Affinity DataKi: 30nMAssay Description:Displacement of [3H]UR-DE257 from Gsalphas-coupled human H2R expressed in Sf9 cell membranes by competitive binding assayMore data for this Ligand-Target Pair
Affinity DataEC50: 72nMAssay Description:Agonist activity at human H2 receptor expressed in Sf9 cell membranes co-exprssing GsalphaS assessed as stimulation of [35S]GTPgammaS binding incubat...More data for this Ligand-Target Pair
Affinity DataKd: 81nMAssay Description:Binding affinity to human H2R expressed in HEK293T-qs5-HA cells by flow cytometry analysisMore data for this Ligand-Target Pair