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Found 3 Enz. Inhib. hit(s) with Target = 'Prothrombin' and Ligand = 'BDBM50432209'
TargetProthrombin(Homo sapiens (Human))
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50432209(BIBR-1048 | BIBR-1048-BS-RS1 | DABIGATRAN ETEXILAT...)
Affinity DataKi:  4.5nMAssay Description:Binding affinity to human thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50432209(BIBR-1048 | BIBR-1048-BS-RS1 | DABIGATRAN ETEXILAT...)
Affinity DataIC50:  2.60nMAssay Description:Inhibition of human thrombin preincubated for 10 mins using Ac-FVR-AMC as substrate by chromogenic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50432209(BIBR-1048 | BIBR-1048-BS-RS1 | DABIGATRAN ETEXILAT...)
Affinity DataIC50:  2.60nMAssay Description:Inhibition of human thrombin preincubated for 10 mins using Ac-FVR-AMC as substrate by chromogenic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed