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Found 75 with Last Name = 'townsend' and Initial = 'lb'
TargetPurine nucleoside phosphorylase(Homo sapiens (Human))
National Defense Medical Center

Curated by ChEMBL
LigandPNGBDBM50005799(2,8-Diamino-9-benzyl-1,9-dihydro-purin-6-one | CHE...)
Affinity DataKi:  200nMAssay Description:PNP activity in human RBCMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPurine nucleoside phosphorylase(Homo sapiens (Human))
National Defense Medical Center

Curated by ChEMBL
LigandPNGBDBM50368825(CHEMBL603291)
Affinity DataKi:  450nMAssay Description:PNP activity in human RBCMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPurine nucleoside phosphorylase(Homo sapiens (Human))
National Defense Medical Center

Curated by ChEMBL
LigandPNGBDBM50022243(2,8-Diamino-1,9-dihydro-purin-6-one | 8-AMINOGUANI...)
Affinity DataKi:  800nMAssay Description:PNP activity in human RBCMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPurine nucleoside phosphorylase(Homo sapiens (Human))
National Defense Medical Center

Curated by ChEMBL
LigandPNGBDBM50368823(CHEMBL606329)
Affinity DataKi:  7.00E+3nMAssay Description:PNP activity in human RBCMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPurine nucleoside phosphorylase(Homo sapiens (Human))
National Defense Medical Center

Curated by ChEMBL
LigandPNGBDBM50404028(CHEMBL2021376)
Affinity DataKi:  7.00E+3nMAssay Description:Compound was evaluated for the inhibitory activity against PNP activity in dialyzed extracts from human erythrocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPurine nucleoside phosphorylase(Homo sapiens (Human))
National Defense Medical Center

Curated by ChEMBL
LigandPNGBDBM50046864(6-(2,8-Diamino-6-oxo-1,6-dihydro-purin-9-yl)-hexan...)
Affinity DataKi:  1.00E+4nMAssay Description:Compound was evaluated for the inhibitory activity against PNP activity in dialyzed extracts from human erythrocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPurine nucleoside phosphorylase(Homo sapiens (Human))
National Defense Medical Center

Curated by ChEMBL
LigandPNGBDBM50046869(2,8-Diamino-9-hexyl-1,9-dihydro-purin-6-one | CHEM...)
Affinity DataKi:  1.24E+4nMAssay Description:Compound was evaluated for the inhibitory activity against PNP activity in dialyzed extracts from human erythrocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPurine nucleoside phosphorylase(Homo sapiens (Human))
National Defense Medical Center

Curated by ChEMBL
LigandPNGBDBM50207253(2,8-Diamino-9-(2-hydroxy-ethoxymethyl)-1,9-dihydro...)
Affinity DataKi:  1.34E+4nMAssay Description:PNP activity in human RBCMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPurine nucleoside phosphorylase(Homo sapiens (Human))
National Defense Medical Center

Curated by ChEMBL
LigandPNGBDBM50046867(2-Amino-9-(2-iodo-ethoxymethyl)-1,9-dihydro-purin-...)
Affinity DataKi:  1.50E+4nMAssay Description:PNP activity in human RBCMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPurine nucleoside phosphorylase(Homo sapiens (Human))
National Defense Medical Center

Curated by ChEMBL
LigandPNGBDBM50207401(2-Amino-8-bromo-9-(2-hydroxy-ethoxymethyl)-1,9-dih...)
Affinity DataKi:  1.87E+4nMAssay Description:PNP activity in human RBCMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPurine nucleoside phosphorylase(Homo sapiens (Human))
National Defense Medical Center

Curated by ChEMBL
LigandPNGBDBM50046868(2,8-Diamino-9-(2-iodo-ethoxymethyl)-1,9-dihydro-pu...)
Affinity DataKi:  2.30E+4nMAssay Description:PNP activity in human RBCMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPurine nucleoside phosphorylase(Homo sapiens (Human))
National Defense Medical Center

Curated by ChEMBL
LigandPNGBDBM50368828(CHEMBL603290)
Affinity DataKi:  2.60E+4nMAssay Description:PNP activity in human RBCMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPurine nucleoside phosphorylase(Homo sapiens (Human))
National Defense Medical Center

Curated by ChEMBL
LigandPNGBDBM50368824(CHEMBL606113)
Affinity DataKi:  3.70E+4nMAssay Description:PNP activity in human RBCMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPurine nucleoside phosphorylase(Homo sapiens (Human))
National Defense Medical Center

Curated by ChEMBL
LigandPNGBDBM50368827(CHEMBL606330)
Affinity DataKi:  9.30E+4nMAssay Description:PNP activity in human RBCMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPurine nucleoside phosphorylase(Homo sapiens (Human))
National Defense Medical Center

Curated by ChEMBL
LigandPNGBDBM50367285(CHEMBL603183)
Affinity DataKi:  1.00E+5nMAssay Description:PNP activity in human RBCMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPurine nucleoside phosphorylase(Homo sapiens (Human))
National Defense Medical Center

Curated by ChEMBL
LigandPNGBDBM50039559(CHEMBL267803 | [5-(2-Amino-6-oxo-1,6-dihydro-purin...)
Affinity DataKi:  1.70E+5nMAssay Description:PNP activity in human RBCMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPurine nucleoside phosphorylase(Homo sapiens (Human))
National Defense Medical Center

Curated by ChEMBL
LigandPNGBDBM50021776(2-Amino-9-(2-hydroxy-ethoxymethyl)-5,9-dihydro-pur...)
Affinity DataKi:  1.80E+5nMAssay Description:PNP activity in human RBCMore data for this Ligand-Target Pair
TargetPurine nucleoside phosphorylase(Homo sapiens (Human))
National Defense Medical Center

Curated by ChEMBL
LigandPNGBDBM50368826(CHEMBL603298)
Affinity DataKi: >3.00E+5nMAssay Description:PNP activity in human RBCMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50002692((AZT) 1-(4-Azido-5-hydroxymethyl-tetrahydro-furan-...)
Affinity DataIC50:  3.10nMAssay Description:Antiviral activity against Human Immunodeficiency Virus by Reverse transcriptase assay in CEM-SS cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50002692((AZT) 1-(4-Azido-5-hydroxymethyl-tetrahydro-furan-...)
Affinity DataIC50:  11nMAssay Description:antiviral activity in Human immunodeficiency virus-1 as reverse transcriptase activity in culture supernatantMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50031364(4-Amino-7-(3-fluoro-4-hydroxy-5-hydroxymethyl-tetr...)
Affinity DataIC50:  20nMAssay Description:antiviral activity in Human immunodeficiency virus-1 as reverse transcriptase activity in culture supernatantMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50369541(CHEMBL608901)
Affinity DataIC50:  35nMAssay Description:Antiviral activity was evaluated by RT (reverse transcriptase) activity in cells acutely infected with HIV-1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50422306(Phosphate Salt Of Tricyclic Nucleoside | TRICIRIBI...)
Affinity DataIC50:  40nMAssay Description:Antiviral activity was tested in cells acutely infected with HIV-1 RT (reverse transcriptase)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50089379((2R,3R,4S,5R)-2-(3-Amino-5-methyl-5H-1,4,5,6,8-pen...)
Affinity DataIC50:  40nMAssay Description:Inhibitory concentration against human immunodeficiency virus type 1 reverse transcriptaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50369528(NSC-154020 | TRICIRIBINE)
Affinity DataIC50:  40nMAssay Description:Antiviral activity was tested in cells acutely infected with HIV-1 RT (reverse transcriptase)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50369528(NSC-154020 | TRICIRIBINE)
Affinity DataIC50:  40nMAssay Description:Antiviral activity was evaluated by RT (reverse transcriptase) activity in cells acutely infected with HIV-1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50422306(Phosphate Salt Of Tricyclic Nucleoside | TRICIRIBI...)
Affinity DataIC50:  40nMAssay Description:Antiviral activity was evaluated by RT (reverse transcriptase) activity in cells acutely infected with HIV-1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50031365(4-Amino-7-(3-fluoro-4-hydroxy-5-hydroxymethyl-tetr...)
Affinity DataIC50:  70nMAssay Description:antiviral activity in Human immunodeficiency virus-1 as reverse transcriptase activity in culture supernatantMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50369542(CHEMBL611850)
Affinity DataIC50:  100nMAssay Description:Antiviral activity was evaluated by Reverse transcriptase activity in cells acutely infected with HIV-1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50369534(CHEMBL607723)
Affinity DataIC50:  250nMAssay Description:Antiviral activity was evaluated by Reverse transcriptase activity in cells acutely infected with HIV-1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGMP synthase [glutamine-hydrolyzing](Mus musculus)
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50042853(CHEMBL127366 | N-(4-Isothiocyanatomethyl-thiazol-2...)
Affinity DataIC50:  350nMAssay Description:In vitro inhibitory activity against partially purified GMP synthetase in L1210 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50369533(CHEMBL611245)
Affinity DataIC50:  350nMAssay Description:Antiviral activity was evaluated by RT (reverse transcriptase) activity in cells acutely infected with HIV-1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50369536(CHEMBL611242)
Affinity DataIC50:  500nMAssay Description:Antiviral activity was evaluated by RT (reverse transcriptase) activity in cells acutely infected with HIV-1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50369535(CHEMBL607724)
Affinity DataIC50:  800nMAssay Description:Antiviral activity was evaluated by Reverse transcriptase activity in cells acutely infected with HIV-1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50369540(CHEMBL608301)
Affinity DataIC50:  800nMAssay Description:Antiviral activity was evaluated by RT (reverse transcriptase) activity in cells acutely infected with HIV-1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50369537(CHEMBL611243)
Affinity DataIC50:  1.00E+3nMAssay Description:Antiviral activity was evaluated by Reverse transcriptase activity in cells acutely infected with HIV-1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50168027((2R,3R,4S,5R)-2-(3-Amino-5-methyl-5H-1,4,5,6,7,8-h...)
Affinity DataIC50:  2.20E+3nMAssay Description:Inhibitory concentration against human immunodeficiency virus type 1 reverse transcriptaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50369539(CHEMBL610949)
Affinity DataIC50:  6.80E+3nMAssay Description:Antiviral activity was evaluated by RT (reverse transcriptase) activity in cells acutely infected with HIV-1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50369532(CHEMBL610657)
Affinity DataIC50:  8.00E+3nMAssay Description:Antiviral activity was evaluated by RT (reverse transcriptase) activity in cells acutely infected with HIV-1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50369538(CHEMBL609191)
Affinity DataIC50:  8.40E+3nMAssay Description:Antiviral activity was evaluated by RT (reverse transcriptase) activity in cells acutely infected with HIV-1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50063941(5,6-Dichloro-1-(4-chloro-benzyl)-1H-benzoimidazol-...)
Affinity DataIC50:  1.00E+4nMAssay Description:Antiviral activity against Human Immunodeficiency Virus by Reverse transcriptase (RT) assay in CEM-SS cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50407560(CHEMBL473686)
Affinity DataIC50:  1.20E+4nMAssay Description:antiviral activity in Human immunodeficiency virus-1 as reverse transcriptase activity in culture supernatantMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50407562(CHEMBL2112687)
Affinity DataIC50:  1.20E+4nMAssay Description:antiviral activity in Human immunodeficiency virus-1 as reverse transcriptase activity in culture supernatantMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50063977(5,6-Dichloro-1-(4-trifluoromethyl-benzyl)-1H-benzo...)
Affinity DataIC50:  2.00E+4nMAssay Description:Antiviral activity against Human Immunodeficiency Virus by Reverse transcriptase assay in CEM-SS cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50408925(CHEMBL2112098)
Affinity DataIC50:  2.10E+4nMAssay Description:Antiviral activity was tested in cells acutely infected with HIV-1 RT (reverse transcriptase)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50407563(CHEMBL2111874)
Affinity DataIC50:  3.20E+4nMAssay Description:antiviral activity in Human immunodeficiency virus-1 as reverse transcriptase activity in culture supernatantMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50063948(2-Bromo-5,6-dichloro-1-(3-nitro-benzyl)-1H-benzoim...)
Affinity DataIC50: >3.20E+4nMAssay Description:Antiviral activity against Human Immunodeficiency Virus by Reverse transcriptase (RT) assay in CEM-SS cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50063945(2-Bromo-5,6-dichloro-1-(3-methyl-benzyl)-1H-benzoi...)
Affinity DataIC50:  6.60E+4nMAssay Description:Antiviral activity against Human Immunodeficiency Virus by Reverse transcriptase assay in CEM-SS cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 15 member 1(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50370614(CHEMBL608788)
Affinity DataIC50:  9.60E+4nMAssay Description:Inhibitory concentration against [3H]glycylsarcosine uptake in HeLa cells expressing human Intestinal peptide transporter PepT1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50063968(1-(3,5-Bis-trifluoromethyl-benzyl)-2-bromo-5,6-dic...)
Affinity DataIC50: >1.00E+5nMAssay Description:Antiviral activity against Human Immunodeficiency Virus by Reverse transcriptase assay in CEM-SS cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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