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Found 59 Enz. Inhib. hit(s) with all data for entry = 50018708
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))TBA
LigandPNGBDBM50110719(5-Methoxymethyl-3-pyrrol-1-yl-oxazolidin-2-one | C...)
Affinity DataKi:  4.90nMAssay Description:Inhibition of recombinant human MAO-A using kynuramine as substrate incubated for 20 mins by spectrophotometry analysisMore data for this Ligand-Target Pair
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TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))TBA
LigandPNGBDBM15611(N-Methyl,N-(propargyl),N-(pyrrol-2-ylmethyl)amine ...)
Affinity DataKi:  5.40nMAssay Description:Inhibition of MAO-A (unknown origin)More data for this Ligand-Target Pair
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TargetAmine oxidase [flavin-containing] B(Rattus norvegicus (rat))TBA
LigandPNGBDBM50028010(AD-810 | CHEBI:10127 | CI-912 | PD-110843 | Zonegr...)
Affinity DataKi:  2.90E+3nMAssay Description:Competitive inhibition of rat MAO-BMore data for this Ligand-Target Pair
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TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))TBA
LigandPNGBDBM50028010(AD-810 | CHEBI:10127 | CI-912 | PD-110843 | Zonegr...)
Affinity DataKi:  3.10E+3nMAssay Description:Competitive inhibition of human MAO-BMore data for this Ligand-Target Pair
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TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))TBA
LigandPNGBDBM50611766(CHEMBL5268461)
Affinity DataKi:  1.50E+4nMAssay Description:Irreversible inhibition of human recombinant MAO-BMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))TBA
LigandPNGBDBM50028010(AD-810 | CHEBI:10127 | CI-912 | PD-110843 | Zonegr...)
Affinity DataKi:  3.08E+4nMAssay Description:Inhibition of MAO-B (unknown origin)More data for this Ligand-Target Pair
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TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))TBA
LigandPNGBDBM50113840(4-Phenyl-butylamine | 4-phenylbutylamine | CHEMBL7...)
Affinity DataKi:  3.10E+4nMAssay Description:Competitive inhibition of human MAO-AMore data for this Ligand-Target Pair
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TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))TBA
LigandPNGBDBM50611765(CHEMBL5283202)
Affinity DataKi:  2.68E+5nMAssay Description:Irreversible inhibition of human recombinant MAO-AMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))TBA
LigandPNGBDBM174835(US9114126, 2027BA1)
Affinity DataIC50:  0.220nMAssay Description:Inhibition of rat MAO-AMore data for this Ligand-Target Pair
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TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))TBA
LigandPNGBDBM50029819(2-{5-[4-(3-Chloro-benzyloxy)-phenyl]-tetrazol-2-yl...)
Affinity DataIC50:  2nMAssay Description:Inhibition of human MAO-BMore data for this Ligand-Target Pair
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TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))TBA
LigandPNGBDBM50029810(2-[5-(4-Benzyloxy-phenyl)-tetrazol-2-yl]-ethanol |...)
Affinity DataIC50:  2nMAssay Description:Inhibition of human MAO-BMore data for this Ligand-Target Pair
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TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))TBA
LigandPNGBDBM50611767(CHEMBL63782)
Affinity DataIC50:  10nMAssay Description:Inhibition of human recombinant MAO-AMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))TBA
LigandPNGBDBM50038938(CHEMBL417566 | N-(6-Ethyl-9,10,10-trioxo-9,10-dihy...)
Affinity DataIC50:  10nMAssay Description:Inhibition of human recombinant MAO-AMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))TBA
LigandPNGBDBM50038939(CHEMBL63678 | N-(5,5-Dioxo-5,10-dihydro-5lambda*6*...)
Affinity DataIC50:  10nMAssay Description:Inhibition of human recombinant MAO-AMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))TBA
LigandPNGBDBM50611768(CHEMBL292052)
Affinity DataIC50:  10nMAssay Description:Inhibition of human recombinant MAO-AMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))TBA
LigandPNGBDBM50038943(CHEMBL66260 | N-(7-Acetylamino-10-methyl-5,5-dioxo...)
Affinity DataIC50:  10nMAssay Description:Inhibition of human recombinant MAO-AMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))TBA
LigandPNGBDBM50611769(CHEMBL65583)
Affinity DataIC50:  10nMAssay Description:Inhibition of human recombinant MAO-AMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))TBA
LigandPNGBDBM50038932(CHEMBL304069 | N-(9,10-Dioxo-9,10-dihydro-anthrace...)
Affinity DataIC50:  10nMAssay Description:Inhibition of human recombinant MAO-AMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))TBA
LigandPNGBDBM50611770(CHEMBL304484)
Affinity DataIC50:  10nMAssay Description:Inhibition of human recombinant MAO-AMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))TBA
LigandPNGBDBM50611771(CHEMBL5270901)
Affinity DataIC50:  10nMAssay Description:Inhibition of human recombinant MAO-AMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))TBA
LigandPNGBDBM50038941(CHEMBL63510 | N-(6-Methyl-9,10,10-trioxo-9,10-dihy...)
Affinity DataIC50:  10nMAssay Description:Inhibition of human recombinant MAO-AMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))TBA
LigandPNGBDBM50038942(CHEMBL63458 | N-(9,10,10-Trioxo-9,10-dihydro-10lam...)
Affinity DataIC50:  10nMAssay Description:Inhibition of human recombinant MAO-AMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))TBA
LigandPNGBDBM50038934(CHEMBL65156 | N-(9,10,10-Trioxo-9,10-dihydro-10lam...)
Affinity DataIC50:  10nMAssay Description:Inhibition of human recombinant MAO-AMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))TBA
LigandPNGBDBM50038947(CHEMBL63934 | N-(10,10-Dioxo-10H-10lambda*6*-pheno...)
Affinity DataIC50:  10nMAssay Description:Inhibition of human recombinant MAO-AMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))TBA
LigandPNGBDBM50038946(CHEMBL63141 | N-(9,10,10-Trioxo-6-propyl-9,10-dihy...)
Affinity DataIC50:  10nMAssay Description:Inhibition of human recombinant MAO-AMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))TBA
LigandPNGBDBM50261815(2-(3,4-dimethoxyphenyl)-3-fluoroprop-2-en-1-amine ...)
Affinity DataIC50:  10nMAssay Description:Inhibition of MAO-B (unknown origin)More data for this Ligand-Target Pair
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TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))TBA
LigandPNGBDBM50428646(CHEMBL2332175)
Affinity DataIC50:  11nMAssay Description:Reversible inhibition of human MAO-BMore data for this Ligand-Target Pair
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TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))TBA
LigandPNGBDBM50029816(5-Chloro-pyridine-2-carboxylic acid (2-amino-ethyl...)
Affinity DataIC50:  30nMAssay Description:Inhibition of human MAO-BMore data for this Ligand-Target Pair
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TargetAmine oxidase [flavin-containing] B(Rattus norvegicus (rat))TBA
LigandPNGBDBM50031048(3-(4-(trifluoromethyl)phenyl)-5H-indeno[1,2-c]pyri...)
Affinity DataIC50:  90nMAssay Description:Inhibition of rat brain MAO-BMore data for this Ligand-Target Pair
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TargetAcetylcholinesterase(Homo sapiens (Human))TBA
LigandPNGBDBM50409091(CHEMBL109085)
Affinity DataIC50:  3.00E+3nMAssay Description:Inhibition of AChE (unknown origin) using acetylthiocholine chloride as substrate incubated for 5 mins by DTNB reagent based Ellman's methodMore data for this Ligand-Target Pair
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TargetAcetylcholinesterase(Homo sapiens (Human))TBA
LigandPNGBDBM50409109(CHEMBL108928)
Affinity DataIC50:  3.00E+3nMAssay Description:Inhibition of AChE (unknown origin) using acetylthiocholine chloride as substrate incubated for 5 mins by DTNB reagent based Ellman's methodMore data for this Ligand-Target Pair
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TargetAcetylcholinesterase(Homo sapiens (Human))TBA
LigandPNGBDBM50409094(CHEMBL107488)
Affinity DataIC50:  3.00E+3nMAssay Description:Inhibition of AChE (unknown origin) using acetylthiocholine chloride as substrate incubated for 5 mins by DTNB reagent based Ellman's methodMore data for this Ligand-Target Pair
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TargetAcetylcholinesterase(Homo sapiens (Human))TBA
LigandPNGBDBM50611773(CHEMBL5290626)
Affinity DataIC50:  3.00E+3nMAssay Description:Inhibition of AChE (unknown origin) using acetylthiocholine chloride as substrate incubated for 5 mins by DTNB reagent based Ellman's methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetAcetylcholinesterase(Homo sapiens (Human))TBA
LigandPNGBDBM50409081(CHEMBL111309)
Affinity DataIC50:  3.00E+3nMAssay Description:Inhibition of AChE (unknown origin) using acetylthiocholine chloride as substrate incubated for 5 mins by DTNB reagent based Ellman's methodMore data for this Ligand-Target Pair
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TargetAcetylcholinesterase(Homo sapiens (Human))TBA
LigandPNGBDBM50611774(CHEMBL5271985)
Affinity DataIC50:  3.00E+3nMAssay Description:Inhibition of AChE (unknown origin) using acetylthiocholine chloride as substrate incubated for 5 mins by DTNB reagent based Ellman's methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetAcetylcholinesterase(Homo sapiens (Human))TBA
LigandPNGBDBM50409112(CHEMBL109084)
Affinity DataIC50:  3.00E+3nMAssay Description:Inhibition of AChE (unknown origin) using acetylthiocholine chloride as substrate incubated for 5 mins by DTNB reagent based Ellman's methodMore data for this Ligand-Target Pair
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TargetAcetylcholinesterase(Homo sapiens (Human))TBA
LigandPNGBDBM50409082(CHEMBL107541)
Affinity DataIC50:  3.00E+3nMAssay Description:Inhibition of AChE (unknown origin) using acetylthiocholine chloride as substrate incubated for 5 mins by DTNB reagent based Ellman's methodMore data for this Ligand-Target Pair
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TargetAcetylcholinesterase(Homo sapiens (Human))TBA
LigandPNGBDBM50282510(7-(4-Chloro-benzyloxy)-3,4-dimethyl-chromen-2-one ...)
Affinity DataIC50:  3.00E+3nMAssay Description:Inhibition of AChE (unknown origin) using acetylthiocholine chloride as substrate incubated for 5 mins by DTNB reagent based Ellman's methodMore data for this Ligand-Target Pair
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TargetAcetylcholinesterase(Homo sapiens (Human))TBA
LigandPNGBDBM50409078(CHEMBL325761)
Affinity DataIC50:  3.00E+3nMAssay Description:Inhibition of AChE (unknown origin) using acetylthiocholine chloride as substrate incubated for 5 mins by DTNB reagent based Ellman's methodMore data for this Ligand-Target Pair
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TargetAcetylcholinesterase(Homo sapiens (Human))TBA
LigandPNGBDBM50282502(7-(4-Fluoro-benzyloxy)-3,4-dimethyl-chromen-2-one ...)
Affinity DataIC50:  3.00E+3nMAssay Description:Inhibition of AChE (unknown origin) using acetylthiocholine chloride as substrate incubated for 5 mins by DTNB reagent based Ellman's methodMore data for this Ligand-Target Pair
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TargetAcetylcholinesterase(Homo sapiens (Human))TBA
LigandPNGBDBM50282514(3,4-dimethyl-7-(4-methyl-benzyloxy)-chromen-2-one ...)
Affinity DataIC50:  3.00E+3nMAssay Description:Inhibition of AChE (unknown origin) using acetylthiocholine chloride as substrate incubated for 5 mins by DTNB reagent based Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAcetylcholinesterase(Homo sapiens (Human))TBA
LigandPNGBDBM50231957(7-(3-Chloro-benzyloxy)-3,4-dimethyl-chromen-2-one ...)
Affinity DataIC50:  3.00E+3nMAssay Description:Inhibition of AChE (unknown origin) using acetylthiocholine chloride as substrate incubated for 5 mins by DTNB reagent based Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAcetylcholinesterase(Homo sapiens (Human))TBA
LigandPNGBDBM50409097(CHEMBL108697)
Affinity DataIC50:  3.00E+3nMAssay Description:Inhibition of AChE (unknown origin) using acetylthiocholine chloride as substrate incubated for 5 mins by DTNB reagent based Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAcetylcholinesterase(Homo sapiens (Human))TBA
LigandPNGBDBM50409069(CHEMBL320251)
Affinity DataIC50:  3.00E+3nMAssay Description:Inhibition of AChE (unknown origin) using acetylthiocholine chloride as substrate incubated for 5 mins by DTNB reagent based Ellman's methodMore data for this Ligand-Target Pair
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TargetAcetylcholinesterase(Homo sapiens (Human))TBA
LigandPNGBDBM50409093(CHEMBL111310)
Affinity DataIC50:  3.00E+3nMAssay Description:Inhibition of AChE (unknown origin) using acetylthiocholine chloride as substrate incubated for 5 mins by DTNB reagent based Ellman's methodMore data for this Ligand-Target Pair
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TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))TBA
LigandPNGBDBM50217942(2-(3,4-dihydroxyphenyl)-5,7-dihydroxy-4-oxo-4H-chr...)
Affinity DataIC50:  3.89E+3nMAssay Description:Inhibition of MAO-A (unknown origin) incubated for 60 mins by fluorometric spectrophotometry analysisMore data for this Ligand-Target Pair
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TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))TBA
LigandPNGBDBM50611772(CHEMBL5281685)
Affinity DataIC50:  5.00E+3nMAssay Description:Inhibition of human MAO-BMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))TBA
LigandPNGBDBM50029835(3-{5-[4-(3-Chloro-benzyloxy)-phenyl]-tetrazol-2-yl...)
Affinity DataIC50:  8.00E+3nMAssay Description:Inhibition of human MAO-BMore data for this Ligand-Target Pair
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TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))TBA
LigandPNGBDBM50029815(3-[5-(4-Benzyloxy-phenyl)-tetrazol-2-yl]-propionit...)
Affinity DataIC50:  8.00E+3nMAssay Description:Inhibition of human MAO-BMore data for this Ligand-Target Pair
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TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))TBA
LigandPNGBDBM7460(2-(3,4-dihydroxyphenyl)-3,5,7-trihydroxy-4H-chrome...)
Affinity DataIC50:  1.09E+4nMAssay Description:Inhibition of MAO-A (unknown origin) incubated for 60 mins by fluorometric spectrophotometry analysisMore data for this Ligand-Target Pair
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