Compile Data Set for Download or QSAR
maximum 50k data
Found 80 of ec50 for UniProtKB: P37230
TargetPeroxisome proliferator-activated receptor alpha(Rattus norvegicus)
Johnson & Johnson

Curated by ChEMBL
LigandPNGBDBM50227669((R)-2-(2-(1-ethyl-3-(4-(trifluoromethoxy)phenyl)ur...)
Affinity DataEC50:  2nMAssay Description:Agonist activity at rat PPARalpha in rat H4IIE cells assessed as gene inductionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Rattus norvegicus)
Johnson & Johnson

Curated by ChEMBL
LigandPNGBDBM50227674(2-(2-(1-ethyl-3-(4-(trifluoromethylthio)phenyl)ure...)
Affinity DataEC50:  23nMAssay Description:Agonist activity at rat PPARalpha in rat H4IIE cells assessed as gene inductionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Rattus norvegicus)
Johnson & Johnson

Curated by ChEMBL
LigandPNGBDBM50227656(2-(2-(1-ethyl-3-(4-isopropylphenyl)ureido)-2,3-dih...)
Affinity DataEC50:  32nMAssay Description:Agonist activity at rat PPARalpha in rat H4IIE cells assessed as gene inductionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Rattus norvegicus)
Johnson & Johnson

Curated by ChEMBL
LigandPNGBDBM50227664(2-(2-(1-ethyl-3-(4-(trifluoromethoxy)phenyl)ureido...)
Affinity DataEC50:  33nMAssay Description:Agonist activity at rat PPARalpha in rat H4IIE cells assessed as gene inductionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Rattus norvegicus)
Johnson & Johnson

Curated by ChEMBL
LigandPNGBDBM50227704(2-methyl-2-(2-(1-pentyl-3-(4-(trifluoromethylthio)...)
Affinity DataEC50:  46nMAssay Description:Agonist activity at rat PPARalpha in rat H4IIE cells assessed as gene inductionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Rattus norvegicus)
Johnson & Johnson

Curated by ChEMBL
LigandPNGBDBM50227696(2-methyl-2-(2-(3-(4-(trifluoromethoxy)phenyl)ureid...)
Affinity DataEC50:  96nMAssay Description:Agonist activity at rat PPARalpha in rat H4IIE cells assessed as gene inductionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Rattus norvegicus)
Johnson & Johnson

Curated by ChEMBL
LigandPNGBDBM50227663(2-methyl-2-(2-(1-pentyl-3-(4-(trifluoromethoxy)phe...)
Affinity DataEC50:  105nMAssay Description:Agonist activity at rat PPARalpha in rat H4IIE cells assessed as gene inductionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Rattus norvegicus)
Johnson & Johnson

Curated by ChEMBL
LigandPNGBDBM50227677(2-(2-(3-(4-(dimethylamino)phenyl)-1-ethylureido)-2...)
Affinity DataEC50:  117nMAssay Description:Agonist activity at rat PPARalpha in rat H4IIE cells assessed as gene inductionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Rattus norvegicus)
Johnson & Johnson

Curated by ChEMBL
LigandPNGBDBM28802(2-{[(5-{[2-(4-chlorophenyl)-5-methyl-1,3-oxazol-4-...)
Affinity DataEC50:  123nMAssay Description:EC50 is the concentration of test compounds needed to induce 50% of the maximum luciferase activity in HEK cells transfected with PPAR and Gal4-lucif...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Rattus norvegicus)
Johnson & Johnson

Curated by ChEMBL
LigandPNGBDBM28802(2-{[(5-{[2-(4-chlorophenyl)-5-methyl-1,3-oxazol-4-...)
Affinity DataEC50:  123nMAssay Description:Agonist activity at rat PPAR-alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Rattus norvegicus)
Johnson & Johnson

Curated by ChEMBL
LigandPNGBDBM50227658(2-(2-(3-(4-(dimethylamino)phenyl)-1-pentylureido)-...)
Affinity DataEC50:  141nMAssay Description:Agonist activity at rat PPARalpha in rat H4IIE cells assessed as gene inductionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Rattus norvegicus)
Johnson & Johnson

Curated by ChEMBL
LigandPNGBDBM50227660((R)-2-methyl-2-(2-(3-(4-(trifluoromethoxy)phenyl)u...)
Affinity DataEC50:  146nMAssay Description:Agonist activity at rat PPARalpha in rat H4IIE cells assessed as gene inductionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Rattus norvegicus)
Johnson & Johnson

Curated by ChEMBL
LigandPNGBDBM50227668(2-methyl-2-(2-(1-propyl-3-(4-(trifluoromethoxy)phe...)
Affinity DataEC50:  158nMAssay Description:Agonist activity at rat PPARalpha in rat H4IIE cells assessed as gene inductionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Rattus norvegicus)
Johnson & Johnson

Curated by ChEMBL
LigandPNGBDBM50227659(2-(2-(3-(4-isopropylphenyl)-1-pentylureido)-2,3-di...)
Affinity DataEC50:  159nMAssay Description:Agonist activity at rat PPARalpha in rat H4IIE cells assessed as gene inductionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Rattus norvegicus)
Johnson & Johnson

Curated by ChEMBL
LigandPNGBDBM50227666(2-(2-(1-butyl-3-(4-(trifluoromethylthio)phenyl)ure...)
Affinity DataEC50:  160nMAssay Description:Agonist activity at rat PPARalpha in rat H4IIE cells assessed as gene inductionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Rattus norvegicus)
Johnson & Johnson

Curated by ChEMBL
LigandPNGBDBM50227675((S)-2-(2-(1-ethyl-3-(4-(trifluoromethoxy)phenyl)ur...)
Affinity DataEC50:  165nMAssay Description:Agonist activity at rat PPARalpha in rat H4IIE cells assessed as gene inductionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Rattus norvegicus)
Johnson & Johnson

Curated by ChEMBL
LigandPNGBDBM50227688(2-(2-(1-hexyl-3-(4-(trifluoromethoxy)phenyl)ureido...)
Affinity DataEC50:  166nMAssay Description:Agonist activity at rat PPARalpha in rat H4IIE cells assessed as gene inductionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Rattus norvegicus)
Johnson & Johnson

Curated by ChEMBL
LigandPNGBDBM28799(2-{[4-(2-{[(2,4-difluorophenyl)carbamoyl](heptyl)a...)
Affinity DataEC50:  166nMAssay Description:Agonist activity at rat PPARalpha in rat H4IIE cells assessed as gene inductionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Rattus norvegicus)
Johnson & Johnson

Curated by ChEMBL
LigandPNGBDBM50227705((R)-2-(2-(1-heptyl-3-(4-(trifluoromethoxy)phenyl)u...)
Affinity DataEC50:  169nMAssay Description:Agonist activity at rat PPARalpha in rat H4IIE cells assessed as gene inductionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Rattus norvegicus)
Johnson & Johnson

Curated by ChEMBL
LigandPNGBDBM50227678(2-(2-(1-hexyl-3-(4-isopropylphenyl)ureido)-2,3-dih...)
Affinity DataEC50:  180nMAssay Description:Agonist activity at rat PPARalpha in rat H4IIE cells assessed as gene inductionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Rattus norvegicus)
Johnson & Johnson

Curated by ChEMBL
LigandPNGBDBM50227661(2-(2-(1-butyl-3-(4-(trifluoromethoxy)phenyl)ureido...)
Affinity DataEC50:  195nMAssay Description:Agonist activity at rat PPARalpha in rat H4IIE cells assessed as gene inductionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Rattus norvegicus)
Johnson & Johnson

Curated by ChEMBL
LigandPNGBDBM50227657(2-(2-(1-heptyl-3-(4-(methylthio)phenyl)ureido)-2,3...)
Affinity DataEC50:  210nMAssay Description:Agonist activity at rat PPARalpha in rat H4IIE cells assessed as gene inductionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Rattus norvegicus)
Johnson & Johnson

Curated by ChEMBL
LigandPNGBDBM50227682(2-(2-(3-(4-(dimethylamino)phenyl)-1-hexylureido)-2...)
Affinity DataEC50:  219nMAssay Description:Agonist activity at rat PPARalpha in rat H4IIE cells assessed as gene inductionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Rattus norvegicus)
Johnson & Johnson

Curated by ChEMBL
LigandPNGBDBM50227703(2-(2-(1-heptyl-3-(4-(trifluoromethylthio)phenyl)ur...)
Affinity DataEC50:  229nMAssay Description:Agonist activity at rat PPARalpha in rat H4IIE cells assessed as gene inductionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Rattus norvegicus)
Johnson & Johnson

Curated by ChEMBL
LigandPNGBDBM50227685(2-(2-(1-hexyl-3-(4-(trifluoromethylthio)phenyl)ure...)
Affinity DataEC50:  249nMAssay Description:Agonist activity at rat PPARalpha in rat H4IIE cells assessed as gene inductionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Rattus norvegicus)
Johnson & Johnson

Curated by ChEMBL
LigandPNGBDBM50227671(2-(2-(1-heptyl-3-(4-isopropylphenyl)ureido)-2,3-di...)
Affinity DataEC50:  252nMAssay Description:Agonist activity at rat PPARalpha in rat H4IIE cells assessed as gene inductionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Rattus norvegicus)
Johnson & Johnson

Curated by ChEMBL
LigandPNGBDBM50227662(2-(2-(3-(4-(dimethylamino)phenyl)-1-heptylureido)-...)
Affinity DataEC50:  252nMAssay Description:Agonist activity at rat PPARalpha in rat H4IIE cells assessed as gene inductionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Rattus norvegicus)
Johnson & Johnson

Curated by ChEMBL
LigandPNGBDBM50227687(2-(2-(1-butyl-3-(4-isopropylphenyl)ureido)-2,3-dih...)
Affinity DataEC50:  260nMAssay Description:Agonist activity at rat PPARalpha in rat H4IIE cells assessed as gene inductionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Rattus norvegicus)
Johnson & Johnson

Curated by ChEMBL
LigandPNGBDBM50227683(2-(2-(1-heptyl-3-(4-(trifluoromethoxy)phenyl)ureid...)
Affinity DataEC50:  294nMAssay Description:Agonist activity at rat PPARalpha in rat H4IIE cells assessed as gene inductionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Rattus norvegicus)
Johnson & Johnson

Curated by ChEMBL
LigandPNGBDBM28800(2-{[(3-{[2-(4-chlorophenyl)-5-methyl-1,3-oxazol-4-...)
Affinity DataEC50:  317nMAssay Description:EC50 is the concentration of test compounds needed to induce 50% of the maximum luciferase activity in HEK cells transfected with PPAR and Gal4-lucif...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Rattus norvegicus)
Johnson & Johnson

Curated by ChEMBL
LigandPNGBDBM28800(2-{[(3-{[2-(4-chlorophenyl)-5-methyl-1,3-oxazol-4-...)
Affinity DataEC50:  317nMAssay Description:Agonist activity at rat PPAR-alphaMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Rattus norvegicus)
Johnson & Johnson

Curated by ChEMBL
LigandPNGBDBM50227692(2-(2-(1-isopentyl-3-(4-(trifluoromethoxy)phenyl)ur...)
Affinity DataEC50:  386nMAssay Description:Agonist activity at rat PPARalpha in rat H4IIE cells assessed as gene inductionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Rattus norvegicus)
Johnson & Johnson

Curated by ChEMBL
LigandPNGBDBM50227690(2-(2-(1-(2-methoxyethyl)-3-(4-(trifluoromethoxy)ph...)
Affinity DataEC50:  425nMAssay Description:Agonist activity at rat PPARalpha in rat H4IIE cells assessed as gene inductionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Rattus norvegicus)
Johnson & Johnson

Curated by ChEMBL
LigandPNGBDBM50227679(2-(2-(1-butyl-3-(4-(dimethylamino)phenyl)ureido)-2...)
Affinity DataEC50:  561nMAssay Description:Agonist activity at rat PPARalpha in rat H4IIE cells assessed as gene inductionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Rattus norvegicus)
Johnson & Johnson

Curated by ChEMBL
LigandPNGBDBM50227697(2-(2-(1-ethyl-3-(2-methyl-4-(trifluoromethoxy)phen...)
Affinity DataEC50:  598nMAssay Description:Agonist activity at rat PPARalpha in rat H4IIE cells assessed as gene inductionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Rattus norvegicus)
Johnson & Johnson

Curated by ChEMBL
LigandPNGBDBM50134840((S)-2-Ethoxy-3-[4-((E)-5-phenyl-pent-2-en-4-ynylox...)
Affinity DataEC50:  700nMAssay Description:In vitro transactivation of rat Peroxisome proliferator activated receptor alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Rattus norvegicus)
Johnson & Johnson

Curated by ChEMBL
LigandPNGBDBM50227689(2-methyl-2-(2-(1-(4,4,4-trifluorobutyl)-3-(4-(trif...)
Affinity DataEC50:  707nMAssay Description:Agonist activity at rat PPARalpha in rat H4IIE cells assessed as gene inductionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Rattus norvegicus)
Johnson & Johnson

Curated by ChEMBL
LigandPNGBDBM50227700(2-(2-(1-heptyl-3-(4-methoxyphenyl)ureido)-2,3-dihy...)
Affinity DataEC50:  910nMAssay Description:Agonist activity at rat PPARalpha in rat H4IIE cells assessed as gene inductionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Rattus norvegicus)
Johnson & Johnson

Curated by ChEMBL
LigandPNGBDBM50227673(2-(2-(3-(2-bromo-4-(trifluoromethoxy)phenyl)-1-eth...)
Affinity DataEC50: >1.00E+3nMAssay Description:Agonist activity at rat PPARalpha in rat H4IIE cells assessed as gene inductionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Rattus norvegicus)
Johnson & Johnson

Curated by ChEMBL
LigandPNGBDBM50227701(2-methyl-2-(2-(1-octyl-3-(4-(trifluoromethoxy)phen...)
Affinity DataEC50:  1.03E+3nMAssay Description:Agonist activity at rat PPARalpha in rat H4IIE cells assessed as gene inductionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Rattus norvegicus)
Johnson & Johnson

Curated by ChEMBL
LigandPNGBDBM50227693(2-(2-(1-heptyl-3-(3-methoxyphenyl)ureido)-2,3-dihy...)
Affinity DataEC50:  1.11E+3nMAssay Description:Agonist activity at rat PPARalpha in rat H4IIE cells assessed as gene inductionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Rattus norvegicus)
Johnson & Johnson

Curated by ChEMBL
LigandPNGBDBM50227670((S)-2-methyl-2-(2-(3-(4-(trifluoromethoxy)phenyl)u...)
Affinity DataEC50:  1.11E+3nMAssay Description:Agonist activity at rat PPARalpha in rat H4IIE cells assessed as gene inductionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Rattus norvegicus)
Johnson & Johnson

Curated by ChEMBL
LigandPNGBDBM50227654(2-(2-(1-heptyl-3-(4-(trifluoromethyl)phenyl)ureido...)
Affinity DataEC50:  1.27E+3nMAssay Description:Agonist activity at rat PPARalpha in rat H4IIE cells assessed as gene inductionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Rattus norvegicus)
Johnson & Johnson

Curated by ChEMBL
LigandPNGBDBM50227681(2-(2-(1-heptyl-3-(2-(trifluoromethylthio)phenyl)ur...)
Affinity DataEC50:  1.96E+3nMAssay Description:Agonist activity at rat PPARalpha in rat H4IIE cells assessed as gene inductionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Rattus norvegicus)
Johnson & Johnson

Curated by ChEMBL
LigandPNGBDBM50227667(2-(2-(3-(3-chlorophenyl)-1-heptylureido)-2,3-dihyd...)
Affinity DataEC50:  2.09E+3nMAssay Description:Agonist activity at rat PPARalpha in rat H4IIE cells assessed as gene inductionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Rattus norvegicus)
Johnson & Johnson

Curated by ChEMBL
LigandPNGBDBM24566(2-({4-chloro-6-[(2,3-dimethylphenyl)amino]pyrimidi...)
Affinity DataEC50:  2.10E+3nMAssay Description:In vitro transactivation of rat Peroxisome proliferator activated receptor alphaMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Rattus norvegicus)
Johnson & Johnson

Curated by ChEMBL
LigandPNGBDBM50277897((2S)-2-methoxy-3-{4-[2-(5-methyl-2-phenyl-1,3-oxaz...)
Affinity DataEC50:  2.26E+3nMAssay Description:Agonist activity at rat PPARalphaMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Rattus norvegicus)
Johnson & Johnson

Curated by ChEMBL
LigandPNGBDBM50227698(2-(2-(1-isobutyl-3-(4-(trifluoromethoxy)phenyl)ure...)
Affinity DataEC50:  2.34E+3nMAssay Description:Agonist activity at rat PPARalpha in rat H4IIE cells assessed as gene inductionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Rattus norvegicus)
Johnson & Johnson

Curated by ChEMBL
LigandPNGBDBM50227665(2-(2-(3-(3-fluorophenyl)-1-heptylureido)-2,3-dihyd...)
Affinity DataEC50:  2.67E+3nMAssay Description:Agonist activity at rat PPARalpha in rat H4IIE cells assessed as gene inductionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Rattus norvegicus)
Johnson & Johnson

Curated by ChEMBL
LigandPNGBDBM50227706(2-(2-(1-heptyl-3-(3-(trifluoromethyl)phenyl)ureido...)
Affinity DataEC50:  2.73E+3nMAssay Description:Agonist activity at rat PPARalpha in rat H4IIE cells assessed as gene inductionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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