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Found 2 Enz. Inhib. hit(s) with Target = 'High affinity choline transporter 1' and Ligand = 'BDBM87576'
TargetHigh affinity choline transporter 1(Homo sapiens (Human))
Johns Hopkins Ion Channel Center

Curated by PubChem BioAssay
LigandPNGBDBM87576(MLS001100779 | N-[(3-ethyl-1,2-oxazol-5-yl)methyl]...)
Affinity DataIC50:  18.9nMAssay Description:Data Source (MLPCN Center Name): Johns Hopkins Ion Channel Center (JHICC) Center Affiliation: Johns Hopkins University, School of Medicine Screening ...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetHigh affinity choline transporter 1(Homo sapiens (Human))
Johns Hopkins Ion Channel Center

Curated by PubChem BioAssay
LigandPNGBDBM87576(MLS001100779 | N-[(3-ethyl-1,2-oxazol-5-yl)methyl]...)
Affinity DataIC50:  600nMAssay Description:Inhibition of human CHT Leu530Ala and Val531Ala mutant expressed in HEK293 cells by membrane depolarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed