Found 2 Enz. Inhib. hit(s) with Target = 'Dual specificity mitogen-activated protein kinase kinase 4' and Ligand = 'BDBM50567686'
TargetDual specificity mitogen-activated protein kinase kinase 4(Homo sapiens (Human))
Eberhard Karls Universit£T
Curated by ChEMBL
Eberhard Karls Universit£T
Curated by ChEMBL
Affinity DataIC50: 146nMAssay Description:Inhibition of MKK4 (unknown origin) by PanQinase assayMore data for this Ligand-Target Pair
TargetDual specificity mitogen-activated protein kinase kinase 4(Homo sapiens (Human))
Eberhard Karls Universit£T
Curated by ChEMBL
Eberhard Karls Universit£T
Curated by ChEMBL
Affinity DataKd: 1.70nMAssay Description:Binding affinity to wild-type human partial length MKK4 (S84 to D399 residues) expressed in mammalian expression system by Kinomescan methodMore data for this Ligand-Target Pair