Affinity DataIC50: 500nMAssay Description:Binding affinity was measured against Opioid receptor mu 1 using [3H]-DAMGO as radioligand.More data for this Ligand-Target Pair
Affinity DataEC50: 1.25E+3nMAssay Description:Tested for electrically induced smooth muscle contractions from guinea pig ileum expressed in mu opioid receptorsMore data for this Ligand-Target Pair