Compile Data Set for Download or QSAR
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Found 2 Enz. Inhib. hit(s) with Target = 'ATP-dependent translocase ABCB1' and Ligand = 'BDBM50572470'
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
Athenex

Curated by ChEMBL
LigandPNGBDBM50572470(CHEMBL4861299)
Affinity DataEC50:  69nMAssay Description:Inhibition of P-gp (unknown origin) expressed in MES-SA/DX5 cells assessed as increase in reversal of resistance to paclitaxel-induced cytotoxicity b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
Athenex

Curated by ChEMBL
LigandPNGBDBM50572470(CHEMBL4861299)
Affinity DataEC50:  5.40nMAssay Description:Inhibition of P-gp (unknown origin) expressed in MCF7 cells assessed as increase in reversal of resistance to paclitaxel-induced cytotoxicity by meas...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed