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Found 3 Enz. Inhib. hit(s) with Target = '5-hydroxytryptamine receptor 1A' and Ligand = 'BDBM50102396'
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Universidad De Navarra

Curated by ChEMBL
LigandPNGBDBM50102396(1-Phenyl-3-(4-pyrimidin-2-yl-piperazin-1-yl)-propa...)
Affinity DataKi:  120nMAssay Description:Binding affinity to 5-hydroxytryptamine 1A receptor (5-HT 1A receptor, serotonin receptor) from rat cortex using [3H]-8-OH-DPAT as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Universidade Federal Da Para£Ba

Curated by ChEMBL
LigandPNGBDBM50102396(1-Phenyl-3-(4-pyrimidin-2-yl-piperazin-1-yl)-propa...)
Affinity DataKi:  120nMAssay Description:Antagonist activity at 5HT1AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Universidade Federal Da Para£Ba

Curated by ChEMBL
LigandPNGBDBM50102396(1-Phenyl-3-(4-pyrimidin-2-yl-piperazin-1-yl)-propa...)
Affinity DataKi:  120nMAssay Description:Binding affinity to 5HT1A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed