Compile Data Set for Download or QSAR
maximum 50k data
Found 4 Enz. Inhib. hit(s) with Target = 'Tyrosine-protein kinase SYK' and Ligand = 'BDBM50431366'
TargetTyrosine-protein kinase SYK(Homo sapiens (Human))
Second Military Medical University

Curated by ChEMBL
LigandPNGBDBM50431366(CHEMBL2347996)
Affinity DataIC50:  26nMAssay Description:Inhibition of [3H]5-HT reuptake at serotonin transporter in rat mid brainMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase SYK(Homo sapiens (Human))
Second Military Medical University

Curated by ChEMBL
LigandPNGBDBM50431366(CHEMBL2347996)
Affinity DataIC50:  26nMAssay Description:Inhibition of human recombinant truncated SYK (360 to 365 amino acid residues) using N-terminally biotinylated EPEGDYEEVLE peptide as substrate asses...More data for this Ligand-Target Pair
TargetTyrosine-protein kinase SYK(Homo sapiens (Human))
Second Military Medical University

Curated by ChEMBL
LigandPNGBDBM50431366(CHEMBL2347996)
Affinity DataIC50:  450nMAssay Description:Inhibition of SYK in human Ramos cellsMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase SYK(Homo sapiens (Human))
Second Military Medical University

Curated by ChEMBL
LigandPNGBDBM50431366(CHEMBL2347996)
Affinity DataIC50:  634nMAssay Description:Inhibition of SYK in human whole bloodMore data for this Ligand-Target Pair