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Found 3 Enz. Inhib. hit(s) with Target = 'Glucagon receptor' and Ligand = 'BDBM50104372'
TargetGlucagon receptor(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50104372(4-[2-(4-Chloro-phenyl)-5-(4-phenoxy-phenyl)-3H-imi...)
Affinity DataIC50:  27nMAssay Description:Binding affinity towards human glucagon receptor in absence of Mg2+ expressed as IC50More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50104372(4-[2-(4-Chloro-phenyl)-5-(4-phenoxy-phenyl)-3H-imi...)
Affinity DataIC50:  110nMAssay Description:Affinity for human glucagon receptor in presence of Mg2+More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50104372(4-[2-(4-Chloro-phenyl)-5-(4-phenoxy-phenyl)-3H-imi...)
Affinity DataIC50:  250nMAssay Description:Inhibition of human glucagon receptor expressed in CHO cell membranes by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails Article