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Found 1 Enz. Inhib. hit(s) with Target = 'Tyrosine-protein kinase Lck' and Ligand = 'BDBM50112913'
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50112913(2-Bromo-N-imidazo[1,5-a]quinoxalin-4-yl-benzamide ...)
Affinity DataIC50:  60nMAssay Description:Inhibitory activity against recombinant p56 Lck tyrosine kinase expressed as a His-tagged protein in insect cells using a baculovirus expression syst...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed