Found 2 Enz. Inhib. hit(s) with Target = 'Transient receptor potential cation channel subfamily V member 2' and Ligand = 'BDBM50511105'
TargetTransient receptor potential cation channel subfamily V member 2(Homo sapiens)
Scientus Pharma
Curated by ChEMBL
Scientus Pharma
Curated by ChEMBL
Affinity DataIC50: 800nMAssay Description:Agonist activity at ionomycin-stimulated TRPV2 (unknown origin) channel desensitization in presence of lysophosphatidylcholineMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 2(Homo sapiens)
Scientus Pharma
Curated by ChEMBL
Scientus Pharma
Curated by ChEMBL
Affinity DataEC50: 4.10E+3nMAssay Description:Agonist activity at ionomycin-stimulated TRPV2 (unknown origin) activationMore data for this Ligand-Target Pair