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Found 2 Enz. Inhib. hit(s) with Target = 'Cannabinoid receptor 1' and Ligand = 'BDBM27339'
TargetCannabinoid receptor 1(Homo sapiens (Human))
Pfizer

LigandPNGBDBM27339(9-(4-chlorophenyl)-N-cyclohexyl-8-(2,4-dichlorophe...)
Affinity DataKi:  7.10nM ΔG°:  -47.3kJ/molepH: 7.4 T: 2°CAssay Description:IC50 values for test compounds were determined from nonlinear regression analysis of data collected from ligand binding experiments. The inhibition c...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Pfizer

LigandPNGBDBM27339(9-(4-chlorophenyl)-N-cyclohexyl-8-(2,4-dichlorophe...)
Affinity DataKi:  12nM ΔG°:  -46.0kJ/molepH: 7.4 T: 2°CAssay Description:IC50 values for test compounds were determined from nonlinear regression analysis of data collected from ligand binding experiments. The inhibition c...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed