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Found 4 Enz. Inhib. hit(s) with Target = 'Alpha-1A adrenergic receptor' and Ligand = 'BDBM50259381'
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50259381(6-phenyl-6,7-di hydro-5H-pyrrolo[1,2-a]imidazole |...)
Affinity DataEC50:  83nMAssay Description:Agonist activity at human cloned adrenergic alpha1A receptor expressed in CHO cells assessed as calcium mobilization by FLIPRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50259381(6-phenyl-6,7-di hydro-5H-pyrrolo[1,2-a]imidazole |...)
Affinity DataEC50:  83nMAssay Description:Agonist activity at human cloned adrenergic alpha1A receptor expressed in CHO cells assessed as calcium mobilization by FLIPRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50259381(6-phenyl-6,7-di hydro-5H-pyrrolo[1,2-a]imidazole |...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human cloned adrenergic alpha1A receptor expressed in CHO cells assessed as calcium mobilization by FLIPRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50259381(6-phenyl-6,7-di hydro-5H-pyrrolo[1,2-a]imidazole |...)
Affinity DataEC50:  83nMAssay Description:Agonist activity at human cloned adrenergic alpha1A receptor expressed in CHO cells assessed as calcium mobilization by FLIPRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed