Compile Data Set for Download or QSAR
maximum 50k data
Found 66 Enz. Inhib. hit(s) with all data for entry = 50036339
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Ciba

Curated by ChEMBL
LigandPNGBDBM50031643(1-(4-Benzyloxy-phenyl)-2-dimethylaminomethyl-prope...)
Affinity DataIC50:  180nMAssay Description:In vitro inhibition of the Epidermal growth factor receptor activity in A431 membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Ciba

Curated by ChEMBL
LigandPNGBDBM50031651(4-[4-(2-Dimethylaminomethyl-acryloyl)-phenoxysulfo...)
Affinity DataIC50:  230nMAssay Description:In vitro inhibition of the Epidermal growth factor receptor activity in A431 membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Ciba

Curated by ChEMBL
LigandPNGBDBM50031655(1-[3-(4-Benzyloxy-phenyl)-3-oxo-propyl]-piperidine...)
Affinity DataIC50:  300nMAssay Description:In vitro inhibition of the Epidermal growth factor receptor activity in A431 membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Ciba

Curated by ChEMBL
LigandPNGBDBM50031657(1-(4-Benzyloxy-3-hydroxy-phenyl)-3-dimethylamino-p...)
Affinity DataIC50:  360nMAssay Description:In vitro inhibition of the Epidermal growth factor receptor activity in A431 membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Ciba

Curated by ChEMBL
LigandPNGBDBM50031659(4-[4-(2-Dimethylaminomethyl-acryloyl)-phenoxysulfo...)
Affinity DataIC50:  470nMAssay Description:In vitro inhibition of the Epidermal growth factor receptor activity in A431 membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Ciba

Curated by ChEMBL
LigandPNGBDBM50031648(1-(4-Benzyloxy-3-hydroxy-phenyl)-2-dimethylaminome...)
Affinity DataIC50:  670nMAssay Description:In vitro inhibition of the Epidermal growth factor receptor activity in A431 membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Ciba

Curated by ChEMBL
LigandPNGBDBM50031642(4-Dimethylcarbamoyl-benzenesulfonic acid 4-(2-dime...)
Affinity DataIC50:  700nMAssay Description:In vitro inhibition of the Epidermal growth factor receptor activity in A431 membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Ciba

Curated by ChEMBL
LigandPNGBDBM19459(5,7-dihydroxy-3-(4-hydroxyphenyl)-4H-chromen-4-one...)
Affinity DataIC50:  1.00E+3nMAssay Description:In vitro inhibition of the Epidermal growth factor receptor activity in A431 membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Ciba

Curated by ChEMBL
LigandPNGBDBM50031662(1-(4-Benzyloxy-phenyl)-2-morpholin-4-ylmethyl-prop...)
Affinity DataIC50:  1.10E+3nMAssay Description:In vitro inhibition of the Epidermal growth factor receptor activity in A431 membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Ciba

Curated by ChEMBL
LigandPNGBDBM50031647(1-(4-Benzyloxy-phenyl)-2-piperidin-1-ylmethyl-prop...)
Affinity DataIC50:  1.10E+3nMAssay Description:In vitro inhibition of the Epidermal growth factor receptor activity in A431 membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Ciba

Curated by ChEMBL
LigandPNGBDBM50031660(1-(4-Benzyloxy-phenyl)-3-dimethylamino-propan-1-on...)
Affinity DataIC50:  1.50E+3nMAssay Description:In vitro inhibition of the Epidermal growth factor receptor activity in A431 membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Ciba

Curated by ChEMBL
LigandPNGBDBM50031661(1-(4-Benzyloxy-phenyl)-3-morpholin-4-yl-propan-1-o...)
Affinity DataIC50:  1.50E+3nMAssay Description:In vitro inhibition of the Epidermal growth factor receptor activity in A431 membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Ciba

Curated by ChEMBL
LigandPNGBDBM50031646(1-(4-Benzyloxy-phenyl)-2-piperazin-1-ylmethyl-prop...)
Affinity DataIC50:  1.50E+3nMAssay Description:In vitro inhibition of the Epidermal growth factor receptor activity in A431 membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Ciba

