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Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
641
hits in this display
Target
5-hydroxytryptamine receptor 7
(GUINEA PIG)
Monash University
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
Ki: 0.100nM
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Target
5-hydroxytryptamine receptor 1A
(Rattus norvegicus (rat))
Emory University
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
Copy SMILES
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Affinity Data
Ki: 0.120nM
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Target
5-hydroxytryptamine receptor 7
(Homo sapiens (Human))
University Of Namur
Curated by
ChEMBL
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
Copy SMILES
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Affinity Data
Ki: 0.130nM
Assay Description:
Displacement of [3H]LSD from human 5HT7 receptor
More data for this Ligand-Target Pair
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Target
5-hydroxytryptamine receptor 7
(Rattus norvegicus (rat))
Monash University
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
Copy SMILES
Copy InChI
Affinity Data
Ki: 0.130nM
More data for this Ligand-Target Pair
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Target
5-hydroxytryptamine receptor 7
(Homo sapiens (Human))
University Of Namur
Curated by
ChEMBL
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
Copy SMILES
Copy InChI
Affinity Data
Ki: 0.170nM
Assay Description:
Displacement of [3H]LSD from human recombinant 5-HT7 receptor expressed in CHO cells after 120 mins by scintillation counting
More data for this Ligand-Target Pair
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Target
5-hydroxytryptamine receptor 7
(GUINEA PIG)
Monash University
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
Copy SMILES
Copy InChI
Affinity Data
Ki: 0.25nM
More data for this Ligand-Target Pair
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Target
5-hydroxytryptamine receptor 7
(GUINEA PIG)
Monash University
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
Copy SMILES
Copy InChI
Affinity Data
Ki: 0.25nM
More data for this Ligand-Target Pair
Target Info
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Target
5-hydroxytryptamine receptor 1A
(Homo sapiens (Human))
University of Alberta
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
Copy SMILES
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Affinity Data
Ki: 0.260nM
More data for this Ligand-Target Pair
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Target
5-hydroxytryptamine receptor 2A
(Rattus norvegicus (rat))
Alcon Research
Curated by
ChEMBL
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
Ki: 0.300nM
Assay Description:
In vitro inhibitory constant against [125I]DOI binding to 5-hydroxytryptamine 2A receptor in rat cerebral cortex
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Target
5-hydroxytryptamine receptor 7
(Homo sapiens (Human))
University Of Namur
Curated by
ChEMBL
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
Copy SMILES
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Affinity Data
Ki: 0.380nM
More data for this Ligand-Target Pair
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Target
5-hydroxytryptamine receptor 7
(Homo sapiens (Human))
University Of Namur
Curated by
ChEMBL
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
Copy SMILES
Copy InChI
Affinity Data
Ki: 0.400nM
More data for this Ligand-Target Pair
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Target
5-hydroxytryptamine receptor 1D
(Homo sapiens (Human))
Theravance
Curated by
ChEMBL
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
Copy SMILES
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Affinity Data
Ki: 0.5nM
Assay Description:
Displacement of [3H]5-hydroxytryptamine from human cloned 5HT1D receptor expressed in CHOK1 cells by liquid scintillation counting
More data for this Ligand-Target Pair
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Target
5-hydroxytryptamine receptor 1B
(Homo sapiens (Human))
University of Alberta
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
Copy SMILES
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Affinity Data
Ki: 0.570nM
More data for this Ligand-Target Pair
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Target
5-hydroxytryptamine receptor 1B
(Rattus norvegicus (Rat))
University of Alberta
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
Copy SMILES
Copy InChI
Affinity Data
Ki: 0.570nM
More data for this Ligand-Target Pair
Target Info
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Target
5-hydroxytryptamine receptor 1B
(Homo sapiens (Human))
University of Alberta
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
Copy SMILES
Copy InChI
Affinity Data
Ki: 0.590nM
More data for this Ligand-Target Pair
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Target
5-hydroxytryptamine receptor 7
(Rattus norvegicus (rat))
Monash University
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
Copy SMILES
Copy InChI
Affinity Data
Ki: 0.600nM
More data for this Ligand-Target Pair
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Target
5-hydroxytryptamine receptor 7
(Rattus norvegicus (rat))
Monash University
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
Copy SMILES
Copy InChI
Affinity Data
Ki: 0.600nM
More data for this Ligand-Target Pair
Target Info
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Target
5-hydroxytryptamine receptor 7
(Rattus norvegicus (rat))
Monash University
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
Copy SMILES
Copy InChI
Affinity Data
Ki: 0.603nM
Assay Description:
Binding affinity at rat 5-hydroxytryptamine 7 receptor.
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Target
5-hydroxytryptamine receptor 1A
(Homo sapiens (Human))
University of Alberta
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
Copy SMILES
Copy InChI
Affinity Data
Ki: 0.620nM
Assay Description:
Displacement of [3H]-8-OH-DPAT from human 5HT1A receptor expressed in HEK293 cells
More data for this Ligand-Target Pair
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Target
5-hydroxytryptamine receptor 7
(Rattus norvegicus (rat))
Monash University
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
Copy SMILES
Copy InChI
Affinity Data
Ki: 0.630nM
More data for this Ligand-Target Pair
Target Info
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Target
5-hydroxytryptamine receptor 2C
(Rattus norvegicus (Rat))
University of Alberta
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
Copy SMILES
Copy InChI
Affinity Data
Ki: 0.700nM
More data for this Ligand-Target Pair
Target Info
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Target
5-hydroxytryptamine receptor 1A
(Homo sapiens (Human))
University of Alberta
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
Copy SMILES
Copy InChI
Affinity Data
Ki: 0.790nM
More data for this Ligand-Target Pair
Target Info
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Target
5-hydroxytryptamine receptor 2B
(Homo sapiens (Human))
Syntex Discovery Research
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
Copy SMILES
Copy InChI
Affinity Data
Ki: 0.790nM
More data for this Ligand-Target Pair
Target Info
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Target
5-hydroxytryptamine receptor 7
(Homo sapiens (Human))
University Of Namur
Curated by
ChEMBL
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
Copy SMILES
Copy InChI
Affinity Data
Ki: 0.800nM
Assay Description:
Displacement of [3H]LSD from human 5-HT7 receptor expressed in CHO cells
More data for this Ligand-Target Pair
Target Info
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Target
5-hydroxytryptamine receptor 7
(Homo sapiens (Human))
University Of Namur
Curated by
ChEMBL
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
Copy SMILES
Copy InChI
Affinity Data
Ki: 0.800nM
Assay Description:
Displacement of [3H]LSD from human recombinant 5-HT7 receptor expressed in CHO cells
More data for this Ligand-Target Pair
Target Info
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KEGG
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Target
5-hydroxytryptamine receptor 1A
(Homo sapiens (Human))
University of Alberta
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
Copy SMILES
Copy InChI
Affinity Data
Ki: 0.900nM
Assay Description:
Displacement of [3H]8-OH-DPAT from 5-HT1A receptor (unknown origin) expressed in HEK293 cells by liquid scintillation counter
More data for this Ligand-Target Pair
Target Info
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Target
5-hydroxytryptamine receptor 1A
(Homo sapiens (Human))
University of Alberta
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
Copy SMILES
Copy InChI
Affinity Data
Ki: 0.910nM
Assay Description:
Displacement of [3H]-8-OH-DPAT from human 5-HT1A receptor expressed in CHOK1 cell membranes after 30 mins by liquid scintillation spectrometry
More data for this Ligand-Target Pair
Target Info
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Copy BDB DOI
Target
5-hydroxytryptamine receptor 1A
(Homo sapiens (Human))
University of Alberta
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
Copy SMILES
Copy InChI
Affinity Data
Ki: 0.910nM
Assay Description:
Displacement of [3H]-8-OH-DPAT from human 5-HT1A receptor expressed in CHOK1 cell membranes after 30 mins by liquid scintillation spectrometry
More data for this Ligand-Target Pair
Target Info
PDB
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Target
5-hydroxytryptamine receptor 7
(GUINEA PIG)
Monash University
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
Copy SMILES
Copy InChI
Affinity Data
Ki: 1nM
More data for this Ligand-Target Pair
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Target
5-hydroxytryptamine receptor 2B
(Homo sapiens (Human))
Syntex Discovery Research
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
Copy SMILES
Copy InChI
Affinity Data
Ki: 1nM
More data for this Ligand-Target Pair
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Target
5-hydroxytryptamine receptor 1B
(Homo sapiens (Human))
University of Alberta
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
Copy SMILES
Copy InChI
Affinity Data
Ki: 1.09nM
More data for this Ligand-Target Pair
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Target
5-hydroxytryptamine receptor 1B
(Rattus norvegicus (Rat))
University of Alberta
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
Copy SMILES
Copy InChI
Affinity Data
Ki: 1.10nM
Assay Description:
Ability to displace [3H]5-HT bound to 5-hydroxytryptamine 1B receptor in rat striatum
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Target
5-hydroxytryptamine receptor 1B
(Rattus norvegicus (Rat))
University of Alberta
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
Copy SMILES
Copy InChI
Affinity Data
Ki: 1.10nM
Assay Description:
Binding affinity against 5-hydroxytryptamine 1B receptor of rat striatum.
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Target
5-hydroxytryptamine receptor 1B
(Homo sapiens (Human))
University of Alberta
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
Copy SMILES
Copy InChI
Affinity Data
Ki: 1.10nM
Assay Description:
Displacement of [3H]5-hydroxytryptamine from human cloned 5HT1B receptor expressed in CHOK1 cells by liquid scintillation counting
More data for this Ligand-Target Pair
Target Info
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Target
5-hydroxytryptamine receptor 2B
(Homo sapiens (Human))
Syntex Discovery Research
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
Copy SMILES
Copy InChI
Affinity Data
Ki: 1.17nM
More data for this Ligand-Target Pair
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Target
5-hydroxytryptamine receptor 1A
(Homo sapiens (Human))
University of Alberta
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
Copy SMILES
Copy InChI
Affinity Data
Ki: 1.20nM
Assay Description:
Displacement of [3H]-8-OH-DPAT from human recombinant 5-HT1A receptor expressed in HEK293 cells incubated for 60 mins by microbeta2 scintillation cou...
More data for this Ligand-Target Pair
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5-hydroxytryptamine receptor 1A
(Homo sapiens (Human))
University of Alberta
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
Ki: 1.20nM
pH: 7.4
Assay Description:
Binding experiments were conducted in 96-well microplates in a total volume of 250 μL of buffer (50 mM Tris-HCl pH 7.4, 10 mM MgCl2, 0.5 mM EDTA...
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5-hydroxytryptamine receptor 1A
(Homo sapiens (Human))
University of Alberta
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
Ki: 1.25nM
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5-hydroxytryptamine receptor 1A
(Homo sapiens (Human))
University of Alberta
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
Copy SMILES
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Affinity Data
Ki: 1.30nM
Assay Description:
Displacement of [3H]8-OH-DPAT from human recombinant 5HT1A receptor
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5-hydroxytryptamine receptor 1A
(Homo sapiens (Human))
University of Alberta
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
Copy SMILES
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Affinity Data
Ki: 1.30nM
Assay Description:
Displacement of [3H]-8-OH-DPAT from human 5-HT1A receptor expressed in CHO-K1 cell membranes after 60 mins by scintillation counting
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Target
5-hydroxytryptamine receptor 1A
(Homo sapiens (Human))
University of Alberta
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
Copy SMILES
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Affinity Data
Ki: 1.30nM
Assay Description:
Displacement of [3H]-8-OH-DPAT from human 5-HT1A receptor expressed in CHO-K1 cell membranes after 60 mins by scintillation counting method
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Target
5-hydroxytryptamine receptor 1A
(Homo sapiens (Human))
University of Alberta
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
Copy SMILES
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Affinity Data
Ki: 1.30nM
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Target
5-hydroxytryptamine receptor 7
(GUINEA PIG)
Monash University
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
Ki: 1.34nM
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5-hydroxytryptamine receptor 1A
(Homo sapiens (Human))
University of Alberta
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
Copy SMILES
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Affinity Data
Ki: 1.40nM
Assay Description:
Displacement of [3H]-8-OH-DPAT from human 5-HT1A receptor expressed in CHO-K1 cell membranes after 60 mins by microbeta scintillation counting analys...
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5-hydroxytryptamine receptor 7
(Homo sapiens (Human))
University Of Namur
Curated by
ChEMBL
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
Copy SMILES
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Affinity Data
Ki: 1.40nM
Assay Description:
Displacement of [3H]5-HT from human 5-HT7 receptor expressed in HEK293 cells after 30 mins by microbeta counting analysis
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5-hydroxytryptamine receptor 7
(Rattus norvegicus (rat))
Monash University
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
Ki: 1.51nM
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5-hydroxytryptamine receptor 7
(Rattus norvegicus (rat))
Monash University
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
Ki: 1.52nM
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5-hydroxytryptamine receptor 1A
(Rattus norvegicus (rat))
Emory University
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
Copy SMILES
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Affinity Data
Ki: 1.60nM
Assay Description:
Displacement of [3H]8-OHDPAT from 5HT1A receptor in rat hippocampus
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5-hydroxytryptamine receptor 1A
(Rattus norvegicus (rat))
Emory University
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
Copy SMILES
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Affinity Data
Ki: 1.60nM
Assay Description:
Displacement of [3H]8-OHDPAT from 5HT1A receptor in rat hippocampus
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5-hydroxytryptamine receptor 1A
(Rattus norvegicus (rat))
Emory University
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
Copy SMILES
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Affinity Data
Ki: 1.70nM
Assay Description:
Binding affinity towards 5-hydroxytryptamine 1A receptor
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Target
5-hydroxytryptamine receptor 1D
(Homo sapiens (Human))
Theravance
Curated by
ChEMBL
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
Ki: 1.70nM
Assay Description:
In vitro affitnity human cloned 5-hydroxytryptamine 1D receptor alpha by [3H]-5-HT displacement.
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Target
5-hydroxytryptamine receptor 1A
(Homo sapiens (Human))
University of Alberta
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
Ki: 1.70nM
Assay Description:
Binding affinity was measured on 5-hydroxytryptamine 1A receptor in AK cells transfected with human 5-HT1A gene labeled with [3H]-8-OH-DPAT
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5-hydroxytryptamine receptor 7
(Rattus norvegicus (rat))
Monash University
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
Ki: 1.81nM
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5-hydroxytryptamine receptor 7
(Rattus norvegicus (rat))
Monash University
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
Ki: 1.83nM
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5-hydroxytryptamine receptor 1A
(Rattus norvegicus (rat))
Emory University
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
Copy SMILES
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Affinity Data
Ki: 1.90nM
Assay Description:
Binding affinity to 5HT1A receptor in rat cortex membrane
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Target
5-hydroxytryptamine 1D receptor
(Bos taurus (Bovine))
Albany Medical College
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Ki: 1.90nM
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5-hydroxytryptamine receptor 2A
(Rattus norvegicus (rat))
Alcon Research
Curated by
ChEMBL
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
Ki: 1.99nM
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5-hydroxytryptamine receptor 7
(Rattus norvegicus (rat))
Monash University
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
Ki: 2nM
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5-hydroxytryptamine receptor 1D
(Homo sapiens (Human))
Theravance
Curated by
ChEMBL
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
Copy SMILES
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Affinity Data
Ki: 2nM
Assay Description:
In vitro receptor binding affinity for cloned human 5-hydroxytryptamine 1D receptor
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5-hydroxytryptamine receptor 1A
(Rattus norvegicus (rat))
Emory University
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
Ki: 2nM
Assay Description:
Binding affinity was determined against 5-hydroxytryptamine 1A receptor was determined in male Sprague-Dawley rat brain.
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Target
5-hydroxytryptamine receptor 1A/1B/1D/1F
(RAT)
TBA
Curated by
ChEMBL
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
Ki: 2nM
Assay Description:
Evaluated for binding affinity towards rat cortical membranes at 5-hydroxytryptamine 1 receptor binding site by using [3H]-5-HT as a radioligand.
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Target
5-hydroxytryptamine receptor 1D
(Homo sapiens (Human))
Theravance
Curated by
ChEMBL
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
Ki: 2.08nM
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Target
5-hydroxytryptamine receptor 2B
(Homo sapiens (Human))
Syntex Discovery Research
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
Ki: 2.09nM
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Target
5-hydroxytryptamine receptor 7
(Homo sapiens (Human))
University Of Namur
Curated by
ChEMBL
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
Copy SMILES
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Affinity Data
Ki: 2.10nM
Assay Description:
Displacement of [3H]5-CT from human recombinant 5-HT7A receptor expressed in HEK cells by radioligand completion assay
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Target
5-hydroxytryptamine receptor 7
(Homo sapiens (Human))
University Of Namur
Curated by
ChEMBL
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
Copy SMILES
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Affinity Data
Ki: 2.10nM
Assay Description:
Displacement of [3H]-5-HT from human 5-HT7 receptor expressed in CHOK1 cell membranes after 30 mins by liquid scintillation spectrometry
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Target
5-hydroxytryptamine receptor 1A
(Homo sapiens (Human))
University of Alberta
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
Copy SMILES
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Affinity Data
Ki: 2.10nM
Assay Description:
Displacement of [3H]8-OH-DPAT from human 5-HT1A receptor transfected in CFO-K1 cells after 30 mins by liquid scintillation spectrometry
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Target
5-hydroxytryptamine receptor 1D
(Homo sapiens (Human))
Theravance
Curated by
ChEMBL
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
Copy SMILES
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Affinity Data
Ki: 2.10nM
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Target
5-hydroxytryptamine receptor 7
(Homo sapiens (Human))
University Of Namur
Curated by
ChEMBL
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
Copy SMILES
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Affinity Data
Ki: 2.10nM
Assay Description:
Displacement of [3H]-5-HT from human 5-HT7 receptor expressed in CHOK1 cell membranes after 30 mins by liquid scintillation spectrometry
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Target
5-hydroxytryptamine receptor 1A
(Rattus norvegicus (rat))
Emory University
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
Copy SMILES
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Affinity Data
Ki: 2.10nM
Assay Description:
The compound was tested for their binding affinity towards 5-hydroxytryptamine 1A receptor from rat hippocampus using [3H]8-OH-DPAT as radioligand.
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Target
5-hydroxytryptamine receptor 1A
(Rattus norvegicus (rat))
Emory University
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
Copy SMILES
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Affinity Data
Ki: 2.30nM
Assay Description:
Displacement of [3H]-8-OH-DPAT from rat cerebral cortex 5HT1A receptor measured after 15 mins by liquid scintillation counter method
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5-hydroxytryptamine receptor 1E
(Homo sapiens (Human))
Janssen Research Foundation
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PDSP K
i
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Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
Ki: 2.30nM
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5-hydroxytryptamine receptor 2C
(Homo sapiens (Human))
Yamanouchi Pharmaceutical
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i
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Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Ki: 2.40nM
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5-hydroxytryptamine receptor 1A
(Homo sapiens (Human))
University of Alberta
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i
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Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Ki: 2.48nM
Assay Description:
Ability to inhibit the forskolin-stimulated c-AMP formation mediated by human 5-hydroxytryptamine 1A receptor in CHO-K1 cells
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5-hydroxytryptamine receptor 1B
(Rattus norvegicus (Rat))
University of Alberta
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PDSP K
i
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Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
Ki: 2.5nM
Assay Description:
The compound was tested for their binding affinity towards 5-hydroxytryptamine 1B receptor from rat striatum using [3H]5-HT as radioligand.
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5-hydroxytryptamine receptor 1A
(Homo sapiens (Human))
University of Alberta
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PDSP K
i
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Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
Ki: 2.5nM
Assay Description:
The compound was tested for binding affinity against cloned human 5-hydroxytryptamine 1A receptor
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5-hydroxytryptamine receptor 1A
(Homo sapiens (Human))
University of Alberta
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PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
Ki: 2.5nM
Assay Description:
Binding affinity of the compound was evaluated at human recombinant 5-hydroxytryptamine 1A receptor using [3H]-8-OH-DPAT as radioligand
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5-hydroxytryptamine receptor 1B
(GUINEA PIG)
Institut De Recherches Servier
Curated by
PDSP K
i
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Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Ki: 2.51nM
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5-hydroxytryptamine receptor 1D
(RAT)
University of Alberta
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i
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Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Ki: 2.51nM
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5-hydroxytryptamine receptor 1B
(Rattus norvegicus (Rat))
University of Alberta
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Ki: 2.60nM
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5-hydroxytryptamine receptor 1A
(Rattus norvegicus (rat))
Emory University
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PDSP K
i
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Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
Ki: 2.60nM
Assay Description:
Displacement of [3H]8OH-DPAT from 5HT1A in rat brain cerebral cortex after 15 mins by scintillation counting
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5-hydroxytryptamine receptor 1A
(Homo sapiens (Human))
University of Alberta
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i
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Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
Ki: 2.80nM
Assay Description:
Compound was tested in vitro for the inhibition of [3H]-5-HT (2 nM) binding to 5-hydroxytryptamine 1A receptor from bovine hippocampus
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5-hydroxytryptamine receptor 2C
(Homo sapiens (Human))
Yamanouchi Pharmaceutical
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PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Ki: 2.90nM
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5-hydroxytryptamine receptor 1A
(Homo sapiens (Human))
University of Alberta
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
Ki: 3nM
Assay Description:
Compound was tested in vitro for the inhibition of [3H]-DPAT (1 nM) binding to 5-hydroxytryptamine 1A receptor from bovine hippocampus
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5-hydroxytryptamine receptor 1A
(Homo sapiens (Human))
University of Alberta
Curated by
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i
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Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
Ki: 3nM ΔG°: -48.6kJ/mole
T: 2°C
Assay Description:
The composition of the assay buffers was as follows: for 5-HT1AR: 50 mM Tris¿HCl, 0.1 mM EDTA, 4 mM MgCl2, 10 lM pargyline, and 0.1% ascorbate; for 5...
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5-hydroxytryptamine receptor 1A
(Rattus norvegicus (rat))
Emory University
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PDSP K
i
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Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
Ki: 3nM
Assay Description:
Evaluated for the binding affinity to hippocampus striatal membranes at 5-hydroxytryptamine 1A receptor binding site by using [3H]-8-OH- DPAT as a ra...
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5-hydroxytryptamine receptor 1A
(Rattus norvegicus (rat))
Emory University
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
Ki: 3nM
Assay Description:
Displacement of [3H]8-OH-DPAT from rat 5HT1A receptor expressed in CHO cells
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5-hydroxytryptamine receptor 1D
(Homo sapiens (Human))
Theravance
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ChEMBL
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
Ki: 3nM
Assay Description:
Binding affinity was determined against 5-hydroxytryptamine 1D receptor in bovine caudate homogenate
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5-hydroxytryptamine receptor 2A
(Rattus norvegicus (rat))
Alcon Research
Curated by
ChEMBL
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Ki: 3nM
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5-hydroxytryptamine receptor 1A
(Homo sapiens (Human))
University of Alberta
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
Ki: 3nM
Assay Description:
Displacement of [3H]-8-OH-DPAT from recombinant human 5HT1A receptor expressed in CHO cell membranes measured after 60 mins by microbeta scintillatio...
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5-hydroxytryptamine receptor 1B
(Rattus norvegicus (Rat))
University of Alberta
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Ki: 3nM
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5-hydroxytryptamine receptor 1B
(Rattus norvegicus (Rat))
University of Alberta
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Ki: 3.01nM
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5-hydroxytryptamine receptor 7
(Homo sapiens (Human))
University Of Namur
Curated by
ChEMBL
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Ki: 3.20nM
Assay Description:
Binding affinity against 5-hydroxytryptamine 7 human receptors
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5-hydroxytryptamine receptor 1D
(Homo sapiens (Human))
Theravance
Curated by
ChEMBL
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Ki: 3.38nM
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Target
5-hydroxytryptamine receptor 1D
(Homo sapiens (Human))
Theravance
Curated by
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Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Ki: 3.40nM
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Target
5-hydroxytryptamine receptor 1B
(Rattus norvegicus (Rat))
University of Alberta
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
Ki: 3.5nM
Assay Description:
Displacement of [3H]5-HT from 5-HT1B receptor of rat frontal cortex homogenate
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5-hydroxytryptamine receptor 1E
(Homo sapiens (Human))
Janssen Research Foundation
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Ki: 3.5nM
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5-hydroxytryptamine receptor 1A
(Homo sapiens (Human))
University of Alberta
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
Ki: 3.60nM
Assay Description:
Displacement of [3H]8-OH-DPAT from human 5-HT1A receptor expressed in CHO-K1 cell membranes incubated for 60 mins by microbeta scintillation counting...
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5-hydroxytryptamine receptor 1D
(Homo sapiens (Human))
Theravance
Curated by
ChEMBL
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Ki: 3.89nM
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5-hydroxytryptamine receptor 1B
(Homo sapiens (Human))
University of Alberta
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Ki: 3.90nM
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5-hydroxytryptamine receptor 1A
(Homo sapiens (Human))
University of Alberta
Curated by
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i
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Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Ki: 3.98nM
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Target
5-hydroxytryptamine receptor 1A
(Homo sapiens (Human))
University of Alberta
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Ki: 3.98nM
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Target
5-hydroxytryptamine receptor 1B
(Homo sapiens (Human))
University of Alberta
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Ki: 3.98nM
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Target
5-hydroxytryptamine receptor 1A
(Homo sapiens (Human))
University of Alberta
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Ki: 3.98nM
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Target
5-hydroxytryptamine receptor 1D
(Homo sapiens (Human))
Theravance
Curated by
ChEMBL
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Ki: 3.98nM
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5-hydroxytryptamine receptor 1A
(Homo sapiens (Human))
University of Alberta
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
Ki: 4nM
Assay Description:
Binding affinity against 5-hydroxytryptamine 1A human cloned receptors in HEK293 cells using [3H]8-OH-DPAT as radioligand
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5-hydroxytryptamine receptor 1E
(Homo sapiens (Human))
Janssen Research Foundation
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
Ki: 4nM
Assay Description:
Binding affinity was determined against 5-hydroxytryptamine 1E receptor in human cortical homogenate
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5-hydroxytryptamine receptor 1B
(Homo sapiens (Human))
University of Alberta
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
Ki: 4nM
Assay Description:
Binding affinity was measured on 5-hydroxytryptamine 1D receptor beta in CHO cells transfected with human 5-HT1D beta gene labeled with [3H]-5-HT
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5-hydroxytryptamine receptor 1B
(Homo sapiens (Human))
University of Alberta
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
Copy SMILES
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Affinity Data
Ki: 4nM
Assay Description:
Binding affinity of the compound towards cloned human 5-hydroxytryptamine 1D receptor beta was determined using [3H]-8-OH-DPAT as radioligand
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5-hydroxytryptamine receptor 7
(Homo sapiens (Human))
University Of Namur
Curated by
ChEMBL
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
Ki: 4nM
Assay Description:
Binding affinity of compound towards rodent 5-hydroxytryptamine 7 receptor
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5-hydroxytryptamine receptor 2B
(Homo sapiens (Human))
Syntex Discovery Research
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Ki: 4nM
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5-hydroxytryptamine 1D receptor
(Bos taurus (Bovine))
Albany Medical College
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Ki: 4nM
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5-hydroxytryptamine receptor 1B
(Homo sapiens (Human))
University of Alberta
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
Ki: 4.07nM
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5-hydroxytryptamine receptor 1A
(Rattus norvegicus (rat))
Emory University
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
Ki: 4.20nM
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5-hydroxytryptamine receptor 1B
(Homo sapiens (Human))
University of Alberta
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
Ki: 4.26nM
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5-hydroxytryptamine receptor 1D
(Homo sapiens (Human))
Theravance
Curated by
ChEMBL
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Ki: 4.30nM
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5-hydroxytryptamine receptor 1A
(Rattus norvegicus (rat))
Emory University
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
Ki: 4.30nM
Assay Description:
Binding affinity towards 5-hydroxytryptamine 1A receptor by the displacement of [125I]trans-8-OH-PIPAT in membrane homogenates of hippocampal tissue ...
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Target
5-hydroxytryptamine receptor 1A
(Homo sapiens (Human))
University of Alberta
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
Copy SMILES
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Affinity Data
Ki: 4.5nM
Assay Description:
Displacement of [3H]8-OH-DAPT from human recombinant 5-HT1A receptor expressed in CHO cells measured after 60 to 90 mins by radioligand completion as...
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5-hydroxytryptamine receptor 1A
(Rattus norvegicus (rat))
Emory University
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
Ki: 4.80nM
Assay Description:
Binding affinity of a compound to rat brain 5-hydroxytryptamine 1A (serotonin) receptor assayed by radiolabeled [3H]-8-OH-DPAT ligand displacement
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5-hydroxytryptamine receptor 1B
(Homo sapiens (Human))
University of Alberta
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
Ki: 4.80nM
Assay Description:
Ability to displace [3H]5-CT (1.5 nM) from HeLa cells of human 5-hydroxytryptamine 1B receptor
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5-hydroxytryptamine receptor 1D
(Homo sapiens (Human))
Theravance
Curated by
ChEMBL
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
Copy SMILES
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Affinity Data
Ki: 4.80nM
Assay Description:
Binding affinity to recombinant human 5-hydroxytryptamine 1D receptor alpha
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5-hydroxytryptamine receptor 7
(Rattus norvegicus (rat))
Monash University
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
Ki: 4.89nM
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5-hydroxytryptamine receptor 1B
(Homo sapiens (Human))
University of Alberta
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
Copy SMILES
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Affinity Data
Ki: 5nM
Assay Description:
Binding affinity against cloned human 5-hydroxytryptamine 1B receptor in CHO cells using [3H]5-CT as radioligand
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5-hydroxytryptamine receptor 1B
(Rattus norvegicus (Rat))
University of Alberta
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
Ki: 5nM
Assay Description:
Binding affinity was determined against 5-hydroxytryptamine 1B receptor was determined in male Sprague-Dawley rat brain.
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5-hydroxytryptamine receptor 7
(Rattus norvegicus (rat))
Monash University
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Ki: 5nM
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5-hydroxytryptamine receptor 7
(Mus musculus (Mouse))
University of Alberta
Curated by
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i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Ki: 5.01nM
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5-hydroxytryptamine receptor 1D
(Dog)
University of Alberta
Curated by
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i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Ki: 5.01nM
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Target
5-hydroxytryptamine receptor 6
(MOUSE)
Cnrs
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Ki: 5.01nM
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Target
5-hydroxytryptamine receptor 1D
(Homo sapiens (Human))
Theravance
Curated by
ChEMBL
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
Copy SMILES
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Affinity Data
Ki: 5.06nM
Assay Description:
Ability to inhibit the forskolin-stimulated c-AMP formation mediated by human 5-hydroxytryptamine 1D receptor in CHO-K1 cells
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Target
5-hydroxytryptamine receptor 1D
(Homo sapiens (Human))
Theravance
Curated by
ChEMBL
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
Copy SMILES
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Affinity Data
Ki: 5.10nM
Assay Description:
Binding affinity of the compound was evaluated at human recombinant 5-hydroxytryptamine 1D receptor using [3H]-5-CT as radioligand
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Target
5-hydroxytryptamine receptor 1B
(Rattus norvegicus (Rat))
University of Alberta
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
Ki: 5.24nM
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Target
5-hydroxytryptamine receptor 1B
(Rattus norvegicus (Rat))
University of Alberta
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
Ki: 5.40nM
Assay Description:
Evaluated for binding affinity towards 5-hydroxytryptamine 1B receptor
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Target
5-hydroxytryptamine receptor 1B
(Rattus norvegicus (Rat))
University of Alberta
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
Ki: 5.40nM
Assay Description:
Binding affinity was measured on 5-hydroxytryptamine 1B receptor in rat striatum labeled with [3H]-5-HT
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Target
5-hydroxytryptamine receptor 1D
(Homo sapiens (Human))
Theravance
Curated by
ChEMBL
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
Copy SMILES
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Affinity Data
Ki: 5.5nM
Assay Description:
Binding affinity was measured on 5-hydroxytryptamine 1D receptor alpha in COS cells transfected with human 5-HT1D alpha gene labeled with [3H]-5-HT
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Target
5-hydroxytryptamine receptor 1A
(Homo sapiens (Human))
University of Alberta
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
Ki: 5.5nM
Assay Description:
Displacement of [3H]-8-OH-DPAT from human 5HT1A receptor expressed in CHO-K1 cell membranes incubated for 60 mins by microbeta scintillation counting...
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Target
5-hydroxytryptamine receptor 2C
(Homo sapiens (Human))
Yamanouchi Pharmaceutical
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
Ki: 5.75nM
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5-hydroxytryptamine receptor 2C
(Homo sapiens (Human))
Yamanouchi Pharmaceutical
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
Ki: 5.75nM
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5-hydroxytryptamine receptor 2A
(Rattus norvegicus (rat))
Alcon Research
Curated by
ChEMBL
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Ki: 5.75nM
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Target
5-hydroxytryptamine receptor 7
(Homo sapiens (Human))
University Of Namur
Curated by
ChEMBL
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
Copy SMILES
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Affinity Data
Ki: 6nM
Assay Description:
Displacement of [3H]D-lysergic acid diethylamide from 5HT7R (unknown origin) expressed in HEK293 cell membranes incubated for 1.5 hrs in absence of l...
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Target
Serotonin 2 (5-HT2) receptor
(RAT)
TBA
Curated by
ChEMBL
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
Ki: 6nM
Assay Description:
Binding affinity to rat cortical membranes at 5-hydroxytryptamine 2 receptor binding site by using [3H]- DOB as a radioligand.
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5-hydroxytryptamine receptor 1E
(Homo sapiens (Human))
Janssen Research Foundation
Curated by
PDSP K
i
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Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
Ki: 6.16nM
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5-hydroxytryptamine receptor 4
(RAT)
Synaptic Pharmaceutical
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PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Ki: 6.30nM
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5-hydroxytryptamine receptor 7
(Homo sapiens (Human))
University Of Namur
Curated by
ChEMBL
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Ki: 6.31nM
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5-hydroxytryptamine receptor 1B
(Homo sapiens (Human))
University of Alberta
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
Ki: 6.80nM
Assay Description:
Binding affinity of the compound was evaluated at human recombinant 5-hydroxytryptamine 1B receptor using [3H]-5-CT as radioligand
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5-hydroxytryptamine receptor 1B
(Homo sapiens (Human))
University of Alberta
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
Ki: 6.80nM
Assay Description:
Ability to inhibit the forskolin-stimulated c-AMP formation mediated by human 5-hydroxytryptamine 1B receptor in CHO-K1 cells
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5-hydroxytryptamine receptor 2C
(Homo sapiens (Human))
Yamanouchi Pharmaceutical
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
Ki: 6.90nM
Assay Description:
Displacement of [3H]5HT from human 5HT2C
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5-hydroxytryptamine receptor 2C
(Homo sapiens (Human))
Yamanouchi Pharmaceutical
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
Ki: 6.90nM
Assay Description:
Affinity for human 5-hydroxytryptamine 2B receptor expressed in mammalian cell line
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5-hydroxytryptamine receptor 1E
(RAT)
The Scripps Research Institute
Curated by
PDSP K
i
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Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Ki: 7nM
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5-hydroxytryptamine receptor 1B
(Homo sapiens (Human))
University of Alberta
Curated by
PDSP K
i
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Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
Ki: 7.10nM
Assay Description:
The compound was tested for binding affinity against cloned human 5-hydroxytryptamine 1D receptor beta
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5-hydroxytryptamine receptor 1E
(Homo sapiens (Human))
Janssen Research Foundation
Curated by
PDSP K
i
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Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
Ki: 7.24nM
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5-hydroxytryptamine receptor 1A
(Rattus norvegicus (rat))
Emory University
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
Ki: 7.30nM
Assay Description:
Ability to displace [3H]- -(OH)-DPAT bound to 5-hydroxytryptamine 1A receptor in rat hippocampus
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5-hydroxytryptamine receptor 1A
(Rattus norvegicus (rat))
Emory University
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
Ki: 7.30nM
Assay Description:
Binding affinity against 5-hydroxytryptamine 1A receptor of rat hippocampus tissue.
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5-hydroxytryptamine receptor 7
(Rattus norvegicus (rat))
Monash University
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
Ki: 7.33nM
Assay Description:
Displacement of [3H]LSD from rat recombinant 5HT7 receptor expressed in HEK293 cells at 10 uM
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5-hydroxytryptamine receptor 5B
(RAT)
University of Alberta
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i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Ki: 7.76nM
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5-hydroxytryptamine receptor 2A
(Homo sapiens (Human))
Eli Lilly
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
Ki: 7.77nM
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Target
Serotonin 2 (5-HT2) receptor
(RAT)
TBA
Curated by
ChEMBL
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
Ki: 7.80nM
Assay Description:
Binding affinity for the Opioid receptor kappa 1
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Target
5-hydroxytryptamine receptor 5B
(RAT)
University of Alberta
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Ki: 7.80nM
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5-hydroxytryptamine receptor 7
(Homo sapiens (Human))
University Of Namur
Curated by
ChEMBL
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
Ki: 7.90nM
Assay Description:
Displacement of [3H]5-HT from recombinant human 5-HT7 receptor expressed in African green monkey COS7 cells
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5-hydroxytryptamine receptor 4
(RAT)
Synaptic Pharmaceutical
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Ki: 7.94nM
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Target
5-hydroxytryptamine receptor 7
(Rattus norvegicus (rat))
Monash University
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Ki: 7.94nM
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5-hydroxytryptamine receptor 7
(Homo sapiens (Human))
University Of Namur
Curated by
ChEMBL
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Ki: 7.94nM
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5-hydroxytryptamine receptor 1B
(Homo sapiens (Human))
University of Alberta
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
Ki: 7.94nM
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5-hydroxytryptamine receptor 7
(Homo sapiens (Human))
University Of Namur
Curated by
ChEMBL
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
Ki: 8.10nM
Assay Description:
Displacement of [3H]5-HT from human 5-hydroxytryptamine 7 receptor
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Target
5-hydroxytryptamine receptor 7
(Homo sapiens (Human))
University Of Namur
Curated by
ChEMBL
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Ki: 8.10nM
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Target
5-hydroxytryptamine receptor 7
(Homo sapiens (Human))
University Of Namur
Curated by
ChEMBL
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
Ki: 8.12nM
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5-hydroxytryptamine receptor 2A
(Homo sapiens (Human))
Eli Lilly
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
Ki: 8.20nM
Assay Description:
Displacement of [125I]DOI from cloned human 5HT2A receptor expressed in CHO cells
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5-hydroxytryptamine receptor 2A
(Homo sapiens (Human))
Eli Lilly
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
Ki: 8.20nM
Assay Description:
Inhibitory constant against cloned human 5-hydroxytryptamine 2A receptor using with [125I]- DOI radioligand
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5-hydroxytryptamine receptor 2C
(Homo sapiens (Human))
Yamanouchi Pharmaceutical
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
Ki: 8.30nM
Assay Description:
Displacement of [125I]DOI from cloned human 5HT2C receptor expressed in CHO cells
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5-hydroxytryptamine receptor 2C
(Homo sapiens (Human))
Yamanouchi Pharmaceutical
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
Ki: 8.30nM
Assay Description:
Inhibitory constant against cloned human 5-hydroxytryptamine 2C receptor using with [125I]- DOI radioligand
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5-hydroxytryptamine receptor 1D
(Homo sapiens (Human))
Theravance
Curated by
ChEMBL
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
Ki: 8.90nM
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Target
5-hydroxytryptamine receptor 1D
(Homo sapiens (Human))
Theravance
Curated by
ChEMBL
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
Ki: 8.91nM
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Target
5-hydroxytryptamine receptor 1B
(Homo sapiens (Human))
University of Alberta
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
Ki: 9nM
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5-hydroxytryptamine receptor 2B
(Homo sapiens (Human))
Syntex Discovery Research
Curated by
PDSP K
i
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Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
Ki: 9.46nM
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Target
5-hydroxytryptamine receptor 2B
(Homo sapiens (Human))
Syntex Discovery Research
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
Ki: 9.80nM
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5-hydroxytryptamine receptor 7
(Rattus norvegicus (rat))
Monash University
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
Ki: 10nM
Assay Description:
Binding affinity towards rat 5-hydroxytryptamine 7 receptor
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5-hydroxytryptamine receptor 1A
(Homo sapiens (Human))
University of Alberta
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
Ki: 10nM
Assay Description:
Displacement of [3H]-8-OH-DPAT from human cloned 5HT1A receptor
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5-hydroxytryptamine receptor 1A
(Homo sapiens (Human))
University of Alberta
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
Copy SMILES
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Affinity Data
Ki: 10nM ΔG°: -47.5kJ/mole
pH: 7.4 T: 2°C
Assay Description:
Human-cloned 5-HT1A serotonin receptors stably expressed in HEK293-EBNA cells (Perkin-Elmer, Waltham, MA) were radiolabeled with 1.0nM [3H]-8-OH-DPAT...
