assayMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetHigh affinity nerve growth factor receptor(Homo sapiens (Human))
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM136597(US10005783, 14 | US10047097, 14 | US10774085, Exam...)
Affinity DataIC50:  3nMAssay Description:Inhibition of TRKA (unknown origin) using TK as substrate in presence of ATP incubated for 30 mins by HTRF KinEASE assayMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetRetinol-binding protein 4(Homo sapiens (Human))
Albany Molecular Research

Curated by ChEMBL
LigandPNGBDBM50026249(CHEMBL3358466)
Affinity DataIC50:  3.10nMAssay Description:Antagonist activity at maltose binding protein-tagged RBP4 (unknown origin) expressed in Escherichia coli assessed as inhibition of retinol-induced p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBDNF/NT-3 growth factors receptor(Homo sapiens (Human))
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM136597(US10005783, 14 | US10047097, 14 | US10774085, Exam...)
Affinity DataIC50:  3.30nMAssay Description:Inhibition of TRKB (unknown origin) incubated for 40 mins in presence of ATP by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetHigh affinity nerve growth factor receptor(Homo sapiens (Human))
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50577766(CHEMBL4856292)
Affinity DataIC50:  3.40nMAssay Description:Inhibition of N-terminal GST-tagged human TRKA (436 to 790 residues) expressed in baculovirus infected Sf21 cells using TK as substrate in presence o...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PLK4(Homo sapiens (Human))
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50591947(CHEMBL5190548)
Affinity DataIC50:  3.70nMAssay Description:Inhibition of recombinant human PLK4 incubated for 60 mins by Lanthascreen Eu kinase binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetSerine/threonine-protein kinase PLK4(Homo sapiens (Human))
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50591942(CHEMBL5207473)
Affinity DataIC50:  3.80nMAssay Description:Inhibition of recombinant human PLK4 incubated for 60 mins by Lanthascreen Eu kinase binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetRetinol-binding protein 4(Homo sapiens (Human))
Albany Molecular Research

Curated by ChEMBL
LigandPNGBDBM50026248(CHEMBL3358465)
Affinity DataIC50:  3.90nMAssay Description:Antagonist activity at maltose binding protein-tagged RBP4 (unknown origin) expressed in Escherichia coli assessed as inhibition of retinol-induced p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PLK4(Homo sapiens (Human))
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50591941(CHEMBL5201909)
Affinity DataIC50:  4nMAssay Description:Inhibition of recombinant human PLK4 incubated for 60 mins by Lanthascreen Eu kinase binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetHigh affinity nerve growth factor receptor(Homo sapiens (Human))
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50577766(CHEMBL4856292)
Affinity DataIC50:  4.10nMAssay Description:Inhibition of N-terminal human TRKA (436 to 790 residues) expressed in baculovirus expression system using TK as substrate measured after 30 mins in ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetNT-3 growth factor receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50598129(CHEMBL5196903)
Affinity DataIC50:  4.5nMAssay Description:Inhibition of N-terminal human TRKC (456 to 825 residues) expressed in baculovirus expression system using TK as substrate measured after 40 mins in ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetHigh affinity nerve growth factor receptor(Homo sapiens (Human))
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50598110(CHEMBL5175892)
Affinity DataIC50:  4.70nMAssay Description:Inhibition of N-terminal human TRKA (436 to 790 residues) expressed in baculovirus expression system using TK as substrate measured after 30 mins in ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetBDNF/NT-3 growth factors receptor(Homo sapiens (Human))
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50577766(CHEMBL4856292)
Affinity DataIC50:  4.70nMAssay Description:Inhibition of N-terminal GST-tagged human TRKB (456 to 822 residues) expressed in baculovirus infected Sf21 cells using TK as substrate in presence o...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
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