Curated by ChEMBL
LigandPNGBDBM50031658(1-(4-Benzyloxy-phenyl)-3-piperidin-1-yl-propan-1-o...)
Affinity DataIC50:  1.80E+3nMAssay Description:In vitro inhibition of the Epidermal growth factor receptor activity in A431 membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Ciba

Curated by ChEMBL
LigandPNGBDBM50031644(1-(4-Benzyloxy-phenyl)-3-dimethylamino-2-(3,4-dime...)
Affinity DataIC50:  2.10E+3nMAssay Description:In vitro inhibition of the Epidermal growth factor receptor activity in A431 membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Ciba

Curated by ChEMBL
LigandPNGBDBM50031649(2-{3-(4-benzyloxy)-2-[(dimethylamino)methyl]-3-oxo...)
Affinity DataIC50:  3.90E+3nMAssay Description:In vitro inhibition of the Epidermal growth factor receptor activity in A431 membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Ciba

Curated by ChEMBL
LigandPNGBDBM50369028(CHEMBL468975)
Affinity DataIC50:  5.60E+3nMAssay Description:In vitro inhibition of the Epidermal growth factor receptor activity in A431 membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Ciba

Curated by ChEMBL
LigandPNGBDBM50031656(1-(4-Benzyloxy-phenyl)-3-dimethylamino-2-phenylsul...)
Affinity DataIC50:  7.30E+3nMAssay Description:In vitro inhibition of the Epidermal growth factor receptor activity in A431 membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Ciba

Curated by ChEMBL
LigandPNGBDBM50031650(2-[3-(4-Benzyloxy-phenyl)-2-dimethylaminomethyl-3-...)
Affinity DataIC50:  8.80E+3nMAssay Description:In vitro inhibition of the Epidermal growth factor receptor activity in A431 membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Ciba

Curated by ChEMBL
LigandPNGBDBM50031653(2-(2-Amino-ethylsulfanylmethyl)-1-(4-benzyloxy-phe...)
Affinity DataIC50:  8.80E+3nMAssay Description:In vitro inhibition of the Epidermal growth factor receptor activity in A431 membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Ciba

Curated by ChEMBL
LigandPNGBDBM19459(5,7-dihydroxy-3-(4-hydroxyphenyl)-4H-chromen-4-one...)
Affinity DataIC50:  1.00E+4nMAssay Description:In vitro inhibition of the v-abl tyrosine kinase activity in A431 membranes using angiotensin II as phosphate acceptor as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Ciba

Curated by ChEMBL
LigandPNGBDBM50031657(1-(4-Benzyloxy-3-hydroxy-phenyl)-3-dimethylamino-p...)
Affinity DataIC50: >5.00E+4nMAssay Description:In vitro inhibition of the c-src tyrosine kinase activity in A431 membranes using angiotensin II as phosphate acceptor as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Ciba

Curated by ChEMBL
LigandPNGBDBM50031651(4-[4-(2-Dimethylaminomethyl-acryloyl)-phenoxysulfo...)
Affinity DataIC50:  5.00E+4nMAssay Description:In vitro inhibition of the v-abl tyrosine kinase activity in A431 membranes using angiotensin II as phosphate acceptor as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Ciba

Curated by ChEMBL
LigandPNGBDBM50031648(1-(4-Benzyloxy-3-hydroxy-phenyl)-2-dimethylaminome...)
Affinity DataIC50:  5.00E+4nMAssay Description:In vitro inhibition of the c-src tyrosine kinase activity in A431 membranes using angiotensin II as phosphate acceptor as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Ciba

Curated by ChEMBL
LigandPNGBDBM50031642(4-Dimethylcarbamoyl-benzenesulfonic acid 4-(2-dime...)
Affinity DataIC50: >5.00E+4nMAssay Description:In vitro inhibition of the c-src tyrosine kinase activity in A431 membranes using angiotensin II as phosphate acceptor as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Ciba

Curated by ChEMBL
LigandPNGBDBM50031648(1-(4-Benzyloxy-3-hydroxy-phenyl)-2-dimethylaminome...)
Affinity DataIC50: >5.00E+4nMAssay Description:In vitro inhibition of the v-abl tyrosine kinase activity in A431 membranes using angiotensin II as phosphate acceptor as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Ciba

Curated by ChEMBL
LigandPNGBDBM50031656(1-(4-Benzyloxy-phenyl)-3-dimethylamino-2-phenylsul...)
Affinity DataIC50: >5.00E+4nMAssay Description:In vitro inhibition of the v-abl tyrosine kinase activity in A431 membranes using angiotensin II as phosphate acceptor as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Ciba

Curated by ChEMBL
LigandPNGBDBM50031653(2-(2-Amino-ethylsulfanylmethyl)-1-(4-benzyloxy-phe...)
Affinity DataIC50: >5.00E+4nMAssay Description:In vitro inhibition of the v-abl tyrosine kinase activity in A431 membranes using angiotensin II as phosphate acceptor as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Ciba

Curated by ChEMBL
LigandPNGBDBM50031659(4-[4-(2-Dimethylaminomethyl-acryloyl)-phenoxysulfo...)
Affinity DataIC50: >5.00E+4nMAssay Description:In vitro inhibition of the v-abl tyrosine kinase activity in A431 membranes using angiotensin II as phosphate acceptor as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Ciba

Curated by ChEMBL
LigandPNGBDBM50031656(1-(4-Benzyloxy-phenyl)-3-dimethylamino-2-phenylsul...)
Affinity DataIC50: >5.00E+4nMAssay Description:In vitro inhibition of the c-src tyrosine kinase activity in A431 membranes using angiotensin II as phosphate acceptor as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Ciba

Curated by ChEMBL
LigandPNGBDBM50031659(4-[4-(2-Dimethylaminomethyl-acryloyl)-phenoxysulfo...)
Affinity DataIC50:  5.00E+4nMAssay Description:In vitro inhibition of the c-src tyrosine kinase activity in A431 membranes using angiotensin II as phosphate acceptor as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Ciba

Curated by ChEMBL
LigandPNGBDBM50031642(4-Dimethylcarbamoyl-benzenesulfonic acid 4-(2-dime...)
Affinity DataIC50:  7.00E+4nMAssay Description:In vitro inhibition of the v-abl tyrosine kinase activity in A431 membranes using angiotensin II as phosphate acceptor as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Ciba

Curated by ChEMBL
LigandPNGBDBM50031654(2-Cyano-2-(3,4-dihydroxy-benzyl)-thioacetamide | C...)
Affinity DataIC50:  7.00E+4nMAssay Description:In vitro inhibition of the Epidermal growth factor receptor activity in A431 membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Ciba

Curated by ChEMBL
LigandPNGBDBM19459(5,7-dihydroxy-3-(4-hydroxyphenyl)-4H-chromen-4-one...)
Affinity DataIC50:  7.50E+4nMAssay Description:In vitro inhibition of the c-src tyrosine kinase activity in A431 membranes using angiotensin II as phosphate acceptor as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Ciba

Curated by ChEMBL
LigandPNGBDBM50031649(2-{3-(4-benzyloxy)-2-[(dimethylamino)methyl]-3-oxo...)
Affinity DataIC50: >1.00E+5nMAssay Description:In vitro inhibition of the c-src tyrosine kinase activity in A431 membranes using angiotensin II as phosphate acceptor as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Ciba

Curated by ChEMBL
LigandPNGBDBM50369028(CHEMBL468975)
Affinity DataIC50: >1.00E+5nMAssay Description:In vitro inhibition of the v-abl tyrosine kinase activity in A431 membranes using angiotensin II as phosphate acceptor as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Ciba

Curated by ChEMBL
LigandPNGBDBM50031645(1-(4-Benzyloxy-phenyl)-4-dimethylamino-butan-1-one...)
Affinity DataIC50: >1.00E+5nMAssay Description:In vitro inhibition of the v-abl tyrosine kinase activity in A431 membranes using angiotensin II as phosphate acceptor as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Ciba

Curated by ChEMBL
LigandPNGBDBM50031653(2-(2-Amino-ethylsulfanylmethyl)-1-(4-benzyloxy-phe...)
Affinity DataIC50: >1.00E+5nMAssay Description:In vitro inhibition of the c-src tyrosine kinase activity in A431 membranes using angiotensin II as phosphate acceptor as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Ciba

Curated by ChEMBL
LigandPNGBDBM50031649(2-{3-(4-benzyloxy)-2-[(dimethylamino)methyl]-3-oxo...)
Affinity DataIC50: >1.00E+5nMAssay Description:In vitro inhibition of the v-abl tyrosine kinase activity in A431 membranes using angiotensin II as phosphate acceptor as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Ciba

Curated by ChEMBL
LigandPNGBDBM50031655(1-[3-(4-Benzyloxy-phenyl)-3-oxo-propyl]-piperidine...)
Affinity DataIC50: >1.00E+5nMAssay Description:In vitro inhibition of the v-abl tyrosine kinase activity in A431 membranes using angiotensin II as phosphate acceptor as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Ciba

Curated by ChEMBL
LigandPNGBDBM50031643(1-(4-Benzyloxy-phenyl)-2-dimethylaminomethyl-prope...)
Affinity DataIC50: >1.00E+5nMAssay Description:In vitro inhibition of the c-src tyrosine kinase activity in A431 membranes using angiotensin II as phosphate acceptor as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Ciba

Curated by ChEMBL
LigandPNGBDBM50031654(2-Cyano-2-(3,4-dihydroxy-benzyl)-thioacetamide | C...)
Affinity DataIC50: >1.00E+5nMAssay Description:In vitro inhibition of the v-abl tyrosine kinase activity in A431 membranes using angiotensin II as phosphate acceptor as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Ciba

Curated by ChEMBL
LigandPNGBDBM50031646(1-(4-Benzyloxy-phenyl)-2-piperazin-1-ylmethyl-prop...)
Affinity DataIC50: >1.00E+5nMAssay Description:In vitro inhibition of the c-src tyrosine kinase activity in A431 membranes using angiotensin II as phosphate acceptor as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Ciba

Curated by ChEMBL
LigandPNGBDBM50031644(1-(4-Benzyloxy-phenyl)-3-dimethylamino-2-(3,4-dime...)
Affinity DataIC50: >1.00E+5nMAssay Description:In vitro inhibition of the c-src tyrosine kinase activity in A431 membranes using angiotensin II as phosphate acceptor as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Ciba

Curated by ChEMBL
LigandPNGBDBM50031647(1-(4-Benzyloxy-phenyl)-2-piperidin-1-ylmethyl-prop...)
Affinity DataIC50: >1.00E+5nMAssay Description:In vitro inhibition of the v-abl tyrosine kinase activity in A431 membranes using angiotensin II as phosphate acceptor as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Ciba

Curated by ChEMBL
LigandPNGBDBM50031644(1-(4-Benzyloxy-phenyl)-3-dimethylamino-2-(3,4-dime...)
Affinity DataIC50: >1.00E+5nMAssay Description:In vitro inhibition of the v-abl tyrosine kinase activity in A431 membranes using angiotensin II as phosphate acceptor as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Ciba

Curated by ChEMBL
LigandPNGBDBM50031660(1-(4-Benzyloxy-phenyl)-3-dimethylamino-propan-1-on...)
Affinity DataIC50: >1.00E+5nMAssay Description:In vitro inhibition of the c-src tyrosine kinase activity in A431 membranes using angiotensin II as phosphate acceptor as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Ciba

Curated by ChEMBL
LigandPNGBDBM50031652(4-[4-(3-Dimethylamino-2-methyl-propionyl)-phenoxys...)
Affinity DataIC50:  1.00E+5nMAssay Description:In vitro inhibition of the Epidermal growth factor receptor activity in A431 membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Ciba

Curated by ChEMBL
LigandPNGBDBM50031651(4-[4-(2-Dimethylaminomethyl-acryloyl)-phenoxysulfo...)
Affinity DataIC50: >1.00E+5nMAssay Description:In vitro inhibition of the c-src tyrosine kinase activity in A431 membranes using angiotensin II as phosphate acceptor as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Ciba

Curated by ChEMBL
LigandPNGBDBM50031650(2-[3-(4-Benzyloxy-phenyl)-2-dimethylaminomethyl-3-...)
Affinity DataIC50: >1.00E+5nMAssay Description:In vitro inhibition of the v-abl tyrosine kinase activity in A431 membranes using angiotensin II as phosphate acceptor as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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