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Found 3 Enz. Inhib. hit(s) with Target = 'Muscarinic acetylcholine receptor M1' and Ligand = 'BDBM50280549'
LigandPNGBDBM50280549((Trans)-(R)-2,7-Dimethyl-1,3-dioxa-7-aza-spiro[4.4...)
Affinity DataKi:  1.75E+3nMAssay Description:In vitro 100 nM cortex affinity to displace [3H]- -CD providing a measure of muscarinic m1 receptor agonist affinityMore data for this Ligand-Target Pair
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LigandPNGBDBM50280549((Trans)-(R)-2,7-Dimethyl-1,3-dioxa-7-aza-spiro[4.4...)
Affinity DataKi:  1.75E+3nMAssay Description:In vitro 100 nM cortex affinity to displace [3H]- -CD providing a measure of muscarinic m1 receptor agonist affinityMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50280549((Trans)-(R)-2,7-Dimethyl-1,3-dioxa-7-aza-spiro[4.4...)
Affinity DataKi: >1.00E+4nMAssay Description:In vitro 100 nM cortex affinity to displace [3H]- -pirenzepine providing a measure of muscarinic m1 receptor antagonist affinityMore data for this Ligand-Target Pair
In DepthDetails Article