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Found 367 with Last Name = 'winegar' and Initial = 'da'
LigandPNGBDBM28691(5-methyl-2-({3-[(7-methyl-1H-indole-1-)sulfonyl]be...)
Affinity DataIC50:  4nM EC50:  79nMAssay Description:Competition-binding curves for test compounds were determined with expressed human PPAR LBD. Plots of inhibitor concentration versus cpm of radioliga...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM28674(2-({3-[(2-carboxy-4-chlorophenyl)carbamoyl]benzene...)
Affinity DataIC50:  4nM EC50:  1.26E+3nMpH: 7.0 T: 2°CAssay Description:Competition-binding curves for test compounds were determined with expressed human PPAR LBD. Plots of inhibitor concentration versus cpm of radioliga...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM28661(2-{2-methyl-4-[({4-methyl-2-[4-(trifluoromethyl)ph...)
Affinity DataIC50:  5nMAssay Description:Displacement of [3H]GW 2433 from human PPARdelta by scintillation proximity assayMore data for this Ligand-Target Pair
LigandPNGBDBM28669(2-{[3-(1,2,3,4-tetrahydroisoquinoline-2-sulfonyl)b...)
Affinity DataIC50:  5nM EC50:  158nMpH: 7.0 T: 2°CAssay Description:Competition-binding curves for test compounds were determined with expressed human PPAR LBD. Plots of inhibitor concentration versus cpm of radioliga...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM28670(4-bromo-2-{[3-(1,2,3,4-tetrahydroisoquinoline-2-su...)
Affinity DataIC50:  5nM EC50:  158nMpH: 7.0 T: 2°CAssay Description:Competition-binding curves for test compounds were determined with expressed human PPAR LBD. Plots of inhibitor concentration versus cpm of radioliga...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM28661(2-{2-methyl-4-[({4-methyl-2-[4-(trifluoromethyl)ph...)
Affinity DataIC50:  5nM EC50:  3nMpH: 7.0 T: 2°CAssay Description:Competition-binding curves for test compounds were determined with expressed human PPAR LBD. Plots of inhibitor concentration versus cpm of radioliga...More data for this Ligand-Target Pair
LigandPNGBDBM28682(5-methyl-2-({3-[(4-methyl-1H-indole-1-)sulfonyl]be...)
Affinity DataIC50:  6nM EC50:  20nMAssay Description:Competition-binding curves for test compounds were determined with expressed human PPAR LBD. Plots of inhibitor concentration versus cpm of radioliga...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM28695(5-chloro-2-({3-[(4-methoxy-1H-indole-1-)sulfonyl]b...)
Affinity DataIC50:  6nM EC50:  158nMAssay Description:Competition-binding curves for test compounds were determined with expressed human PPAR LBD. Plots of inhibitor concentration versus cpm of radioliga...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50418124(CHEMBL1760428)
Affinity DataIC50:  6.30nMAssay Description:Displacement of [3H]GW 2433 from human PPARdelta by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50418148(CHEMBL1760411)
Affinity DataIC50:  7.90nMAssay Description:Displacement of [3H]GW 2433 from human PPARdelta by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM28666(5-chloro-2-{[3-(1,2,3,4-tetrahydroisoquinoline-2-s...)
Affinity DataIC50:  8nM EC50:  126nMpH: 7.0 T: 2°CAssay Description:Competition-binding curves for test compounds were determined with expressed human PPAR LBD. Plots of inhibitor concentration versus cpm of radioliga...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM28667(5-bromo-2-{[3-(1,2,3,4-tetrahydroisoquinoline-2-su...)
Affinity DataIC50:  8nM EC50:  200nMpH: 7.0 T: 2°CAssay Description:Competition-binding curves for test compounds were determined with expressed human PPAR LBD. Plots of inhibitor concentration versus cpm of radioliga...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM28675(2-[(3-{[5-(carboxymethoxy)-1,2,3,4-tetrahydroisoqu...)
Affinity DataIC50:  10nM EC50: >1.00E+4nMpH: 7.0 T: 2°CAssay Description:Competition-binding curves for test compounds were determined with expressed human PPAR LBD. Plots of inhibitor concentration versus cpm of radioliga...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM28676(5-chloro-2-({3-[(6-methoxy-1,2,3,4-tetrahydroisoqu...)
Affinity DataIC50:  10nM EC50:  794nMpH: 7.0 T: 2°CAssay Description:Competition-binding curves for test compounds were determined with expressed human PPAR LBD. Plots of inhibitor concentration versus cpm of radioliga...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM28684(2-({3-[(4-methoxy-1H-indole-1-)sulfonyl]benzene}am...)
Affinity DataIC50:  10nM EC50:  40nMAssay Description:Competition-binding curves for test compounds were determined with expressed human PPAR LBD. Plots of inhibitor concentration versus cpm of radioliga...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM28688(5-methyl-2-({3-[(6-methyl-1H-indole-1-)sulfonyl]be...)
Affinity DataIC50:  10nM EC50:  50nMAssay Description:Competition-binding curves for test compounds were determined with expressed human PPAR LBD. Plots of inhibitor concentration versus cpm of radioliga...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM28685(5-methyl-2-({3-[(5-methyl-1H-indole-1-)sulfonyl]be...)
Affinity DataIC50:  10nM EC50:  32nMAssay Description:Competition-binding curves for test compounds were determined with expressed human PPAR LBD. Plots of inhibitor concentration versus cpm of radioliga...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM28683(2-({3-[(4-bromo-1H-indole-1-)sulfonyl]benzene}amid...)
Affinity DataIC50:  10nM EC50:  13nMAssay Description:Competition-binding curves for test compounds were determined with expressed human PPAR LBD. Plots of inhibitor concentration versus cpm of radioliga...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM28672(5-chloro-2-({3-[(5-methoxy-1,2,3,4-tetrahydroisoqu...)
Affinity DataIC50:  13nM EC50:  1.26E+3nMpH: 7.0 T: 2°CAssay Description:Competition-binding curves for test compounds were determined with expressed human PPAR LBD. Plots of inhibitor concentration versus cpm of radioliga...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM28665(5-methyl-2-{[3-(1,2,3,4-tetrahydroisoquinoline-2-s...)
Affinity DataIC50:  13nM EC50:  200nMpH: 7.0 T: 2°CAssay Description:Competition-binding curves for test compounds were determined with expressed human PPAR LBD. Plots of inhibitor concentration versus cpm of radioliga...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM28697(5-chloro-2-({3-[(6-methoxy-1H-indole-1-)sulfonyl]b...)
Affinity DataIC50:  13nM EC50:  100nMAssay Description:Competition-binding curves for test compounds were determined with expressed human PPAR LBD. Plots of inhibitor concentration versus cpm of radioliga...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM28696(5-chloro-2-({3-[(5-methoxy-1H-indole-1-)sulfonyl]b...)
Affinity DataIC50:  13nM EC50:  158nMAssay Description:Competition-binding curves for test compounds were determined with expressed human PPAR LBD. Plots of inhibitor concentration versus cpm of radioliga...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50418129(CHEMBL1760268)
Affinity DataIC50:  13nMAssay Description:Displacement of [3H]GW 2433 from human PPARdelta by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM28677(5-chloro-2-({3-[(7-fluoro-1,2,3,4-tetrahydroisoqui...)
Affinity DataIC50:  16nM EC50:  1.00E+3nMpH: 7.0 T: 2°CAssay Description:Competition-binding curves for test compounds were determined with expressed human PPAR LBD. Plots of inhibitor concentration versus cpm of radioliga...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM28692(2-({3-[(7-chloro-1H-indole-1-)sulfonyl]benzene}ami...)
Affinity DataIC50:  16nM EC50:  158nMAssay Description:Competition-binding curves for test compounds were determined with expressed human PPAR LBD. Plots of inhibitor concentration versus cpm of radioliga...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50418161(CHEMBL1760424)
Affinity DataIC50:  16nMAssay Description:Displacement of [3H]GW 2433 from human PPARdelta by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM28679(5-chloro-2-({3-[(7-chloro-8-methyl-1,2,3,4-tetrahy...)
Affinity DataIC50:  16nM EC50:  316nMpH: 7.0 T: 2°CAssay Description:Competition-binding curves for test compounds were determined with expressed human PPAR LBD. Plots of inhibitor concentration versus cpm of radioliga...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50418135(CHEMBL1760274)
Affinity DataIC50:  16nMAssay Description:Displacement of [3H]GW 2433 from human PPARdelta by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50418123(CHEMBL1760005)
Affinity DataIC50:  16nMAssay Description:Displacement of [3H]GW 2433 from human PPARdelta by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM28698(5-chloro-2-({3-[(5-methoxy-4-methyl-1H-indole-1-)s...)
Affinity DataIC50:  16nM EC50:  16nMAssay Description:Competition-binding curves for test compounds were determined with expressed human PPAR LBD. Plots of inhibitor concentration versus cpm of radioliga...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM28686(2-({3-[(5-chloro-1H-indole-1-)sulfonyl]benzene}ami...)
Affinity DataIC50:  20nM EC50:  50nMAssay Description:Competition-binding curves for test compounds were determined with expressed human PPAR LBD. Plots of inhibitor concentration versus cpm of radioliga...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM28694(2-({3-[(5-methoxy-4-methyl-1H-indole-1-)sulfonyl]b...)
Affinity DataIC50:  20nM EC50:  13nMAssay Description:Competition-binding curves for test compounds were determined with expressed human PPAR LBD. Plots of inhibitor concentration versus cpm of radioliga...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM28673(5-chloro-2-({3-[(5-hydroxy-1,2,3,4-tetrahydroisoqu...)
Affinity DataIC50:  20nM EC50:  2.00E+3nMpH: 7.0 T: 2°CAssay Description:Competition-binding curves for test compounds were determined with expressed human PPAR LBD. Plots of inhibitor concentration versus cpm of radioliga...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50418134(CHEMBL1760273)
Affinity DataIC50:  25nMAssay Description:Displacement of [3H]GW 2433 from human PPARdelta by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM28678(5-chloro-2-({3-[(7-chloro-1,2,3,4-tetrahydroisoqui...)
Affinity DataIC50:  25nM EC50:  794nMpH: 7.0 T: 2°CAssay Description:Competition-binding curves for test compounds were determined with expressed human PPAR LBD. Plots of inhibitor concentration versus cpm of radioliga...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50418149(CHEMBL1760412)
Affinity DataIC50:  25nMAssay Description:Displacement of [3H]GW 2433 from human PPARdelta by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM28668(5-fluoro-2-{[3-(1,2,3,4-tetrahydroisoquinoline-2-s...)
Affinity DataIC50:  25nM EC50:  501nMpH: 7.0 T: 2°CAssay Description:Competition-binding curves for test compounds were determined with expressed human PPAR LBD. Plots of inhibitor concentration versus cpm of radioliga...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM28690(2-({3-[(6-methoxy-1H-indole-1-)sulfonyl]benzene}am...)
Affinity DataIC50:  32nM EC50:  100nMAssay Description:Competition-binding curves for test compounds were determined with expressed human PPAR LBD. Plots of inhibitor concentration versus cpm of radioliga...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM28693(2-({3-[(7-methoxy-1H-indole-1-)sulfonyl]benzene}am...)
Affinity DataIC50:  50nM EC50:  631nMAssay Description:Competition-binding curves for test compounds were determined with expressed human PPAR LBD. Plots of inhibitor concentration versus cpm of radioliga...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50418128(CHEMBL1760267)
Affinity DataIC50:  50nMAssay Description:Displacement of [3H]GW 2433 from human PPARdelta by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50418130(CHEMBL1760269)
Affinity DataIC50:  63nMAssay Description:Displacement of [3H]GW 2433 from human PPARdelta by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50418150(CHEMBL1760413)
Affinity DataIC50:  63nMAssay Description:Displacement of [3H]GW 2433 from human PPARdelta by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM28689(2-({3-[(6-chloro-1H-indole-1-)sulfonyl]benzene}ami...)
Affinity DataIC50:  63nM EC50:  200nMAssay Description:Competition-binding curves for test compounds were determined with expressed human PPAR LBD. Plots of inhibitor concentration versus cpm of radioliga...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50418162(CHEMBL1760425)
Affinity DataIC50:  79nMAssay Description:Displacement of [3H]GW 2433 from human PPARdelta by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50418136(CHEMBL1760399)
Affinity DataIC50:  79nMAssay Description:Displacement of [3H]GW 2433 from human PPARdelta by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50418125(CHEMBL1760426)
Affinity DataIC50:  79nMAssay Description:Displacement of [3H]GW 2433 from human PPARdelta by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50418126(CHEMBL1760427)
Affinity DataIC50:  100nMAssay Description:Displacement of [3H]GW 2433 from human PPARdelta by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM28663(2-{[3-(1,2,3,4-tetrahydroisoquinoline-2-sulfonyl)b...)
Affinity DataIC50:  126nM EC50:  1.26E+3nMpH: 7.0 T: 2°CAssay Description:Competition-binding curves for test compounds were determined with expressed human PPAR LBD. Plots of inhibitor concentration versus cpm of radioliga...More data for this Ligand-Target Pair
LigandPNGBDBM50418142(CHEMBL1760405)
Affinity DataIC50:  126nMAssay Description:Displacement of [3H]GW 2433 from human PPARdelta by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50418159(CHEMBL1760422)
Affinity DataIC50:  126nMAssay Description:Displacement of [3H]GW 2433 from human PPARdelta by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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