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5-hydroxytryptamine receptor 2C
(Rattus norvegicus (Rat))
University of Alberta
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
Copy SMILES
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Affinity Data
Ki: 10nM
Assay Description:
Binding affinity was determined against 5-hydroxytryptamine 1C receptor was determined in male Sprague-Dawley rat brain.
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5-hydroxytryptamine receptor 1F
(Homo sapiens (Human))
Janssen Research Foundation
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Ki: 10nM
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5-hydroxytryptamine receptor 1F
(Homo sapiens (Human))
Janssen Research Foundation
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
Copy SMILES
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Ki: 10nM
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Target
5-hydroxytryptamine receptor 1F
(Homo sapiens (Human))
Janssen Research Foundation
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
Copy SMILES
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Affinity Data
Ki: 10nM
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Target
5-hydroxytryptamine receptor 2B
(RAT)
Syntex Discovery Research
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
Copy SMILES
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Ki: 10nM
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Target
5-hydroxytryptamine receptor 2B
(RAT)
Syntex Discovery Research
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
Copy SMILES
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Ki: 10.2nM
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Target
5-hydroxytryptamine receptor 2B
(RAT)
Syntex Discovery Research
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
Copy SMILES
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Ki: 10.2nM
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5-hydroxytryptamine receptor 1E
(Homo sapiens (Human))
Janssen Research Foundation
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
Ki: 11.0nM
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5-hydroxytryptamine receptor 2A
(Rattus norvegicus (rat))
Alcon Research
Curated by
ChEMBL
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
Ki: 11nM
Assay Description:
Displacement of [3H]DOI-HCL from 5HT2A in Sprague-Dawley rat frontal cortex membranes measured after 20 mins
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5-hydroxytryptamine receptor 2B
(Homo sapiens (Human))
Syntex Discovery Research
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
Ki: 11nM
Assay Description:
Displacement of [3H]LSD from human recombinant 5-HT2B receptor expressed in HEK cells by radioligand completion assay relative to control
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5-hydroxytryptamine receptor 1E
(Homo sapiens (Human))
Janssen Research Foundation
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
Ki: 11nM
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5-hydroxytryptamine receptor 2C
(Rattus norvegicus (Rat))
University of Alberta
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
Copy SMILES
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Affinity Data
Ki: 11nM
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5-hydroxytryptamine receptor 2C
(Rattus norvegicus (Rat))
University of Alberta
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
Copy SMILES
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Affinity Data
Ki: 11nM
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Target
5-hydroxytryptamine receptor 2B
(RAT)
Syntex Discovery Research
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Ki: 11.3nM
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5-hydroxytryptamine receptor 2A
(Homo sapiens (Human))
Eli Lilly
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
Copy SMILES
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Affinity Data
Ki: 12nM
Assay Description:
Displacement of [125I]DOI from human 5HT2A receptor expressed in HEK293 cell membranes
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Target
5-hydroxytryptamine receptor 2B
(Homo sapiens (Human))
Syntex Discovery Research
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
Copy SMILES
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Affinity Data
Ki: 12nM
Assay Description:
Affinity for human 5-hydroxytryptamine 2B receptor expressed in mammalian cell line
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Target
5-hydroxytryptamine receptor 2B
(Homo sapiens (Human))
Syntex Discovery Research
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
Copy SMILES
Copy InChI
Affinity Data
Ki: 12nM
Assay Description:
Displacement of [3H]5HT from human 5HT2B
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5-hydroxytryptamine receptor 2A
(Homo sapiens (Human))
Eli Lilly
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
Ki: 12.0nM
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Target
5-hydroxytryptamine receptor 2C
(Rattus norvegicus (Rat))
University of Alberta
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
Copy SMILES
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Affinity Data
Ki: 12.2nM
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Target
5-hydroxytryptamine receptor 1A
(Homo sapiens (Human))
University of Alberta
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
Copy SMILES
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Affinity Data
Ki: 12.6nM
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Target
5-hydroxytryptamine receptor 6
(RAT)
F. Hoffmann-La Roche
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
Copy SMILES
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Ki: 12.6nM
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Target
5-hydroxytryptamine receptor 2B
(Homo sapiens (Human))
Syntex Discovery Research
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
Copy SMILES
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Affinity Data
Ki: 13nM
Assay Description:
Displacement of [125I]DOI from cloned human 5HT2B receptor expressed in CHO cells
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Target
5-hydroxytryptamine receptor 2B
(Homo sapiens (Human))
Syntex Discovery Research
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
Copy SMILES
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Affinity Data
Ki: 13nM
Assay Description:
Inhibitory constant against cloned human 5-hydroxytryptamine 2B receptor using with [125I]- DOI radioligand
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Target
5-hydroxytryptamine receptor 2B
(Homo sapiens (Human))
Syntex Discovery Research
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
Copy SMILES
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Affinity Data
Ki: 13.5nM
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Target
5-hydroxytryptamine receptor 1B
(Homo sapiens (Human))
University of Alberta
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
Copy SMILES
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Affinity Data
Ki: 14nM
Assay Description:
Displacement of [125I]CYP from human 5HT1B receptor
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Target
5-hydroxytryptamine receptor 1B
(Rattus norvegicus (Rat))
University of Alberta
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
Copy SMILES
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Affinity Data
Ki: 14nM
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5-hydroxytryptamine receptor 2A
(Homo sapiens (Human))
Eli Lilly
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
Copy SMILES
Copy InChI
Affinity Data
Ki: 14nM
Assay Description:
Displacement of [125I]DOI from human 5HT2A
More data for this Ligand-Target Pair
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Target
5-hydroxytryptamine receptor 2A
(Homo sapiens (Human))
Eli Lilly
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
Copy SMILES
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Affinity Data
Ki: 14nM
Assay Description:
Functional activity against human 5-hydroxytryptamine 2A receptor expressed in CHO cells using fluorometricimaging plate reader
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Target
5-hydroxytryptamine receptor 2C
(Homo sapiens (Human))
Yamanouchi Pharmaceutical
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
Copy SMILES
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Affinity Data
Ki: 15.5nM
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Target
5-hydroxytryptamine receptor 1B
(Homo sapiens (Human))
University of Alberta
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
Copy SMILES
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Affinity Data
Ki: 15.8nM
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5-hydroxytryptamine receptor 1D
(Dog)
University of Alberta
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
Copy SMILES
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Ki: 15.8nM
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Target
5-hydroxytryptamine receptor 1B
(Rattus norvegicus (Rat))
University of Alberta
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
Copy SMILES
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Ki: 15.8nM
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5-hydroxytryptamine receptor 2A
(Homo sapiens (Human))
Eli Lilly
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
Copy SMILES
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Affinity Data
Ki: 16.2nM
More data for this Ligand-Target Pair
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Target
5-hydroxytryptamine receptor 2A
(Homo sapiens (Human))
Eli Lilly
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
Copy SMILES
Copy InChI
Affinity Data
Ki: 17nM
Assay Description:
Displacement of [3H]LSD from human recombinant 5-HT2A receptor expressed in HEK cells by radioligand completion assay relative to control
More data for this Ligand-Target Pair
Target Info
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5-hydroxytryptamine receptor 1D
(RAT)
University of Alberta
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
Ki: 18nM
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5-hydroxytryptamine receptor 2C
(Homo sapiens (Human))
Yamanouchi Pharmaceutical
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
Ki: 18.2nM
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5-hydroxytryptamine receptor 2B
(Homo sapiens (Human))
Syntex Discovery Research
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
Ki: 19nM
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5-hydroxytryptamine receptor 2C
(Homo sapiens (Human))
Yamanouchi Pharmaceutical
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
Copy SMILES
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Affinity Data
Ki: 20nM
Assay Description:
Displacement of [N-methyl-3H]LSD from human 5HT2C receptor expressed in HEK293 cells
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5-hydroxytryptamine receptor 2A
(Homo sapiens (Human))
Eli Lilly
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
Ki: 21nM
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5-hydroxytryptamine receptor 2C
(Rattus norvegicus (Rat))
University of Alberta
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
Ki: 22.9nM
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5-hydroxytryptamine receptor 2C
(Rattus norvegicus (Rat))
University of Alberta
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
Ki: 23nM
Assay Description:
Binding affinity was measured on 5-hydroxytryptamine 2C receptor in J1 cells transfected with rat 5-HT2C gene labeled with [3H]-mesulergine
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5-hydroxytryptamine receptor 1B
(Rattus norvegicus (Rat))
University of Alberta
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
Ki: 25nM
Assay Description:
Binding affinity (Ki) to rat cortical membranes at 5-HT1B binding site by using [125 I] ICYP as a radioligand.
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5-hydroxytryptamine receptor 7
(Rattus norvegicus (rat))
Monash University
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
Ki: 25.1nM
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Target
5-hydroxytryptamine receptor 2B
(RAT)
Syntex Discovery Research
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Ki: 28.2nM
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5-hydroxytryptamine receptor 4
(Homo sapiens (Human))
Monash University
Curated by
ChEMBL
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
Copy SMILES
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Affinity Data
Ki: 29.5nM
Assay Description:
Displacement of [3H]GR-113808 from human 5HT4b receptor expressed in COS7 cell membrane by scintillation counting
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Target
5-hydroxytryptamine receptor 2A
(Homo sapiens (Human))
Eli Lilly
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
Copy SMILES
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Affinity Data
Ki: 30.9nM
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5-hydroxytryptamine receptor 6
(Homo sapiens (Human))
Jagiellonian University Collegium Medicum
Curated by
ChEMBL
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
Copy SMILES
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Affinity Data
Ki: 33nM
Assay Description:
Displacement of [3H]LSD from human recombinant 5-HT6 receptor expressed in HEK-293 cells incubated for 60 mins by scintillation counting method
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Target
5-hydroxytryptamine receptor 6
(Homo sapiens (Human))
Jagiellonian University Collegium Medicum
Curated by
ChEMBL
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
Copy SMILES
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Affinity Data
Ki: 33nM
Assay Description:
Displacement of [3H]LSD from human recombinant 5-HT6 receptor expressed in CHO cells
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Target
5-hydroxytryptamine receptor 2C
(Homo sapiens (Human))
Yamanouchi Pharmaceutical
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
Copy SMILES
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Affinity Data
Ki: 35nM
Assay Description:
Evaluated for the binding affinity to porcine choroid plexus at 5-hydroxytryptamine 2C receptor binding site by using [3H]-MES as a radioligand.
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Target
5-hydroxytryptamine receptor 4
(RAT)
Synaptic Pharmaceutical
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
Copy SMILES
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Affinity Data
Ki: 37nM
Assay Description:
Binding affinity at 5-hydroxytryptamine 4 receptor in rat striatum by [3H]GR-113808 displacement.
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Target
5-hydroxytryptamine receptor 1B
(Homo sapiens (Human))
University of Alberta
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
Copy SMILES
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Affinity Data
Ki: 38nM
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Target
5-hydroxytryptamine receptor 4
(RAT)
Synaptic Pharmaceutical
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
Copy SMILES
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Affinity Data
Ki: 38.9nM
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Target
5-hydroxytryptamine receptor 4
(GUINEA PIG)
Janssen Research Foundation
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
Ki: 39.8nM
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Target
5-hydroxytryptamine receptor 1B
(Mus musculus (Mouse))
University of Alberta
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
Ki: 39.8nM
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Target
5-hydroxytryptamine receptor 6
(MOUSE)
Cnrs
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
Copy SMILES
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Affinity Data
Ki: 39.8nM
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Target
5-hydroxytryptamine receptor 2C
(Rattus norvegicus (Rat))
University of Alberta
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
Copy SMILES
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Affinity Data
Ki: 44nM
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5-hydroxytryptamine receptor 1A
(Rattus norvegicus (rat))
Emory University
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
Ki: 46.8nM
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Target
5-hydroxytryptamine receptor 2C
(Homo sapiens (Human))
Yamanouchi Pharmaceutical
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
Copy SMILES
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Affinity Data
Ki: 50nM
Assay Description:
Binding affinity against 5-hydroxytryptamine 2C receptor human cloned receptors in HEK 293 cells using [3H]mesulergine as radioligand
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Target
5-hydroxytryptamine receptor 4
(GUINEA PIG)
Janssen Research Foundation
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
Copy SMILES
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Affinity Data
Ki: 50.1nM
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Target
5-hydroxytryptamine receptor 4
(GUINEA PIG)
Janssen Research Foundation
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
Copy SMILES
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Affinity Data
Ki: 50.1nM
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Target
5-hydroxytryptamine receptor 4
(GUINEA PIG)
Janssen Research Foundation
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
Copy SMILES
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Affinity Data
Ki: 50.1nM
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Target
5-hydroxytryptamine receptor 6
(RAT)
F. Hoffmann-La Roche
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
Copy SMILES
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Affinity Data
Ki: 56nM
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Target
5-hydroxytryptamine receptor 6
(Homo sapiens (Human))
Jagiellonian University Collegium Medicum
Curated by
ChEMBL
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
Copy SMILES
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Affinity Data
Ki: 56nM
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Target
5-hydroxytryptamine receptor 6
(RAT)
F. Hoffmann-La Roche
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
Copy SMILES
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Affinity Data
Ki: 56.2nM
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Target
5-hydroxytryptamine receptor 4
(MOUSE)
Cnrs Upr 9023
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
Copy SMILES
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Affinity Data
Ki: 56.2nM
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Target
5-hydroxytryptamine receptor 2C
(Homo sapiens (Human))
Yamanouchi Pharmaceutical
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
Copy SMILES
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Affinity Data
Ki: 56.2nM
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Target
5-hydroxytryptamine receptor 4
(Homo sapiens (Human))
Monash University
Curated by
ChEMBL
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
Copy SMILES
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Affinity Data
Ki: 56.2nM
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Target
5-hydroxytryptamine receptor 6
(Homo sapiens (Human))
Jagiellonian University Collegium Medicum
Curated by
ChEMBL
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
Copy SMILES
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Affinity Data
Ki: 61nM
Assay Description:
Displacement of [3H]LSD from human recombinant 5-HT6 receptor expressed in CHO cells after 120 mins by scintillation counting
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Target
5-hydroxytryptamine receptor 2A
(Homo sapiens (Human))
Eli Lilly
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
Copy SMILES
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Affinity Data
Ki: 63.1nM
More data for this Ligand-Target Pair
Target Info
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Target
5-hydroxytryptamine receptor 6
(Homo sapiens (Human))
Jagiellonian University Collegium Medicum
Curated by
ChEMBL
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
Copy SMILES
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Affinity Data
Ki: 65nM
More data for this Ligand-Target Pair
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5-hydroxytryptamine receptor 6
(Homo sapiens (Human))
Jagiellonian University Collegium Medicum
Curated by
ChEMBL
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
Copy SMILES
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Affinity Data
Ki: 65nM
Assay Description:
Binding affinity towards human 5-hydroxytryptamine 6 receptor was evaluated using [3H]-LSD as radioligand
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5-hydroxytryptamine receptor 3A/3B
(Rattus norvegicus)
Universit£
Curated by
ChEMBL
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
Ki: 66nM
Assay Description:
Binding affinity for 5-hydroxytryptamine 3 receptor from rat cortex using [3H]BRL-43694 as radioligand
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5-hydroxytryptamine receptor 1F
(RAT)
University of Alberta
Curated by
PDSP K
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Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Ki: 67.6nM
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5-hydroxytryptamine receptor 6
(Homo sapiens (Human))
Jagiellonian University Collegium Medicum
Curated by
ChEMBL
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
Ki: 70nM
Assay Description:
Binding affinity to Homo sapiens (human) 5-HT6 receptor
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5-hydroxytryptamine receptor 6
(Homo sapiens (Human))
Jagiellonian University Collegium Medicum
Curated by
ChEMBL
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
Copy SMILES
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Affinity Data
Ki: 75nM
Assay Description:
Binding affinity for human 5-hydroxytryptamine 6 receptor expressed in HEK 293 human embryonic kidney cells, [3H]-lysergic acid diethylamide as radio...
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Target
5-hydroxytryptamine receptor 6
(Homo sapiens (Human))
Jagiellonian University Collegium Medicum
Curated by
ChEMBL
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
Ki: 78nM
Assay Description:
Binding affinity against human 5-hydroxytryptamine 6 receptor stably transfected to HEK 293 human embryonic kidney cells using [3H]-lysergic acid die...
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Target
5-hydroxytryptamine receptor 2C
(Homo sapiens (Human))
Yamanouchi Pharmaceutical
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
Ki: 79nM
Assay Description:
Displacement of [3H]mesulergine from human 5HT2C receptor expressed in tsA201 cell membranes after 1 hr by scintillation counting analysis
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Target
5-hydroxytryptamine receptor 4
(MOUSE)
Cnrs Upr 9023
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Ki: 79.4nM
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Target
5-hydroxytryptamine receptor 4
(GUINEA PIG)
Janssen Research Foundation
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Ki: 79.4nM
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Target
5-hydroxytryptamine receptor 4
(GUINEA PIG)
Janssen Research Foundation
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
Copy SMILES
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Ki: 79.4nM
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Target
5-hydroxytryptamine receptor 6
(RAT)
F. Hoffmann-La Roche
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
Copy SMILES
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Ki: 79.4nM
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Target
5-hydroxytryptamine receptor 4
(MOUSE)
Cnrs Upr 9023
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
Copy SMILES
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Ki: 79.4nM
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Target
5-hydroxytryptamine receptor 4
(MOUSE)
Cnrs Upr 9023
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
Copy SMILES
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Ki: 79.4nM
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5-hydroxytryptamine receptor 2A
(Rattus norvegicus (rat))
Alcon Research
Curated by
ChEMBL
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Ki: 83nM
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5-hydroxytryptamine receptor 6
(Homo sapiens (Human))
Jagiellonian University Collegium Medicum
Curated by
ChEMBL
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
Ki: 84nM
Assay Description:
Displacement of [3H]LSD from human 5HT6 receptor
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5-hydroxytryptamine receptor 3A/3B
(Rattus norvegicus)
Universit£
Curated by
ChEMBL
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
Ki: 87nM
Assay Description:
In vitro relaxation of carbachol pre-contracted rat oesophageal TMM.
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5-hydroxytryptamine receptor 2C
(Rattus norvegicus (Rat))
University of Alberta
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
Ki: 87.1nM
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5-hydroxytryptamine receptor 1A
(Rattus norvegicus (rat))
Emory University
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
Ki: 90nM
Assay Description:
Radioligand receptor binding studies were conducted in the rat brain.
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Target
5-hydroxytryptamine receptor 6
(MOUSE)
Cnrs
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
Ki: 95.5nM
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Target
5-hydroxytryptamine receptor 2A
(Rattus norvegicus (rat))
Alcon Research
Curated by
ChEMBL
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Ki: 96nM
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5-hydroxytryptamine receptor 6
(Homo sapiens (Human))
Jagiellonian University Collegium Medicum
Curated by
ChEMBL
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
Copy SMILES
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Affinity Data
Ki: 100nM
Assay Description:
Binding affinity to 5-Ht6 receptor (unknown origin)
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Target
5-hydroxytryptamine receptor 4
(GUINEA PIG)
Janssen Research Foundation
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
Ki: 100nM
Assay Description:
Displacement of [3H]GR-113808 from 5HT4 receptor in guinea pig striatum
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Target
5-hydroxytryptamine receptor 4
(GUINEA PIG)
Janssen Research Foundation
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
Copy SMILES
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Affinity Data
Ki: 100nM
Assay Description:
Displacement of [3H]GR113808 from 5HT4 receptor in guinea pig striatum
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Target
5-hydroxytryptamine receptor 4
(Homo sapiens (Human))
Monash University
Curated by
ChEMBL
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
Copy SMILES
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Ki: 100nM
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Target
5-hydroxytryptamine receptor 6
(Homo sapiens (Human))
Jagiellonian University Collegium Medicum
Curated by
ChEMBL
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
Copy SMILES
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Affinity Data
Ki: 100nM
Assay Description:
Binding affinity against 5-hydroxytryptamine 6 receptor
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Target
5-hydroxytryptamine receptor 1A
(Homo sapiens (Human))
University of Alberta
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Ki: 102nM
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Target
5-hydroxytryptamine receptor 1A
(Homo sapiens (Human))
University of Alberta
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
Copy SMILES
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Ki: 102nM
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Target
5-hydroxytryptamine receptor 4
(Homo sapiens (Human))
Monash University
Curated by
ChEMBL
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
Copy SMILES
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Affinity Data
Ki: 110nM
Assay Description:
Displacement of [3H]GR-113808 from human recombinant 5HT4b receptor expressed in HEK293 cells by scintillation counting
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Target
5-hydroxytryptamine receptor 3A/3B
(Rattus norvegicus)
Universit£
Curated by
ChEMBL
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
Copy SMILES
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Affinity Data
Ki: 120nM
Assay Description:
Inhibition of [3H]granisetron binding to 5-hydroxytryptamine 3 receptor of rat cortical membrane
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Target
5-hydroxytryptamine receptor 3A/3B
(Rattus norvegicus)
Universit£
Curated by
ChEMBL
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
Copy SMILES
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Affinity Data
Ki: 120nM
Assay Description:
Ability to displace [3H]granisetron specifically bound to 5-hydroxytryptamine 3 receptor in rat cortical membrane
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Target
5-hydroxytryptamine receptor 2A
(Homo sapiens (Human))
Eli Lilly
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
Copy SMILES
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Affinity Data
Ki: 120nM
Assay Description:
Displacement of [3H]ketanserin from human 5HT2A receptor expressed in human A549 cells
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Target
5-hydroxytryptamine receptor 2A
(Rattus norvegicus (rat))
Alcon Research
Curated by
ChEMBL
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Ki: 120nM
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Target
5-hydroxytryptamine receptor 2A
(Rattus norvegicus (rat))
Alcon Research
Curated by
ChEMBL
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
Copy SMILES
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Ki: 126nM
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Target
5-hydroxytryptamine receptor 1F
(MOUSE)
University of Alberta
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
Copy SMILES
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Affinity Data
Ki: 126nM
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Target
5-hydroxytryptamine receptor 4
(RAT)
Synaptic Pharmaceutical
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
Copy SMILES
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Ki: 126nM
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Target
5-hydroxytryptamine receptor 5A
(Homo sapiens (Human))
Virginia Commonwealth University
Curated by
ChEMBL
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
Copy SMILES
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Affinity Data
Ki: 126nM
Assay Description:
Binding affinity towards human 5-hydroxytryptamine 5A receptor was evaluated using [3H]-5-CT as radioligand
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5-hydroxytryptamine receptor 6
(Homo sapiens (Human))
Jagiellonian University Collegium Medicum
Curated by
ChEMBL
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
Copy SMILES
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Affinity Data
Ki: 126nM
Assay Description:
Binding affinity against 5-hydroxytryptamine 6 human cloned receptors in HeLa cells using [3H]LSD as radioligand
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Target
5-hydroxytryptamine receptor 5A
(Homo sapiens (Human))
Virginia Commonwealth University
Curated by
ChEMBL
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
Copy SMILES
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Affinity Data
Ki: 130nM
Assay Description:
Displacement of [3H]LSD from human recombinant 5-HT5a receptor in HEK293 cells after 120 mins by scintillation counting
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5-hydroxytryptamine receptor 2A
(Homo sapiens (Human))
Eli Lilly
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
Copy SMILES
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Affinity Data
Ki: 130nM
Assay Description:
Displacement of [3H]ketanserin from human 5HT2A receptor expressed in human HEK293 cells
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5-hydroxytryptamine receptor 2C
(Homo sapiens (Human))
Yamanouchi Pharmaceutical
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
Copy SMILES
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Affinity Data
Ki: 130nM
Assay Description:
Displacement of [3H]mesulergine form human cloned 5HT2C receptor expressed in african green monkey COS7 cells by scintillation spectroscopy
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Target
5-hydroxytryptamine receptor 1A
(Rattus norvegicus (rat))
Emory University
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
Copy SMILES
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Ki: 134nM
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Target
5-hydroxytryptamine receptor 4
(RAT)
Synaptic Pharmaceutical
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
Copy SMILES
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Ki: 145nM
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Target
5-hydroxytryptamine receptor 4
(RAT)
Synaptic Pharmaceutical
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
Copy SMILES
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Affinity Data
Ki: 145nM
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Target
5-hydroxytryptamine receptor 2A
(Homo sapiens (Human))
Eli Lilly
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
Copy SMILES
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Affinity Data
Ki: 150nM
Assay Description:
Displacement of [3H]INBMeO from human 5HT2A receptor expressed in human HEK293 cells
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Target
5-hydroxytryptamine receptor 5A
(MOUSE)
Virginia Commonwealth University
Curated by
ChEMBL
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
Copy SMILES
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Affinity Data
Ki: 150nM
Assay Description:
Binding affinity towards mouse 5-hydroxytryptamine 5A receptor
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Target
5-hydroxytryptamine receptor 6
(RAT)
F. Hoffmann-La Roche
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
Copy SMILES
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Affinity Data
Ki: 151nM
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Target
5-hydroxytryptamine receptor 6
(RAT)
F. Hoffmann-La Roche
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
Copy SMILES
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Ki: 151nM
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Target
5-hydroxytryptamine receptor 4
(RAT)
Synaptic Pharmaceutical
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
Copy SMILES
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Affinity Data
Ki: 158nM
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Target
5-hydroxytryptamine receptor 4
(Homo sapiens (Human))
Monash University
Curated by
ChEMBL
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
Copy SMILES
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Affinity Data
Ki: 159nM
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Target
5-hydroxytryptamine receptor 2C
(Rattus norvegicus (Rat))
University of Alberta
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
Copy SMILES
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Affinity Data
Ki: 159nM
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Target
5-hydroxytryptamine receptor 2C
(Rattus norvegicus (Rat))
University of Alberta
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
Copy SMILES
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Affinity Data
Ki: 159nM
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Target
5-hydroxytryptamine receptor 2A
(Homo sapiens (Human))
Eli Lilly
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
Copy SMILES
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Affinity Data
Ki: 160nM
Assay Description:
Displacement of [3H]INBMeO from human 5HT2A receptor expressed in human A549 cells
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Target
5-hydroxytryptamine receptor 5A
(Homo sapiens (Human))
Virginia Commonwealth University
Curated by
ChEMBL
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
Copy SMILES
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Affinity Data
Ki: 170nM
Assay Description:
Displacement of [3H]LSD from human 5HT5A receptor
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Target
5-hydroxytryptamine receptor 4
(RAT)
Synaptic Pharmaceutical
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
Copy SMILES
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Affinity Data
Ki: 187nM
Assay Description:
Binding affinity towards 5-hydroxytryptamine 4 receptor was determined in rat striatal membranes using [3H]GR-113808 as radioligand
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Target
5-hydroxytryptamine receptor 4
(RAT)
Synaptic Pharmaceutical
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
Copy SMILES
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Ki: 200nM
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Target
5-hydroxytryptamine receptor 4
(RAT)
Synaptic Pharmaceutical
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
Copy SMILES
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Affinity Data
Ki: 200nM
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Target
5-hydroxytryptamine receptor 2C
(Homo sapiens (Human))
Yamanouchi Pharmaceutical
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
Copy SMILES
Copy InChI
Affinity Data
Ki: 214nM
Assay Description:
Displacement of [3H]-mesulergine from 5HT2C receptor expressed in CHO cell membranes after 90 mins by scintillation counting
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Target
5-hydroxytryptamine receptor 2A
(Homo sapiens (Human))
Eli Lilly
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
Copy SMILES
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Affinity Data
Ki: 219nM
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Target
5-hydroxytryptamine receptor 4
(GUINEA PIG)
Janssen Research Foundation
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
Copy SMILES
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Affinity Data
Ki: 230nM
Assay Description:
The compound was tested for their binding affinity towards 5-hydroxytryptamine 4 receptor from guinea pig striatum using [3H]GR-113808 as radioligand...
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Target
5-hydroxytryptamine receptor 6
(RAT)
F. Hoffmann-La Roche
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
Copy SMILES
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Ki: 234nM
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Target
5-hydroxytryptamine receptor 5B
(RAT)
University of Alberta
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
Copy SMILES
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Ki: 239nM
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Target
5-hydroxytryptamine receptor 5A
(RAT)
University of Alberta
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
Copy SMILES
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Ki: 240nM
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Target
5-hydroxytryptamine receptor 4
(Homo sapiens (Human))
Monash University
Curated by
ChEMBL
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
Copy SMILES
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Affinity Data
Ki: 246nM
Assay Description:
Binding affinity to recombinant human brain 5HT4 receptor by radio ligand binding assay
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Target
5-hydroxytryptamine receptor 5A
(Homo sapiens (Human))
Virginia Commonwealth University
Curated by
ChEMBL
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
Copy SMILES
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Affinity Data
Ki: 250nM
Assay Description:
Binding affinity for rodent 5-hydroxytryptamine 5A receptor
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Target
5-hydroxytryptamine receptor 5A
(MOUSE)
Virginia Commonwealth University
Curated by
ChEMBL
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
Copy SMILES
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Affinity Data
Ki: 251nM
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Target
5-hydroxytryptamine receptor 2A
(Rattus norvegicus (rat))
Alcon Research
Curated by
ChEMBL
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
Copy SMILES
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Ki: 251nM
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Target
5-hydroxytryptamine receptor 5A
(MOUSE)
Virginia Commonwealth University
Curated by
ChEMBL
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
Copy SMILES
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Affinity Data
Ki: 251nM
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Target
5-hydroxytryptamine receptor 5A
(MOUSE)
Virginia Commonwealth University
Curated by
ChEMBL
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
Copy SMILES
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Affinity Data
Ki: 251nM
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Target
5-hydroxytryptamine receptor 5B
(MOUSE)
University of Alberta
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
Copy SMILES
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Affinity Data
Ki: 251nM
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Target
5-hydroxytryptamine receptor 5A
(MOUSE)
Virginia Commonwealth University
Curated by
ChEMBL
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
Copy SMILES
Copy InChI
Affinity Data
Ki: 251nM
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Target
5-hydroxytryptamine receptor 5B
(MOUSE)
University of Alberta
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
Copy SMILES
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Affinity Data
Ki: 251nM
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Target
5-hydroxytryptamine receptor 4
(Homo sapiens (Human))
Monash University
Curated by
ChEMBL
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
Copy SMILES
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Ki: 251nM
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5-hydroxytryptamine receptor 3A
(Mus musculus (house mouse))
University of Alberta
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Ki: 269nM
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5-hydroxytryptamine receptor 2A
(Rattus norvegicus (rat))
Alcon Research
Curated by
ChEMBL
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Ki: 270nM
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5-hydroxytryptamine receptor 3A
(Mus musculus (house mouse))
University of Alberta
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Ki: 292nM
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5-hydroxytryptamine receptor 4
(Homo sapiens (Human))
Monash University
Curated by
ChEMBL
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Ki: 316nM
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5-hydroxytryptamine receptor 4
(Homo sapiens (Human))
Monash University
Curated by
ChEMBL
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Ki: 316nM
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5-hydroxytryptamine receptor 4
(Homo sapiens (Human))
Monash University
Curated by
ChEMBL
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Ki: 316nM
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5-hydroxytryptamine receptor 2A
(Homo sapiens (Human))
Eli Lilly
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
Ki: 320nM
Assay Description:
Displacement of [3H]ketanserin from human 5HT2A receptor expressed in tsA201 cell membranes after 1 hr by scintillation counting analysis
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5-hydroxytryptamine receptor 2A
(Homo sapiens (Human))
Eli Lilly
Curated by
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i
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Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
Ki: 320nM
Assay Description:
Displacement of [3H]methylspiperone form human cloned 5HT2A receptor expressed in african green monkey COS7 cells by scintillation spectroscopy
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5-hydroxytryptamine receptor 3A/3B
(Rattus norvegicus)
Universit£
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ChEMBL
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Ki: 320nM
Assay Description:
Binding affinity of the compound was measured on 5-hydroxytryptamine 3 receptor in NG-108 cells labeled with [3H]-GR-65,630
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5-hydroxytryptamine receptor 4
(Homo sapiens (Human))
Monash University
Curated by
ChEMBL
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Ki: 330nM
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5-hydroxytryptamine receptor 2A
(Homo sapiens (Human))
Eli Lilly
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Ki: 341nM
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Target
5-hydroxytryptamine receptor 3A
(Mus musculus (house mouse))
University of Alberta
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
Ki: 361nM
Assay Description:
The binding affinity was measured for 5-hydroxytryptamine 3 receptor on NG 108-15 cell line of mouse neuroblastoma-glioma cells in presence of [3H]5 ...
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5-hydroxytryptamine receptor 3A/3B
(Rattus norvegicus)
Universit£
Curated by
ChEMBL
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
Ki: 390nM
Assay Description:
The ability to inhibit [3H]GR-65630 binding to 5-hydroxytryptamine 3 receptor in rat brain cortices
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5-hydroxytryptamine receptor 2A
(Homo sapiens (Human))
Eli Lilly
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
Ki: 398nM
Assay Description:
Binding affinity against 5-hydroxytryptamine 2A receptor human cloned receptors in HEK 293 cells using [3H]ketanserin as radioligand
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5-hydroxytryptamine receptor 2C
(Homo sapiens (Human))
Yamanouchi Pharmaceutical
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Ki: 445nM
Assay Description:
Displacement of [3H]-mesulergine from 5HT2C receptor expressed in CHO cell membranes using 11 concentration of ligand after 90 mins by scintillation ...
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5-hydroxytryptamine receptor 2A
(Rattus norvegicus (rat))
Alcon Research
Curated by
ChEMBL
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Ki: 479nM
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5-hydroxytryptamine receptor 4
(Homo sapiens (Human))
Monash University
Curated by
ChEMBL
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Ki: 482nM
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Target
5-hydroxytryptamine receptor 3A
(GUINEA PIG)
Syntex Discovery Research
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Ki: 495nM
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5-hydroxytryptamine receptor 2A/2B/2C
(Mus musculus (Mouse))
Polytechnic University
Curated by
ChEMBL
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Ki: 500nM
Assay Description:
Binding affinity towards 5-hydroxytryptamine 2 receptor by the displacement of [3H]-ketanserin in mouse cerebral cortex
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5-hydroxytryptamine receptor 4
(Homo sapiens (Human))
Monash University
Curated by
ChEMBL
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Ki: 500nM
Assay Description:
Displacement of [N-methyl-3H]GR113808 from human 5HT4 receptor expressed in HEK293 cells
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Target
5-hydroxytryptamine receptor 2A
(Homo sapiens (Human))
Eli Lilly
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
Ki: 510nM
Assay Description:
Binding affinity was measured on 5-hydroxytryptamine 2A receptor in GF6 cells transfected with human 5-HT2A gene labeled with [3H]-ketanserin
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Target
Serotonin 2 (5-HT2) receptor
(RAT)
TBA
Curated by
ChEMBL
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Ki: 560nM
Assay Description:
Binding affinity to rat cortical membranes at 5-hydroxytryptamine 2 (5-HT2) receptor using [3H]KET as a radioligand
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5-hydroxytryptamine receptor 2A
(Rattus norvegicus (rat))
Alcon Research
Curated by
ChEMBL
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Ki: 600nM
Assay Description:
Binding affinity against human progesterone receptor (hPR) in a competitive binding assay
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5-hydroxytryptamine receptor 2A
(Homo sapiens (Human))
Eli Lilly
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Ki: 603nM
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5-hydroxytryptamine receptor 2C
(Homo sapiens (Human))
Yamanouchi Pharmaceutical
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Ki: 656nM
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5-hydroxytryptamine receptor 2A
(Homo sapiens (Human))
Eli Lilly
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
Ki: 690nM
Assay Description:
Displacement of [N-methyl-3H]LSD from human 5HT2A receptor expressed in HEK293 cells
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5-hydroxytryptamine receptor 2A
(Rattus norvegicus (rat))
Alcon Research
Curated by
ChEMBL
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Ki: 708nM
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Target
Sodium-dependent serotonin transporter
(Rattus norvegicus (rat))
Universit£
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ChEMBL
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Ki: 740nM
Assay Description:
Ability to displace [3H]paroxetine bound to Serotonin transporter receptor in rat forebrain
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Target
Sodium-dependent serotonin transporter
(Rattus norvegicus (rat))
Universit£
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ChEMBL
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Ki: 740nM
Assay Description:
Binding affinity towards Serotonin transporter was determined in rat forebrain membrane
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Target
5-hydroxytryptamine receptor 2B
(BOVINE)
Stanford University
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Ki: 750nM
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Target
Serotonin 2 (5-HT2) receptor
(RAT)
TBA
Curated by
ChEMBL
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
Ki: 930nM
Assay Description:
Effect on plasma amine oxidase (0.1 uM) after 15 min of incubation at pH 7.2
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Target
Serotonin 2 (5-HT2) receptor
(RAT)
TBA
Curated by
ChEMBL
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
Ki: 950nM
Assay Description:
Binding affinity was determined against 5-hydroxytryptamine 2 receptor from male Sprague-Dawley rat brain.
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Target
Serotonin 2 (5-HT2) receptor
(RAT)
TBA
Curated by
ChEMBL
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
Ki: 977nM
Assay Description:
Displacement of [3H]ketanserin from 5-hydroxytryptamine 2 receptor of rat frontal cortex homogenate
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Target
Norepinephrine transporter
(RAT)
Novo Industri
Curated by
PDSP K
i
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Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Ki: 1.00E+3nM
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Target
5-hydroxytryptamine receptor 4
(Homo sapiens (Human))
Monash University
Curated by
ChEMBL
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
Ki: 1.05E+3nM ΔG°: -34.1kJ/mole EC50: 12nM
pH: 7.4 T: 2°C
Assay Description:
Radioligand binding studies were performed in buffer contains test compound, [3H]-GR113808, and receptor C6 glial cell membrane preparation. Nonspeci...
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Target
5-hydroxytryptamine receptor 5A
(MOUSE)
Virginia Commonwealth University
Curated by
ChEMBL
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Ki: 1.10E+3nM
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Target
5-hydroxytryptamine receptor 4
(Homo sapiens (Human))
Monash University
Curated by
ChEMBL
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Ki: 1.15E+3nM
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Target
5-hydroxytryptamine receptor 2A
(Rattus norvegicus (rat))
Alcon Research
Curated by
ChEMBL
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
Ki: 1.26E+3nM
Assay Description:
Displacement of [3H]ketanserin from 5HT2A receptor in rat cortex
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Target
5-hydroxytryptamine receptor 2A
(Rattus norvegicus (rat))
Alcon Research
Curated by
ChEMBL
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
Ki: 1.26E+3nM
Assay Description:
Displacement of [3H]ketanserin from 5HT2A receptor in rat cortex
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Target
5-hydroxytryptamine receptor 2B
(Mus musculus (Mouse))
University of Alberta
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Ki: 1.26E+3nM
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Target
5-hydroxytryptamine receptor 5B
(RAT)
University of Alberta
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Ki: 1.32E+3nM
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Target
5-hydroxytryptamine receptor 5A
(RAT)
University of Alberta
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Ki: 1.33E+3nM
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Target
D(2) dopamine receptor
(Rattus norvegicus (rat))
Schering-Plough
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
Ki: 1.66E+3nM
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Target
Synaptic vesicular amine transporter
(Homo sapiens (Human))
Organix
Curated by
ChEMBL
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
Ki: 2.29E+3nM
Assay Description:
Displacement of [3H](+)-syn-Ethyl 1-(2-(2,4-Dioxo-1,2-dihydroquinazolin-3(4H)-yl)ethyl)-4-(4-fluorophenyl)piperidine-3-carboxylate from human VMAT2 e...
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Target
D(3) dopamine receptor
(Rattus norvegicus (Rat))
University Of Pennsylvania
Curated by
ChEMBL
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
Ki: 2.34E+3nM
Assay Description:
Tested for binding affinity against dopamine receptor D3 expressed in Sf9 cells.
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Target
Sodium-dependent dopamine transporter
(Rattus norvegicus (rat))
Nih
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Ki: 2.70E+3nM
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Target
Serotonin 2 (5-HT2) receptor
(RAT)
TBA
Curated by
ChEMBL
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
Ki: 2.95E+3nM
Assay Description:
Binding affinity to 5-hydroxytryptamine 2 receptor in rat frontal cortical membranes by [3H]- KET displacement.
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Target
5-hydroxytryptamine receptor 2A
(Rattus norvegicus (rat))
Alcon Research
Curated by
ChEMBL
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Ki: 2.96E+3nM
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Target
D(1B) dopamine receptor
(Homo sapiens (Human))
University of Toronto
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
Ki: 3.00E+3nM
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Target
Norepinephrine transporter
(RAT)
Novo Industri
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Ki: 3.01E+3nM
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Target
Dopamine receptor D4
(CANINE)
University of Toronto
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Ki: 4.18E+3nM
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Target
D(1A) dopamine receptor
(RAT)
UniversitÉ
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
Ki: 5.00E+3nM
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Target
Synaptic vesicular amine transporter
(Homo sapiens (Human))
Organix
Curated by
ChEMBL
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
Ki: 7.69E+3nM
Assay Description:
Displacement of [3H]reserpine from human VMAT2 expressed in HEK293 cell membranes incubated for 60 mins by scintillation counting method
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Target
D(2) dopamine receptor
(Rattus norvegicus (rat))
Schering-Plough
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
Ki: 7.95E+3nM
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Target
D(2) dopamine receptor
(Homo sapiens (Human))
University of Toronto
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
Ki: >1.00E+4nM
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Target
D(2) dopamine receptor
(Rattus norvegicus (rat))
Schering-Plough
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
Copy SMILES
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Affinity Data
Ki: >1.00E+4nM
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Target
D(1A) dopamine receptor
(Homo sapiens (Human))
Sri International
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
Ki: >1.00E+4nM
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Target
D(2) dopamine receptor
(Homo sapiens (Human))
University of Toronto
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
Copy SMILES
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Affinity Data
Ki: >1.00E+4nM
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Target
Sodium-dependent dopamine transporter
(Rattus norvegicus (rat))
Nih
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
Copy SMILES
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Affinity Data
Ki: >1.00E+4nM
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Target
Norepinephrine transporter
(RAT)
Novo Industri
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
Copy SMILES
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Affinity Data
Ki: >1.00E+4nM
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Target
Sodium-dependent dopamine transporter
(Homo sapiens (Human))
University of Toronto
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
Copy SMILES
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Affinity Data
Ki: >1.00E+4nM
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Target
Sodium-dependent dopamine transporter
(Homo sapiens (Human))
University of Toronto
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
Copy SMILES
Copy InChI
Affinity Data
Ki: >1.00E+4nM
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Target
Sodium-dependent dopamine transporter
(Homo sapiens (Human))
University of Toronto
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
Copy SMILES
Copy InChI
Affinity Data
Ki: >1.00E+4nM
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Target
5-hydroxytryptamine receptor 1F
(Homo sapiens (Human))
Janssen Research Foundation
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
Copy SMILES
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Affinity Data
Ki: >1.00E+4nM
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Target
Melatonin receptor type 1A
(Sheep)
Massachusetts General Hospital
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
Copy SMILES
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Ki: >1.00E+4nM
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Target
D(2) dopamine receptor
(Rattus norvegicus (rat))
Schering-Plough
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
Copy SMILES
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Affinity Data
Ki: >1.00E+4nM
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Target
5-hydroxytryptamine receptor 3A
(GUINEA PIG)
Syntex Discovery Research
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
Copy SMILES
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Affinity Data
Ki: >1.00E+4nM
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Target
5-hydroxytryptamine receptor 3A
(GUINEA PIG)
Syntex Discovery Research
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
Copy SMILES
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Affinity Data
Ki: >1.00E+4nM
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Target
Melatonin receptor type 1B
(Homo sapiens (Human))
Massachusetts General Hospital
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
Copy SMILES
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Affinity Data
Ki: >1.00E+4nM
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Target
D(2) dopamine receptor
(CANINE)
University of Pennsylvania
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
Copy SMILES
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Affinity Data
Ki: >1.00E+4nM
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Target
Alpha-2C adrenergic receptor
(RAT)
University of California
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
Copy SMILES
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Affinity Data
Ki: >1.00E+4nM
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Target
Sodium-dependent dopamine transporter
(Rattus norvegicus (rat))
Nih
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
Copy SMILES
Copy InChI
Affinity Data
Ki: >1.00E+4nM
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Target
D(2) dopamine receptor
(Rattus norvegicus (rat))
Schering-Plough
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
Copy SMILES
Copy InChI
Affinity Data
Ki: >1.00E+4nM
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Target Info
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Target
5-hydroxytryptamine receptor 1A
(Homo sapiens (Human))
University of Alberta
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
Copy SMILES
Copy InChI
Affinity Data
Ki: 1.00E+4nM
Assay Description:
Displacement of [3H]WAY100635 from human recombinant 5HT1A receptor
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Alpha-1A adrenergic receptor
(Rattus norvegicus (Rat))
TBA
Curated by
PDSP K
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Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Ki: 1.80E+4nM
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Target
Alpha-1A adrenergic receptor
(Rattus norvegicus (Rat))
TBA
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Ki: 2.30E+4nM
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Melatonin receptor type 1B
(Homo sapiens (Human))
Massachusetts General Hospital
Curated by
PDSP K
i
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Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
Ki: >1.00E+5nM
Assay Description:
Inhibition of 2-[125I]-Iodomelatonin binding to human Melatonin receptor type 1B expressed in CHO cells
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Melatonin receptor type 1A
(Homo sapiens (Human))
TBA
Curated by
ChEMBL
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Ki: >1.00E+5nM
Assay Description:
Displacement of 2-[125I]-Iodomelatonin from human Melatonin receptor type 1A expressed in CHO cells
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Solute carrier family 22 member 2
(RAT)
Kyoto University Hospital
Curated by
ChEMBL
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
Ki: 2.42E+5nM
Assay Description:
TP_TRANSPORTER: inhibition of TEA uptake in OCT2-expressing MDCK cells
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Solute carrier family 22 member 1
(RAT)
Kyoto University Hospital
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ChEMBL
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
Ki: 3.90E+5nM
Assay Description:
TP_TRANSPORTER: inhibition of TEA uptake in OCT1-expressing MDCK cells
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Target
Synaptic vesicular amine transporter
(Homo sapiens (Human))
Organix
Curated by
ChEMBL
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
Ki: 6.40E+5nM
Assay Description:
Displacement of [3H]DHTB from human VMAT2 expressed in HEK293 cell membranes incubated for 90 mins by microbeta scintillation counting method
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D(2) dopamine receptor
(Homo sapiens (Human))
University of Toronto
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PDSP K
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Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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IC50: 0nM
Assay Description:
Agonist required to inhibit Dopamine receptor D2 photoinactivation by 50% with Iodazidoclebopride using [3H]-Spiperone
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5-hydroxytryptamine receptor 7
(Homo sapiens (Human))
University Of Namur
Curated by
ChEMBL
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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IC50: 0.25nM
Assay Description:
Displacement of [3H]LSD from human recombinant 5-HT7 receptor expressed in CHO cells
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5-hydroxytryptamine receptor 7
(Homo sapiens (Human))
University Of Namur
Curated by
ChEMBL
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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IC50: 0.25nM
Assay Description:
Displacement of [3H]LSD from human recombinant 5HT7 receptor expressed in CHO cells measured after 120 mins by scintillation counting method
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5-hydroxytryptamine receptor 7
(Homo sapiens (Human))
University Of Namur
Curated by
ChEMBL
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
IC50: 0.470nM
Assay Description:
Displacement of [3H]LSD from human recombinant 5-HT7 receptor expressed in CHO cells after 120 mins by scintillation counting
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5-hydroxytryptamine receptor 2A
(Rattus norvegicus (rat))
Alcon Research
Curated by
ChEMBL
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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IC50: 0.900nM
Assay Description:
In vitro inhibition of [125I]DOI binding to 5-hydroxytryptamine 2A receptor in rat cerebral cortex
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5-hydroxytryptamine receptor 2A
(Rattus norvegicus (rat))
Alcon Research
Curated by
ChEMBL
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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IC50: 0.940nM
Assay Description:
Inhibition of [125I]DOI binding to 5HT2A receptor in rat cerebral cortex
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5-hydroxytryptamine receptor 1A
(Homo sapiens (Human))
University of Alberta
Curated by
PDSP K
i
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Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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IC50: 1.20nM
Assay Description:
In vitro inhibitory concentration required against [3H]8-OH-DPAT binding to cloned human 5-hydroxytryptamine 1A receptor
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5-hydroxytryptamine receptor 2C
(Homo sapiens (Human))
Yamanouchi Pharmaceutical
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PDSP K
i
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Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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IC50: 1.30nM
Assay Description:
Antagonist activity at recombinant human 5-HT2C expressed in human U2OS cells by pathhunter beta-arrestin assay
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5-hydroxytryptamine receptor 1A
(Homo sapiens (Human))
University of Alberta
Curated by
PDSP K
i
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Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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IC50: 2nM
Assay Description:
Compound was tested in vitro for the inhibition of [3H]-DPAT (1 nM) binding to 5-hydroxytryptamine 1A receptor from bovine hippocampus
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5-hydroxytryptamine receptor 1A
(Homo sapiens (Human))
University of Alberta
Curated by
PDSP K
i
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Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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IC50: 2nM
Assay Description:
Compound was tested in vitro for the inhibition of azido-[125I]-IPAPP (0.25 nM) binding to 5-HT1A receptor from bovine hippocampus
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5-hydroxytryptamine receptor 7
(Homo sapiens (Human))
University Of Namur
Curated by
ChEMBL
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
IC50: 2.55nM
Assay Description:
Displacement of [3H]LSD from human 5HT7 receptor expressed in CHO cells
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5-hydroxytryptamine receptor 1A
(Rattus norvegicus (rat))
Emory University
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
IC50: 2.60nM
Assay Description:
Inhibition of radiolabeled [3H]-8-OH-DPAT ligand binding to 5-hydroxytryptamine 1A receptor
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5-hydroxytryptamine receptor 1D
(RAT)
University of Alberta
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PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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IC50: 3nM
Assay Description:
Binding affinity of the compound was measured against serotonin 5-hydroxytryptamine 1D receptor
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5-hydroxytryptamine receptor 1A
(Rattus norvegicus (rat))
Emory University
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
IC50: 3nM
Assay Description:
In vitro inhibitory concentration against radioligand [3H]-8-OH-DPAT binding to 5-hydroxytryptamine 1A receptor in rat hippocampal membrane.
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Target
5-hydroxytryptamine receptor 1D
(Homo sapiens (Human))
Theravance
Curated by
ChEMBL
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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IC50: 3nM
Assay Description:
Tested in vitro for receptor binding affinity to 5-hydroxytryptamine 1D receptor in bovine caudate using [3H]-5-HT radioligand
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5-hydroxytryptamine receptor 1D
(GUINEA PIG)
Pfizer
Curated by
ChEMBL
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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IC50: 3nM
Assay Description:
Effect of the compound on forskolin stimulated adenylate cyclase activity at 5-hydroxytryptamine 1A receptor of guinea pig hippocampus.
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5-hydroxytryptamine receptor 1D
(Homo sapiens (Human))
Theravance
Curated by
ChEMBL
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
IC50: 3nM
Assay Description:
Inhibitory activity against 5-hydroxytryptamine 1D receptor of bovine caudate using [3H]-5-HT as the radioligand
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Target
5-hydroxytryptamine receptor 4
(RAT)
Synaptic Pharmaceutical
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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IC50: 3.70nM
Assay Description:
5-hydroxytryptamine 4 receptor agonist activity was determined by the relaxation of the carbachol-contracted rat esophageal tunica muscularis mucosae
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5-hydroxytryptamine receptor 1B
(Rattus norvegicus (Rat))
University of Alberta
Curated by
PDSP K
i
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Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
IC50: 4.60nM
Assay Description:
Inhibition of radiolabeled [3H]-5-HT ligand binding to 5-hydroxytryptamine 1B receptor
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5-hydroxytryptamine receptor 1B
(Rattus norvegicus (Rat))
University of Alberta
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
IC50: 4.90nM
Assay Description:
Displacement of [125I]CYP from rat cerebral cortex 5HT1B receptor measured after 120 mins by scintillation counting method
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5-hydroxytryptamine receptor 1B
(Rattus norvegicus (Rat))
University of Alberta
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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IC50: 4.90nM
Assay Description:
Displacement of [125I]CYP from rat cerebral cortex 5-HT1B receptor in the presence of isoproternol
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5-hydroxytryptamine receptor 1B
(Homo sapiens (Human))
University of Alberta
Curated by
PDSP K
i
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Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
IC50: 5nM
Assay Description:
Binding affinity of the compound against 5-hydroxytryptamine 1B receptor
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5-hydroxytryptamine receptor 1A
(Mus musculus (Mouse))
Polytechnic University
Curated by
ChEMBL
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
IC50: 5nM
Assay Description:
Inhibitory activity towards 5-hydroxytryptamine 1A receptor by the displacement of [3H]-8-OH-DPAT in mouse hippocampus
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5-hydroxytryptamine receptor 1B
(Rattus norvegicus (Rat))
University of Alberta
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
IC50: 5nM
Assay Description:
Inhibitory activity against 5-hydroxytryptamine 1B receptor of rat cortex using [3H]-5-HT as the radioligand.
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5-hydroxytryptamine receptor 1A
(Homo sapiens (Human))
University of Alberta
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
IC50: 5.20nM
Assay Description:
Binding affinity of the compound against 5-hydroxytryptamine 1A receptor
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5-hydroxytryptamine receptor 1A
(Rattus norvegicus (rat))
Emory University
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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IC50: 5.20nM
Assay Description:
Binding affinity of the compound was measured against serotonin 5-hydroxytryptamine 1A receptor
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5-hydroxytryptamine receptor 1A
(Rattus norvegicus (rat))
Emory University
Curated by
PDSP K
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Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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IC50: 5.20nM
Assay Description:
Tested in vitro for receptor binding affinity to 5-hydroxytryptamine 1A receptor in rat cortex using [3H]-OH-DPAT radioligand
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5-hydroxytryptamine receptor 1A
(Rattus norvegicus (rat))
Emory University
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PDSP K
i
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Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
IC50: 5.20nM
Assay Description:
Displacement of [3H]-8-OH-DPAT from rat cortex 5-hydroxytryptamine 1A receptor
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5-hydroxytryptamine receptor 1A
(Homo sapiens (Human))
University of Alberta
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Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
IC50: 5.60nM
Assay Description:
Compound was tested in vitro for the inhibition of [125I]-IPAPP (0.25 nM) binding to 5-HT1A receptor from bovine hippocampus
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5-hydroxytryptamine receptor 1A
(Homo sapiens (Human))
University of Alberta
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i
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Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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IC50: 6nM
Assay Description:
Compound was tested in vitro for the inhibition of [3H]-5-HT (2 nM) binding to 5-hydroxytryptamine 1A receptor from bovine hippocampus
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Target
5-hydroxytryptamine receptor 1D
(Sus scrofa)
Merck Sharp & Dohme Research Laboratories
Curated by
ChEMBL
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
IC50: 10nM
Assay Description:
Binding activity against 5-hydroxytryptamine 1D receptor from pig caudate membrane using [3H]5-HT as radioligand
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5-hydroxytryptamine receptor 1D
(Sus scrofa)
Merck Sharp & Dohme Research Laboratories
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ChEMBL
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
IC50: 10nM
Assay Description:
Compound was tested for the displacement of [3H]-5-HT to 5-hydroxytryptamine 1D receptor recognition sites in pig caudate membranes
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5-hydroxytryptamine receptor 1D
(Sus scrofa)
Merck Sharp & Dohme Research Laboratories
Curated by
ChEMBL
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
IC50: 10nM
Assay Description:
Displacement of radioligand [3H]5-HT binding to 5-hydroxytryptamine 1D receptor in pig caudate membrane
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Target
5-hydroxytryptamine receptor 1A/1B/1D/1F
(RAT)
TBA
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ChEMBL
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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IC50: 20nM
Assay Description:
Inhibition of human erythrocyte carbonic anhydrase II
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Target
Serotonin 2 (5-HT2) receptor
(RAT)
TBA
Curated by
ChEMBL
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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IC50: 20nM
Assay Description:
Binding affinity of the compound against 5-hydroxytryptamine 1A receptor
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5-hydroxytryptamine receptor 6
(Homo sapiens (Human))
Jagiellonian University Collegium Medicum
Curated by
ChEMBL
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
IC50: 27.5nM
Assay Description:
Displacement of [3H]LSD from human 5HT6 receptor by scintillation counting
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5-hydroxytryptamine receptor 2A
(Homo sapiens (Human))
Eli Lilly
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Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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IC50: 28nM
Assay Description:
Antagonist activity at recombinant human 5-HT2A expressed in human U2OS cells by pathhunter beta-arrestin assay
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5-hydroxytryptamine receptor 2C
(Rattus norvegicus (Rat))
University of Alberta
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Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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IC50: 42nM
Assay Description:
Inhibition of radiolabeled [3H]mesulergine ligand binding to 5-hydroxytryptamine 2C receptor
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5-hydroxytryptamine receptor 5A
(Homo sapiens (Human))
Virginia Commonwealth University
Curated by
ChEMBL
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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IC50: 79nM
Assay Description:
Inhibitory concentration against human Adenosine A3 receptor expressed in HEK293 cells using 0.1 nM [3H]AB-MECA
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5-hydroxytryptamine receptor 2C
(Homo sapiens (Human))
Yamanouchi Pharmaceutical
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PDSP K
i
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Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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IC50: 81nM
Assay Description:
inhibitory activity against 5-hydroxytryptamine 1C receptor of pig choroid plexus using [3H]-mesulergine as the radioligand
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5-hydroxytryptamine receptor 2C
(Rattus norvegicus (Rat))
University of Alberta
Curated by
PDSP K
i
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Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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IC50: 81nM
Assay Description:
Binding affinity of the compound against 5-hydroxytryptamine 1C receptor
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Synaptic vesicular amine transporter
(Mus musculus)
Organix
Curated by
ChEMBL
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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IC50: 98nM
Assay Description:
Inhibition of VMAT2 in C57Bl/6J mouse striatal membranes assessed as reduction in [3H[-5HT uptake pre-incubated for 10 mins before [3H[-5HT addition ...
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5-hydroxytryptamine receptor 6
(Homo sapiens (Human))
Jagiellonian University Collegium Medicum
Curated by
ChEMBL
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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IC50: 120nM
Assay Description:
Displacement of [3H]LSD from human recombinant 5-HT6 receptor expressed in CHO cells
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5-hydroxytryptamine receptor 6
(Homo sapiens (Human))
Jagiellonian University Collegium Medicum
Curated by
ChEMBL
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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IC50: 120nM
Assay Description:
Displacement of [3H]LSD from human recombinant 5HT6 receptor expressed in CHO cells measured after 120 mins by scintillation counting method
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5-hydroxytryptamine receptor 6
(Homo sapiens (Human))
Jagiellonian University Collegium Medicum
Curated by
ChEMBL
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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IC50: 130nM
Assay Description:
Displacement of [3H]LSD from human recombinant 5-HT6 receptor expressed in CHO cells after 120 mins by scintillation counting
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Target
5-hydroxytryptamine receptor 4
(RAT)
Synaptic Pharmaceutical
Curated by
PDSP K
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Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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IC50: 147nM
Assay Description:
Inhibition of radiolabeled [3H]GR-113808 ligand binding to 5-hydroxytryptamine 4 receptor
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5-hydroxytryptamine receptor 5A
(Homo sapiens (Human))
Virginia Commonwealth University
Curated by
ChEMBL
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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IC50: 180nM
Assay Description:
Displacement of [3H]LSD from human recombinant 5-HT5A receptor expressed in HEK293 cells
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5-hydroxytryptamine receptor 5A
(Homo sapiens (Human))
Virginia Commonwealth University
Curated by
ChEMBL
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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IC50: 180nM
Assay Description:
Displacement of [3H]LSD from human recombinant 5HT5A receptor expressed in HEK293 cells measured after 120 mins by scintillation counting method
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5-hydroxytryptamine receptor 5A
(Homo sapiens (Human))
Virginia Commonwealth University
Curated by
ChEMBL
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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IC50: 260nM
Assay Description:
Displacement of [3H]LSD from human recombinant 5-HT5a receptor in HEK293 cells after 120 mins by scintillation counting
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5-hydroxytryptamine receptor 4
(Homo sapiens (Human))
Monash University
Curated by
ChEMBL
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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IC50: 323nM
Assay Description:
Displacement of [3H]-GR 113808 from recombinant human brain 5HT4 receptor measured after 60 mins by radio ligand binding assay
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5-hydroxytryptamine receptor 2A
(Rattus norvegicus (rat))
Alcon Research
Curated by
ChEMBL
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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IC50: 600nM
Assay Description:
Displacement of [3H]-ketanserin from 5HT2A receptor high affinity component in rat brain cortical membranes after 15 mins by competition assay
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5-hydroxytryptamine receptor 2A/2B/2C
(Mus musculus (Mouse))
Polytechnic University
Curated by
ChEMBL
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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IC50: 680nM
Assay Description:
Inhibitory activity towards 5-hydroxytryptamine 2 receptor by the displacement of [3H]ketanserin in mouse cerebral cortex
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5-hydroxytryptamine receptor 3A/3B
(Rattus norvegicus)
Universit£
Curated by
ChEMBL
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
IC50: 727nM
Assay Description:
Inhibition of [3H]BRL-43694 binding to 5-hydroxytryptamine 3 receptor of rat cortical homogenate.
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Target
Synaptic vesicular amine transporter
(Homo sapiens (Human))
Organix
Curated by
ChEMBL
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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IC50: 1.43E+3nM
Assay Description:
Inhibition of human VMAT2 expressed in HEK293 cell membranes assessed as reduction in [3H[-5HT uptake pre-incubated for 10 mins before [3H[-5HT addit...
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Target
5-hydroxytryptamine receptor 2A
(Rattus norvegicus (rat))
Alcon Research
Curated by
ChEMBL
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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IC50: 2.35E+3nM
Assay Description:
Inhibition of radiolabeled [3H]-Ketanserin ligand binding to 5-hydroxytryptamine 2A receptor
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MAP/microtubule affinity-regulating kinase 4
(Homo sapiens (Human))
Jamia Millia Islamia
Curated by
ChEMBL
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
IC50: 2.99E+3nM
Assay Description:
Inhibition of MARK4 (unknown origin) ATPase activity using ATP as substrate incubated for 1.5 hr in presence of MgCl2 by Biomol green reagent based E...
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Target
Serotonin 2 (5-HT2) receptor
(RAT)
TBA
Curated by
ChEMBL
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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IC50: 3.60E+3nM
Assay Description:
Binding affinity against 5-hydroxytryptamine 2 receptor using [3H]ket as radioligand.
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Target
Serotonin 2 (5-HT2) receptor
(RAT)
TBA
Curated by
ChEMBL
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
IC50: 4.60E+3nM
Assay Description:
Compound was evaluated for its inhibitory activity against 5-hydroxytryptamine 2 receptor of rat anterior cortex using [3H]ketanserin as the radiolig...
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5-hydroxytryptamine receptor 2A
(Rattus norvegicus (rat))
Alcon Research
Curated by
ChEMBL
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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IC50: 1.30E+4nM
Assay Description:
Displacement of [3H]-ketanserin from 5HT2A receptor in rat brain cortical membranes after 15 mins by competition assay in presence of Gpp(NH)p
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5-hydroxytryptamine receptor 2A
(Rattus norvegicus (rat))
Alcon Research
Curated by
ChEMBL
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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IC50: 3.06E+4nM
Assay Description:
Displacement of [3H]-ketanserin from 5HT2A receptor low affinity component in rat brain cortical membranes after 15 mins by competition assay
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Epidermal growth factor receptor
(Homo sapiens (Human))
Universit£T Leipzig
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ChEMBL
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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IC50: >5.00E+4nM
Assay Description:
Inhibition of EGFR after 30 mins by chemiluminescence ELISA
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Vascular endothelial growth factor receptor 2
(Homo sapiens (Human))
Universit£T Leipzig
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Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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IC50: >5.00E+4nM
Assay Description:
Noncompetitive inhibition of VEGFR2 after 30 mins by chemiluminescence ELISA in presence of 25 uM ATP
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Insulin-like growth factor 1 receptor
(Homo sapiens (Human))
Universit£T Leipzig
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ChEMBL
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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IC50: >5.00E+4nM
Assay Description:
Noncompetitive inhibition of IGF1R after 30 mins by chemiluminescence ELISA in presence of 50 uM ATP
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Vascular endothelial growth factor receptor 3
(Homo sapiens (Human))
Universit£T Leipzig
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ChEMBL
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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IC50: >5.00E+4nM
Assay Description:
Inhibition of VEGFR3 after 30 mins by chemiluminescence ELISA
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Ribosyldihydronicotinamide dehydrogenase [quinone]
(Homo sapiens (Human))
University of Illinois At Chicago
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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IC50: 5.39E+4nM
pH: 8.0 T: 2°C
Assay Description:
The activity of recombinant human QR2 under steady-state conditions was evaluated on a MolecularDevices SpectraMax Plus 384 UV-visible spectrophotome...
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Solute carrier family 22 member 3
(Rattus norvegicus)
Medical College Of Georgia
Curated by
ChEMBL
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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IC50: 9.70E+4nM
Assay Description:
TP_TRANSPORTER: inhibition of MPP+ uptake (MPP+: 1 uM) in OCT3-expressing HRPE cells
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Alpha-glucosidase MAL62
(Saccharomyces cerevisiae)
TBA
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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IC50: >3.00E+5nM
Assay Description:
Inhibition of yeast alpha-glucosidase using p-nitrophenyl-alpha-D-glucopyranoside as substrate preincubated for 10 min before substrate addition and ...
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Isocitrate lyase
(Candida albicans)
Institute
Curated by
ChEMBL
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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IC50: 3.01E+5nM
Assay Description:
Inhibition of Candida albicans isocitrate lyase
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Isocitrate lyase
(Candida albicans)
Institute
Curated by
ChEMBL
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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IC50: 3.01E+5nM
Assay Description:
Inhibition of Candida albicans isocitrate lyase
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Polyphenol oxidase 2
(Agaricus bisporus (Common mushroom))
Kinki University
Curated by
ChEMBL
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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IC50: >3.50E+5nM
Assay Description:
Inhibition of mushroom tyrosinase after 25 mins by spectrophotometry
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Macrophage migration inhibitory factor
(Homo sapiens (Human))
Wuhan University
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ChEMBL
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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IC50: >4.00E+5nM
Assay Description:
Inhibition of MIF tautomerase (unknown origin) using 4-HPP as substrate preincubated for 1 hr followed by substrate addition
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Prostaglandin G/H synthase 2
(Homo sapiens (Human))
Kinki University
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Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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IC50: >4.00E+5nM
Assay Description:
Inhibition of COX2 after 5 mins by spectrophotometric analysis
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Prostaglandin G/H synthase 1
(Homo sapiens (Human))
Kinki University
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ChEMBL
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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IC50: >4.00E+5nM
Assay Description:
Inhibition of COX1 after 5 mins by spectrophotometric analysis
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Tyrosinase
(Mus musculus (Mouse))
National Institute Of Advanced Industrial Science And Technology
Curated by
ChEMBL
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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IC50: 5.50E+5nM
Assay Description:
Inhibition of catecholase activity of tyrosinase in mouse B16 cells assessed as dopachrome formation
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5-hydroxytryptamine receptor 1D
(GUINEA PIG)
Pfizer
Curated by
ChEMBL
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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EC50: 5.20nM
Assay Description:
Effect on forskolin stimulated adenylate cyclase activity at 5-HT1D receptor of guinea pig substantia nigra.
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5-hydroxytryptamine receptor 1D
(GUINEA PIG)
Pfizer
Curated by
ChEMBL
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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EC50: 8.5nM
Assay Description:
Compound was tested for the inhibition of forskolin-stimulated adenylate cyclase at 5-hydroxytryptamine 1D receptor in guinea pig substantia nigra
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5-hydroxytryptamine receptor 4
(GUINEA PIG)
Janssen Research Foundation
Curated by
PDSP K
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Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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EC50: 5nM
Assay Description:
5-hydroxytryptamine 4 receptor agonist activity as increased response to electrical stimulation in guinea pig ileum
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5-hydroxytryptamine receptor 4
(RAT)
Synaptic Pharmaceutical
Curated by
PDSP K
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Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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EC50: 17nM
Assay Description:
In vitro relaxation of carbachol pre-contracted rat oesophageal TMM.
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5-hydroxytryptamine receptor 1B
(Homo sapiens (Human))
University of Alberta
Curated by
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Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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EC50: 30nM
Assay Description:
Inhibition of Forskolin-stimulated adenylate cyclase activity against 5-hydroxytryptamine 1A receptor of guinea pig hippocampus
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5-hydroxytryptamine receptor 1D
(GUINEA PIG)
Pfizer
Curated by
ChEMBL
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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EC50: 16nM
Assay Description:
Inhibition of Forskolin-stimulated adenylate cyclase activity against 5-hydroxytryptamine 1D receptor of guinea pig substantia nigra
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5-hydroxytryptamine receptor 2B
(Homo sapiens (Human))
Syntex Discovery Research
Curated by
PDSP K
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Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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EC50: 1.5nM
Assay Description:
Functional activity against human 5-hydroxytryptamine 2B receptor expressed in CHO cells using fluorometricimaging plate reader
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5-hydroxytryptamine receptor 2C
(Homo sapiens (Human))
Yamanouchi Pharmaceutical
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Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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EC50: 1.70nM
Assay Description:
Functional activity against human 5-hydroxytryptamine 2C receptor expressed in CHO cells using fluorometricimaging plate reader
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5-hydroxytryptamine receptor 1D
(RAT)
University of Alberta
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Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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EC50: 5.20nM
Assay Description:
Inhibition of forskolin stimulated adenylate cyclase at 5-hydroxytryptamine 1D receptor
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5-hydroxytryptamine receptor 1A
(Rattus norvegicus (rat))
Emory University
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PDSP K
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Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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EC50: 10nM
Assay Description:
Inhibition of forskolin stimulated adenylate cyclase at 5-hydroxytryptamine 1A receptor
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5-hydroxytryptamine receptor 4
(GUINEA PIG)
Janssen Research Foundation
Curated by
PDSP K
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Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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EC50: 5nM
Assay Description:
5-hydroxytryptamine 4 receptor agonist activity, concentration which gave 50% increase in the response to electrically-stimulated myenteric plexus an...
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5-hydroxytryptamine receptor 1B
(Homo sapiens (Human))
University of Alberta
Curated by
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Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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EC50: 4.82nM
Assay Description:
Inhibition of forskolin-stimulated c-AMP formation by human 5-hydroxytryptamine 1B receptor expressed in CHO-K1 cells
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5-hydroxytryptamine receptor 1B
(Homo sapiens (Human))
University of Alberta
Curated by
PDSP K
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Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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EC50: 4.70nM
Assay Description:
The intrinsic activity of the compound was evaluated for its ability to inhibit forskolin-stimulated c-AMP formation mediated by cloned 5-hydroxytryp...
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5-hydroxytryptamine receptor 1A
(Homo sapiens (Human))
University of Alberta
Curated by
PDSP K
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Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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EC50: 1nM
Assay Description:
Agonistic activity at human 5HT1A in CHO cells by the inhibition of forskolin-stimulated cAMP accumulation
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5-hydroxytryptamine receptor 1A
(Homo sapiens (Human))
University of Alberta
Curated by
PDSP K
i
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Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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EC50: 3nM
Assay Description:
Agonist activity at 5HT1A receptor (unknown origin) after 20 mins by [35S]GTP-gammaS binding assay
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5-hydroxytryptamine receptor 2A
(Homo sapiens (Human))
Eli Lilly
Curated by
PDSP K
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Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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EC50: 11nM
Assay Description:
Functional activity against human 5-hydroxytryptamine 2A receptor expressed in CHO cells using fluorometricimaging plate reader
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5-hydroxytryptamine receptor 7
(Homo sapiens (Human))
University Of Namur
Curated by
ChEMBL
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Kd: 4nM
Assay Description:
Displacement of [3H]5-HT from human 5HT7 receptor transfected in CFO-K1 cells after 30 mins by liquid scintillation spectrometry
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5-hydroxytryptamine receptor 7
(Homo sapiens (Human))
University Of Namur
Curated by
ChEMBL
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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EC50: 17nM
Assay Description:
Agonist activity at human 5-HT7 expressed in HEK-293 cells assessed as increase in cAMP level after 45 mins by HTRF assay
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5-hydroxytryptamine receptor 2B
(Homo sapiens (Human))
Syntex Discovery Research
Curated by
PDSP K
i
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Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
EC50: 1.5nM
Assay Description:
Binding to human 5HT2B receptor expressed in CHO cells
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5-hydroxytryptamine receptor 2A
(Homo sapiens (Human))
Eli Lilly
Curated by
PDSP K
i
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Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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EC50: 11nM
Assay Description:
Binding to human 5HT2A receptor expressed in CHO cells
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5-hydroxytryptamine receptor 2C
(Homo sapiens (Human))
Yamanouchi Pharmaceutical
Curated by
PDSP K
i
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Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
EC50: 1.70nM
Assay Description:
Binding to human 5HT2C receptor expressed in CHO cells
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5-hydroxytryptamine receptor 2B
(Homo sapiens (Human))
Syntex Discovery Research
Curated by
PDSP K
i
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Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
EC50: 0.920nM
Assay Description:
Agonist activity at human 5-HT2B receptor expressed in HEK293 cells assessed as calcium flux by FLIPR assay
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5-hydroxytryptamine receptor 2C
(Homo sapiens (Human))
Yamanouchi Pharmaceutical
Curated by
PDSP K
i
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Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
EC50: 0.210nM
Assay Description:
Agonist activity at human 5-HT2C receptor expressed in HEK293 cells assessed as calcium flux by FLIPR assay
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5-hydroxytryptamine receptor 2A
(Homo sapiens (Human))
Eli Lilly
Curated by
PDSP K
i
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Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
EC50: 1.90nM
Assay Description:
Agonist activity at human 5-HT2A receptor expressed in HEK293 cells assessed as calcium flux by FLIPR assay
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5-hydroxytryptamine receptor 1A
(Homo sapiens (Human))
University of Alberta
Curated by
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i
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Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
EC50: 0.700nM
Assay Description:
Agonist activity assessed by stimulation of [35S]GTPgammaS binding to human 5HT1A receptor expressed in CHO cells
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5-hydroxytryptamine receptor 1A
(Homo sapiens (Human))
University of Alberta
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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EC50: 1nM
Assay Description:
Agonistic activity at human 5HT1A in CHO cells by the inhibition of forskolin-stimulated cAMP accumulation
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5-hydroxytryptamine receptor 2A
(Rattus norvegicus (rat))
Alcon Research
Curated by
ChEMBL
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
EC50: 58nM
Assay Description:
Activity against 5HT2A mediated intracellular calcium mobilization by FLIPR in rat vascular smooth muscle cells
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5-hydroxytryptamine receptor 2C
(Rattus norvegicus (Rat))
University of Alberta
Curated by
PDSP K
i
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Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
EC50: 2.80nM
Assay Description:
Activity against recombinant rat 5HT2C mediated intracellular calcium mobilization by FLIPR in SR3T3 cells
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5-hydroxytryptamine receptor 2B
(RAT)
Syntex Discovery Research
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
EC50: 3.5nM
Assay Description:
Activity against 5HT2B receptor in longitudinal stomach fundus strips in wistar rats
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5-hydroxytryptamine receptor 1A
(Homo sapiens (Human))
University of Alberta
Curated by
PDSP K
i
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Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
EC50: 28nM
Assay Description:
Agonist activity at human 5-HT1A receptor expressed in CHO cells assessed as inhibition of forskolin-stimulated cAMP accumulation after 15 mins by EL...
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5-hydroxytryptamine receptor 1A
(Homo sapiens (Human))
University of Alberta
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
EC50: 170nM
Assay Description:
Agonist activity at human 5-HT1A receptor expressed in CHO cells after 90 mins by beta-arrestin-2 recruitment assay
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5-hydroxytryptamine receptor 2A
(Homo sapiens (Human))
Eli Lilly
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
EC50: 302nM
T: 2°C
Assay Description:
Partial agonist activity at human 5-HT2A receptor expressed in HEK293 cells preincubated for 1 hr at 37 degC followed by incubated for 15 mins at roo...
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5-hydroxytryptamine receptor 2C
(Homo sapiens (Human))
Yamanouchi Pharmaceutical
Curated by
PDSP K
i
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Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
EC50: 191nM
T: 2°C
Assay Description:
Partial agonist activity at human 5-HT2C receptor expressed in HEK293 cells preincubated for 1 hr at 37 degC followed by incubated for 15 mins at roo...
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5-hydroxytryptamine receptor 1A
(Rattus norvegicus (rat))
Emory University
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
EC50: 323nM
Assay Description:
Agonist activity at 5HT1A receptor in CRL:CD(SD)BR-COBS rat hippocampus assessed as increase in [35S]GTPgammaS binding
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5-hydroxytryptamine receptor 2C
(Homo sapiens (Human))
Yamanouchi Pharmaceutical
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
EC50: 0.0900nM
Assay Description:
Agonist activity at human 5HT2C receptor expressed in HEK293 cells assessed as calcium flux by FLIPR assay
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5-hydroxytryptamine receptor 2B
(Homo sapiens (Human))
Syntex Discovery Research
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
Copy SMILES
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Affinity Data
EC50: 0.5nM
Assay Description:
Agonist activity at human 5HT2B receptor expressed in HEK293 cells assessed as calcium flux by FLIPR assay
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5-hydroxytryptamine receptor 2A
(Homo sapiens (Human))
Eli Lilly
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
EC50: 5.80nM
Assay Description:
Agonist activity at human 5HT2A receptor expressed in HEK293 cells assessed as calcium flux by FLIPR assay
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5-hydroxytryptamine receptor 7
(Homo sapiens (Human))
University Of Namur
Curated by
ChEMBL
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
EC50: 15nM
Assay Description:
Agonist activity at human recombinant 5HT7 receptor expressed in CHOK1 cells assessed as increase in cAMP levels by HTRF assay
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5-hydroxytryptamine receptor 1A
(Homo sapiens (Human))
University of Alberta
Curated by
PDSP K
i
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Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
EC50: 43nM
Assay Description:
Compound was tested for the inhibition of forskolin-stimulated adenylate cyclase at 5-hydroxytryptamine 1A receptor in guinea pig
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5-hydroxytryptamine receptor 2C
(Homo sapiens (Human))
Yamanouchi Pharmaceutical
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
EC50: 25nM
Assay Description:
Agonist activity at human recombinant 5HT2C receptor expressed in CHO K1 cells assessed as induction of calcium mobilization by FLIPR assay
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5-hydroxytryptamine receptor 7
(Homo sapiens (Human))
University Of Namur
Curated by
ChEMBL
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
EC50: 7nM
Assay Description:
Agonist activity at human 5-HT7 receptor expressed in CHO-K1 cells assessed as increase in serotonin-induced cAMP level after 1 hr by TR-FRET assay
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5-hydroxytryptamine receptor 1A
(Homo sapiens (Human))
University of Alberta
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
EC50: 229nM
Assay Description:
Agonist activity at human 5HT1A receptor expressed in C6 cells assessed as stimulation of [35S]GTPgammaS binding
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5-hydroxytryptamine receptor 1A
(Homo sapiens (Human))
University of Alberta
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
EC50: 8.70nM
Assay Description:
Binding affinity against human 5-hydroxytryptamine 1A receptors HEK 293 cell membranes using [35S]GTP gamma-S
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5-hydroxytryptamine receptor 6
(Homo sapiens (Human))
Jagiellonian University Collegium Medicum
Curated by
ChEMBL
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
EC50: 44nM
Assay Description:
Agonist activity at serotonin 5-HT6R receptor (unknown origin) expressed in HEK293 cells assessed as induction of calcium flux after 60 mins by calci...
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5-hydroxytryptamine receptor 2A
(Homo sapiens (Human))
Eli Lilly
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
EC50: 1.60nM
Assay Description:
Agonist activity at serotonin 5-HT2A receptor (unknown origin) expressed in HEK293 cells assessed as induction of calcium flux after 60 mins by calci...
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5-hydroxytryptamine receptor 1A
(Homo sapiens (Human))
University of Alberta
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
EC50: 19nM
Assay Description:
Agonist activity at serotonin 5-HT1A receptor (unknown origin) expressed in HEK293 cells assessed as induction of calcium flux after 60 mins by calci...
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5-hydroxytryptamine receptor 2B
(Homo sapiens (Human))
Syntex Discovery Research
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
EC50: 25nM
Assay Description:
Agonist activity at human 5HT2B receptor expressed in HEK293 cells assessed as intracellular IP3 accumulation
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5-hydroxytryptamine receptor 2C
(Homo sapiens (Human))
Yamanouchi Pharmaceutical
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
EC50: 25nM
Assay Description:
Agonist activity at human 5HT2C receptor expressed in HEK293 cells assessed as intracellular IP3 accumulation
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5-hydroxytryptamine receptor 2A
(Homo sapiens (Human))
Eli Lilly
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
EC50: 126nM
Assay Description:
Agonist activity at human 5HT2A receptor expressed in HEK293 cells assessed as intracellular IP3 accumulation
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Target
5-hydroxytryptamine receptor 2B
(RAT)
Syntex Discovery Research
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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EC50: 4.20nM
Assay Description:
Agonist activity at 5HT2b receptor in Wistar rat fundus measured for 90 secs
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5-hydroxytryptamine receptor 1A
(Homo sapiens (Human))
University of Alberta
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
EC50: 5.60nM
Assay Description:
Agonist activity at human recombinant 5-HT1A receptor expressed in CHOK1 cells measured after 1 hr by microbeta2 scintillation counter
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5-hydroxytryptamine receptor 7
(Homo sapiens (Human))
University Of Namur
Curated by
ChEMBL
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
EC50: 5.40nM
Assay Description:
Agonist activity at human recombinant 5-HT7 receptor expressed in CHOK1 cells by LANCE TR-FRET assay
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5-hydroxytryptamine receptor 1A
(Homo sapiens (Human))
University of Alberta
Curated by
PDSP K
i
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Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
EC50: 5.61nM
Assay Description:
Agonist activity at human recombinant 5-HT1A receptor expressed in CHOK1 cells measured after 1 hr by microbeta2 scintillation counter
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5-hydroxytryptamine receptor 7
(Homo sapiens (Human))
University Of Namur
Curated by
ChEMBL
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
EC50: 5.70nM
Assay Description:
Agonist activity at human recombinant 5-HT7 receptor expressed in CHOK1 cells by LANCE TR-FRET assay
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5-hydroxytryptamine receptor 2A
(Homo sapiens (Human))
Eli Lilly
Curated by
PDSP K
i
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Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
EC50: 0.275nM
Assay Description:
Agonist activity at recombinant human 5HT2A receptor expressed in Flp-In-293 cells assessed as increase in calcium influx measured for 300 secs by Fl...
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5-hydroxytryptamine receptor 2C
(Homo sapiens (Human))
Yamanouchi Pharmaceutical
Curated by
PDSP K
i
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Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
EC50: 0.191nM
Assay Description:
Agonist activity at recombinant human unedited 5HT2C receptor isoform INI expressed in Flp-In-293 cells assessed as increase in calcium influx measur...
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5-hydroxytryptamine receptor 2C
(Homo sapiens (Human))
Yamanouchi Pharmaceutical
Curated by
PDSP K
i
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Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
EC50: 0.190nM
Assay Description:
Agonist activity at recombinant human unedited 5HT2C receptor isoform INI expressed in Flp-In-293 cells assessed as increase in calcium influx measur...
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5-hydroxytryptamine receptor 2B
(Homo sapiens (Human))
Syntex Discovery Research
Curated by
PDSP K
i
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Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
EC50: 0.860nM
Assay Description:
Agonist activity at recombinant human 5HT2B receptor expressed in Flp-In-293 cells assessed as increase in calcium influx measured for 300 secs by Fl...
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5-hydroxytryptamine receptor 2A
(Homo sapiens (Human))
Eli Lilly
Curated by
PDSP K
i
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Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
EC50: 0.270nM
Assay Description:
Agonist activity at recombinant human 5HT2A receptor expressed in Flp-In-293 cells assessed as increase in calcium influx measured for 300 secs by Fl...
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5-hydroxytryptamine receptor 2B
(Homo sapiens (Human))
Syntex Discovery Research
Curated by
PDSP K
i
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Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
EC50: 0.851nM
Assay Description:
Agonist activity at recombinant human 5HT2B receptor expressed in Flp-In-293 cells assessed as increase in calcium influx measured for 300 secs by Fl...
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5-hydroxytryptamine receptor 1A
(Homo sapiens (Human))
University of Alberta
Curated by
PDSP K
i
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Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
EC50: 1.80E+3nM
Assay Description:
Agonist activity at human 5HT1A receptor expressed in CHOK1 cells incubated for 16 hrs followed by forskolin-stimulation and measured after 2 hrs by ...
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Target
5-hydroxytryptamine receptor 1A
(Homo sapiens (Human))
University of Alberta
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
EC50: 1.80E+3nM
Assay Description:
Agonist activity at human 5HT1A receptor expressed in CHOK1 cells incubated for 16 hrs followed by forskolin-stimulation and measured after 2 hrs by ...
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5-hydroxytryptamine receptor 2C
(Homo sapiens (Human))
Yamanouchi Pharmaceutical
Curated by
PDSP K
i
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Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
EC50: 0.410nM
Assay Description:
Agonist activity at human 5HT2C receptor stably expressed in HEK293 cells co-expressing Gq assessed as induction of calcium mobilization measured at ...
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5-hydroxytryptamine receptor 1A
(Homo sapiens (Human))
University of Alberta
Curated by
PDSP K
i
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Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
EC50: 18nM
Assay Description:
Agonist activity at human recombinant 5HT1A receptor (unknown origin) stably expressed in CHO-K1 incubated for 30 mins by [35S]GTPgammaS binding assa...
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5-hydroxytryptamine receptor 2B
(Homo sapiens (Human))
Syntex Discovery Research
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
EC50: 4.5nM
Assay Description:
Agonist activity at recombinant human 5-HT2B receptor expressed in CHOK1 cells assessed as increase in inositol1-phosphate accumulation measured afte...
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5-hydroxytryptamine receptor 2A
(Homo sapiens (Human))
Eli Lilly
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
EC50: 0.510nM
Assay Description:
Agonist activity at human 5-HT2A receptor expressed in Flp-In T-REx 293 cells assessed as induction of Gq-mediated calcium flux incubated for 1 hr by...
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5-hydroxytryptamine receptor 2A
(Homo sapiens (Human))
Eli Lilly
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
EC50: 0.513nM
Assay Description:
Agonist activity at human 5-HT2A receptor expressed in Flp-In T-REx 293 cells assessed as induction of Gq-mediated calcium flux incubated for 1 hr by...
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5-hydroxytryptamine receptor 2A
(Mus musculus (Mouse))
Usona Institute
Curated by
ChEMBL
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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EC50: 0.525nM
Assay Description:
Agonist activity at mouse 5-HT2A receptor expressed in Flp-In T-REx 293 cells assessed as induction of Gq-mediated calcium flux incubated for 1 hr by...
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5-hydroxytryptamine receptor 2A
(Mus musculus (Mouse))
Usona Institute
Curated by
ChEMBL
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
EC50: 0.530nM
Assay Description:
Agonist activity at mouse 5-HT2A receptor expressed in Flp-In T-REx 293 cells assessed as induction of Gq-mediated calcium flux incubated for 1 hr by...
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5-hydroxytryptamine receptor 2B
(Homo sapiens (Human))
Syntex Discovery Research
Curated by
PDSP K
i
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Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
EC50: 11nM
Assay Description:
Agonist activity at human recombinant 5HT2B receptor assessed as induction of calcium mobilization by FLIPR assay
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5-hydroxytryptamine receptor 3A
(Homo sapiens (Human))
Amri
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ChEMBL
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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EC50: 141nM
Assay Description:
Partial agonist activity at human 5HT3A receptor expressed in HEK293 cells assessed as decrease in 10 uM 5-chloroindole-induced increase in intracell...
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Target
5-hydroxytryptamine receptor 3A
(Homo sapiens (Human))
Amri
Curated by
ChEMBL
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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EC50: 178nM
Assay Description:
Partial agonist activity at human 5HT3A receptor expressed in HEK293 cells assessed as effect on serotonin-induced response
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5-hydroxytryptamine receptor 3A
(RAT)
University Of Florida
Curated by
ChEMBL
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
EC50: 1.20E+4nM
Assay Description:
Response at rat 5-hydroxytryptamine 3a receptor expressed in xenopus oocytes
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D(1A) dopamine receptor
(Homo sapiens (Human))
Sri International
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
Kd: 9.69E+3nM
Assay Description:
Equilibrium dissociation constant against recombinant Dopamine receptor D1A expressed in COS7 cells
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5-hydroxytryptamine receptor 1F
(Homo sapiens (Human))
Janssen Research Foundation
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
EC50: 7.90nM
Assay Description:
In vitro effective concentration for inhibition of skolin-stimulated adenylate cyclase in cell line expressing human 5-hydroxytryptamine 1F receptor
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5-hydroxytryptamine receptor 2A
(Rattus norvegicus (rat))
Alcon Research
Curated by
ChEMBL
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
EC50: 55.8nM
Assay Description:
The receptor (5-hydroxytryptamine 2A ) mediated mobilization of intracellular calcium [Ca2+] was studied in rat smooth muscle cells
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5-hydroxytryptamine receptor 2A
(Rattus norvegicus (rat))
Alcon Research
Curated by
ChEMBL
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
EC50: 351nM
Assay Description:
In vitro relative agonist activity against 5-hydroxytryptamine 2A using PI assay in rat vascular smooth muscle cells
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5-hydroxytryptamine receptor 1A
(Homo sapiens (Human))
University of Alberta
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
EC50: 3.70nM
Assay Description:
Tested for functional response on CHO cells expressing cloned human 5-hydroxytryptamine 1A receptor
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D(3) dopamine receptor
(Homo sapiens (Human))
Universit£
Curated by
ChEMBL
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
EC50: 523nM
Assay Description:
Basal binding towards Dopamine receptor D3 was evaluated using [35S]- GTP-gamma S radioligand
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5-hydroxytryptamine receptor 2A
(Homo sapiens (Human))
Eli Lilly
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
EC50: 47nM
Assay Description:
Agonist activity at 5-HT2A receptor (unknown origin) expressed in CHOK1 cells co-expressing G-alpha 15 by Fluo-4 dye based FLIPR assay
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5-hydroxytryptamine receptor 1A
(Homo sapiens (Human))
University of Alberta
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
EC50: 15nM
Assay Description:
Agonist activity at 5-HT1A receptor (unknown origin) expressed in CHOK1 cells co-expressing G-alpha 15 by Fluo-4 dye based FLIPR assay
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5-hydroxytryptamine receptor 3A
(Homo sapiens (Human))
Amri
Curated by
ChEMBL
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
EC50: 457nM
Assay Description:
Antagonist activity at human 5HT3A receptor expressed in HEK293 cells by FMP assay
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5-hydroxytryptamine receptor 1A
(Homo sapiens (Human))
University of Alberta
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
EC50: 3.80nM
Assay Description:
Agonist activity at 5-HT1A receptor (unknown origin) expressed in HEK293 cells assessed as inhibition of [35S]GTPgammaS binding by scintillation prox...
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5-hydroxytryptamine receptor 4
(GUINEA PIG)
Janssen Research Foundation
Curated by
PDSP K
i
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Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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EC50: 10nM
Assay Description:
Agonist activity at 5HT4 receptor in guinea pig colon assessed as longitudinal muscle plexus contraction
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5-hydroxytryptamine receptor 2C
(Homo sapiens (Human))
Yamanouchi Pharmaceutical
Curated by
PDSP K
i
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Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
EC50: 0.870nM
Assay Description:
Agonist activity at human 5HT2C receptor expressed in HEK293 cells assessed as induction of intracellular calcium release measured for 90 secs by flu...
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5-hydroxytryptamine receptor 2A
(Homo sapiens (Human))
Eli Lilly
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
EC50: 2.60nM
Assay Description:
Agonist activity at human 5HT2A receptor expressed in HEK293 cells assessed as induction of intracellular calcium release measured for 90 secs by flu...
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5-hydroxytryptamine receptor 2C
(Homo sapiens (Human))
Yamanouchi Pharmaceutical
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
EC50: 44nM
Assay Description:
Agonist activity at human 5HT2C receptor expressed in HEK293 cells assessed as accumulation of IP1 incubated for 1 hr at 37 degC followed by 15 mins ...
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5-hydroxytryptamine receptor 2A
(Homo sapiens (Human))
Eli Lilly
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
EC50: 150nM
Assay Description:
Agonist activity at human 5HT2A receptor expressed in HEK293 cells assessed as accumulation of IP1 incubated for 1 hr at 37 degC followed by 15 mins ...
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5-hydroxytryptamine receptor 3A
(Mus musculus (house mouse))
University of Alberta
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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EC50: 3.40E+3nM
Assay Description:
Agonist activity at wild type mouse 5HT3A receptor expressed in Xenopus oocyte by two-electrode voltage patch clamp method
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5-hydroxytryptamine receptor 4
(Homo sapiens (Human))
Monash University
Curated by
ChEMBL
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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EC50: 100nM
Assay Description:
Activity at SER4 receptor expressed in HEK293 cells assessed as increase in calcium by calcium imaging assay
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5-hydroxytryptamine receptor 1A
(Homo sapiens (Human))
University of Alberta
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
EC50: 150nM
Assay Description:
Agonist activity at 5HT1A receptor expressed in CHO cells by [35S]GTPgammaS binding assay
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5-hydroxytryptamine receptor 1A
(Homo sapiens (Human))
University of Alberta
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
EC50: 147nM
Assay Description:
Agonist activity at 5HT1A receptor expressed in CHO cells assessed as stimulation of [35S]GTPgamma binding
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5-hydroxytryptamine receptor 2C
(Homo sapiens (Human))
Yamanouchi Pharmaceutical
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
EC50: 24nM
Assay Description:
Agonist activity at human cloned 5HT2C receptor expressed in CHO cells assessed as myo-[3H]inositol hydrolysis
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5-hydroxytryptamine receptor 2B
(Homo sapiens (Human))
Syntex Discovery Research
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
EC50: 5.80nM
Assay Description:
Agonist activity at human cloned 5HT2B receptor expressed in HEK293-EBNA cells assessed as myo-[3H]inositol hydrolysis
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5-hydroxytryptamine receptor 2A
(Homo sapiens (Human))
Eli Lilly
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
EC50: 70nM
Assay Description:
Agonist activity at human cloned 5HT2A receptor expressed in CHO cells assessed as myo-[3H]inositol hydrolysis
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5-hydroxytryptamine receptor 1B
(Rattus norvegicus (Rat))
University of Alberta
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
EC50: 26nM
Assay Description:
Inhibition of Forskolin-stimulated adenylate cyclase activity against 5-hydroxytryptamine 1B receptor of rat substantia nigra
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Serotonin 2 (5-HT2) receptor
(Homo sapiens (Human))
Smithkline Beecham Pharmaceuticals
Curated by
ChEMBL
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
Kd: 3.16E+3nM
Assay Description:
Binding affinity for 5-hydroxytryptamine 2 receptor was determined
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5-hydroxytryptamine receptor 1D
(Homo sapiens (Human))
Theravance
Curated by
ChEMBL
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
Kd: 13nM
Assay Description:
Binding affinity for 5-hydroxytryptamine 1D receptor was determined
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5-hydroxytryptamine receptor 2C
(Rattus norvegicus (Rat))
University of Alberta
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
Kd: 32nM
Assay Description:
Binding affinity for 5-hydroxytryptamine 1C receptor was determined
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5-hydroxytryptamine receptor 1A
(Homo sapiens (Human))
University of Alberta
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
Kd: 3.20nM
Assay Description:
Binding affinity for 5-hydroxytryptamine 1A receptor was determined
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5-hydroxytryptamine receptor 2C
(Homo sapiens (Human))
Yamanouchi Pharmaceutical
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
EC50: 1.63nM
Assay Description:
Agonist activity at 5HT2C receptor expressed in CHO cells by fluorescence based calcium mobilization assay
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5-hydroxytryptamine receptor 2B
(Homo sapiens (Human))
Syntex Discovery Research
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
EC50: 0.860nM
Assay Description:
Agonist activity at human 5HT2B receptor expressed in HEK293 cells assessed as calcium flux measured every sec for 3 mins by FLIPR assay
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5-hydroxytryptamine receptor 2C
(Homo sapiens (Human))
Yamanouchi Pharmaceutical
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
EC50: 0.0900nM
Assay Description:
Agonist activity at human 5HT2C receptor expressed in HEK293 cells assessed as calcium flux measured every sec for 3 mins by FLIPR assay
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5-hydroxytryptamine receptor 2A
(Homo sapiens (Human))
Eli Lilly
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
EC50: 7.60nM
Assay Description:
Agonist activity at human 5HT2A receptor expressed in HEK293 cells assessed as calcium flux measured every sec for 3 mins by FLIPR assay
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5-hydroxytryptamine receptor 1A
(Homo sapiens (Human))
University of Alberta
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
EC50: 45nM
Assay Description:
Partial agonist activity at recombinant human 5-HT1A expressed in CHO-K1 cells by pathhunter beta-arrestin assay
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5-hydroxytryptamine receptor 7
(Homo sapiens (Human))
University Of Namur
Curated by
ChEMBL
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
EC50: 70nM
Assay Description:
Agonist activity at human recombinant 5-HT7 receptor expressed in CHOK1 Hunter cell incubated for 30 to 60 mins by hit-hunter cAMP assay based chemil...
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5-hydroxytryptamine receptor 2C
(Homo sapiens (Human))
Yamanouchi Pharmaceutical
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
EC50: 0.166nM
Assay Description:
Agonist activity at human 5-HT2C receptor expressed in human Flp-In-293 cells assessed as induction of calcium flux incubated for 1 hr by Fluo-4 dire...
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5-hydroxytryptamine receptor 2C
(Homo sapiens (Human))
Yamanouchi Pharmaceutical
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
EC50: 0.170nM
Assay Description:
Agonist activity at human 5-HT2C receptor expressed in human Flp-In-293 cells assessed as induction of calcium flux incubated for 1 hr by Fluo-4 dire...
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5-hydroxytryptamine receptor 2B
(Homo sapiens (Human))
Syntex Discovery Research
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
EC50: 1.40nM
Assay Description:
Agonist activity at human 5-HT2B receptor expressed in human Flp-In-293 cells assessed as induction of calcium flux incubated for 1 hr by Fluo-4 dire...
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5-hydroxytryptamine receptor 2B
(Homo sapiens (Human))
Syntex Discovery Research
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
EC50: 1.5nM
Assay Description:
Agonist activity at human 5-HT2B receptor expressed in human Flp-In-293 cells assessed as induction of calcium flux incubated for 1 hr by Fluo-4 dire...
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5-hydroxytryptamine receptor 2A
(Homo sapiens (Human))
Eli Lilly
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
EC50: 2.30nM
Assay Description:
Agonist activity at human 5-HT2A receptor expressed in human Flp-In-293 cells assessed as induction of calcium flux incubated for 1 hr by Fluo-4 dire...
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Target
5-hydroxytryptamine receptor 2A
(Homo sapiens (Human))
Eli Lilly
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
Copy SMILES
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Affinity Data
EC50: 2.40nM
Assay Description:
Agonist activity at human 5-HT2A receptor expressed in human Flp-In-293 cells assessed as induction of calcium flux incubated for 1 hr by Fluo-4 dire...
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5-hydroxytryptamine receptor 2C
(Homo sapiens (Human))
Yamanouchi Pharmaceutical
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
EC50: 0.135nM
Assay Description:
Agonist activity at human 5-HT2C INI receptor expressed in human Flp-In-293 cells assessed as induction of calcium flux incubated for 1 hr by Fluo-4 ...
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5-hydroxytryptamine receptor 2C
(Homo sapiens (Human))
Yamanouchi Pharmaceutical
Curated by
PDSP K
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Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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EC50: 0.140nM
Assay Description:
Agonist activity at human 5-HT2C INI receptor expressed in human Flp-In-293 cells assessed as induction of calcium flux incubated for 1 hr by Fluo-4 ...
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5-hydroxytryptamine receptor 2C
(Homo sapiens (Human))
Yamanouchi Pharmaceutical
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Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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EC50: 22nM
Assay Description:
Agonist activity at human 5-HT2C INI receptor expressed in human HEK293 cells assessed as induction of beta-arrestin-2 recruitment incubated for 20 h...
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5-hydroxytryptamine receptor 2C
(Homo sapiens (Human))
Yamanouchi Pharmaceutical
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Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
EC50: 21nM
Assay Description:
Agonist activity at human 5-HT2C INI receptor expressed in human HEK293 cells assessed as induction of beta-arrestin-2 recruitment incubated for 20 h...
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5-hydroxytryptamine receptor 1A
(Homo sapiens (Human))
University of Alberta
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i
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BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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EC50: 33nM
Assay Description:
Biased agonist activity at human recombinant 5-HT1A receptor stably expressed in CHO-K1 cells assessed as increase in ERK1/2 phosphorylation levels i...
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5-hydroxytryptamine receptor 1A
(Homo sapiens (Human))
University of Alberta
Curated by
PDSP K
i
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Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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EC50: 31nM
Assay Description:
Biased agonist activity at human recombinant 5-HT1A receptor stably expressed in CHO-K1 cells assessed as inhibition of forskolin-induced cAMP accumu...
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5-hydroxytryptamine receptor 1A
(Homo sapiens (Human))
University of Alberta
Curated by
PDSP K
i
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Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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EC50: 129nM
Assay Description:
Biased agonist activity at Gal4-VP16 transcription factor linked human 5-HT1A receptor expressed in human U2OS cells assessed as stimulation of beta-...
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5-hydroxytryptamine receptor 1A
(Homo sapiens (Human))
University of Alberta
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PDSP K
i
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Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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EC50: 50nM
Assay Description:
Biased agonist activity at human recombinant 5-HT1A receptor stably expressed in CHO-K1 cells assessed as increase in calcium mobilization measured a...
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5-hydroxytryptamine receptor 2B
(Homo sapiens (Human))
Syntex Discovery Research
Curated by
PDSP K
i
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Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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EC50: 0.0708nM
Assay Description:
Agonist activity at 5-HT2B receptor (unknown origin) by calcium mobilization assay
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5-hydroxytryptamine receptor 1A
(Homo sapiens (Human))
University of Alberta
Curated by
PDSP K
i
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Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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EC50: 5.80nM
Assay Description:
Agonist activity at human 5HT1A receptor expressed in CHO-K1 cells by calcium 4 dye based FLIPR assay
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5-hydroxytryptamine receptor 2A
(Homo sapiens (Human))
Eli Lilly
Curated by
PDSP K
i
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Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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EC50: 1.10nM
Assay Description:
Agonist activity at human 5HT2A receptor expressed in CHO-K1 cells by calcium 4 dye based FLIPR assay
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5-hydroxytryptamine receptor 6
(Homo sapiens (Human))
Jagiellonian University Collegium Medicum
Curated by
ChEMBL
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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EC50: 42nM
Assay Description:
Agonist activity at human 5HT6 receptor expressed in CHO-K1 cells by calcium 4 dye based FLIPR assay
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5-hydroxytryptamine receptor 1A
(Homo sapiens (Human))
University of Alberta
Curated by
PDSP K
i
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Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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EC50: 33nM
Assay Description:
Biased agonist activity at human 5-HT1A receptor stably expressed in CHO-K1 cells assessed as increase in ERK1/2 phosphorylation after 15 mins by Alp...
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5-hydroxytryptamine receptor 1A
(Homo sapiens (Human))
University of Alberta
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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EC50: 31nM
Assay Description:
Biased agonist activity at human 5-HT1A receptor stably expressed in CHO-K1 cells assessed as inhibition of forskolin-induced cAMP accumulation after...
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5-hydroxytryptamine receptor 1A
(Homo sapiens (Human))
University of Alberta
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
EC50: 129nM
Assay Description:
Biased agonist activity at Gal4-VP16 transcription factor linked human 5-HT1A receptor expressed in human U2OS cells assessed as induction of beta-ar...
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5-hydroxytryptamine receptor 1A
(Homo sapiens (Human))
University of Alberta
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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EC50: 59nM
Assay Description:
Biased agonist activity at human 5-HT1A receptor stably expressed in CHO-K1 cells co-expressing Galpha16/GPCR assessed as increase in calcium mobiliz...
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5-hydroxytryptamine receptor 1A
(Homo sapiens (Human))
University of Alberta
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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EC50: 2nM
Assay Description:
Agonist activity at human 5-HT1A receptor expressed in HEK cell membranes incubated for 60 mins by [35S]GTPgammaS binding assay
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5-hydroxytryptamine receptor 7
(Homo sapiens (Human))
University Of Namur
Curated by
ChEMBL
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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EC50: 3.70nM
Assay Description:
Agonist activity at human 5-HT7A receptor expressed in HEK cell membranes incubated for 20 mins by cAMP functional assay
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5-hydroxytryptamine receptor 7
(Homo sapiens (Human))
University Of Namur
Curated by
ChEMBL
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
EC50: 9.30nM
Assay Description:
Agonist activity at human 5-HT7R transfected in HEK293 cells assessed as Gs-mediated cAMP accumulation incubated for 30 mins by microplate reader ana...
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5-hydroxytryptamine receptor 7
(Homo sapiens (Human))
University Of Namur
Curated by
ChEMBL
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
EC50: 9.33nM
Assay Description:
Agonist activity at human 5-HT7R transfected in HEK293 cells assessed as Gs-mediated cAMP accumulation incubated for 30 mins by microplate reader ana...
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5-hydroxytryptamine receptor 7
(Homo sapiens (Human))
University Of Namur
Curated by
ChEMBL
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
EC50: 112nM
Assay Description:
Agonist activity at 5-HT7R (unknown origin) transfected in HEK293 cells expressing tTA-dependent luciferase reporter and beta arrestin 2-TEV fusion g...
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5-hydroxytryptamine receptor 7
(Homo sapiens (Human))
University Of Namur
Curated by
ChEMBL
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
EC50: 110nM
Assay Description:
Agonist activity at 5-HT7R (unknown origin) transfected in HEK293 cells expressing tTA-dependent luciferase reporter and beta arrestin 2-TEV fusion g...
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Trace amine-associated receptor 1
(Homo sapiens (Human))
Sunovion Pharmaceuticals
Curated by
ChEMBL
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
EC50: 3.51E+4nM
Assay Description:
Agonist activity at recombinant human TAAR1 expressed in CHO-K1 cells assessed as increase in intracellular cAMP incubated for 30 mins by HTRF analys...
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5-hydroxytryptamine receptor 1A
(Homo sapiens (Human))
University of Alberta
Curated by
PDSP K
i
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Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
EC50: 10nM
Assay Description:
Agonist activity at human 5-HT1A receptor expressed in CHO-K1 cells assessed as stimulation of ERK1/2 phosphorylation incubated for 15 mins by Alpha ...
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5-hydroxytryptamine receptor 1A
(Homo sapiens (Human))
University of Alberta
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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EC50: 11nM
Assay Description:
Agonist activity at human 5-HT1A receptor expressed in CHO-K1 cells assessed as inhibition of forskolin-induced cAMP production incubated for 40 mins...
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5-hydroxytryptamine receptor 1A
(Homo sapiens (Human))
University of Alberta
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
EC50: 398nM
Assay Description:
Agonist activity at human 5-HT1A receptor expressed in U2OS cells assessed as beta-arrestin recruitment incubated for 5 hrs by Tango assay
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5-hydroxytryptamine receptor 2A
(Homo sapiens (Human))
Eli Lilly
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
EC50: 12nM
Assay Description:
Agonist activity at human 5HT2A receptor transfected in HEK293T cells assessed as beta arrestin-2 recruitment measured for 2 hrs by luminescent assay
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5-hydroxytryptamine receptor 2A
(Homo sapiens (Human))
Eli Lilly
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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EC50: 130nM
Assay Description:
Agonist activity at human 5HT2A receptor transfected in HEK293T cells assessed as mini Galphaq recruitment measured for 2 hrs by luminescent assay
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5-hydroxytryptamine receptor 2A
(Homo sapiens (Human))
Eli Lilly
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
EC50: 661nM
Assay Description:
Agonist activity at human 5HT2A S159A mutant transfected in HEK293T cells assessed as beta arrestin-2 recruitment measured for 2 hrs by luminescent a...
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5-hydroxytryptamine receptor 2A
(Homo sapiens (Human))
Eli Lilly
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
EC50: 1.67E+3nM
Assay Description:
Agonist activity at human 5HT2A S159A mutant transfected in HEK293T cells assessed as mini Galphaq recruitment measured for 2 hrs by luminescent assa...
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5-hydroxytryptamine receptor 2A
(Homo sapiens (Human))
Eli Lilly
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
EC50: 0.350nM
Assay Description:
Agonist activity at human 5HT2A receptor stably expressed in Flp-In-T-REx-293 cells assessed as increase in Gq-mediated calcium flux by Fluo-4 direct...
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5-hydroxytryptamine receptor 2A
(Homo sapiens (Human))
Eli Lilly
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
EC50: 0.347nM
Assay Description:
Agonist activity at human 5HT2A receptor stably expressed in Flp-In-T-REx-293 cells assessed as increase in Gq-mediated calcium flux by Fluo-4 direct...
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5-hydroxytryptamine receptor 2C
(Homo sapiens (Human))
Yamanouchi Pharmaceutical
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
EC50: 0.320nM
Assay Description:
Agonist activity at human 5HT2C receptor stably expressed in Flp-In-T-REx-293 cells assessed as increase in Gq-mediated calcium flux by Fluo-4 direct...
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Target
5-hydroxytryptamine receptor 2C
(Homo sapiens (Human))
Yamanouchi Pharmaceutical
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
EC50: 0.324nM
Assay Description:
Agonist activity at human 5HT2C receptor stably expressed in Flp-In-T-REx-293 cells assessed as increase in Gq-mediated calcium flux by Fluo-4 direct...
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5-hydroxytryptamine receptor 2B
(Homo sapiens (Human))
Syntex Discovery Research
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
EC50: 0.363nM
Assay Description:
Agonist activity at human 5HT2B receptor stably expressed in Flp-In-T-REx-293 cells assessed as increase in Gq-mediated calcium flux by Fluo-4 direct...
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Target
5-hydroxytryptamine receptor 2B
(Homo sapiens (Human))
Syntex Discovery Research
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
EC50: 0.360nM
Assay Description:
Agonist activity at human 5HT2B receptor stably expressed in Flp-In-T-REx-293 cells assessed as increase in Gq-mediated calcium flux by Fluo-4 direct...
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5-hydroxytryptamine receptor 2A
(Homo sapiens (Human))
Eli Lilly
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
EC50: 3nM
Assay Description:
Agonist activity at 5-HT2AR (unknown origin) stably expressed in HEK293 cells measured after 1 hr by fluorescence based Ca2+/Fluo-4 assay
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5-hydroxytryptamine receptor 2C
(Homo sapiens (Human))
Yamanouchi Pharmaceutical
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
EC50: 1.20nM
Assay Description:
Agonist activity at 5-HT2CR (unknown origin) stably expressed in HEK293 cells measured after 1 hr by fluorescence based Ca2+/Fluo-4 assay
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5-hydroxytryptamine receptor 1A
(Homo sapiens (Human))
University of Alberta
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
EC50: 10nM
Assay Description:
Binding affinity of the compound against 5-hydroxytryptamine 1D receptor
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Target
5-hydroxytryptamine receptor 7
(Homo sapiens (Human))
University Of Namur
Curated by
ChEMBL
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
EC50: 5.80nM
Assay Description:
Agonist activity at human 5-HT7R expressed in HEK293 cells assessed as induction of cAMP levels treated for 10 mins measured after 30 mins by D2-dye ...
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Target
5-hydroxytryptamine receptor 7
(Homo sapiens (Human))
University Of Namur
Curated by
ChEMBL
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
EC50: 5.80nM
Assay Description:
Agonist activity at human 5-HT7R expressed in HEK293 cells assessed as induction of cAMP levels treated for 10 mins measured after 30 mins by D2-dye ...
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Target
5-hydroxytryptamine receptor 4
(RAT)
Synaptic Pharmaceutical
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
EC50: 6.30nM
Assay Description:
5-hydroxytryptamine 4 receptor agonist activity in the rat esophageal muscularis mucosae
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Target
5-hydroxytryptamine receptor 2C
(Homo sapiens (Human))
Yamanouchi Pharmaceutical
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
EC50: 15nM
Assay Description:
Agonist activity at tTA containing TEV cleavage site-fused 5-HT2C-INI receptor isoform (unknown origin) expressed in TEV-fused beta-arrestin2 express...
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Target
5-hydroxytryptamine receptor 2B
(Homo sapiens (Human))
Syntex Discovery Research
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
EC50: 1.5nM
Assay Description:
Agonist activity at human 5-HT2B receptor expressed in Flp-IN HEK293 cells assessed as induction of calcium flux measured every second for 5 mins by ...
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Target
5-hydroxytryptamine receptor 2A
(Homo sapiens (Human))
Eli Lilly
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
EC50: 2.30nM
Assay Description:
Agonist activity at human 5-HT2A receptor expressed in Flp-IN HEK293 cells assessed as induction of calcium flux measured every second for 5 mins by ...
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5-hydroxytryptamine receptor 2C
(Homo sapiens (Human))
Yamanouchi Pharmaceutical
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
EC50: 15nM
Assay Description:
Agonist activity at tTA containing TEV cleavage site-fused 5-HT2C-INI receptor isoform (unknown origin) expressed in TEV-fused beta-arrestin2 express...
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Target
5-hydroxytryptamine receptor 2B
(Homo sapiens (Human))
Syntex Discovery Research
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
EC50: 1.40nM
Assay Description:
Agonist activity at human 5-HT2B receptor expressed in Flp-IN HEK293 cells assessed as induction of calcium flux measured every second for 5 mins by ...
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Target
5-hydroxytryptamine receptor 2A
(Homo sapiens (Human))
Eli Lilly
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
Copy SMILES
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Affinity Data
EC50: 2.40nM
Assay Description:
Agonist activity at human 5-HT2A receptor expressed in Flp-IN HEK293 cells assessed as induction of calcium flux measured every second for 5 mins by ...
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Target
5-hydroxytryptamine receptor 2C
(Homo sapiens (Human))
Yamanouchi Pharmaceutical
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
EC50: 0.170nM
Assay Description:
Agonist activity at human 5-HT2C-INI receptor isoform expressed in Flp-IN HEK293 cells assessed as induction of Gq-mediated calcium flux measured eve...
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Target
5-hydroxytryptamine receptor 2C
(Homo sapiens (Human))
Yamanouchi Pharmaceutical
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
EC50: 0.182nM
Assay Description:
Agonist activity at human 5-HT2C-INI receptor isoform expressed in Flp-IN HEK293 cells assessed as induction of Gq-mediated calcium flux measured eve...
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Target
5-hydroxytryptamine receptor 1A
(Homo sapiens (Human))
University of Alberta
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
EC50: 69nM
Assay Description:
Agonist activity at human 5-HT1A receptor expressed in CHO-K1 cells assessed as increase in calcium mobilization measured for 30 secs by aequorin-der...
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Target
5-hydroxytryptamine receptor 1A
(Homo sapiens (Human))
University of Alberta
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
EC50: 98nM
Assay Description:
Agonist activity at human 5-HT1A receptor expressed in CHO-K1 cells co-expressing Galpha16 assessed as increase in calcium mobilization measured for ...
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Target
5-hydroxytryptamine receptor 7
(Homo sapiens (Human))
University Of Namur
Curated by
ChEMBL
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
Copy SMILES
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Affinity Data
EC50: 48nM
Assay Description:
Agonist activity at tTA containing TCS cleavage site-fused 5-HT7 receptor (unknown origin) expressed in tTA-dependent luciferase reporter/TEV-fused b...
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Target
5-hydroxytryptamine receptor 7
(Homo sapiens (Human))
University Of Namur
Curated by
ChEMBL
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
Copy SMILES
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Affinity Data
EC50: 48nM
Assay Description:
Agonist activity at tTA containing TCS cleavage site-fused 5-HT7 receptor (unknown origin) expressed in tTA-dependent luciferase reporter/TEV-fused b...
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Target
5-hydroxytryptamine receptor 2B
(Homo sapiens (Human))
Syntex Discovery Research
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
Copy SMILES
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Affinity Data
EC50: 4.5nM
Assay Description:
Agonist activity at human 5-HT2BR expressed in CHO cells assessed as induction of IP1 accumulation after 30 mins by HTRF method
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Target
5-hydroxytryptamine receptor 1A
(Homo sapiens (Human))
University of Alberta
Curated by
PDSP K
i
Database
Ligand
BDBM10755
(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
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Affinity Data
EC50: 5.70nM
Assay Description:
Agonist activity at human 5-HT1AR expressed in CHO-K1 cells assessed as increase in calcium flux by fluorimetric method
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