Compile Data Set for Download or QSAR
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Found 2 Enz. Inhib. hit(s) with Target = 'Dimer of Protein farnesyltransferase subunit beta' and Ligand = 'BDBM50177643'
TargetDimer of Protein farnesyltransferase subunit beta(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50177643((R)-[8-chloro-6-(1-piperazinyl)-1H-benzo[5,6]]cycl...)
Affinity DataIC50:  7nMAssay Description:Inhibition of farnesyltransferase activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDimer of Protein farnesyltransferase subunit beta(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50177643((R)-[8-chloro-6-(1-piperazinyl)-1H-benzo[5,6]]cycl...)
Affinity DataIC50:  72nMAssay Description:Inhibition of farnesyltransferase activity in COS7 cells transfected with Ras gene in soft agar proliferationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed