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Found 5 Enz. Inhib. hit(s) with Target = 'Cruzipain' and Ligand = 'BDBM50295154'
TargetCruzipain(Trypanosoma cruzi)
University Of California

Curated by ChEMBL
LigandPNGBDBM50295154(2-(2,5-dichlorophenylamino)-2-oxoethyl 2-aminonico...)
Affinity DataKi:  3.20E+4nMAssay Description:Competitive inhibition of Trypanosoma cruzi cruzain by Lineaweaver-Burk plot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCruzipain(Trypanosoma cruzi)
University Of California

Curated by ChEMBL
LigandPNGBDBM50295154(2-(2,5-dichlorophenylamino)-2-oxoethyl 2-aminonico...)
Affinity DataIC50:  2.70E+4nMAssay Description:Inhibition of Trypanosoma cruzi cruzain preincubated for 5 mins before substrate addition in presence of 0.001% Triton X-100More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCruzipain(Trypanosoma cruzi)
University Of California

Curated by ChEMBL
LigandPNGBDBM50295154(2-(2,5-dichlorophenylamino)-2-oxoethyl 2-aminonico...)
Affinity DataIC50:  2.70E+4nMAssay Description:Inhibition of Trypanosoma cruzi cruzain preincubated for 5 mins before substrate addition in presence of 0.01% Triton X-100More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCruzipain(Trypanosoma cruzi)
University Of California

Curated by ChEMBL
LigandPNGBDBM50295154(2-(2,5-dichlorophenylamino)-2-oxoethyl 2-aminonico...)
Affinity DataIC50:  7.70E+4nMAssay Description:Inhibition of Trypanosoma cruzi cruzain preincubated for 5 mins before substrate additionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCruzipain(Trypanosoma cruzi)
University Of California

Curated by ChEMBL
LigandPNGBDBM50295154(2-(2,5-dichlorophenylamino)-2-oxoethyl 2-aminonico...)
Affinity DataIC50:  1.16E+5nMAssay Description:Inhibition of Trypanosoma cruzi cruzain preincubated for 5 mins before substrate addition in presence of 0.001% bovine serum albuminMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed