Found 4 Enz. Inhib. hit(s) with Target = 'Transient receptor potential cation channel subfamily V member 2' and Ligand = 'BDBM50318487'
TargetTransient receptor potential cation channel subfamily V member 2(Rattus norvegicus)
Universita` Del Piemonte Orientale
Curated by ChEMBL
Universita` Del Piemonte Orientale
Curated by ChEMBL
Affinity DataIC50: 1.50E+3nMAssay Description:Agonist activity at rat recombinant TRPV2 receptor expressed in HEK293 cells assessed as stimulation of intracellular calcium level using Fluo4-AM dy...More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 2(Homo sapiens)
Scientus Pharma
Curated by ChEMBL
Scientus Pharma
Curated by ChEMBL
Affinity DataIC50: 1.50E+3nMAssay Description:Agonist activity at ionomycin-stimulated TRPV2 (unknown origin) channel desensitization in presence of lysophosphatidylcholineMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 2(Homo sapiens)
Scientus Pharma
Curated by ChEMBL
Scientus Pharma
Curated by ChEMBL
Affinity DataEC50: 1.70E+3nMAssay Description:Agonist activity at ionomycin-stimulated TRPV2 (unknown origin) activationMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 2(Rattus norvegicus)
Universita` Del Piemonte Orientale
Curated by ChEMBL
Universita` Del Piemonte Orientale
Curated by ChEMBL
Affinity DataEC50: 1.70E+3nMAssay Description:Agonist activity at rat recombinant TRPV2 receptor expressed in HEK293 cells assessed as stimulation of intracellular calcium level using Fluo4-AM dy...More data for this Ligand-Target Pair