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Found 69 with Last Name = 'simonnet' and Initial = 'g'
TargetNeuropeptide FF receptor 2(RAT)
Cnrs

Curated by ChEMBL
LigandPNGBDBM50037567(2-[(Pyrrolidine-2-carbonyl)-amino]-pentanedioic ac...)
Affinity DataKi:  0.160nMAssay Description:Binding affinity for NPPF receptor in rat spinal cord membranes using the radioligand [125I]-[Tyr1]NPFFMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide FF receptor 2(RAT)
Cnrs

Curated by ChEMBL
LigandPNGBDBM50037568(2-{[1-(2-{2-[2-(2-Amino-3-(p-hydroxyphenyl)-propio...)
Affinity DataKi:  0.190nMAssay Description:Binding affinity for NPPF receptor in rat spinal cord membranes using the radioligand [125I]-[Tyr1]NPFFMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide FF receptor 2(RAT)
Cnrs

Curated by ChEMBL
LigandPNGBDBM50037559((S)-2-[((S)-1-{(S)-2-[(S)-2-((S)-2-Amino-4-methyl-...)
Affinity DataKi:  0.200nMAssay Description:Binding affinity for NPPF receptor in rat spinal cord membranes using the radioligand [125I]-[Tyr1]NPFFMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide FF receptor 2(RAT)
Cnrs

Curated by ChEMBL
LigandPNGBDBM50037575(2-Amino-pentanedioic acid 5-amide 1-{[1-(1-carbamo...)
Affinity DataKi:  0.200nMAssay Description:Binding affinity for NPPF receptor in rat spinal cord membranes using the radioligand [125I]-[Tyr1]NPFFMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide FF receptor 2(RAT)
Cnrs

Curated by ChEMBL
LigandPNGBDBM50037557(2-{[1-(2-{2-[2-(2-Amino-3-phenyl-propionylamino)-4...)
Affinity DataKi:  0.210nMAssay Description:Binding affinity for NPPF receptor in rat spinal cord membranes using the radioligand [125I]-[Tyr1]NPFFMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide FF receptor 2(RAT)
Cnrs

Curated by ChEMBL
LigandPNGBDBM50037572(2-{[1-(2-{2-[2-(2-Amino-3-(p-hydroxyphenyl)-propio...)
Affinity DataKi:  0.220nMAssay Description:Binding affinity for NPPF receptor in rat spinal cord membranes using the radioligand [125I]-[Tyr1]NPFFMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide FF receptor 1(Homo sapiens (Human))
University Of Strasbourg

Curated by ChEMBL
LigandPNGBDBM50402454(CHEMBL2208337)
Affinity DataKi:  0.320nMAssay Description:Displacement of [3H]FFRF-NH2 from human flag-tagged NPFF1 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide FF receptor 2(RAT)
Cnrs

Curated by ChEMBL
LigandPNGBDBM50037565((S)-2-({(S)-1-[(S)-2-((S)-2-Amino-3-phenyl-propion...)
Affinity DataKi:  0.430nMAssay Description:Binding affinity for NPPF receptor in rat spinal cord membranes using the radioligand [125I]-[Tyr1]NPFFMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide FF receptor 2(RAT)
Cnrs

Curated by ChEMBL
LigandPNGBDBM50037563(2-{[1-(2-{2-[2-(2-Amino-3-(p-hydroxyphenyl)-propio...)
Affinity DataKi:  0.5nMAssay Description:Binding affinity for NPPF receptor in rat spinal cord membranes using the radioligand [125I]-[Tyr1]NPFFMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide FF receptor 2(RAT)
Cnrs

Curated by ChEMBL
LigandPNGBDBM50037576(1-(2-{2-[2-(2-Amino-3-phenyl-propionylamino)-4-met...)
Affinity DataKi:  0.600nMAssay Description:Binding affinity for NPPF receptor in rat spinal cord membranes using the radioligand [125I]-[Tyr1]NPFFMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide FF receptor 1(Homo sapiens (Human))
University Of Strasbourg

Curated by ChEMBL
LigandPNGBDBM50402442(CHEMBL2208303)
Affinity DataKi:  0.800nMAssay Description:Displacement of [3H]FFRF-NH2 from human flag-tagged NPFF1 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide FF receptor 1(Homo sapiens (Human))
University Of Strasbourg

Curated by ChEMBL
LigandPNGBDBM50402459(CHEMBL2208301)
Affinity DataKi:  0.900nMAssay Description:Displacement of [3H]FFRF-NH2 from human flag-tagged NPFF1 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide FF receptor 2(RAT)
Cnrs

Curated by ChEMBL
LigandPNGBDBM50037564(2-{[1-(2-{2-[2-(2-Amino-3-(p-hydroxyphenyl)-propio...)
Affinity DataKi:  1nMAssay Description:Binding affinity for NPPF receptor in rat spinal cord membranes using the radioligand [125I]-[Tyr1]NPFFMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide FF receptor 2(RAT)
Cnrs

Curated by ChEMBL
LigandPNGBDBM50037569(2-(2-Amino-3-phenyl-propionylamino)-4-methyl-penta...)
Affinity DataKi:  1.20nMAssay Description:Binding affinity for NPPF receptor in rat spinal cord membranes using the radioligand [125I]-[Tyr1]NPFFMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide FF receptor 1(Homo sapiens (Human))
University Of Strasbourg

Curated by ChEMBL
LigandPNGBDBM50402453(CHEMBL2208338)
Affinity DataKi:  2nMAssay Description:Displacement of [3H]FFRF-NH2 from human flag-tagged NPFF1 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide FF receptor 1(Homo sapiens (Human))
University Of Strasbourg

Curated by ChEMBL
LigandPNGBDBM50402449(CHEMBL2208325)
Affinity DataKi:  2nMAssay Description:Displacement of [3H]FFRF-NH2 from human flag-tagged NPFF1 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide FF receptor 2(Homo sapiens (Human))
University Of Strasbourg

Curated by ChEMBL
LigandPNGBDBM50402444(CHEMBL2208319)
Affinity DataKi:  4nMAssay Description:Displacement of [3H]FFRF-NH2 from human flag-tagged NPFF2 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide FF receptor 2(Homo sapiens (Human))
University Of Strasbourg

Curated by ChEMBL
LigandPNGBDBM50402453(CHEMBL2208338)
Affinity DataKi:  4nMAssay Description:Displacement of [3H]FFRF-NH2 from human flag-tagged NPFF2 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide FF receptor 1(Homo sapiens (Human))
University Of Strasbourg

Curated by ChEMBL
LigandPNGBDBM50402452(CHEMBL2208320)
Affinity DataKi:  5nMAssay Description:Displacement of [3H]FFRF-NH2 from human flag-tagged NPFF1 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide FF receptor 1(Homo sapiens (Human))
University Of Strasbourg

Curated by ChEMBL
LigandPNGBDBM50402451(CHEMBL2208322)
Affinity DataKi:  6nMAssay Description:Displacement of [3H]FFRF-NH2 from human flag-tagged NPFF1 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide FF receptor 2(Homo sapiens (Human))
University Of Strasbourg

Curated by ChEMBL
LigandPNGBDBM50402451(CHEMBL2208322)
Affinity DataKi:  9nMAssay Description:Displacement of [3H]FFRF-NH2 from human flag-tagged NPFF2 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide FF receptor 2(RAT)
Cnrs

Curated by ChEMBL
LigandPNGBDBM50037558(2-{[1-(2-{2-[2-(2-Amino-3-phenyl-propionylamino)-4...)
Affinity DataKi:  10nMAssay Description:Binding affinity for NPPF receptor in rat spinal cord membranes using the radioligand [125I]-[Tyr1]NPFFMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide FF receptor 1(Homo sapiens (Human))
University Of Strasbourg

Curated by ChEMBL
LigandPNGBDBM50402444(CHEMBL2208319)
Affinity DataKi:  10nMAssay Description:Displacement of [3H]FFRF-NH2 from human flag-tagged NPFF1 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide FF receptor 1(Homo sapiens (Human))
University Of Strasbourg

Curated by ChEMBL
LigandPNGBDBM50402457(CHEMBL2208340)
Affinity DataKi:  11nMAssay Description:Displacement of [3H]FFRF-NH2 from human flag-tagged NPFF1 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide FF receptor 1(Homo sapiens (Human))
University Of Strasbourg

