Found 2 Enz. Inhib. hit(s) with Target = 'DNA-dependent protein kinase catalytic subunit' and Ligand = 'BDBM50398037'
TargetDNA-dependent protein kinase catalytic subunit(Homo sapiens (Human))
University Hospital Hradec Kralove
Curated by ChEMBL
University Hospital Hradec Kralove
Curated by ChEMBL
Affinity DataIC50: 400nMAssay Description:Inhibition of DNA-PK purified from HeLa nuclear extracts assessed as EPPLSQEAFADLWKKR peptide substrate phosphorylationMore data for this Ligand-Target Pair
TargetDNA-dependent protein kinase catalytic subunit(Homo sapiens (Human))
University Hospital Hradec Kralove
Curated by ChEMBL
University Hospital Hradec Kralove
Curated by ChEMBL
Affinity DataIC50: 400nMAssay Description:Inhibition of DNA-PK isolated from human HeLa cell extract assessed as inhibition of p53 peptide fragment phosphorylation after 10 minsMore data for this Ligand-Target Pair