Compile Data Set for Download or QSAR
maximum 50k data
Found 3 Enz. Inhib. hit(s) with Target = 'RAC-alpha serine/threonine-protein kinase' and Ligand = 'BDBM24867'
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

LigandPNGBDBM24867(1-(2-aminophenyl)-3-[({4-[2-(methylsulfanyl)-6-phe...)
Affinity DataIC50:  15nMpH: 7.5 T: 2°CAssay Description:Purified recombinant human Akt kinase was monitored for kinase activity in the presence or absence of inhibitors in a 96-well format. Detection was d...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

LigandPNGBDBM24867(1-(2-aminophenyl)-3-[({4-[2-(methylsulfanyl)-6-phe...)
Affinity DataIC50:  15nMAssay Description:Inhibition of Akt1 (unknown origin) phosphorylation by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

LigandPNGBDBM24867(1-(2-aminophenyl)-3-[({4-[2-(methylsulfanyl)-6-phe...)
Affinity DataIC50:  78nMAssay Description:Inhibition of Akt1 (unknown origin) phosphorylation in human by C33a cells by IPKA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed