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Found 2 Enz. Inhib. hit(s) with Target = 'Kappa-type opioid receptor' and Ligand = 'BDBM50257767'
TargetKappa-type opioid receptor(Homo sapiens (Human))
Alkem Laboratories

Curated by ChEMBL
LigandPNGBDBM50257767(CHEMBL4097541)
Affinity DataIC50:  800nMAssay Description:Agonist activity at recombinant human KOR expressed in HEK293T cells assessed as inhibition of forskolin-stimulated cAMP level preincubated for 15 to...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
Alkem Laboratories

Curated by ChEMBL
LigandPNGBDBM50257767(CHEMBL4097541)
Affinity DataIC50:  813nMAssay Description:Antagonist activity at recombinant human MOR expressed in HEK293T cells assessed as reduction in DAMGO-induced inhibition of forskolin-stimulated cAM...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed