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Found 2 Enz. Inhib. hit(s) with Target = 'Kappa-type opioid receptor' and Ligand = 'BDBM50143602'
TargetKappa-type opioid receptor(Homo sapiens (Human))
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50143602(20-cyclopropylmethyl-(1R,12R)-7-thia-5,20-diazapen...)
Affinity DataKi:  0.0490nMAssay Description:Inhibition of [3H]U-69593 binding to Opioid receptor kappa 1 of Chinese hamster ovary membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50143602(20-cyclopropylmethyl-(1R,12R)-7-thia-5,20-diazapen...)
Affinity DataEC50:  2.40nMAssay Description:Agonistic activity against kappa opioid receptor in Chinese hamster ovary membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed