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Found 4 Enz. Inhib. hit(s) with Target = 'Sodium-dependent serotonin transporter' and Ligand = 'BDBM50076047'
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Organix

Curated by ChEMBL
LigandPNGBDBM50076047((1R/1S)-methyl 3-(3,4-dichlorophenyl)-8-oxa-bicycl...)
Affinity DataIC50:  1.90E+3nMAssay Description:Inhibition of [3H]citalopram binding to human serotonin transporter (hSERT)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Organix

Curated by ChEMBL
LigandPNGBDBM50076047((1R/1S)-methyl 3-(3,4-dichlorophenyl)-8-oxa-bicycl...)
Affinity DataIC50:  1.96E+3nMAssay Description:Inhibition of [3H]citalopram binding to serotonin transporter (SERT) of cynomolgus monkey caudate-putamenMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Organix

Curated by ChEMBL
LigandPNGBDBM50076047((1R/1S)-methyl 3-(3,4-dichlorophenyl)-8-oxa-bicycl...)
Affinity DataIC50:  2.12E+3nMAssay Description:Inhibition of [3H]citalopram binding to serotonin transporter (SERT) of cynomolgus monkey caudate-putamenMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Macaca mulatta)
Organix

Curated by ChEMBL
LigandPNGBDBM50076047((1R/1S)-methyl 3-(3,4-dichlorophenyl)-8-oxa-bicycl...)
Affinity DataIC50:  6.00E+3nMAssay Description:Displacement of [3H]citalopram from SERT in rhesus monkey caudate-putamenMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed