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Found 52 with Last Name = 'yui' and Initial = 'j'
TargetTranslocator protein(Rattus norvegicus (rat))
National Institute Of Radiological Sciences

Curated by ChEMBL
LigandPNGBDBM50122294(CHEMBL292092 | N-(5-fluoro-2-phenoxyphenyl)-N-(2-(...)
Affinity DataKi:  0.0800nMAssay Description:Displacement of [11C]DAA1106 from PBR receptor in rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
National Institute Of Radiological Sciences

Curated by ChEMBL
LigandPNGBDBM50266889(CHEMBL513922 | N-benzyl-N-ethyl-2-(7-methyl-8-oxo-...)
Affinity DataKi:  0.200nMAssay Description:Displacement of [11C]PK11195 from PBR receptor in rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Rattus norvegicus (Rat))
National Institute Of Radiological Sciences

Curated by ChEMBL
LigandPNGBDBM50312840(CHEMBL1076680 | US9139546, 16 | [11C](3',5'-dichlo...)
Affinity DataKi:  0.270nMAssay Description:Binding affinity to rat brain CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
National Institute Of Radiological Sciences

Curated by ChEMBL
LigandPNGBDBM22032(1-(2-chlorophenyl)-N-methyl-N-(1-methylpropyl)isoq...)
Affinity DataKi:  0.310nMAssay Description:Displacement of [11C]PK11195 from PBR receptor in rat brain membraneMore data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 1(Homo sapiens (Human))
National Institute Of Radiological Sciences

Curated by ChEMBL
LigandPNGBDBM50163592((3,4-Dihydro-2H-1-oxa-9-aza-anthracen-6-yl)-(4-met...)
Affinity DataKi:  0.340nMAssay Description:Binding affinity to mGluR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 1(Homo sapiens (Human))
National Institute Of Radiological Sciences

Curated by ChEMBL
LigandPNGBDBM50301822(5-(1-(2-fluoropyridin-3-yl)-5-methyl-1H-1,2,3-tria...)
Affinity DataKi:  0.400nMAssay Description:Binding affinity to mGluR1 by PET analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 1(Homo sapiens (Human))
National Institute Of Radiological Sciences

Curated by ChEMBL
LigandPNGBDBM50301822(5-(1-(2-fluoropyridin-3-yl)-5-methyl-1H-1,2,3-tria...)
Affinity DataKi:  0.400nMAssay Description:Binding affinity to mGluR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
National Institute Of Radiological Sciences

Curated by ChEMBL
LigandPNGBDBM50266861(CHEMBL515622 | N-benzyl-N-ethyl-2-(7-(2-fluoroethy...)
Affinity DataKi:  0.490nMAssay Description:Displacement of [11C]PK11195 from PBR receptor in rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
National Institute Of Radiological Sciences

Curated by ChEMBL
LigandPNGBDBM50266863(CHEMBL476811 | N-benzyl-N-(2-fluoroethyl)-2-(7-met...)
Affinity DataKi:  0.510nMAssay Description:Displacement of [11C]PK11195 from PBR receptor in rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
National Institute Of Radiological Sciences

Curated by ChEMBL
LigandPNGBDBM50266889(CHEMBL513922 | N-benzyl-N-ethyl-2-(7-methyl-8-oxo-...)
Affinity DataKi:  0.600nMAssay Description:Displacement of [11C]-PK-11195 from TPSO in Sprague-Dawley rat brain homogenate after 30 mins by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
National Institute Of Radiological Sciences

Curated by ChEMBL
LigandPNGBDBM50054139((R)1-(2-Chloro-phenyl)-isoquinoline-3-carboxylic a...)
Affinity DataKi:  0.700nMAssay Description:Displacement of [11C]-PK-11195 from TPSO in Sprague-Dawley rat brain homogenate after 30 mins by gamma countingMore data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 1(Homo sapiens (Human))
National Institute Of Radiological Sciences

Curated by ChEMBL
LigandPNGBDBM50333368(CHEMBL1645348 | [11C]-cis-(3-ethyl-2-methylquinoli...)
Affinity DataKi:  0.870nMAssay Description:Binding affinity to mGluR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 1(Homo sapiens (Human))
National Institute Of Radiological Sciences

Curated by ChEMBL
LigandPNGBDBM50333368(CHEMBL1645348 | [11C]-cis-(3-ethyl-2-methylquinoli...)
Affinity DataKi:  0.870nMAssay Description:Binding affinity to mGluR1 by PET analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
National Institute Of Radiological Sciences

Curated by ChEMBL
LigandPNGBDBM50266862(CHEMBL476607 | N-benzyl-2-(7-(2-fluoroethyl)-8-oxo...)
Affinity DataKi:  1.34nMAssay Description:Displacement of [11C]PK11195 from PBR receptor in rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 1(Homo sapiens (Human))
National Institute Of Radiological Sciences

Curated by ChEMBL
LigandPNGBDBM50273942(4-(1-(2-fluoropyridin-3-yl)-5-methyl-1H-1,2,3-tria...)
Affinity DataKi:  2nMAssay Description:Binding affinity to mGluR1 by PET analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Rattus norvegicus (Rat))
National Institute Of Radiological Sciences

Curated by ChEMBL
LigandPNGBDBM50312841(CHEMBL1081609 | US9139546, 30 | [11C](3',5'-dichlo...)
Affinity DataKi:  2.30nMAssay Description:Binding affinity to rat brain CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Rattus norvegicus (rat))
National Institute Of Radiological Sciences

Curated by ChEMBL
LigandPNGBDBM50395192(CHEMBL2164336)
Affinity DataKi:  2.60nMAssay Description:Binding affinity to 5-HT7 in rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 1(Homo sapiens (Human))
National Institute Of Radiological Sciences

Curated by ChEMBL
LigandPNGBDBM50273942(4-(1-(2-fluoropyridin-3-yl)-5-methyl-1H-1,2,3-tria...)
Affinity DataKi:  3.90nMAssay Description:Binding affinity to mGluR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
National Institute Of Radiological Sciences

Curated by ChEMBL
LigandPNGBDBM50312838(CHEMBL1081623 | SCH-225336 | [11C]N-(1-(4-(4-metho...)
Affinity DataKi:  4.5nMAssay Description:Binding affinity to human CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 1(Homo sapiens (Human))
National Institute Of Radiological Sciences

Curated by ChEMBL
LigandPNGBDBM50333371(CHEMBL1645351 | CHEMBL1771388 | [11C]-6-N-cyclohex...)
Affinity DataKi:  4.80nMAssay Description:Binding affinity to mGluR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 1(Homo sapiens (Human))
National Institute Of Radiological Sciences

Curated by ChEMBL
LigandPNGBDBM50333371(CHEMBL1645351 | CHEMBL1771388 | [11C]-6-N-cyclohex...)
Affinity DataKi:  4.80nMAssay Description:Binding affinity to mGluR1 by PET analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
National Institute Of Radiological Sciences

Curated by ChEMBL
LigandPNGBDBM50401000(CHEMBL2206282)
Affinity DataKi:  5.10nMAssay Description:Displacement of [11C]-PK-11195 from TPSO in Sprague-Dawley rat brain homogenate after 30 mins by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 1(RAT)
National Institute Of Radiological Sciences

Curated by ChEMBL
LigandPNGBDBM50301520(4-fluoro-N-(4-(6-(isopropylamino)pyrimidin-4-yl)th...)
Affinity DataKi:  5.40nMAssay Description:Displacement of 4-[18F]fluoro-N-[4-(6-(isopropylamino)pyrimidin-4-yl)-1,3-thiazol-2-yl]-N-methylbenzamide from mGluR1 in Sprague-Dawley rat brain hom...More data for this Ligand-Target Pair
TargetCannabinoid receptor 2(Homo sapiens (Human))
National Institute Of Radiological Sciences

Curated by ChEMBL
LigandPNGBDBM50312837(CHEMBL1081610 | [11C]8-butoxy-N-cyclohexyl-7-metho...)
Affinity DataKi:  9.60nMAssay Description:Binding affinity to human CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
National Institute Of Radiological Sciences

Curated by ChEMBL
LigandPNGBDBM50492860(CHEMBL2413451)
Affinity DataKi:  9.70nMAssay Description:Binding affinity to 5-HT7 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 1(RAT)
National Institute Of Radiological Sciences

Curated by ChEMBL
LigandPNGBDBM50388957(CHEMBL2063722)
Affinity DataKi:  12.6nMAssay Description:Displacement of 4-[18F]fluoro-N-[4-(6-(isopropylamino)pyrimidin-4-yl)-1,3-thiazol-2-yl]-N-methylbenzamide from mGluR1 in Sprague-Dawley rat brain hom...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
National Institute Of Radiological Sciences

Curated by ChEMBL
LigandPNGBDBM50400999(CHEMBL2206283)
Affinity DataKi:  13.2nMAssay Description:Displacement of [11C]-PK-11195 from TPSO in Sprague-Dawley rat brain homogenate after 30 mins by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 1(RAT)
National Institute Of Radiological Sciences

Curated by ChEMBL
LigandPNGBDBM50400331(CHEMBL2181520)
Affinity DataKi:  13.6nMAssay Description:Displacement of [18F]FITM from mGlu1 receptor in rat brain homogenates after 1 hr by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 1(RAT)
National Institute Of Radiological Sciences

Curated by ChEMBL
LigandPNGBDBM50400332(CHEMBL2181521)
Affinity DataKi:  22.2nMAssay Description:Displacement of [18F]FITM from mGlu1 receptor in rat brain homogenates after 1 hr by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 1(RAT)
National Institute Of Radiological Sciences

Curated by ChEMBL
LigandPNGBDBM50400330(CHEMBL2181519)
Affinity DataKi:  27.3nMAssay Description:Displacement of [18F]FITM from mGlu1 receptor in rat brain homogenates after 1 hr by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
National Institute Of Radiological Sciences

Curated by ChEMBL
LigandPNGBDBM50312839(CHEMBL1081622 | [18F]8-butoxy-N-cyclohexyl-7-(2-fl...)
Affinity DataKi:  36nMAssay Description:Binding affinity to human CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
National Institute Of Radiological Sciences

Curated by ChEMBL
LigandPNGBDBM50400998(CHEMBL2206284)
Affinity DataKi:  40nMAssay Description:Displacement of [11C]-PK-11195 from TPSO in Sprague-Dawley rat brain homogenate after 30 mins by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 1(RAT)
National Institute Of Radiological Sciences

Curated by ChEMBL
LigandPNGBDBM50388958(CHEMBL2063723)
Affinity DataKi:  153nMAssay Description:Displacement of 4-[18F]fluoro-N-[4-(6-(isopropylamino)pyrimidin-4-yl)-1,3-thiazol-2-yl]-N-methylbenzamide from mGluR1 in Sprague-Dawley rat brain hom...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
National Institute Of Radiological Sciences

Curated by ChEMBL
LigandPNGBDBM50312841(CHEMBL1081609 | US9139546, 30 | [11C](3',5'-dichlo...)
Affinity DataKi:  503nMAssay Description:Binding affinity to CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
National Institute Of Radiological Sciences

Curated by ChEMBL
LigandPNGBDBM50312840(CHEMBL1076680 | US9139546, 16 | [11C](3',5'-dichlo...)
Affinity DataKi: >1.00E+3nMAssay Description:Binding affinity to CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 1(RAT)
National Institute Of Radiological Sciences

Curated by ChEMBL
LigandPNGBDBM50388959(CHEMBL2063724)
Affinity DataKi: >5.00E+3nMAssay Description:Displacement of 4-[18F]fluoro-N-[4-(6-(isopropylamino)pyrimidin-4-yl)-1,3-thiazol-2-yl]-N-methylbenzamide from mGluR1 in Sprague-Dawley rat brain hom...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 1(Mus musculus)
National Institute Of Radiological Sciences

Curated by ChEMBL
LigandPNGBDBM50333367(6-(1-(2-fluoropyridin-3-yl)-5-methyl-1H-1,2,3-tria...)
Affinity DataIC50:  1.40nMAssay Description:Binding affinity to mouse mGluR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 1(Homo sapiens (Human))
National Institute Of Radiological Sciences

Curated by ChEMBL
LigandPNGBDBM50333367(6-(1-(2-fluoropyridin-3-yl)-5-methyl-1H-1,2,3-tria...)
Affinity DataIC50:  3.60nMAssay Description:Binding affinity to human mGluR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 1(RAT)
National Institute Of Radiological Sciences

Curated by ChEMBL
LigandPNGBDBM50301520(4-fluoro-N-(4-(6-(isopropylamino)pyrimidin-4-yl)th...)
Affinity DataIC50:  13.9nMAssay Description:Displacement of 4-[18F]fluoro-N-[4-(6-(isopropylamino)pyrimidin-4-yl)-1,3-thiazol-2-yl]-N-methylbenzamide from mGluR1 in Sprague-Dawley rat brain hom...More data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 1(RAT)
National Institute Of Radiological Sciences

Curated by ChEMBL
LigandPNGBDBM50400331(CHEMBL2181520)
Affinity DataIC50:  26.5nMAssay Description:Displacement of [18F]FITM from mGlu1 receptor in rat brain homogenates after 1 hr by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 1(RAT)
National Institute Of Radiological Sciences

Curated by ChEMBL
LigandPNGBDBM50388957(CHEMBL2063722)
Affinity DataIC50:  32.7nMAssay Description:Displacement of 4-[18F]fluoro-N-[4-(6-(isopropylamino)pyrimidin-4-yl)-1,3-thiazol-2-yl]-N-methylbenzamide from mGluR1 in Sprague-Dawley rat brain hom...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 1(RAT)
National Institute Of Radiological Sciences

Curated by ChEMBL
LigandPNGBDBM50400332(CHEMBL2181521)
Affinity DataIC50:  47nMAssay Description:Displacement of [18F]FITM from mGlu1 receptor in rat brain homogenates after 1 hr by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 1(RAT)
National Institute Of Radiological Sciences

Curated by ChEMBL
LigandPNGBDBM50400330(CHEMBL2181519)
Affinity DataIC50:  64.7nMAssay Description:Displacement of [18F]FITM from mGlu1 receptor in rat brain homogenates after 1 hr by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 1(RAT)
National Institute Of Radiological Sciences

Curated by ChEMBL
LigandPNGBDBM50388958(CHEMBL2063723)
Affinity DataIC50:  395nMAssay Description:Displacement of 4-[18F]fluoro-N-[4-(6-(isopropylamino)pyrimidin-4-yl)-1,3-thiazol-2-yl]-N-methylbenzamide from mGluR1 in Sprague-Dawley rat brain hom...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 5(Rattus norvegicus (Rat))
National Institute Of Radiological Sciences

Curated by ChEMBL
LigandPNGBDBM50400331(CHEMBL2181520)
Affinity DataIC50: >1.00E+4nMAssay Description:Displacement of [11C]-ABP688 from mGlu5 receptor in rat brain homogenates after 1 hr by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 5(Rattus norvegicus (Rat))
National Institute Of Radiological Sciences

Curated by ChEMBL
LigandPNGBDBM50400330(CHEMBL2181519)
Affinity DataIC50: >1.00E+4nMAssay Description:Displacement of [11C]-ABP688 from mGlu5 receptor in rat brain homogenates after 1 hr by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 5(Rattus norvegicus (Rat))
National Institute Of Radiological Sciences

Curated by ChEMBL
LigandPNGBDBM50301520(4-fluoro-N-(4-(6-(isopropylamino)pyrimidin-4-yl)th...)
Affinity DataIC50: >1.00E+4nMAssay Description:Displacement of [11C]-ABP688 from mGluR5 in Sprague-Dawley rat brain homogenates after 1 hr by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 5(Rattus norvegicus (Rat))
National Institute Of Radiological Sciences

Curated by ChEMBL
LigandPNGBDBM50388959(CHEMBL2063724)
Affinity DataIC50: >1.00E+4nMAssay Description:Displacement of [11C]-ABP688 from mGluR5 in Sprague-Dawley rat brain homogenates after 1 hr by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 5(Rattus norvegicus (Rat))
National Institute Of Radiological Sciences

Curated by ChEMBL
LigandPNGBDBM50388958(CHEMBL2063723)
Affinity DataIC50: >1.00E+4nMAssay Description:Displacement of [11C]-ABP688 from mGluR5 in Sprague-Dawley rat brain homogenates after 1 hr by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 5(Rattus norvegicus (Rat))
National Institute Of Radiological Sciences

Curated by ChEMBL
LigandPNGBDBM50388957(CHEMBL2063722)
Affinity DataIC50: >1.00E+4nMAssay Description:Displacement of [11C]-ABP688 from mGluR5 in Sprague-Dawley rat brain homogenates after 1 hr by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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