Curated by ChEMBL
LigandPNGBDBM50402443(CHEMBL2208299)
Affinity DataKi:  15nMAssay Description:Displacement of [3H]FFRF-NH2 from human flag-tagged NPFF1 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide FF receptor 2(RAT)
Cnrs

Curated by ChEMBL
LigandPNGBDBM50037573((S)-2-[((S)-Pyrrolidine-2-carbonyl)-amino]-pentane...)
Affinity DataKi:  15.5nMAssay Description:Binding affinity for NPPF receptor in rat spinal cord membranes using the radioligand [125I]-[Tyr1]NPFFMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide FF receptor 2(RAT)
Cnrs

Curated by ChEMBL
LigandPNGBDBM50037562((S)-2-{[(S)-1-((S)-2-Amino-4-carbamoyl-butyryl)-py...)
Affinity DataKi:  20.9nMAssay Description:Binding affinity for NPPF receptor in rat spinal cord membranes using the radioligand [125I]-[Tyr1]NPFFMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide FF receptor 2(Homo sapiens (Human))
University Of Strasbourg

Curated by ChEMBL
LigandPNGBDBM50402457(CHEMBL2208340)
Affinity DataKi:  22nMAssay Description:Displacement of [3H]FFRF-NH2 from human flag-tagged NPFF2 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide FF receptor 1(Homo sapiens (Human))
University Of Strasbourg

Curated by ChEMBL
LigandPNGBDBM50336912(Adamantane-1-carboxylic acid [(S)-1-((S)-1-carbamo...)
Affinity DataKi:  22nMAssay Description:Displacement of [3H]FFRF-NH2 from human flag-tagged NPFF1 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide FF receptor 1(Homo sapiens (Human))
University Of Strasbourg

Curated by ChEMBL
LigandPNGBDBM50402458(CHEMBL2208339)
Affinity DataKi:  23nMAssay Description:Displacement of [3H]FFRF-NH2 from human flag-tagged NPFF1 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide FF receptor 1(Homo sapiens (Human))
University Of Strasbourg

Curated by ChEMBL
LigandPNGBDBM50402440(CHEMBL2208305)
Affinity DataKi:  29nMAssay Description:Displacement of [3H]FFRF-NH2 from human flag-tagged NPFF1 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide FF receptor 2(RAT)
Cnrs

Curated by ChEMBL
LigandPNGBDBM50037561(2-{[1-(2-{2-[2-(2-Amino-3-(p-hydroxyphenyl)-propio...)
Affinity DataKi:  30nMAssay Description:Binding affinity for NPPF receptor in rat spinal cord membranes using the radioligand [125I]-[Tyr1]NPFFMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide FF receptor 2(RAT)
Cnrs

Curated by ChEMBL
LigandPNGBDBM50037570((S)-2-[((R)-1-{(S)-2-[(S)-2-((S)-2-Amino-4-methyl-...)
Affinity DataKi:  33nMAssay Description:Binding affinity for NPPF receptor in rat spinal cord membranes using the radioligand [125I]-[Tyr1]NPFFMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide FF receptor 1(Homo sapiens (Human))
University Of Strasbourg

Curated by ChEMBL
LigandPNGBDBM50402446(CHEMBL2208316)
Affinity DataKi:  35nMAssay Description:Displacement of [3H]FFRF-NH2 from human flag-tagged NPFF1 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide FF receptor 2(Homo sapiens (Human))
University Of Strasbourg

Curated by ChEMBL
LigandPNGBDBM50336912(Adamantane-1-carboxylic acid [(S)-1-((S)-1-carbamo...)
Affinity DataKi:  43nMAssay Description:Displacement of [3H]FFRF-NH2 from human flag-tagged NPFF2 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide FF receptor 2(RAT)
Cnrs

Curated by ChEMBL
LigandPNGBDBM50037560((S)-2-({(R)-1-[(S)-2-((S)-2-Amino-3-phenyl-propion...)
Affinity DataKi:  45nMAssay Description:Binding affinity for NPPF receptor in rat spinal cord membranes using the radioligand [125I]-[Tyr1]NPFFMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide FF receptor 2(Homo sapiens (Human))
University Of Strasbourg

Curated by ChEMBL
LigandPNGBDBM50402447(CHEMBL2208312)
Affinity DataKi:  47nMAssay Description:Displacement of [3H]FFRF-NH2 from human flag-tagged NPFF2 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide FF receptor 1(Homo sapiens (Human))
University Of Strasbourg

Curated by ChEMBL
LigandPNGBDBM50402438(CHEMBL2208307)
Affinity DataKi:  51nMAssay Description:Displacement of [3H]FFRF-NH2 from human flag-tagged NPFF1 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide FF receptor 2(RAT)
Cnrs

Curated by ChEMBL
LigandPNGBDBM50037566((S)-2-{[(R)-1-((S)-2-Amino-4-carbamoyl-butyryl)-py...)
Affinity DataKi:  64nMAssay Description:Binding affinity for NPPF receptor in rat spinal cord membranes using the radioligand [125I]-[Tyr1]NPFFMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide FF receptor 1(Homo sapiens (Human))
University Of Strasbourg

Curated by ChEMBL
LigandPNGBDBM50402441(CHEMBL2208304)
Affinity DataKi:  84nMAssay Description:Displacement of [3H]FFRF-NH2 from human flag-tagged NPFF1 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide FF receptor 1(Homo sapiens (Human))
University Of Strasbourg

Curated by ChEMBL
LigandPNGBDBM50402437(CHEMBL2208294)
Affinity DataKi:  87nMAssay Description:Displacement of [3H]FFRF-NH2 from human flag-tagged NPFF1 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide FF receptor 2(Homo sapiens (Human))
University Of Strasbourg

Curated by ChEMBL
LigandPNGBDBM50402458(CHEMBL2208339)
Affinity DataKi:  92nMAssay Description:Displacement of [3H]FFRF-NH2 from human flag-tagged NPFF2 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide FF receptor 2(RAT)
Cnrs

Curated by ChEMBL
LigandPNGBDBM50037574((S)-2-[((R)-Pyrrolidine-2-carbonyl)-amino]-pentane...)
Affinity DataKi:  94nMAssay Description:Binding affinity for NPPF receptor in rat spinal cord membranes using the radioligand [125I]-[Tyr1]NPFFMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide FF receptor 2(Homo sapiens (Human))
University Of Strasbourg

Curated by ChEMBL
LigandPNGBDBM50402449(CHEMBL2208325)
Affinity DataKi:  94nMAssay Description:Displacement of [3H]FFRF-NH2 from human flag-tagged NPFF2 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide FF receptor 1(Homo sapiens (Human))
University Of Strasbourg

Curated by ChEMBL
LigandPNGBDBM50402455(CHEMBL2208334)
Affinity DataKi:  106nMAssay Description:Displacement of [3H]FFRF-NH2 from human flag-tagged NPFF1 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide FF receptor 1(Homo sapiens (Human))
University Of Strasbourg

Curated by ChEMBL
LigandPNGBDBM50402450(CHEMBL2208323)
Affinity DataKi:  110nMAssay Description:Displacement of [3H]FFRF-NH2 from human flag-tagged NPFF1 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide FF receptor 1(Homo sapiens (Human))
University Of Strasbourg

Curated by ChEMBL
LigandPNGBDBM50402439(CHEMBL2208306)
Affinity DataKi:  114nMAssay Description:Displacement of [3H]FFRF-NH2 from human flag-tagged NPFF1 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide FF receptor 2(Homo sapiens (Human))
University Of Strasbourg

Curated by ChEMBL
LigandPNGBDBM50402442(CHEMBL2208303)
Affinity DataKi:  117nMAssay Description:Displacement of [3H]FFRF-NH2 from human flag-tagged NPFF2 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide FF receptor 1(Homo sapiens (Human))
University Of Strasbourg

Curated by ChEMBL
LigandPNGBDBM50402447(CHEMBL2208312)
Affinity DataKi:  121nMAssay Description:Displacement of [3H]FFRF-NH2 from human flag-tagged NPFF1 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide FF receptor 2(Homo sapiens (Human))
University Of Strasbourg

Curated by ChEMBL
LigandPNGBDBM50402436(CHEMBL2208296)
Affinity DataKi:  136nMAssay Description:Displacement of [3H]FFRF-NH2 from human flag-tagged NPFF2 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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