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Found 4 Enz. Inhib. hit(s) with Target = 'Sigma non-opioid intracellular receptor 1' and Ligand = 'BDBM50040287'
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
University Of North Carolina

Curated by ChEMBL
LigandPNGBDBM50040287((1R,3S)Dimethyl-(2-methyl-4-phenyl-1,2,3,4-tetrahy...)
Affinity DataIC50:  0.510nMAssay Description:Binding affinity against sigma receptor from guinea pig brain (minus cerebellum) homogenates, using the novel [3H]-(+/-)-4 as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
University Of North Carolina

Curated by ChEMBL
LigandPNGBDBM50040287((1R,3S)Dimethyl-(2-methyl-4-phenyl-1,2,3,4-tetrahy...)
Affinity DataIC50:  0.510nMAssay Description:Binding affinity against dopamine receptor D1 from rat striatal homogenates, using [3H]SCH-23390 as radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
University Of North Carolina

Curated by ChEMBL
LigandPNGBDBM50040287((1R,3S)Dimethyl-(2-methyl-4-phenyl-1,2,3,4-tetrahy...)
Affinity DataIC50:  5.31E+3nMAssay Description:Binding affinity against dopamine receptor D2 from rat striatal homogenates using [3H]YM-09151-2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
University Of North Carolina

Curated by ChEMBL
LigandPNGBDBM50040287((1R,3S)Dimethyl-(2-methyl-4-phenyl-1,2,3,4-tetrahy...)
Affinity DataIC50:  5.31E+3nMAssay Description:Binding affinity against sigma receptor from guinea pig brain (minus cerebellum) homogenates, using the novel [3H]-(+/-)-4 as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed