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Found 53 with Last Name = 'rodrigues' and Initial = 'da'
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Universidade Federal De Goi£S

Curated by ChEMBL
LigandPNGBDBM50001884(2-[4-(4-Methyl-benzyl)-piperazin-1-yl]-1-(2-methyl...)
Affinity DataKi:  20nMAssay Description:Displacement of [3H]-ketanserin from 5HT2A receptor in Wistar rat cortical membrane after 15 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
Universidade Federal De Goi£S

Curated by ChEMBL
LigandPNGBDBM50001884(2-[4-(4-Methyl-benzyl)-piperazin-1-yl]-1-(2-methyl...)
Affinity DataKi:  24nMAssay Description:Displacement of [3H]-mesulergine from human 5HT2C receptor after 60 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetAlpha-1B adrenergic receptor(Rattus norvegicus (rat))
Universidade Federal De Goi£S

Curated by ChEMBL
LigandPNGBDBM50001884(2-[4-(4-Methyl-benzyl)-piperazin-1-yl]-1-(2-methyl...)
Affinity DataKi:  29nMAssay Description:Displacement of [3H]-prazosin from alpha1B adrenergic receptor in Wistar rat liver membrane after 45 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Universidade Federal De Goi£S

Curated by ChEMBL
LigandPNGBDBM50429260(CHEMBL2333732)
Affinity DataKi:  34nMAssay Description:Displacement of [3H]-YM-09151-2 from human D4 dopamine receptor after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Universidade Federal De Goi£S

Curated by ChEMBL
LigandPNGBDBM50001884(2-[4-(4-Methyl-benzyl)-piperazin-1-yl]-1-(2-methyl...)
Affinity DataKi:  60nMAssay Description:Displacement of [3H]-YM-09151-2 from human D4 dopamine receptor after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetAlpha-2A adrenergic receptor [16-465](Rattus norvegicus (rat))
Universidade Federal De Goi£S

Curated by ChEMBL
LigandPNGBDBM50001884(2-[4-(4-Methyl-benzyl)-piperazin-1-yl]-1-(2-methyl...)
Affinity DataKi:  100nMAssay Description:Displacement of [3H]-RX821002 from alpha2A adrenergic receptor in Wistar rat cortical membrane after 45 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Universidade Federal De Goi£S

Curated by ChEMBL
LigandPNGBDBM50001884(2-[4-(4-Methyl-benzyl)-piperazin-1-yl]-1-(2-methyl...)
Affinity DataKi:  130nMAssay Description:Displacement of [3H]-YM-09151-2 from D2 dopamine receptor in Wistar rat brain striatal membrane after 60 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Universidade Federal De Goi£S

Curated by ChEMBL
LigandPNGBDBM50308002(1-[(1-(4-Chlorophenyl)-1H-pyrazol-4-yl)methyl]-4-p...)
Affinity DataKi:  170nMAssay Description:Displacement of [3H]-YM-09151-2 from human D4 dopamine receptor after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Universidade Federal De Goi£S

Curated by ChEMBL
LigandPNGBDBM50308002(1-[(1-(4-Chlorophenyl)-1H-pyrazol-4-yl)methyl]-4-p...)
Affinity DataKi:  210nMAssay Description:Displacement of [3H]-OH-8-DPAT from 5HT1A receptor in Wistar rat hippocampal membrane after 15 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Universidade Federal De Goi£S

Curated by ChEMBL
LigandPNGBDBM50001884(2-[4-(4-Methyl-benzyl)-piperazin-1-yl]-1-(2-methyl...)
Affinity DataKi:  260nMAssay Description:Displacement of [3H]-OH-8-DPAT from 5HT1A receptor in Wistar rat hippocampal membrane after 15 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Universidade Federal De Goi£S

Curated by ChEMBL
LigandPNGBDBM50308002(1-[(1-(4-Chlorophenyl)-1H-pyrazol-4-yl)methyl]-4-p...)
Affinity DataKi:  380nMAssay Description:Displacement of [3H]-YM-09151-2 from D2 dopamine receptor in Wistar rat brain striatal membrane after 60 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Universidade Federal De Goi£S

Curated by ChEMBL
LigandPNGBDBM50429260(CHEMBL2333732)
Affinity DataKi:  530nMAssay Description:Displacement of [3H]-YM-09151-2 from D2 dopamine receptor in Wistar rat brain striatal membrane after 60 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(Rattus norvegicus (rat))
Universidade Federal De Goi£S

Curated by ChEMBL
LigandPNGBDBM50429260(CHEMBL2333732)
Affinity DataKi:  1.15E+3nMAssay Description:Displacement of [3H]-prazosin from alpha1B adrenergic receptor in Wistar rat liver membrane after 45 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2A adrenergic receptor [16-465](Rattus norvegicus (rat))
Universidade Federal De Goi£S

Curated by ChEMBL
LigandPNGBDBM50308002(1-[(1-(4-Chlorophenyl)-1H-pyrazol-4-yl)methyl]-4-p...)
Affinity DataKi:  2.49E+3nMAssay Description:Displacement of [3H]-RX821002 from alpha2A adrenergic receptor in Wistar rat cortical membrane after 45 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(Rattus norvegicus (rat))
Universidade Federal De Goi£S

Curated by ChEMBL
LigandPNGBDBM50308002(1-[(1-(4-Chlorophenyl)-1H-pyrazol-4-yl)methyl]-4-p...)
Affinity DataKi:  3.00E+3nMAssay Description:Displacement of [3H]-prazosin from alpha1B adrenergic receptor in Wistar rat liver membrane after 45 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Universidade Federal De Goi£S

Curated by ChEMBL
LigandPNGBDBM50429260(CHEMBL2333732)
Affinity DataKi:  5.87E+3nMAssay Description:Displacement of [3H]-OH-8-DPAT from 5HT1A receptor in Wistar rat hippocampal membrane after 15 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2A adrenergic receptor [16-465](Rattus norvegicus (rat))
Universidade Federal De Goi£S

Curated by ChEMBL
LigandPNGBDBM50429260(CHEMBL2333732)
Affinity DataKi:  6.45E+3nMAssay Description:Displacement of [3H]-RX821002 from alpha2A adrenergic receptor in Wistar rat cortical membrane after 45 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Universidade Federal De Goi£S

Curated by ChEMBL
LigandPNGBDBM50308002(1-[(1-(4-Chlorophenyl)-1H-pyrazol-4-yl)methyl]-4-p...)
Affinity DataKi:  6.82E+3nMAssay Description:Displacement of [3H]-ketanserin from 5HT2A receptor in Wistar rat cortical membrane after 15 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Universidade Federal De Goi£S

Curated by ChEMBL
LigandPNGBDBM50429260(CHEMBL2333732)
Affinity DataKi:  8.22E+3nMAssay Description:Displacement of [3H]-ketanserin from 5HT2A receptor in Wistar rat cortical membrane after 15 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
Universidade Federal De Goi£S

Curated by ChEMBL
LigandPNGBDBM50308002(1-[(1-(4-Chlorophenyl)-1H-pyrazol-4-yl)methyl]-4-p...)
Affinity DataKi:  8.44E+3nMAssay Description:Displacement of [3H]-mesulergine from human 5HT2C receptor after 60 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
Universidade Federal De Goi£S

Curated by ChEMBL
LigandPNGBDBM50429260(CHEMBL2333732)
Affinity DataKi:  1.23E+4nMAssay Description:Displacement of [3H]-mesulergine from human 5HT2C receptor after 60 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Universidade Federal De Alfenas

Curated by ChEMBL
LigandPNGBDBM50005711(CHEBI:46024 | GNF-Pf-1011 | TRICHOSTATIN | Trichos...)
Affinity DataIC50:  8.5nMAssay Description:Inhibition of recombinant human HDAC1 by fluorimetryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 6(Homo sapiens (Human))
Universidade Federal De Alfenas

Curated by ChEMBL
LigandPNGBDBM50005711(CHEBI:46024 | GNF-Pf-1011 | TRICHOSTATIN | Trichos...)
Affinity DataIC50:  9nMAssay Description:Inhibition of recombinant human HDAC6 by fluorimetryMore data for this Ligand-Target Pair
TargetHistone deacetylase 6(Homo sapiens (Human))
Universidade Federal De Alfenas

Curated by ChEMBL
LigandPNGBDBM50146076(CHEMBL3764525)
Affinity DataIC50:  15nMAssay Description:Inhibition of recombinant human HDAC6 by fluorimetryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase(Rattus norvegicus)
Universidade Federal De Alfenas

Curated by ChEMBL
LigandPNGBDBM50146077(CHEMBL3763388)
Affinity DataIC50:  18nMAssay Description:Inhibition of HDAC in rat liver by fluorimetryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase(Rattus norvegicus)
Universidade Federal De Alfenas

Curated by ChEMBL
LigandPNGBDBM50146076(CHEMBL3764525)
Affinity DataIC50:  21nMAssay Description:Inhibition of HDAC in rat liver by fluorimetryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 6(Homo sapiens (Human))
Universidade Federal De Alfenas

Curated by ChEMBL
LigandPNGBDBM50146077(CHEMBL3763388)
Affinity DataIC50:  27nMAssay Description:Inhibition of recombinant human HDAC6 by fluorimetryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 2(Homo sapiens (Human))
Universidade Federal De Alfenas

Curated by ChEMBL
LigandPNGBDBM50005711(CHEBI:46024 | GNF-Pf-1011 | TRICHOSTATIN | Trichos...)
Affinity DataIC50:  52nMAssay Description:Inhibition of recombinant human HDAC2 by fluorimetryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 8(Homo sapiens (Human))
Universidade Federal De Alfenas

Curated by ChEMBL
LigandPNGBDBM50146080(CHEMBL3763386)
Affinity DataIC50:  54nMAssay Description:Inhibition of recombinant human HDAC8 by fluorimetryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 6(Homo sapiens (Human))
Universidade Federal De Alfenas

Curated by ChEMBL
LigandPNGBDBM50146079(CHEMBL3764728)
Affinity DataIC50:  56nMAssay Description:Inhibition of recombinant human HDAC6 by fluorimetryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 6(Homo sapiens (Human))
Universidade Federal De Alfenas

Curated by ChEMBL
LigandPNGBDBM50146080(CHEMBL3763386)
Affinity DataIC50:  97nMAssay Description:Inhibition of recombinant human HDAC6 by fluorimetryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 8(Homo sapiens (Human))
Universidade Federal De Alfenas

Curated by ChEMBL
LigandPNGBDBM50146079(CHEMBL3764728)
Affinity DataIC50:  110nMAssay Description:Inhibition of recombinant human HDAC8 by fluorimetryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 8(Homo sapiens (Human))
Universidade Federal De Alfenas

Curated by ChEMBL
LigandPNGBDBM50146077(CHEMBL3763388)
Affinity DataIC50:  130nMAssay Description:Inhibition of recombinant human HDAC8 by fluorimetryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 8(Homo sapiens (Human))
Universidade Federal De Alfenas

Curated by ChEMBL
LigandPNGBDBM50146076(CHEMBL3764525)
Affinity DataIC50:  230nMAssay Description:Inhibition of recombinant human HDAC8 by fluorimetryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(RAT)
National Institute For Science And Technology On Innovation On Neglected Diseases (Inct/Idn)

Curated by ChEMBL
LigandPNGBDBM50462906(CHEMBL3211778)
Affinity DataIC50:  350nMAssay Description:Agonist activity at endothelial M3 receptor in Wistar-Kyoto rat thoracic aortic rings assessed as inhibition of phenylephrine-induced contractionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 8(Homo sapiens (Human))
Universidade Federal De Alfenas

Curated by ChEMBL
LigandPNGBDBM50005711(CHEBI:46024 | GNF-Pf-1011 | TRICHOSTATIN | Trichos...)
Affinity DataIC50:  360nMAssay Description:Inhibition of recombinant human HDAC8 by fluorimetryMore data for this Ligand-Target Pair
TargetHistone deacetylase 6(Homo sapiens (Human))
Universidade Federal De Alfenas

Curated by ChEMBL
LigandPNGBDBM50146075(CHEMBL3765502)
Affinity DataIC50:  390nMAssay Description:Inhibition of recombinant human HDAC6 by fluorimetryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase(Rattus norvegicus)
Universidade Federal De Alfenas

Curated by ChEMBL
LigandPNGBDBM50146075(CHEMBL3765502)
Affinity DataIC50:  1.20E+3nMAssay Description:Inhibition of HDAC in rat liver by fluorimetryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 8(Homo sapiens (Human))
Universidade Federal De Alfenas

Curated by ChEMBL
LigandPNGBDBM50146078(CHEMBL3764442)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibition of recombinant human HDAC8 by fluorimetryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 8(Homo sapiens (Human))
Universidade Federal De Alfenas

Curated by ChEMBL
LigandPNGBDBM50146075(CHEMBL3765502)
Affinity DataIC50:  2.20E+3nMAssay Description:Inhibition of recombinant human HDAC8 by fluorimetryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 6(Homo sapiens (Human))
Universidade Federal De Alfenas

Curated by ChEMBL
LigandPNGBDBM50146078(CHEMBL3764442)
Affinity DataIC50:  2.50E+3nMAssay Description:Inhibition of recombinant human HDAC6 by fluorimetryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 2(Homo sapiens (Human))
Universidade Federal De Alfenas

Curated by ChEMBL
LigandPNGBDBM50146076(CHEMBL3764525)
Affinity DataIC50: >3.00E+3nMAssay Description:Inhibition of recombinant human HDAC2 by fluorimetryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 2(Homo sapiens (Human))
Universidade Federal De Alfenas

Curated by ChEMBL
LigandPNGBDBM50146077(CHEMBL3763388)
Affinity DataIC50: >3.00E+3nMAssay Description:Inhibition of recombinant human HDAC2 by fluorimetryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 2(Homo sapiens (Human))
Universidade Federal De Alfenas

Curated by ChEMBL
LigandPNGBDBM50146079(CHEMBL3764728)
Affinity DataIC50: >3.00E+3nMAssay Description:Inhibition of recombinant human HDAC2 by fluorimetryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 2(Homo sapiens (Human))
Universidade Federal De Alfenas

Curated by ChEMBL
LigandPNGBDBM50146080(CHEMBL3763386)
Affinity DataIC50: >3.00E+3nMAssay Description:Inhibition of recombinant human HDAC2 by fluorimetryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Universidade Federal De Alfenas

Curated by ChEMBL
LigandPNGBDBM50146076(CHEMBL3764525)
Affinity DataIC50: >3.00E+3nMAssay Description:Inhibition of recombinant human HDAC1 by fluorimetryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Universidade Federal De Alfenas

Curated by ChEMBL
LigandPNGBDBM50146077(CHEMBL3763388)
Affinity DataIC50: >3.00E+3nMAssay Description:Inhibition of recombinant human HDAC1 by fluorimetryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Universidade Federal De Alfenas

Curated by ChEMBL
LigandPNGBDBM50146079(CHEMBL3764728)
Affinity DataIC50: >3.00E+3nMAssay Description:Inhibition of recombinant human HDAC1 by fluorimetryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Universidade Federal De Alfenas

Curated by ChEMBL
LigandPNGBDBM50146080(CHEMBL3763386)
Affinity DataIC50: >3.00E+3nMAssay Description:Inhibition of recombinant human HDAC1 by fluorimetryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Universidade Federal De Alfenas

Curated by ChEMBL
LigandPNGBDBM50146075(CHEMBL3765502)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of recombinant human HDAC1 by fluorimetryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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