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Found 92 with Last Name = 'thorberg' and Initial = 'so'
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Preclinical R & D, Astra Arcus

Curated by PDSP Ki Database
LigandPNGBDBM86708(CAS_146714-97-8 | CHEMBL31354 | CHEMBL514874 | CHE...)
Affinity DataKi:  0.240nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Preclinical R & D, Astra Arcus

Curated by PDSP Ki Database
LigandPNGBDBM50090771((R)-1-[3-(Isopropyl-propyl-amino)-chroman-5-yl]-et...)
Affinity DataKi:  0.300nMAssay Description:In vitro binding affinity at 5-HT1A receptors assayed by displacement of [3H]-8-OH-DPAT from 5-hydroxytryptamine 1A receptor in rat hippocampal membr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Preclinical R & D, Astra Arcus

Curated by PDSP Ki Database
LigandPNGBDBM50090762((R)-3-(Isopropyl-propyl-amino)-chroman-5-carboxyli...)
Affinity DataKi:  0.320nMAssay Description:In vitro binding affinity at 5-HT1A receptors assayed by displacement of [3H]-8-OH-DPAT from 5-hydroxytryptamine 1A receptor in rat hippocampal membr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Preclinical R & D, Astra Arcus

Curated by PDSP Ki Database
LigandPNGBDBM50090763((R)-3-{[4-(7,9-Dioxo-8-aza-spiro[4.5]dec-8-yl)-but...)
Affinity DataKi:  0.340nMAssay Description:In vitro binding affinity at 5-HT1A receptors assayed by displacement of [3H]-8-OH-DPAT from 5-hydroxytryptamine 1A receptor in rat hippocampal membr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Preclinical R & D, Astra Arcus

Curated by PDSP Ki Database
LigandPNGBDBM50090756((R)-3-(Cyclopentyl-propyl-amino)-chroman-5-carboxy...)
Affinity DataKi:  0.410nMAssay Description:In vitro binding affinity at 5-HT1A receptors assayed by displacement of [3H]-8-OH-DPAT from 5-hydroxytryptamine 1A receptor in rat hippocampal membr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Preclinical R & D, Astra Arcus

Curated by PDSP Ki Database
LigandPNGBDBM50090764((R)-3-(Isopropyl-propyl-amino)-chroman-5-carboxyli...)
Affinity DataKi:  0.480nMAssay Description:In vitro binding affinity at 5-HT1A receptors assayed by displacement of [3H]-8-OH-DPAT from 5-hydroxytryptamine 1A receptor in rat hippocampal membr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Preclinical R & D, Astra Arcus

Curated by PDSP Ki Database
LigandPNGBDBM85190(CAS_3055171 | NAD-299 | NSC_3055171)
Affinity DataKi:  0.590nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Preclinical R & D, Astra Arcus

Curated by PDSP Ki Database
LigandPNGBDBM50090772((R)-3-(Isobutyl-propyl-amino)-chroman-5-carboxylic...)
Affinity DataKi:  2.37nMAssay Description:In vitro binding affinity at 5-HT1A receptors assayed by displacement of [3H]-8-OH-DPAT from 5-hydroxytryptamine 1A receptor in rat hippocampal membr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Preclinical R & D, Astra Arcus

Curated by PDSP Ki Database
LigandPNGBDBM50090770((R)-Isopropyl-(5-methoxy-chroman-3-yl)-propyl-amin...)
Affinity DataKi:  3.10nMAssay Description:In vitro binding affinity at 5-HT1A receptor by measuring its ability to displace [3H]-8-OH-DPAT from 5-hydroxytryptamine 1A receptor in rat hippocam...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Preclinical R & D, Astra Arcus

Curated by PDSP Ki Database
LigandPNGBDBM50090771((R)-1-[3-(Isopropyl-propyl-amino)-chroman-5-yl]-et...)
Affinity DataKi:  11.9nMAssay Description:In vitro binding affinity at 5-HT1A receptors assayed by displacement of [3H]-8-OH-DPAT from 5-hydroxytryptamine 1A receptor in rat hippocampal membr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Preclinical R & D, Astra Arcus

Curated by PDSP Ki Database
LigandPNGBDBM50090759((R)-3-Dipropylamino-chroman-5-carboxylic acid isop...)
Affinity DataKi:  14nMAssay Description:In vitro binding affinity at 5-HT1A receptors assayed by displacement of [3H]-8-OH-DPAT from 5-hydroxytryptamine 1A receptor in rat hippocampal membr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Preclinical R & D, Astra Arcus

Curated by PDSP Ki Database
LigandPNGBDBM50090761((R)-3-(Cyclopentyl-propyl-amino)-chroman-5-carboxy...)
Affinity DataKi:  18.5nMAssay Description:In vitro binding affinity at 5-HT1A receptors assayed by displacement of [3H]-8-OH-DPAT from 5-hydroxytryptamine 1A receptor in rat hippocampal membr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Preclinical R & D, Astra Arcus

Curated by PDSP Ki Database
LigandPNGBDBM86708(CAS_146714-97-8 | CHEMBL31354 | CHEMBL514874 | CHE...)
Affinity DataKi:  45nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
Target5-hydroxytryptamine receptor 1B(Rattus norvegicus (Rat))
Astra Arcus

Curated by ChEMBL
LigandPNGBDBM50369356(CHEMBL1744087)
Affinity DataKi:  47nMAssay Description:Binding affinity against 5-hydroxytryptamine 1B receptor in membranes of Rat cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1B(Rattus norvegicus (Rat))
Astra Arcus

Curated by ChEMBL
LigandPNGBDBM50369357(CHEMBL1201939)
Affinity DataKi:  60nMAssay Description:Binding affinity against 5-hydroxytryptamine 1B receptor in membranes of Rat cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Preclinical R & D, Astra Arcus

Curated by PDSP Ki Database
LigandPNGBDBM50090759((R)-3-Dipropylamino-chroman-5-carboxylic acid isop...)
Affinity DataKi:  64nMAssay Description:In vitro binding affinity at 5-HT1A receptor by measuring its ability to displace [3H]-8-OH-DPAT from 5-hydroxytryptamine 1A receptor in rat hippocam...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Preclinical R & D, Astra Arcus

Curated by PDSP Ki Database
LigandPNGBDBM86708(CAS_146714-97-8 | CHEMBL31354 | CHEMBL514874 | CHE...)
Affinity DataKi:  67nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Preclinical R & D, Astra Arcus

Curated by PDSP Ki Database
LigandPNGBDBM86708(CAS_146714-97-8 | CHEMBL31354 | CHEMBL514874 | CHE...)
Affinity DataKi:  79nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Preclinical R & D, Astra Arcus

Curated by PDSP Ki Database
LigandPNGBDBM50090754((R)-3-Propylamino-chroman-5-carboxylic acid amide ...)
Affinity DataKi:  98.4nMAssay Description:In vitro binding affinity at 5-HT1A receptors assayed by displacement of [3H]-8-OH-DPAT from 5-hydroxytryptamine 1A receptor in rat hippocampal membr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Preclinical R & D, Astra Arcus

Curated by PDSP Ki Database
LigandPNGBDBM50090770((R)-Isopropyl-(5-methoxy-chroman-3-yl)-propyl-amin...)
Affinity DataKi:  134nMAssay Description:In vitro binding affinity at 5-HT1A receptor by measuring its ability to displace [3H]-8-OH-DPAT from 5-hydroxytryptamine 1A receptor in rat hippocam...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1B(Rattus norvegicus (Rat))
Astra Arcus

Curated by ChEMBL
LigandPNGBDBM50064466(CHEMBL58961 | Morpholin-4-yl-[8-(morpholin-2-ylmet...)
Affinity DataKi:  240nMAssay Description:Binding affinity against 5-hydroxytryptamine 1B receptor in membranes of Rat cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1B(Rattus norvegicus (Rat))
Astra Arcus

Curated by ChEMBL
LigandPNGBDBM50064462(8-(Morpholin-2-ylmethoxy)-2H-chromene-3-carbonitri...)
Affinity DataKi:  250nMAssay Description:Binding affinity against 5-hydroxytryptamine 1B receptor in membranes of Rat cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Preclinical R & D, Astra Arcus

Curated by PDSP Ki Database
LigandPNGBDBM85190(CAS_3055171 | NAD-299 | NSC_3055171)
Affinity DataKi:  260nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
Target5-hydroxytryptamine receptor 1B(Rattus norvegicus (Rat))
Astra Arcus

Curated by ChEMBL
LigandPNGBDBM50369355(CHEMBL1202783)
Affinity DataKi:  275nMAssay Description:Binding affinity against 5-hydroxytryptamine 1B receptor in membranes of Rat cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(Rattus norvegicus)
Preclinical R & D, Astra Arcus

Curated by PDSP Ki Database
LigandPNGBDBM85190(CAS_3055171 | NAD-299 | NSC_3055171)
Affinity DataKi:  340nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Preclinical R & D, Astra Arcus

Curated by PDSP Ki Database
LigandPNGBDBM50090757((R)-3-Isopropylamino-chroman-5-carboxylic acid ami...)
Affinity DataKi:  397nMAssay Description:In vitro binding affinity at 5-HT1A receptors assayed by displacement of [3H]-8-OH-DPAT from 5-hydroxytryptamine 1A receptor in rat hippocampal membr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1B(Rattus norvegicus (Rat))
Astra Arcus

Curated by ChEMBL
LigandPNGBDBM50064464(5-(Morpholin-2-ylmethoxy)-3,4-dihydro-naphthalene-...)
Affinity DataKi:  445nMAssay Description:Binding affinity against 5-hydroxytryptamine 1B receptor in membranes of Rat cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2C adrenergic receptor(RAT)
Preclinical R & D, Astra Arcus

Curated by PDSP Ki Database
LigandPNGBDBM86708(CAS_146714-97-8 | CHEMBL31354 | CHEMBL514874 | CHE...)
Affinity DataKi:  1.00E+3nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Preclinical R & D, Astra Arcus

Curated by PDSP Ki Database
LigandPNGBDBM85190(CAS_3055171 | NAD-299 | NSC_3055171)
Affinity DataKi:  1.00E+3nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAlpha-2C adrenergic receptor(RAT)
Preclinical R & D, Astra Arcus

Curated by PDSP Ki Database
LigandPNGBDBM85190(CAS_3055171 | NAD-299 | NSC_3055171)
Affinity DataKi:  1.00E+3nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Preclinical R & D, Astra Arcus

Curated by PDSP Ki Database
LigandPNGBDBM50090754((R)-3-Propylamino-chroman-5-carboxylic acid amide ...)
Affinity DataKi: >1.00E+3nMAssay Description:In vitro binding affinity at human cloned Dopamine receptor D2A measured by ability to displace [3H]-raclopride from D2A receptor expressed in mouse ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(RAT)
Astrazeneca R&D SöDertäLje

Curated by ChEMBL
LigandPNGBDBM50090759((R)-3-Dipropylamino-chroman-5-carboxylic acid isop...)
Affinity DataKi: >1.00E+3nMAssay Description:In vitro binding affinity at D1 receptor by measuring its ability to displace [3H]-SCH-23,390 from Dopamine receptor D1 in rat striatumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Preclinical R & D, Astra Arcus

Curated by PDSP Ki Database
LigandPNGBDBM50090758((R)-3-(Cyclopentyl-propyl-amino)-chroman-5-carboxy...)
Affinity DataKi: >1.00E+3nMAssay Description:In vitro binding affinity at human cloned Dopamine receptor D2A measured by ability to displace [3H]-raclopride from D2A receptor expressed in mouse ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Preclinical R & D, Astra Arcus

Curated by PDSP Ki Database
LigandPNGBDBM85190(CAS_3055171 | NAD-299 | NSC_3055171)
Affinity DataKi:  1.00E+3nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetD(1A) dopamine receptor(RAT)
Astrazeneca R&D SöDertäLje

Curated by ChEMBL
LigandPNGBDBM86708(CAS_146714-97-8 | CHEMBL31354 | CHEMBL514874 | CHE...)
Affinity DataKi:  1.00E+3nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetD(1A) dopamine receptor(RAT)
Astrazeneca R&D SöDertäLje

Curated by ChEMBL
LigandPNGBDBM85190(CAS_3055171 | NAD-299 | NSC_3055171)
Affinity DataKi:  1.00E+3nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMuscarinic acetylcholine receptor M2(RAT)
Preclinical R & D, Astra Arcus

Curated by PDSP Ki Database
LigandPNGBDBM86708(CAS_146714-97-8 | CHEMBL31354 | CHEMBL514874 | CHE...)
Affinity DataKi:  1.00E+3nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetBeta-2 adrenergic receptor(Rattus norvegicus)
Preclinical R & D, Astra Arcus

Curated by PDSP Ki Database
LigandPNGBDBM86708(CAS_146714-97-8 | CHEMBL31354 | CHEMBL514874 | CHE...)
Affinity DataKi:  1.00E+3nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMuscarinic acetylcholine receptor M2(RAT)
Preclinical R & D, Astra Arcus

Curated by PDSP Ki Database
LigandPNGBDBM85190(CAS_3055171 | NAD-299 | NSC_3055171)
Affinity DataKi:  1.00E+3nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Astrazeneca R&D SöDertäLje

Curated by ChEMBL
LigandPNGBDBM50090764((R)-3-(Isopropyl-propyl-amino)-chroman-5-carboxyli...)
Affinity DataKi: >1.00E+3nMAssay Description:In vitro binding affinity at 5-hydroxytryptamine 2A receptor by displacement of [3H]-ketanserin from rat cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(RAT)
Astra Arcus

Curated by ChEMBL
LigandPNGBDBM50369356(CHEMBL1744087)
Affinity DataKi: >1.00E+3nMAssay Description:Binding affinity against Muscarinic acetylcholine receptor using [3H]QNB as the radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Astrazeneca R&D SöDertäLje

Curated by ChEMBL
LigandPNGBDBM50090754((R)-3-Propylamino-chroman-5-carboxylic acid amide ...)
Affinity DataKi: >1.00E+3nMAssay Description:In vitro binding affinity at 5-hydroxytryptamine 2A receptor by displacement of [3H]-ketanserin from rat cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Astrazeneca R&D SöDertäLje

Curated by ChEMBL
LigandPNGBDBM50090759((R)-3-Dipropylamino-chroman-5-carboxylic acid isop...)
Affinity DataKi: >1.00E+3nMAssay Description:In vitro binding affinity at 5-hydroxytryptamine 2A receptor by displacement of [3H]-ketanserin from rat cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(RAT)
Astrazeneca R&D SöDertäLje

Curated by ChEMBL
LigandPNGBDBM50090754((R)-3-Propylamino-chroman-5-carboxylic acid amide ...)
Affinity DataKi: >1.00E+3nMAssay Description:In vitro binding affinity at D1 receptor by measuring its ability to displace [3H]-SCH-23,390 from Dopamine receptor D1 in rat striatumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Preclinical R & D, Astra Arcus

Curated by PDSP Ki Database
LigandPNGBDBM50090759((R)-3-Dipropylamino-chroman-5-carboxylic acid isop...)
Affinity DataKi: >1.00E+3nMAssay Description:In vitro binding affinity at human cloned Dopamine receptor D2A measured by ability to displace [3H]-raclopride from D2A receptor expressed in mouse ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Astrazeneca R&D SöDertäLje

Curated by ChEMBL
LigandPNGBDBM50090758((R)-3-(Cyclopentyl-propyl-amino)-chroman-5-carboxy...)
Affinity DataKi: >1.00E+3nMAssay Description:In vitro binding affinity at 5-hydroxytryptamine 2A receptor by displacement of [3H]-ketanserin from rat cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(RAT)
Astrazeneca R&D SöDertäLje

Curated by ChEMBL
LigandPNGBDBM50090764((R)-3-(Isopropyl-propyl-amino)-chroman-5-carboxyli...)
Affinity DataKi: >1.00E+3nMAssay Description:In vitro binding affinity at D1 receptor by measuring its ability to displace [3H]-SCH-23,390 from Dopamine receptor D1 in rat striatumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Preclinical R & D, Astra Arcus

Curated by PDSP Ki Database
LigandPNGBDBM50090757((R)-3-Isopropylamino-chroman-5-carboxylic acid ami...)
Affinity DataKi: >1.00E+3nMAssay Description:In vitro binding affinity at human cloned Dopamine receptor D2A measured by ability to displace [3H]-raclopride from D2A receptor expressed in mouse ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Astrazeneca R&D SöDertäLje

Curated by ChEMBL
LigandPNGBDBM50090757((R)-3-Isopropylamino-chroman-5-carboxylic acid ami...)
Affinity DataKi: >1.00E+3nMAssay Description:In vitro binding affinity at 5-hydroxytryptamine 2A receptor by displacement of [3H]-ketanserin from rat cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(RAT)
Astrazeneca R&D SöDertäLje

Curated by ChEMBL
LigandPNGBDBM50090757((R)-3-Isopropylamino-chroman-5-carboxylic acid ami...)
Affinity DataKi: >1.00E+3nMAssay Description:In vitro binding affinity at D1 receptor by measuring its ability to displace [3H]-SCH-23,390 from Dopamine receptor D1 in rat striatumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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