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Found 2 Enz. Inhib. hit(s) with Target = 'Thyrotropin-releasing hormone receptor' and Ligand = 'BDBM50072395'
TargetThyrotropin-releasing hormone receptor(MOUSE)
Washington University

Curated by ChEMBL
LigandPNGBDBM50072395(1-[3-cyclohexyl-2-(5-oxotetrahydro-1H-2-pyrrolylca...)
Affinity DataKi:  6.50E+3nMAssay Description:Ability to bind thyroliberin endocrine receptor (TRH-R) using AtT-20 mouse pituitary tumor cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThyrotropin-releasing hormone receptor(MOUSE)
Washington University

Curated by ChEMBL
LigandPNGBDBM50072395(1-[3-cyclohexyl-2-(5-oxotetrahydro-1H-2-pyrrolylca...)
Affinity DataEC50:  430nMAssay Description:Ability to activate thyroliberin endocrine receptor (TRH-R) using AtT-20 mouse pituitary tumor cells prelabelled with myo-[3H] inositolMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed