Affinity DataKi: 0.590nMAssay Description:Displacement of [3H]U69593 from human KOP stably expressed in CHO cells by competitive binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 0.600nMAssay Description:Displacement of [3H]U69593 from kappa opioid receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataEC50: 0.0770nMAssay Description:Agonist activity at human KOP stably expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKd: 0.590nMAssay Description:Binding affinity to kappa opioid receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataEC50: 1.13E+3nMAssay Description:Agonist activity at kappa opioid receptor (unknown origin) assessed as increase in venus-tagged N-terminal beta-arrestin-2 recruitment by BRET assayMore data for this Ligand-Target Pair
Affinity DataEC50: 5.20nMAssay Description:Agonist activity at kappa opioid receptor (unknown origin) expressed in HEK cells co-expressing luciferase based cAMP biosensor assessed as increase ...More data for this Ligand-Target Pair
Affinity DataEC50: 0.0770nMAssay Description:Inhibition of kappa opioid receptor (unknown origin)More data for this Ligand-Target Pair