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Found 50 with Last Name = 'rizner' and Initial = 'tl'
Target11-beta-hydroxysteroid dehydrogenase 1(Homo sapiens (Human))
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50335199(3-Acetyl-7-(4-hydroxyphenyl)-2H-chromen-2-one | CH...)
Affinity DataKi:  143nMAssay Description:Displacement of [3H]estrone human recombinant 17beta-HSD1 expressed in Escherichia coli BL21 (DE3)-RIL by competitive inhibition assay in presence of...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Homo sapiens (Human))
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50335195(3-Acetyl-2-oxo-2H-chromen-7-yl trifluoromethanesul...)
Affinity DataKi:  173nMAssay Description:Displacement of [3H]estrone human recombinant 17beta-HSD1 expressed in Escherichia coli BL21 (DE3)-RIL by competitive inhibition assay in presence of...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Homo sapiens (Human))
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50335198(3-Acetyl-7-(4-methoxyphenyl)-2H-chromen-2-one | CH...)
Affinity DataKi:  585nMAssay Description:Displacement of [3H]estrone human recombinant 17beta-HSD1 expressed in Escherichia coli BL21 (DE3)-RIL by competitive inhibition assay in presence of...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Homo sapiens (Human))
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50335197(3-Acetyl-7-para-tolyl-2H-chromen-2-one | CHEMBL165...)
Affinity DataKi:  585nMAssay Description:Displacement of [3H]estrone human recombinant 17beta-HSD1 expressed in Escherichia coli BL21 (DE3)-RIL by competitive inhibition assay in presence of...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Homo sapiens (Human))
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50335196(3-Acetyl-7-phenyl-2H-chromen-2-one | CHEMBL1650699)
Affinity DataKi:  911nMAssay Description:Displacement of [3H]estrone human recombinant 17beta-HSD1 expressed in Escherichia coli BL21 (DE3)-RIL by competitive inhibition assay in presence of...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAldo-keto reductase family 1 member C3(Homo sapiens (Human))
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50293439(2-(4-chlorobenzylidene)cyclopentylmethyl ether | C...)
Affinity DataKi:  1.62E+4nMAssay Description:Inhibition of human recombinant GST-tagged AKR1C3 expressed in Escherichia coli BL21More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAldo-keto reductase family 1 member C1(Homo sapiens (Human))
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50293435(2-(4-Chlorobenzylidene)cyclopentanone | CHEMBL5623...)
Affinity DataKi:  1.72E+4nMAssay Description:Inhibition of human recombinant GST-tagged AKR1C1 expressed in Escherichia coli BL21More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAldo-keto reductase family 1 member C1(Homo sapiens (Human))
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50293435(2-(4-Chlorobenzylidene)cyclopentanone | CHEMBL5623...)
Affinity DataKi:  1.72E+4nMAssay Description:Inhibition of human recombinant GST-tagged AKR1C1 expressed in Escherichia coli BL21More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAldo-keto reductase family 1 member C3(Homo sapiens (Human))
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50293436(2-(4-chlorobenzylidene)cyclopentyl ethyl ether | C...)
Affinity DataKi:  2.05E+4nMAssay Description:Inhibition of human recombinant GST-tagged AKR1C3 expressed in Escherichia coli BL21More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAldo-keto reductase family 1 member C1(Homo sapiens (Human))
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50293436(2-(4-chlorobenzylidene)cyclopentyl ethyl ether | C...)
Affinity DataKi:  3.05E+4nMAssay Description:Inhibition of human recombinant GST-tagged AKR1C1 expressed in Escherichia coli BL21More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAldo-keto reductase family 1 member C1(Homo sapiens (Human))
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50293436(2-(4-chlorobenzylidene)cyclopentyl ethyl ether | C...)
Affinity DataKi:  3.05E+4nMAssay Description:Inhibition of human recombinant GST-tagged AKR1C1 expressed in Escherichia coli BL21More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAldo-keto reductase family 1 member C3(Homo sapiens (Human))
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50293435(2-(4-Chlorobenzylidene)cyclopentanone | CHEMBL5623...)
Affinity DataKi:  3.34E+4nMAssay Description:Inhibition of human recombinant GST-tagged AKR1C3 expressed in Escherichia coli BL21More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAldo-keto reductase family 1 member C1(Homo sapiens (Human))
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50293438(1-phenylcyclopentanecarboxylic acid | CHEMBL554543)
Affinity DataKi:  3.58E+4nMAssay Description:Inhibition of human recombinant GST-tagged AKR1C1 expressed in Escherichia coli BL21More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAldo-keto reductase family 1 member C1(Homo sapiens (Human))
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50293438(1-phenylcyclopentanecarboxylic acid | CHEMBL554543)
Affinity DataKi:  3.58E+4nMAssay Description:Inhibition of human recombinant GST-tagged AKR1C1 expressed in Escherichia coli BL21More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAldo-keto reductase family 1 member C1(Homo sapiens (Human))
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50293437(3-Phenylcyclopentanecarboxylic acid | CHEMBL554283)
Affinity DataKi:  4.85E+4nMAssay Description:Inhibition of human recombinant GST-tagged AKR1C1 expressed in Escherichia coli BL21More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAldo-keto reductase family 1 member C3(Homo sapiens (Human))
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50293437(3-Phenylcyclopentanecarboxylic acid | CHEMBL554283)
Affinity DataKi:  6.96E+4nMAssay Description:Inhibition of human recombinant GST-tagged AKR1C3 expressed in Escherichia coli BL21More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Homo sapiens (Human))
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50335200(3-Benzyl-2-(2-bromo-3,4,5-trimethoxy-phenyl)-8-hyd...)
Affinity DataIC50:  5nMAssay Description:Inhibition of 17beta-HSD1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Homo sapiens (Human))
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50335199(3-Acetyl-7-(4-hydroxyphenyl)-2H-chromen-2-one | CH...)
Affinity DataIC50:  270nMAssay Description:Displacement of [3H]estrone human recombinant 17beta-HSD1 expressed in Escherichia coli BL21 (DE3)-RIL by scintillation counting in presence of bacte...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Homo sapiens (Human))
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50335195(3-Acetyl-2-oxo-2H-chromen-7-yl trifluoromethanesul...)
Affinity DataIC50:  360nMAssay Description:Displacement of [3H]estrone human recombinant 17beta-HSD1 expressed in Escherichia coli BL21 (DE3)-RIL by scintillation counting in presence of bacte...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAldo-keto reductase family 1 member C3(Homo sapiens (Human))
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50339185((2S)-2-(6-methoxynaphthalen-2-yl)propanoic acid | ...)
Affinity DataIC50:  480nMAssay Description:Inhibition of recombinant human AKR1C3More data for this Ligand-Target Pair
TargetAldo-keto reductase family 1 member C3(Homo sapiens (Human))
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50060998(3-Phenoxy-benzoic acid | 3-phenoxybenzoic acid | C...)
Affinity DataIC50:  680nMAssay Description:Inhibition of recombinant human AKR1C3More data for this Ligand-Target Pair
Target17beta-hydroxysteroid dehydrogenase(Curvularia lunata)
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50149609((E)-3-Phenyl-acrylic acid benzyl ester | CHEMBL361...)
Affinity DataIC50:  700nMAssay Description:Inhibitory activity against 17 beta-hydroxysteroid dehydrogenase catalysed oxidation reactionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Homo sapiens (Human))
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50335198(3-Acetyl-7-(4-methoxyphenyl)-2H-chromen-2-one | CH...)
Affinity DataIC50:  1.14E+3nMAssay Description:Displacement of [3H]estrone human recombinant 17beta-HSD1 expressed in Escherichia coli BL21 (DE3)-RIL by scintillation counting in presence of bacte...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Homo sapiens (Human))
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50335197(3-Acetyl-7-para-tolyl-2H-chromen-2-one | CHEMBL165...)
Affinity DataIC50:  1.24E+3nMAssay Description:Displacement of [3H]estrone human recombinant 17beta-HSD1 expressed in Escherichia coli BL21 (DE3)-RIL by scintillation counting in presence of bacte...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Homo sapiens (Human))
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50335196(3-Acetyl-7-phenyl-2H-chromen-2-one | CHEMBL1650699)
Affinity DataIC50:  1.93E+3nMAssay Description:Displacement of [3H]estrone human recombinant 17beta-HSD1 expressed in Escherichia coli BL21 (DE3)-RIL by scintillation counting in presence of bacte...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAldo-keto reductase family 1 member C3(Homo sapiens (Human))
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50174201(ARTHROTEC | GP 45840 | SOLARAZE | Sodium; [2-(2,6-...)
Affinity DataIC50:  2.60E+3nMAssay Description:Inhibition of recombinant human AKR1C3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target17beta-hydroxysteroid dehydrogenase(Curvularia lunata)
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50149607(2-Oxo-2H-chromene-3-carboxylic acid benzyl ester |...)
Affinity DataIC50:  2.70E+3nMAssay Description:Inhibitory activity against 17 beta-hydroxysteroid dehydrogenase catalysed oxidation reactionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target17beta-hydroxysteroid dehydrogenase(Curvularia lunata)
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50149603((E)-3-Phenyl-acrylic acid 2-(1,3-dioxo-1,3-dihydro...)
Affinity DataIC50:  5.00E+3nMAssay Description:Inhibitory activity against 17 beta-hydroxysteroid dehydrogenase catalysed oxidation reactionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target17beta-hydroxysteroid dehydrogenase(Curvularia lunata)
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50149609((E)-3-Phenyl-acrylic acid benzyl ester | CHEMBL361...)
Affinity DataIC50:  7.00E+3nMAssay Description:Inhibitory activity against 17 beta-hydroxysteroid dehydrogenase catalysed reduction reactionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target17beta-hydroxysteroid dehydrogenase(Curvularia lunata)
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50149607(2-Oxo-2H-chromene-3-carboxylic acid benzyl ester |...)
Affinity DataIC50:  8.00E+3nMAssay Description:Inhibitory activity against 17 beta-hydroxysteroid dehydrogenase catalysed reduction reactionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target17beta-hydroxysteroid dehydrogenase(Curvularia lunata)
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50149614((E)-3-Phenyl-acrylic acid 1,3-dioxo-1,3-dihydro-is...)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibitory activity against 17 beta-hydroxysteroid dehydrogenase catalysed oxidation reactionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target17beta-hydroxysteroid dehydrogenase(Curvularia lunata)
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50149613((E)-3-Phenyl-acrylic acid naphthalen-1-yl ester | ...)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibitory activity against 17 beta-hydroxysteroid dehydrogenase catalysed oxidation reactionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAldo-keto reductase family 1 member C3(Homo sapiens (Human))
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50174204(2-[(2,2-diphenylacetyl)amino]benzoic acid | CHEMBL...)
Affinity DataIC50:  1.10E+4nMAssay Description:Inhibition of recombinant human AKR1C3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target17beta-hydroxysteroid dehydrogenase(Curvularia lunata)
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50149606((E)-3-Phenyl-acrylic acid 4-cyano-phenyl ester | C...)
Affinity DataIC50:  1.30E+4nMAssay Description:Inhibitory activity against 17 beta-hydroxysteroid dehydrogenase catalysed oxidation reactionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target17beta-hydroxysteroid dehydrogenase(Curvularia lunata)
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50149611((E)-3-Phenyl-acrylic acid 3,4,5-trimethoxy-benzyl ...)
Affinity DataIC50:  1.40E+4nMAssay Description:Inhibitory activity against 17 beta-hydroxysteroid dehydrogenase catalysed oxidation reactionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target17beta-hydroxysteroid dehydrogenase(Curvularia lunata)
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50149612((E)-3-Phenyl-acrylic acid phenyl ester | CHEMBL182...)
Affinity DataIC50:  2.60E+4nMAssay Description:Inhibitory activity against 17 beta-hydroxysteroid dehydrogenase catalysed oxidation reactionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAldo-keto reductase family 1 member C3(Homo sapiens (Human))
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50009859((+-)-2-(p-isobutylphenyl)propionic acid | (+-)-alp...)
Affinity DataIC50:  3.30E+4nMAssay Description:Inhibition of recombinant human AKR1C3More data for this Ligand-Target Pair
TargetAldo-keto reductase family 1 member C3(Homo sapiens (Human))
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50174203(2-(4-bromobenzoyl)benzoic acid | CHEMBL198745)
Affinity DataIC50:  3.90E+4nMAssay Description:Inhibition of recombinant human AKR1C3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAldo-keto reductase family 1 member C3(Homo sapiens (Human))
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50145840(2-(4-Methyl-benzoyl)-benzoic acid | 2-(4-methylben...)
Affinity DataIC50:  4.40E+4nMAssay Description:Inhibition of recombinant human AKR1C3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAldo-keto reductase family 1 member C3(Homo sapiens (Human))
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50174202(2-benzoylbenzoic acid | CHEMBL196812)
Affinity DataIC50:  7.00E+4nMAssay Description:Inhibition of recombinant human AKR1C3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target17beta-hydroxysteroid dehydrogenase(Curvularia lunata)
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50149603((E)-3-Phenyl-acrylic acid 2-(1,3-dioxo-1,3-dihydro...)
Affinity DataIC50:  9.00E+4nMAssay Description:Inhibitory activity against 17 beta-hydroxysteroid dehydrogenase catalysed reduction reactionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAldo-keto reductase family 1 member C1(Homo sapiens (Human))
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50293437(3-Phenylcyclopentanecarboxylic acid | CHEMBL554283)
Affinity DataIC50:  9.86E+4nMAssay Description:Inhibition of human recombinant GST-tagged AKR1C1 expressed in Escherichia coli BL21More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target17beta-hydroxysteroid dehydrogenase(Curvularia lunata)
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50149604((E)-3-Phenyl-acrylic acid 3-phenoxy-benzyl ester |...)
Affinity DataIC50:  1.30E+5nMAssay Description:Inhibitory activity against 17 beta-hydroxysteroid dehydrogenase catalysed oxidation reactionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target17beta-hydroxysteroid dehydrogenase(Curvularia lunata)
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50149610((E)-3-Phenyl-acrylic acid 3-methoxy-phenyl ester |...)
Affinity DataIC50:  1.35E+5nMAssay Description:Inhibitory activity against 17 beta-hydroxysteroid dehydrogenase catalysed oxidation reactionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAldo-keto reductase family 1 member C3(Homo sapiens (Human))
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50174205(4-methoxybenzophenone | CHEMBL198085 | cid_69146)
Affinity DataIC50:  1.80E+5nMAssay Description:Inhibition of recombinant human AKR1C3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target17beta-hydroxysteroid dehydrogenase(Curvularia lunata)
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50149605((E)-3-Phenyl-acrylic acid 4-octanoylamino-phenyl e...)
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibitory activity against 17 beta-hydroxysteroid dehydrogenase catalysed oxidation reactionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target17beta-hydroxysteroid dehydrogenase(Curvularia lunata)
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50149608((E)-3-Phenyl-acrylic acid 4-acetylamino-phenyl est...)
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibitory activity against 17 beta-hydroxysteroid dehydrogenase catalysed oxidation reactionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target17beta-hydroxysteroid dehydrogenase(Curvularia lunata)
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50149608((E)-3-Phenyl-acrylic acid 4-acetylamino-phenyl est...)
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibitory activity against 17 beta-hydroxysteroid dehydrogenase catalysed reduction reactionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target17beta-hydroxysteroid dehydrogenase(Curvularia lunata)
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50149612((E)-3-Phenyl-acrylic acid phenyl ester | CHEMBL182...)
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibitory activity against 17 beta-hydroxysteroid dehydrogenase catalysed reduction reactionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target17beta-hydroxysteroid dehydrogenase(Curvularia lunata)
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50149605((E)-3-Phenyl-acrylic acid 4-octanoylamino-phenyl e...)
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibitory activity against 17 beta-hydroxysteroid dehydrogenase catalysed reduction reactionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed