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Found 2 Enz. Inhib. hit(s) with Target = 'Lysine-specific histone demethylase 1A' and Ligand = 'BDBM225266'
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
Taipei Medical University

Curated by ChEMBL
LigandPNGBDBM225266(2-((5-Chloro-2-hydroxyphenyl)(methyl)amino)-N-(3-(...)
Affinity DataIC50:  9.50E+3nMAssay Description:Inhibition of human LSD1 (158 to end residues) expressed in Escherichia coli preincubated for 15 mins followed by H3K4me2 peptide addition and measur...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
Taipei Medical University

Curated by ChEMBL
LigandPNGBDBM225266(2-((5-Chloro-2-hydroxyphenyl)(methyl)amino)-N-(3-(...)
Affinity DataIC50:  9.50E+3nMpH: 7.5 T: 2°CAssay Description:The LSD1 screening biochemical assay was performed by Shanghai ChemPartner Co. Ltd and the detailed protocol was shown as followed. The AlphaLISA ass...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed