5953 SMILES Strings for High affinity nerve growth factor receptor

Compound Name
SMILES String
Cc1cc(CNc2ncc(Br)c(Nc3cc(n[nH]3)C3CC3)n2)on1
Brc1cnc(NCc2ccccc2)nc1Nc1cc(n[nH]1)C1CC1
COc1cccc(CNc2ncc(Br)c(Nc3cc(n[nH]3)C3CC3)n2)c1
Clc1ccccc1CNc1ncc(Br)c(Nc2cc(n[nH]2)C2CC2)n1
COc1ccccc1CNc1ncc(Br)c(Nc2cc(n[nH]2)C2CC2)n1
Fc1ccc(CNc2ncc(Br)c(Nc3cc(n[nH]3)C3CC3)n2)cc1
Clc1ccc(CNc2ncc(Br)c(Nc3cc(n[nH]3)C3CC3)n2)cc1
C[C@H](Nc1ncc(Br)c(Nc2cc(n[nH]2)C2CC2)n1)c1ccccc1 |r|
C[C@@H](Nc1ncc(Br)c(Nc2cc(n[nH]2)C2CC2)n1)c1ccccc1 |r|
OC[C@@H](Nc1ncc(Br)c(Nc2cc(n[nH]2)C2CC2)n1)c1ccccc1 |r|
OC[C@H](Nc1ncc(Br)c(Nc2cc(n[nH]2)C2CC2)n1)c1ccccc1 |r|
C[C@H](Nc1ncc(Br)c(Nc2cc(n[nH]2)C2CC2)n1)c1ccc(F)cc1 |r|
OC[C@H](Nc1ncc(Cl)c(Nc2cc(n[nH]2)C2CC2)n1)c1ccc(F)cc1 |r|
CN(C)C(=O)C[C@H](Nc1ncc(Cl)c(Nc2cc(n[nH]2)C2CC2)n1)c1ccc(F)cc1 |r|
CNC(=O)C[C@H](Nc1ncc(Cl)c(Nc2cc(n[nH]2)C2CC2)n1)c1ccc(F)cc1 |r|
CNC(=O)Nc1snc(SCc2ccc(Cl)cc2)c1C(N)=O
CNC(=O)Nc1snc(SC(C)c2ccc(Cl)cc2)c1C(N)=O
CCC(Sc1nsc(NC(=O)NC)c1C(N)=O)c1ccc(Cl)cc1
CC[C@@H](Sc1nsc(NC(=O)NC)c1C(N)=O)c1ccc(Cl)cc1 |r|
CC[C@H](Sc1nsc(NC(=O)NC)c1C(N)=O)c1ccc(Cl)cc1 |r|
CNC(=O)Nc1snc(SC(C(C)C)c2ccc(Cl)cc2)c1C(N)=O
CCCC(Sc1nsc(NC(=O)NC)c1C(N)=O)c1ccc(Cl)cc1
CNC(=O)Nc1snc(SC(c2ccc(Cl)cc2)C(F)(F)F)c1C(N)=O
CNC(=O)Nc1snc(SC(c2ccccc2)c2ccc(Cl)cc2)c1C(N)=O
CNC(=O)Nc1snc(SCc2ccc(Cl)cc2)c1C#N
NC(=O)c1c(N)snc1SCc1ccc(Cl)cc1
NC(=O)c1c(SCc2ccc(Cl)cc2)nsc1Nc1ccccn1
NC(=O)c1c(SCc2ccc(Cl)cc2)nsc1Nc1cccnc1
CC(Sc1nsc(Nc2cccnc2)c1C(N)=O)c1ccc(Cl)cc1
NC(=O)c1c(SCC2CCCCC2)nsc1Nc1cccnc1
NC(=O)c1c(SCc2ccc(Cl)cc2)nsc1Nc1ccncc1
NC(=O)c1c(SCc2ccccc2Cl)nsc1Nc1ccncc1
NC(=O)c1c(SCc2ccc(Cl)cc2)nsc1Nc1ccncn1
COc1ccc(Nc2snc(SCc3ccc(Cl)cc3)c2C(N)=O)cn1
NC(=O)c1c(SCc2ccc(Cl)cc2)nsc1Nc1ccc(=O)[nH]c1
NC(=O)Nc1snc(SC2CCc3cc(Cl)ccc23)c1C(N)=O
CNC(=O)Nc1snc(SC2CCc3cc(Cl)ccc23)c1C(N)=O
NC(=O)Nc1snc(SC2CCCc3ccccc23)c1C(N)=O
CNC(=O)Nc1snc(SC2CCCc3ccccc23)c1C(N)=O
NC(=O)Nc1snc(SC2CCCCc3ccccc23)c1C(N)=O
NC(=O)Nc1snc(S[C@@H]2CCCCc3ccccc23)c1C(N)=O |r|
NC(=O)Nc1snc(S[C@H]2CCCCc3ccccc23)c1C(N)=O |r|
COc1ccc-2c(CCc3c-2c2C(=O)NCc2c2c4ccccc4n(CCO)c32)c1
CC(C)Oc1ccc-2c(CCc3c-2c2C(=O)NCc2c2c4ccccc4n(CCO)c32)c1
CNC(=O)c1nn(C)c-2c1C(C)(C)Cc1cnc(Nc3ccc(cc3)N3CCN(C)CC3)nc-21
Cc1ccc(F)c(NC(=O)Nc2ccc(cc2)-c2cccc3[nH]nc(N)c23)c1
CCN1CCN(Cc2ccc(NC(=O)Nc3ccc(Oc4cc(NC)ncn4)cc3)cc2C(F)(F)F)CC1
Cc1ccc(cc1)-n1nc(cc1NC(=O)Nc1ccc(OCCN2CCOCC2)c2ccccc12)C(C)(C)C
CN1CCN(CC1)c1ccc2nc([nH]c2c1)-c1c(N)c2c(F)cccc2[nH]c1=O
COc1ccc(cc1)COc2ccc(cc2OC)Cc3cnc(nc3N)N
COc1cc2c(ncnc2cc1OCCCN1CCCCC1)N1CCN(CC1)C(=O)Nc1ccc(OC(C)C)cc1
[H][C@@]12C[C@@H]([C@H](OC)[C@@](C)(O1)n1c3ccccc3c3c4CNC(=O)c4c4c5ccccc5n2c4c13)N(C)C(=O)c1ccccc1 |TLB:11:10:9:4.3.2,17:33:9:4.3.2,THB:24:32:9:4.3.2,5:4:9:10.31.33.32,30:31:9:4.3.2|
Cc1[nH]c(\C=C2/C(=O)Nc3ccc(F)cc23)c(C)c1C(=O)NC[C@H](O)CN1CCOCC1
CNC(=O)c1cc(ccn1)Oc2ccc(cc2)NC(=O)Nc3ccc(c(c3)C(F)(F)F)Cl
CN[C@H]1C[C@@H]2O[C@](C)([C@H]1OC)n1c3ccccc3c3c4CNC(=O)c4c4c5ccccc5n2c4c13
CCN(CC)CCNC(=O)c1c(C)[nH]c(\C=C2/C(=O)Nc3ccc(F)cc23)c1C
CN1CCN(CC1)c1cc(Nc2cc(C)n[nH]2)nc(Sc2ccc(NC(=O)C3CC3)cc2)n1
CC(C)n1cc(C(=O)c2cncc(NC(=O)Cc3ccc(cn3)C#N)c2)c2cnc(N)nc12
CC(CO)(CO)n1cc(C(=O)c2cncc(NC(=O)c3cccc(OC(F)(F)F)c3)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)[C@H](N)Cc3ccc(cc3)C(=O)c3ccccc3)c2)c2cncnc12 |r|
COCc1ccc(CC(=O)Nc2cncc(c2)C(=O)c2cn(C)c3ncncc23)cc1
Cn1cc(C(=O)c2cncc(NC(=O)Cn3cnc(Cl)c3Cl)c2)c2cncnc12
Cn1cc(C(=O)c2cncc(c2)N(N)C(=O)Cc2n[nH]c3CCCc23)c2cncnc12
Cn1cc(cn1)-n1nc(cc1NC(=O)Nc1cncc(c1)C(=O)c1cn(C)c2ncncc12)C(C)(C)C
CS(=O)(=O)c1cccc(CC(=O)Nc2cncc(c2)C(=O)c2cn(c3nc(N)ncc23)C23CC(C2)C3)c1
Nc1ncc2c(cn(c2n1)C12CC(C1)C2)C(=O)c1cncc(NC(=O)Cn2ccc(n2)C(F)(F)F)c1
Nc1ncc2c(cn(c2n1)C12CC(C1)C2)C(=O)c1cncc(NC(=O)Cn2cc(nn2)C(F)(F)F)c1
Nc1ncc2c(cn(c2n1)C12CC(C1)C2)C(=O)c1cncc(NC(=O)Cc2ccc(cc2)C#N)c1
Nc1ncc2c(cn(c2n1)C12CC(C1)C2)C(=O)c1cncc(NC(=O)Cc2ccc(Cl)cn2)c1
CC(C)n1cc(C(=O)c2cncc(NC(=O)c3cn4ncc(Cl)cc4n3)c2)c2cncnc12
CCOc1ccc(CC(=O)Nc2cncc(c2)C(=O)c2cn(c3nc(N)ncc23)C(C)(C)CO)nc1
CC(=O)Nc1cc(Oc2ccc(NC(=O)N3CCN(C3=O)c3ccccc3)cc2)ccn1
Nc1cc(Oc2ccc(NC(=O)N3CCN(C3=O)c3ccccc3)cc2)ccn1
CC(=O)Nc1cc(Oc2ccc(NC(=O)N3CCN(C3=O)c3ccc(F)cc3)cc2)ccn1
CNC(=O)Nc1cc(Oc2ccc(NC(=O)N3CCN(C3=O)c3ccccc3)cc2)ccn1
CNC(=O)Nc1cc(Oc2ccc(NC(=O)N3CCN(C3=O)c3ccc(F)cc3)cc2)ccn1
Fc1ccc(cc1)N1CCN(C(=O)Nc2ccc(Oc3ccnc(NC(=O)NCCN4CCCC4)c3)cc2)C1=O
CC(C)Oc1cc(n[nH]1)-n1cnc2ccc(N[C@@H](C)c3ccc(F)cn3)nc12 |r|
C[C@H](Nc1ccc2ncn(-c3cc([nH]n3)C3CC3)c2n1)c1ccc(F)cn1 |r|
C[C@H](Nc1ccc2ncn(-c3cc([nH]n3)C3CC3)c2n1)c1ncc(F)cn1 |r|
C[C@H](Nc1ncc2ncn(-c3cc([nH]n3)C3CC3)c2n1)c1ncc(F)cn1 |r|
C[C@H](Nc1ncc2ncn(-c3cc([nH]n3)C3CC3)c2n1)c1ccc(F)cn1 |r|
CC(C)Oc1cc(n[nH]1)-n1cnc2ccc(N[C@@H](C)c3ncc(F)cn3)nc12 |r|
CC(C)Oc1cc(n[nH]1)-n1cnc2ccc(N[C@@H](CO)c3ccc(F)cn3)nc12 |r|
CCOc1cc(n[nH]1)-n1cnc2ccc(N[C@@H](CO)c3ccc(F)cn3)nc12 |r|
CCOc1cc(n[nH]1)-n1cnc2ccc(N[C@@H](C)c3ncc(F)cn3)nc12 |r|
CCOc1cc(n[nH]1)-n1cnc2ccc(N[C@@H](C)c3ccc(F)cn3)nc12 |r|
CC(C)Oc1cc(n[nH]1)-n1cnc2cnc(N[C@@H](C)c3ncc(F)cn3)nc12 |r|
CC[C@H](Nc1ccc2ncn(-c3cc(OC(C)C)[nH]n3)c2n1)c1ccc(F)cn1 |r|
CC(C)Oc1cc(n[nH]1)-n1cnc2cc(Cl)c(N[C@@H](C)c3ccc(F)cn3)nc12 |r|
C[C@H](Nc1nc2n(cnc2cc1F)-c1cc(C)[nH]n1)c1ncc(F)cn1 |r|
C[C@H](Nc1ccc2ncn(-c3cc(C)[nH]n3)c2n1)c1ncc(F)cn1 |r|
C[C@H](Nc1ccc2ncn(-c3cc(C)[nH]n3)c2n1)c1ccc(F)cn1 |r|
C[C@H](Nc1ncc2ncn(-c3cc(C)[nH]n3)c2n1)c1ccc(F)cn1 |r|
C[C@H](Nc1nc(C(=O)N2CCOCC2)c2ncn(-c3cc(C)[nH]n3)c2n1)c1ncc(F)cn1 |r|
C[C@H](Nc1nc(NC2CCOCC2)c2ncn(-c3cc(C)[nH]n3)c2n1)c1ccc(F)cn1 |r|
COc1nc(N[C@@H](C)c2ccc(F)cn2)nc2n(cnc12)-c1cc(C)[nH]n1 |r|
C[C@H](Nc1nc(N2CCOCC2)c2ncn(-c3cc(C)[nH]n3)c2n1)c1ccc(F)cn1 |r|
CCOc1cc(n[nH]1)-n1cnc2ccc(N[C@@H](CC)c3ccc(F)cn3)nc12 |r|
CC(C)(C)NC(=O)c1cnn2ccc(nc12)N1CCC[C@@H]1c1cc(F)ccc1F |r|
Fc1ccc(F)c(c1)[C@H]1CCCN1c1ccn2ncc(C(=O)Nc3ccccn3)c2n1 |r|
Cc1cccnc1NC(=O)c1cnn2ccc(nc12)N1CCC[C@@H]1c1cc(F)ccc1F |r|
Fc1ccc(F)c(c1)[C@H]1CCCN1c1ccn2ncc(C(=O)NCCN3CCOCC3)c2n1 |r|
Cc1ccc(CNC(=O)c2cnn3ccc(nc23)N2CCC[C@@H]2c2cc(F)ccc2F)o1 |r|
Cn1ccc(NC(=O)c2cnn3ccc(nc23)N2CCC[C@@H]2c2cc(F)ccc2F)n1 |r|
O[C@H]1CC[C@@H](CC1)NC(=O)c1cnn2ccc(nc12)N1CCC[C@@H]1c1cc(F)ccc1F |r,wU:4.7,wD:23.27,1.0,(6.35,-6.59,;5.95,-5.1,;7.04,-4.01,;6.64,-2.52,;5.15,-2.12,;4.06,-3.21,;4.46,-4.7,;4.75,-.64,;3.27,-.24,;2.18,-1.33,;2.87,1.25,;3.77,2.5,;2.87,3.74,;1.4,3.27,;.07,4.04,;-1.26,3.27,;-1.26,1.73,;.07,.96,;1.4,1.73,;-2.6,.96,;-2.6,-.58,;-4.06,-1.06,;-4.97,.19,;-4.06,1.43,;-4.46,2.92,;-3.37,4.01,;-3.77,5.5,;-2.68,6.59,;-5.26,5.9,;-6.35,4.81,;-5.95,3.32,;-7.04,2.23,)|
CC(C)(CO)NC(=O)c1cnn2ccc(nc12)N1CCC[C@@H]1c1cc(F)ccc1F |r|
CC(C)(CN1CCOCC1)NC(=O)c1cnn2ccc(nc12)N1CCC[C@@H]1c1cc(F)ccc1F |r|
CNC(=O)c1cnn2ccc(nc12)N1CCC[C@@H]1c1cc(F)ccc1F |r|
OC(=O)C1CCN(CC1)C(=O)c1cnn2ccc(nc12)N1CCCC1c1cc(F)ccc1F
OC(=O)CC1CCN(CC1)C(=O)c1cnn2ccc(nc12)N1CCCC1c1cc(F)ccc1F
Fc1ccc(F)c(c1)[C@H]1CCCN1c1ccn2ncc(C(=O)NC3CC3)c2n1 |r|
Fc1ccc(F)c(c1)[C@H]1CCCN1c1ccn2ncc(C(=O)NC3CCC3)c2n1 |r|
Fc1ccc(F)c(c1)[C@H]1CCCN1c1ccn2ncc(C(=O)N[C@H]3CC4CCC3C4)c2n1 |r,THB:22:23:26.27:29|
OCC1(CC1)NC(=O)c1cnn2ccc(nc12)N1CCC[C@@H]1c1cc(F)ccc1F |r|
CC(C)(O)CNC(=O)c1cnn2ccc(nc12)N1CCC[C@@H]1c1cc(F)ccc1F |r|
O[C@H]1CCN(C1)C(=O)c1cnn2ccc(nc12)N1CCC[C@@H]1c1cc(F)ccc1F |r|
O[C@@H]1CCN(C1)C(=O)c1cnn2ccc(nc12)N1CCC[C@@H]1c1cc(F)ccc1F |r|
Fc1ccc(F)c(c1)[C@H]1CCCN1c1ccn2ncc(C(=O)NC3CCOCC3)c2n1 |r|
Cn1cnc(CNC(=O)c2cnn3ccc(nc23)N2CCC[C@@H]2c2cc(F)ccc2F)c1 |r|
Cn1cc(CNC(=O)c2cnn3ccc(nc23)N2CCC[C@@H]2c2cc(F)ccc2F)cn1 |r|
Cn1cncc1CCNC(=O)c1cnn2ccc(nc12)N1CCC[C@@H]1c1cc(F)ccc1F |r|
Fc1ccc(F)c(c1)[C@H]1CCCN1c1ccn2ncc(C(=O)NCCN3CCNC3=O)c2n1 |r|
Fc1ccc(F)c(c1)[C@H]1CCCN1c1ccn2ncc(C(=O)NCCc3cnc[nH]3)c2n1 |r|
OC[C@H](O)CNC(=O)c1cnn2ccc(nc12)N1CCC[C@@H]1c1cc(F)ccc1F |r|
CN(C)C(=O)c1cnn2ccc(nc12)N1CCC[C@@H]1c1cc(F)ccc1F |r|
Fc1ccc(F)c(c1)[C@H]1CCCN1c1ccn2ncc(C(=O)NCCn3ccnc3)c2n1 |r|
OC[C@@H](O)CNC(=O)c1cnn2ccc(nc12)N1CCC[C@@H]1c1cc(F)ccc1F |r|
NC(=O)c1cnn2ccc(nc12)N1CCC[C@@H]1c1cc(F)ccc1F |r|
OC1CN(C1)C(=O)c1cnn2ccc(nc12)N1CCC[C@@H]1c1cc(F)ccc1F |r|
CC1(O)CN(C1)C(=O)c1cnn2ccc(nc12)N1CCC[C@@H]1c1cc(F)ccc1F |r|
OC(=O)C1CCC(CC1)NC(=O)c1cnn2ccc(nc12)N1CCCC1c1cc(F)ccc1F |(4.86,-7.13,;5.95,-6.04,;7.44,-6.44,;5.55,-4.55,;4.06,-4.15,;3.66,-2.67,;4.75,-1.58,;6.24,-1.98,;6.64,-3.46,;4.35,-.09,;2.87,.31,;1.78,-.78,;2.47,1.8,;3.37,3.04,;2.47,4.29,;1,3.81,;-.33,4.58,;-1.66,3.81,;-1.66,2.27,;-.33,1.5,;1,2.27,;-3,1.5,;-3,-.04,;-4.46,-.51,;-5.37,.73,;-4.46,1.98,;-4.86,3.46,;-3.77,4.55,;-4.17,6.04,;-3.08,7.13,;-5.66,6.44,;-6.75,5.35,;-6.35,3.86,;-7.44,2.77,)|
OCc1ccc(F)cc1C1CCCN1c1ccn2ncc(C(=O)NC3CCC(O)CC3)c2n1 |(-6.64,.74,;-7.04,2.23,;-5.95,3.32,;-6.35,4.81,;-5.26,5.9,;-3.77,5.5,;-2.68,6.59,;-3.37,4.01,;-4.46,2.92,;-4.06,1.43,;-4.97,.19,;-4.06,-1.06,;-2.6,-.58,;-2.6,.96,;-1.26,1.73,;-1.26,3.27,;.07,4.04,;1.4,3.27,;2.87,3.74,;3.77,2.5,;2.87,1.25,;3.27,-.24,;2.18,-1.33,;4.75,-.64,;5.15,-2.12,;4.06,-3.21,;4.46,-4.7,;5.95,-5.1,;6.35,-6.59,;7.04,-4.01,;6.64,-2.52,;1.4,1.73,;.07,.96,)|
O[C@H]1CC[C@@H](CC1)NC(=O)c1cnn2ccc(nc12)N1CCC[C@@H]1c1cccc(F)c1 |r,wU:4.7,wD:23.27,1.0,(6,-6.59,;5.6,-5.1,;6.69,-4.01,;6.29,-2.52,;4.81,-2.12,;3.72,-3.21,;4.12,-4.7,;4.41,-.64,;2.92,-.24,;1.83,-1.33,;2.52,1.25,;3.43,2.5,;2.52,3.74,;1.06,3.27,;-.28,4.04,;-1.61,3.27,;-1.61,1.73,;-.28,.96,;1.06,1.73,;-2.94,.96,;-2.94,-.58,;-4.41,-1.06,;-5.31,.19,;-4.41,1.43,;-4.81,2.92,;-6.29,3.32,;-6.69,4.81,;-5.6,5.9,;-4.12,5.5,;-3.03,6.59,;-3.72,4.01,)|
CC(C)(C)NC(=O)c1cnn2ccc(nc12)N1CCC[C@@H]1c1cccc(F)c1 |r|
Fc1cccc(c1)[C@H]1CCCN1c1ccn2ncc(C(=O)NC3CC3)c2n1 |r|
CC(C)(NC(=O)c1cnn2ccc(nc12)N1CCCC1c1cc(F)ccc1F)C#N
Fc1ccc(F)c(c1)C1CCCN1c1ccn2ncc(C(=O)NCC#N)c2n1
CC(C)(CF)NC(=O)c1cnn2ccc(nc12)N1CCC[C@@H]1c1cc(F)ccc1F |r|
O[C@@H]1C[C@@H](N(C1)c1ccn2ncc(C(=O)NC3CC3)c2n1)c1cccc(F)c1 |r|
CC(C)(C)NC(=O)c1cnn2ccc(nc12)N1C[C@H](O)C[C@@H]1c1cccc(F)c1 |r|
CNC(=O)c1cnn2ccc(nc12)N1C[C@H](O)C[C@@H]1c1cccc(F)c1 |r|
CS(=O)(=O)N1CCC(CC1)NC(=O)c1cnn2ccc(nc12)N1CCCC1c1cc(F)ccc1F
NS(=O)(=O)N1CCC(CC1)NC(=O)c1cnn2ccc(nc12)N1CCCC1c1cc(F)ccc1F
CS(=O)(=O)NCCNC(=O)c1cnn2ccc(nc12)N1CCCC1c1cc(F)ccc1F
NS(=O)(=O)CCNC(=O)c1cnn2ccc(nc12)N1CCCC1c1cc(F)ccc1F
OCc1ccc(F)cc1C1CCCN1c1ccn2ncc(C(=O)NC3CC3)c2n1
CC(C)(O)CNC(=O)c1cnn2ccc(nc12)N1CCCC1c1cc(F)ccc1CO
C[C@@]1(O)CCC(CC1)NC(=O)c1cnn2ccc(nc12)N1CCC[C@@H]1c1cc(F)ccc1F |r,w:8.8,wU:1.0,wD:24.28,1.1,(7.04,-6.19,;5.95,-5.1,;5.55,-6.59,;4.46,-4.7,;4.06,-3.21,;5.15,-2.12,;6.64,-2.52,;7.04,-4.01,;4.75,-.64,;3.27,-.24,;2.18,-1.33,;2.87,1.25,;3.77,2.5,;2.87,3.74,;1.4,3.27,;.07,4.04,;-1.26,3.27,;-1.26,1.73,;.07,.96,;1.4,1.73,;-2.6,.96,;-2.6,-.58,;-4.06,-1.06,;-4.97,.19,;-4.06,1.43,;-4.46,2.92,;-3.37,4.01,;-3.77,5.5,;-2.68,6.59,;-5.26,5.9,;-6.35,4.81,;-5.95,3.32,;-7.04,2.23,)|
C[C@@]1(O)CCC(CC1)NC(=O)c1cnn2ccc(nc12)N1CCC[C@@H]1c1cc(F)ccc1F |r,w:8.8,wU:1.1,wD:24.28,1.0,(5.55,-6.59,;5.95,-5.1,;7.04,-6.19,;7.04,-4.01,;6.64,-2.52,;5.15,-2.12,;4.06,-3.21,;4.46,-4.7,;4.75,-.64,;3.27,-.24,;2.18,-1.33,;2.87,1.25,;3.77,2.5,;2.87,3.74,;1.4,3.27,;.07,4.04,;-1.26,3.27,;-1.26,1.73,;.07,.96,;1.4,1.73,;-2.6,.96,;-2.6,-.58,;-4.06,-1.06,;-4.97,.19,;-4.06,1.43,;-4.46,2.92,;-3.37,4.01,;-3.77,5.5,;-2.68,6.59,;-5.26,5.9,;-6.35,4.81,;-5.95,3.32,;-7.04,2.23,)|
Fc1cncc(c1)[C@H]1CCCN1c1ccn2ncc(C(=O)NC3CC3)c2n1 |r|
CC(C)(C)NC(=O)c1cnn2ccc(nc12)N1CCC[C@@H]1c1cncc(F)c1 |r|
OCc1ccc(F)cc1C1CCCN1c1ccn2ncc(C(=O)NCCN3CCOCC3)c2n1
OCC(O)CNC(=O)c1cnn2ccc(nc12)N1CCCC1c1cc(F)ccc1CO
CC(C)(CNS(C)(=O)=O)NC(=O)c1cnn2ccc(nc12)N1CCCC1c1cc(F)ccc1F
CC(C)(N)CNC(=O)c1cnn2ccc(nc12)N1CCC[C@@H]1c1cc(F)ccc1F |r|
CC(C)(C)NC(=O)c1cnn2ccc(nc12)N1CC(F)(F)C[C@@H]1c1cccc(F)c1 |r|
CC(CO)(CO)NC(=O)c1cnn2ccc(nc12)N1CCC[C@@H]1c1cc(F)ccc1F |r|
F[C@H]1CNCC[C@H]1NC(=O)c1cnn2ccc(nc12)N1CCC[C@@H]1c1cc(F)ccc1F |r|
OC[C@@H](O)CNC(=O)c1cnn2ccc(nc12)N1CCC[C@@H]1c1cc(F)ccc1C(F)(F)F |r|
OC[C@H](O)CNC(=O)c1cnn2ccc(nc12)N1CCC[C@@H]1c1cc(F)ccc1C(F)(F)F |r|
NC(=O)c1cnn2ccc(nc12)N1CCC[C@@H]1c1cc(F)ccc1C(F)(F)F |r|
CONC(=O)c1cnn2ccc(nc12)N1CCC[C@@H]1c1cc(F)ccc1F |r|
Fc1ccc(F)c(c1)[C@H]1CCCN1c1ccn2ncc(C(=O)NOCC3CC3)c2n1 |r|
CC1(C)CC[C@@H](N1c1ccn2ncc(C(N)=O)c2n1)c1cc(F)ccc1F |r|
CC1(C)CC[C@@H](N1c1ccn2ncc(C(=O)NC3CC3)c2n1)c1cc(F)ccc1F |r|
CC(C)(NC(=O)c1cnn2ccc(nc12)N1CCCC1c1cncc(F)c1)C#N
CS(=O)(=O)N1CCC(CC1)NC(=O)c1cnn2ccc(nc12)N1CCCC1c1cncc(F)c1
CC(C)(CF)NC(=O)c1cnn2ccc(nc12)N1CCC[C@@H]1c1cncc(F)c1 |r|
Fc1cncc(c1)[C@H]1CCCN1c1ccn2ncc(C(=O)NC3CCOCC3)c2n1 |r|
CONC(=O)c1cnn2ccc(nc12)N1CCC[C@@H]1c1cncc(F)c1 |r|
NC(=O)c1cnn2ccc(nc12)N1CCC[C@@H]1c1cccc(F)c1 |r|
CONC(=O)c1cnn2ccc(nc12)N1CCC[C@@H]1c1cccc(F)c1 |r|
NC(=O)c1cnn2ccc(nc12)N1CCC[C@@H]1c1cc(F)cc(OCCN2CCOCC2)c1 |r|
COCCOc1cc(F)cc(c1)[C@H]1CCCN1c1ccn2ncc(C(=O)NC3CC3)c2n1 |r|
COCCOc1cc(F)cc(c1)[C@H]1CCCN1c1ccn2ncc(C(N)=O)c2n1 |r|
OCc1ncc(F)cc1C1CCCN1c1ccn2ncc(C(=O)NC3CC3)c2n1
CC(C)(C)NC(=O)c1cnn2ccc(nc12)N1CCCC1c1cc(F)cnc1CO
CC(C)(CF)NC(=O)c1cnn2ccc(nc12)N1CCCC1c1cc(F)cnc1CO
NC(=O)c1cnn2ccc(nc12)N1CCCC1c1cc(F)cnc1CO
CONC(=O)c1cnn2ccc(nc12)N1CCCC1c1cc(F)cnc1CO
OC(=O)C1(CC1)NC(=O)c1cnn2ccc(nc12)N1CCCC1c1cc(F)ccc1F
Fc1cc(OCCN2CCOCC2)cc(c1)[C@H]1CCCN1c1ccn2ncc(C(=O)NC3CC3)c2n1 |r|
NC(=O)c1cnn2ccc(nc12)N1CCC[C@@H]1c1cc(F)ccc1OCCN1CCOCC1 |r|
Fc1ccc(OCCN2CCOCC2)c(c1)[C@H]1CCCN1c1ccn2ncc(C(=O)NC3CC3)c2n1 |r|
OC[C@H](O)CONC(=O)c1cnn2ccc(nc12)N1CCC[C@@H]1c1cc(F)ccc1F |r|
COCCOc1ccc(F)cc1[C@H]1CCCN1c1ccn2ncc(C(N)=O)c2n1 |r|
COCCOc1ccc(F)cc1[C@H]1CCCN1c1ccn2ncc(C(=O)NC3CC3)c2n1 |r|
CC1(CC1)NC(=O)c1cnn2ccc(nc12)N1CCC[C@@H]1c1cncc(F)c1 |r|
CC1(O)CN(C1)C(=O)c1cnn2ccc(nc12)N1CCC[C@@H]1c1cncc(F)c1 |r|
CC(C)NC(=O)c1cnn2ccc(nc12)N1CCC[C@@H]1c1cncc(F)c1 |r|
Fc1cncc(c1)[C@H]1CCCN1c1ccn2ncc(C(=O)N3CCCC3)c2n1 |r|
Fc1ccc(NC(=O)c2cnn3ccc(nc23)N2CCC[C@@H]2c2cncc(F)c2)nc1 |r|
COC1CN(C1)C(=O)c1cnn2ccc(nc12)N1CCC[C@@H]1c1cncc(F)c1 |r|
FC(CCl)CNC(=O)c1cnn2ccc(nc12)N1CCC[C@@H]1c1cncc(F)c1 |r|
Fc1cncc(c1)[C@H]1CCCN1c1ccn2ncc(C(=O)NC3(CC3)C(F)(F)F)c2n1 |r|
O[C@H]1CCC(CC1)NC(=O)c1cnn2ccc(nc12)N1CCC[C@@H]1c1cncc(F)c1 |r,wD:23.27,1.0,(7.01,-5.81,;6.24,-4.48,;7.01,-3.14,;6.24,-1.81,;4.7,-1.81,;3.93,-3.14,;4.7,-4.48,;3.93,-.47,;5.02,.61,;6.5,.22,;4.62,2.1,;5.52,3.35,;4.62,4.59,;3.15,4.12,;1.82,4.89,;.49,4.12,;.49,2.58,;1.82,1.81,;3.15,2.58,;-.85,1.81,;-.37,.34,;-1.62,-.56,;-2.86,.34,;-2.39,1.81,;-3.16,3.14,;-2.39,4.48,;-3.16,5.81,;-4.7,5.81,;-5.47,4.48,;-7.01,4.48,;-4.7,3.14,)|
O[C@H]1CCC(CC1)NC(=O)c1cnn2ccc(nc12)N1CCC[C@@H]1c1cncc(F)c1 |r,wU:1.0,wD:23.27,(7.01,-5.81,;6.24,-4.48,;4.7,-4.48,;3.93,-3.14,;4.7,-1.81,;6.24,-1.81,;7.01,-3.14,;3.93,-.47,;5.02,.61,;6.5,.22,;4.62,2.1,;5.52,3.35,;4.62,4.59,;3.15,4.12,;1.82,4.89,;.49,4.12,;.49,2.58,;1.82,1.81,;3.15,2.58,;-.85,1.81,;-.37,.34,;-1.62,-.56,;-2.86,.34,;-2.39,1.81,;-3.16,3.14,;-2.39,4.48,;-3.16,5.81,;-4.7,5.81,;-5.47,4.48,;-7.01,4.48,;-4.7,3.14,)|
Fc1cncc(c1)[C@H]1CCCN1c1ccn2ncc(C(=O)NC3CCC3)c2n1 |r|
CC1(CCC1)NC(=O)c1cnn2ccc(nc12)N1CCCC1c1cncc(F)c1
O[C@H]1CCC[C@@H]1NC(=O)c1cnn2ccc(nc12)N1CCCC1c1cncc(F)c1 |r|
O[C@@H]1CCC[C@@H]1NC(=O)c1cnn2ccc(nc12)N1CCCC1c1cncc(F)c1 |r|
O[C@H]1CC[C@@H](C1)NC(=O)c1cnn2ccc(nc12)N1CCCC1c1cncc(F)c1 |r|
Fc1cncc(c1)C1CCCN1c1ccn2ncc(C(=O)NCC3CC3)c2n1
OCC1(CC1)NC(=O)c1cnn2ccc(nc12)N1CCCC1c1cncc(F)c1
OC1CN(C1)C(=O)c1cnn2ccc(nc12)N1CCCC1c1cncc(F)c1
C[C@H](O)CNC(=O)c1cnn2ccc(nc12)N1CCCC1c1cncc(F)c1 |r|
C[C@@H](O)CNC(=O)c1cnn2ccc(nc12)N1CCCC1c1cncc(F)c1 |r|
CC(C)(O)CNC(=O)c1cnn2ccc(nc12)N1CCCC1c1cncc(F)c1
OCCNC(=O)c1cnn2ccc(nc12)N1CCCC1c1cncc(F)c1
CC(NC(=O)c1cnn2ccc(nc12)N1CCCC1c1cncc(F)c1)C1CC1
CNC(=O)c1cnn2ccc(nc12)N1CCCC1c1cncc(F)c1
C[C@H](CO)NC(=O)c1cnn2ccc(nc12)N1CCCC1c1cncc(F)c1 |r|
C[C@@H](CO)NC(=O)c1cnn2ccc(nc12)N1CCCC1c1cncc(F)c1 |r|
NC(=O)c1cnn2ccc(nc12)N1CCCC1c1cncc(F)c1
COCC(C)NC(=O)c1cnn2ccc(nc12)N1CCCC1c1cncc(F)c1
COCC(O)CNC(=O)c1cnn2ccc(nc12)N1CCCC1c1cncc(F)c1
O[C@H]1CCCC1NC(=O)c1cnn2ccc(nc12)N1CCCC1c1cncc(F)c1 |r|
CC(C)[C@@H](CO)NC(=O)c1cnn2ccc(nc12)N1CCCC1c1cncc(F)c1 |r|
CC(C)[C@H](CO)NC(=O)c1cnn2ccc(nc12)N1CCCC1c1cncc(F)c1 |r|
C[C@@H](NC(=O)c1cnn2ccc(nc12)N1CCC[C@@H]1c1cncc(F)c1)C1CC1 |r|
C[C@H](NC(=O)c1cnn2ccc(nc12)N1CCC[C@@H]1c1cncc(F)c1)C1CC1 |r|
CC(C)(CO)CNC(=O)c1cnn2ccc(nc12)N1CCC[C@@H]1c1cncc(F)c1 |r|
Fc1cncc(c1)[C@H]1CCCN1c1ccn2ncc(C(=O)N3CCC3)c2n1 |r|
OCC1CN(C1)C(=O)c1cnn2ccc(nc12)N1CCC[C@@H]1c1cncc(F)c1 |r|
O[C@H]1CCN(C1)C(=O)c1cnn2ccc(nc12)N1CCC[C@@H]1c1cncc(F)c1 |r|
C[C@@H](NC(=O)c1cnn2ccc(nc12)N1CCCC1c1cncc(F)c1)C(F)(F)F |r|
C[C@H](NC(=O)c1cnn2ccc(nc12)N1CCCC1c1cncc(F)c1)C(F)(F)F |r|
Fc1cncc(c1)[C@H]1CCCN1c1ccn2ncc(C(=O)NCC(F)(F)F)c2n1 |r|
CC(C)(CO)NC(=O)c1cnn2ccc(nc12)N1CCC[C@@H]1c1cncc(F)c1 |r|
O[C@@H]1CCC[C@H]1NC(=O)c1cnn2ccc(nc12)N1CCC[C@@H]1c1cncc(F)c1 |r|
FC(F)CNC(=O)c1cnn2ccc(nc12)N1CCC[C@@H]1c1cncc(F)c1 |r|
O[C@H]1CCC[C@H]1NC(=O)c1cnn2ccc(nc12)N1CCC[C@@H]1c1cncc(F)c1 |r|
O[C@@H]1CCCC[C@H]1NC(=O)c1cnn2ccc(nc12)N1CCC[C@@H]1c1cncc(F)c1 |r|
Fc1cncc(c1)[C@H]1CCCN1c1ccn2ncc(C(=O)N3CCCCC3)c2n1 |r|
OC[C@H]1[C@H]2CCC(C2)[C@H]1NC(=O)c1cnn2ccc(nc12)N1CCCC1c1cncc(F)c1 |r,TLB:1:2:4.5:7,THB:9:8:4.5:7|
COc1ncc(F)cc1[C@H]1CCCN1c1ccn2ncc(C(=O)N3CC(O)C3)c2n1 |r|
COc1ncc(F)cc1[C@H]1CCCN1c1ccn2ncc(C(=O)NC3CC[C@H](O)CC3)c2n1 |r,wD:9.9,27.29,(-7.78,2.63,;-6.29,2.23,;-5.21,3.32,;-5.6,4.81,;-4.51,5.9,;-3.03,5.5,;-1.94,6.59,;-2.63,4.01,;-3.72,2.92,;-3.32,1.43,;-4.22,.19,;-3.32,-1.06,;-1.85,-.58,;-1.85,.96,;-.52,1.73,;-.52,3.27,;.81,4.04,;2.15,3.27,;3.61,3.74,;4.52,2.5,;3.61,1.25,;4.01,-.24,;2.92,-1.33,;5.5,-.64,;5.9,-2.12,;7.38,-2.52,;7.78,-4.01,;6.69,-5.1,;7.09,-6.59,;5.21,-4.7,;4.81,-3.21,;2.15,1.73,;.81,.96,)|
COc1ncc(F)cc1[C@H]1CCCN1c1ccn2ncc(C(=O)NCCCNC(=O)OC(C)(C)C)c2n1 |r|
NCCCNC(=O)c1cnn2ccc(nc12)N1CCC[C@@H]1c1cc(F)c[nH]c1=O |r|
COc1ncc(F)cc1[C@H]1CCCN1c1ccn2ncc(C(=O)NC[C@H](O)CO)c2n1 |r|
COc1ncc(F)cc1[C@H]1CCCN1c1ccn2ncc(C(=O)N3CC(C)(O)C3)c2n1 |r|
COc1ncc(F)cc1[C@H]1CCCN1c1ccn2ncc(C(=O)NCCCO)c2n1 |r|
COc1ncc(F)cc1[C@H]1CCCN1c1ccn2ncc(C(=O)NCC(O)CO)c2n1 |r|
COc1ncc(F)cc1[C@H]1CCCN1c1ccn2ncc(C(=O)NC[C@@H](O)CO)c2n1 |r|
COc1ncc(F)cc1[C@H]1CCCN1c1ccn2ncc(C(=O)NCCCCO)c2n1 |r|
COc1ncc(F)cc1[C@H]1CCCN1c1ccn2ncc(C(=O)NOCCOC(C)(C)C)c2n1 |r|
CNC(=O)c1cnn2ccc(nc12)N1CCC[C@@H]1c1cc(F)cnc1OC |r|
COc1ncc(F)cc1[C@H]1CCCN1c1ccn2ncc(C(=O)N[C@H]3CC[C@H](O)C3)c2n1 |r|
COc1ncc(F)cc1[C@H]1CCCN1c1ccn2ncc(C(=O)NCCO)c2n1 |r|
COc1ncc(F)cc1[C@H]1CCCN1c1ccn2ncc(C(=O)NC[C@H](C)O)c2n1 |r|
COc1ncc(F)cc1[C@H]1CCCN1c1ccn2ncc(C(=O)NC[C@@H](C)O)c2n1 |r|
COc1ncc(F)cc1[C@H]1CCCN1c1ccn2ncc(C(=O)NCC(C)(C)O)c2n1 |r|
COc1ncc(F)cc1[C@H]1CCCN1c1ccn2ncc(C(=O)NC3CCN(CCO)CC3)c2n1 |r|
COc1ncc(F)cc1[C@H]1CCCN1c1ccn2ncc(C(=O)NC(CO)CO)c2n1 |r|
COc1ncc(F)cc1[C@H]1CCCN1c1ccn2ncc(C(=O)Nc3ccc(=O)[nH]c3)c2n1 |r|
COc1ncc(F)cc1[C@H]1CCCN1c1ccn2ncc(C(=O)NC3CCN(CC3)S(C)(=O)=O)c2n1 |r|
OCCNC(=O)c1cnn2ccc(nc12)N1CCCC1c1cc(F)ccc1F
C[C@H](O)CNC(=O)c1cnn2ccc(nc12)N1CCC[C@@H]1c1cc(F)ccc1F |r|
C[C@@H](O)CNC(=O)c1cnn2ccc(nc12)N1CCCC1c1cc(F)ccc1F |r|
CC(C)(CO)CNC(=O)c1cnn2ccc(nc12)N1CCCC1c1cc(F)ccc1F
O[C@H]1CC[C@@H](C1)NC(=O)c1cnn2ccc(nc12)N1CCC[C@@H]1c1cc(F)ccc1F |r|
OC1CCN(CCNC(=O)c2cnn3ccc(nc23)N2CCC[C@@H]2c2cc(F)ccc2F)CC1 |r|
CN1CCN(CCNC(=O)c2cnn3ccc(nc23)N2CCCC2c2cc(F)ccc2F)CC1
COCCNC(=O)c1cnn2ccc(nc12)N1CCCC1c1cc(F)ccc1F
OCC(CO)NC(=O)c1cnn2ccc(nc12)N1CCC[C@@H]1c1cc(F)ccc1F |r|
C[C@@H](O)[C@H](CO)NC(=O)c1cnn2ccc(nc12)N1CCCC1c1cc(F)ccc1F |r|
C[C@H](O)[C@H](CO)NC(=O)c1cnn2ccc(nc12)N1CCCC1c1cc(F)ccc1F |r|
C[C@H](O)[C@@H](CO)NC(=O)c1cnn2ccc(nc12)N1CCCC1c1cc(F)ccc1F |r|
C[C@@H](CO)NC(=O)c1cnn2ccc(nc12)N1CCC[C@@H]1c1cc(F)ccc1F |r|
CC[C@@H](CO)NC(=O)c1cnn2ccc(nc12)N1CCC[C@@H]1c1cc(F)ccc1F |r|
CC(C)[C@@H](CO)NC(=O)c1cnn2ccc(nc12)N1CCCC1c1cc(F)ccc1F |r|
CC(C)(C)[C@@H](CO)NC(=O)c1cnn2ccc(nc12)N1CCC[C@@H]1c1cc(F)ccc1F |r|
Cc1ncc(F)cc1[C@H]1CCCN1c1ccn2ncc(C(=O)NC3CC3)c2n1 |r|
CCc1ncc(F)cc1[C@H]1CCCN1c1ccn2ncc(C(=O)NC3CC3)c2n1 |r|
Cc1ncc(F)cc1[C@H]1CCCN1c1ccn2ncc(C(=O)NC(C)(C)C)c2n1 |r|
CC(C)NC(=O)c1cnn2ccc(nc12)N1CCC[C@@H]1c1cc(F)cnc1C |r|
Cc1ncc(F)cc1C1CCCN1c1ccn2ncc(C(=O)NC3CCC3)c2n1
CNC(=O)c1cnn2ccc(nc12)N1CCC[C@@H]1c1cc(F)cnc1C |r|
Cc1ncc(F)cc1C1CCCN1c1ccn2ncc(C(N)=O)c2n1
Cc1ncc(F)cc1[C@H]1CCCN1c1ccn2ncc(C(=O)NCCO)c2n1 |r|
C[C@@H](O)CNC(=O)c1cnn2ccc(nc12)N1CCC[C@@H]1c1cc(F)cnc1C |r|
Cc1ncc(F)cc1C1CCCN1c1ccn2ncc(C(=O)NC3(C)CC3)c2n1
COCCNC(=O)c1cnn2ccc(nc12)N1CCCC1c1cc(F)cnc1C
Cc1ncc(F)cc1C1CCCN1c1ccn2ncc(C(=O)N3CC(O)C3)c2n1
Cc1ncc(F)cc1C1CCCN1c1ccn2ncc(C(=O)NC3(CO)CC3)c2n1
Cc1ncc(F)cc1C1CCCN1c1ccn2ncc(C(=O)NC3CC[C@H](O)CC3)c2n1 |r,wD:26.28,(-7.38,2.87,;-6.05,3.64,;-6.05,5.18,;-4.72,5.95,;-3.38,5.18,;-2.05,5.95,;-3.38,3.64,;-4.72,2.87,;-4.72,1.33,;-5.96,.42,;-5.49,-1.04,;-3.95,-1.04,;-3.47,.42,;-2.14,1.19,;-2.14,2.73,;-.8,3.5,;.53,2.73,;1.99,3.21,;2.9,1.96,;1.99,.72,;2.76,-.62,;1.99,-1.95,;4.3,-.62,;5.07,-1.95,;6.61,-1.95,;7.38,-3.28,;6.61,-4.62,;7.38,-5.95,;5.07,-4.62,;4.3,-3.28,;.53,1.19,;-.8,.42,)|
Cc1ncc(F)cc1C1CCCN1c1ccn2ncc(C(=O)NC3CC[C@H](O)CC3)c2n1 |r,wU:26.28,(-7.38,2.87,;-6.05,3.64,;-6.05,5.18,;-4.72,5.95,;-3.38,5.18,;-2.05,5.95,;-3.38,3.64,;-4.72,2.87,;-4.72,1.33,;-5.96,.42,;-5.49,-1.04,;-3.95,-1.04,;-3.47,.42,;-2.14,1.19,;-2.14,2.73,;-.8,3.5,;.53,2.73,;1.99,3.21,;2.9,1.96,;1.99,.72,;2.76,-.62,;1.99,-1.95,;4.3,-.62,;5.07,-1.95,;4.3,-3.28,;5.07,-4.62,;6.61,-4.62,;7.38,-5.95,;7.38,-3.28,;6.61,-1.95,;.53,1.19,;-.8,.42,)|
Cc1ncc(F)cc1C1CCCN1c1ccn2ncc(C(=O)N[C@H]3CC[C@H](O)C3)c2n1 |r|
Cc1ncc(F)cc1C1CCCN1c1ccn2ncc(C(=O)N[C@@H]3CCC[C@H]3O)c2n1 |r|
Cc1ncc(F)cc1C1CCCN1c1ccn2ncc(C(=O)N[C@H]3CN4CCC3CC4)c2n1 |r,wU:23.24,(-8.26,.87,;-6.93,1.64,;-6.93,3.18,;-5.59,3.95,;-4.26,3.18,;-2.93,3.95,;-4.26,1.64,;-5.59,.87,;-5.59,-.67,;-6.84,-1.58,;-6.36,-3.04,;-4.82,-3.04,;-4.35,-1.58,;-3.02,-.81,;-3.02,.73,;-1.68,1.5,;-.35,.73,;1.12,1.21,;2.02,-.04,;1.12,-1.28,;1.89,-2.62,;1.12,-3.95,;3.22,-3.39,;4.55,-2.62,;5.36,-1.4,;6.99,-.68,;6.99,1.03,;6.13,-.11,;6.13,-2.12,;7.46,-2.72,;8.26,-1.4,;-.35,-.81,;-1.68,-1.58,)|
CCc1ncc(F)cc1[C@H]1CCCN1c1ccn2ncc(C(=O)NC3CC[C@H](O)CC3)c2n1 |r,wD:9.9,27.29,(-8.05,3.64,;-6.72,2.87,;-5.38,3.64,;-5.38,5.18,;-4.05,5.95,;-2.72,5.18,;-1.38,5.95,;-2.72,3.64,;-4.05,2.87,;-4.05,1.33,;-5.3,.42,;-4.82,-1.04,;-3.28,-1.04,;-2.8,.42,;-1.47,1.19,;-1.47,2.73,;-.14,3.5,;1.2,2.73,;2.66,3.21,;3.57,1.96,;2.66,.72,;3.43,-.62,;2.66,-1.95,;4.97,-.62,;5.74,-1.95,;7.28,-1.95,;8.05,-3.28,;7.28,-4.62,;8.05,-5.95,;5.74,-4.62,;4.97,-3.28,;1.2,1.19,;-.14,.42,)|
CCc1ncc(F)cc1C1CCCN1c1ccn2ncc(C(=O)N[C@H]3CC[C@H](O)C3)c2n1 |r|
CCc1ncc(F)cc1C1CCCN1c1ccn2ncc(C(=O)NCC(C)(C)O)c2n1
CC(C)(C)NC(=O)c1cnn2ccc(nc12)N1CCC[C@@H]1c1cc(F)c[nH]c1=O |r|
CC1(C)OCC(COc2ccc(F)cc2[C@H]2CCCN2c2ccn3ncc(C(=O)NC4CC4)c3n2)O1 |r|
CC1(C)OCC(COc2ccc(F)cc2[C@H]2CCCN2c2ccn3ncc(C(N)=O)c3n2)O1 |r|
CC1(C)OCC(COc2cc(F)cc(c2)[C@H]2CCCN2c2ccn3ncc(C(=O)NC4CC4)c3n2)O1 |r|
CC1(C)OCC(COc2cc(F)cc(c2)[C@H]2CCCN2c2ccn3ncc(C(N)=O)c3n2)O1 |r|
OCC(O)COc1cc(F)cc(c1)[C@H]1CCCN1c1ccn2ncc(C(=O)NC3CC3)c2n1 |r|
NC(=O)c1cnn2ccc(nc12)N1CCC[C@@H]1c1cc(F)cc(OCC(O)CO)c1 |r|
OCC(O)COc1ccc(F)cc1[C@H]1CCCN1c1ccn2ncc(C(=O)NC3CC3)c2n1 |r|
NC(=O)c1cnn2ccc(nc12)N1CCC[C@@H]1c1cc(F)ccc1OCC(O)CO |r|
CC(NC(=O)c1cnn2ccc(nc12)N1C(CO)CCC1c1cncc(F)c1)C(F)(F)F
CC1(CC1)NC(=O)c1cnn2ccc(nc12)N1[C@H](CO)CC[C@@H]1c1cncc(F)c1 |r|
CC(C)NC(=O)c1cnn2ccc(nc12)N1[C@H](CO)CC[C@@H]1c1cncc(F)c1 |r|
CC(NC(=O)c1cnn2ccc(nc12)N1CC(O)CC1c1cccc(F)c1)C(F)(F)F
CC(C)NC(=O)c1cnn2ccc(nc12)N1C[C@@H](O)C[C@@H]1c1cccc(F)c1 |r|
CNC(=O)c1cnn2ccc(nc12)N1C[C@@H](O)C[C@@H]1c1cccc(F)c1 |r|
CC(C)NC(=O)c1cnn2ccc(nc12)N1[C@H](CC[C@@]1(C)CO)c1cncc(F)c1 |r|
CC(NC(=O)c1cnn2ccc(nc12)N1C(CCC1(C)CO)c1cncc(F)c1)C(F)(F)F
Nc1ncc(F)cc1[C@H]1CCCN1c1ccn2ncc(C(=O)N3CCC3)c2n1 |r|
OCCONC(=O)c1cnn2ccc(nc12)N1CCC[C@@H]1c1cc(F)cnc1Cl |r|
Cn1cc(F)cc([C@H]2CCCN2c2ccn3ncc(C(=O)NC(C)(C)C)c3n2)c1=O |r|
CC(C)NC(=O)c1cnn2ccc(nc12)N1CCC[C@@H]1c1cc(F)cn(C)c1=O |r|
Cn1cc(F)cc([C@H]2CCCN2c2ccn3ncc(C(=O)NC4CC4)c3n2)c1=O |r|
Cc1ccc(NC(=O)c2cnn3ccc(nc23)N2CCC[C@@H]2c2cc(F)cn(C)c2=O)cn1 |r|
Cn1cc(F)cc([C@H]2CCCN2c2ccn3ncc(C(=O)NC4CCC4)c3n2)c1=O |r|
Cn1cc(F)cc([C@H]2CCCN2c2ccn3ncc(C(=O)Nc4cccnc4)c3n2)c1=O |r|
Cn1cc(F)cc([C@H]2CCCN2c2ccn3ncc(C(=O)NCC4CC4)c3n2)c1=O |r|
Cn1cc(F)cc([C@H]2CCCN2c2ccn3ncc(C(=O)N[C@H](CO)C(C)(C)C)c3n2)c1=O |r|
Cn1cc(F)cc([C@H]2CCCN2c2ccn3ncc(C(=O)N[C@@H]4CCCC[C@H]4O)c3n2)c1=O |r|
C[C@@H](NC(=O)c1cnn2ccc(nc12)N1CCC[C@@H]1c1cc(F)cn(C)c1=O)C1CC1 |r|
C[C@H](NC(=O)c1cnn2ccc(nc12)N1CCC[C@@H]1c1cc(F)cn(C)c1=O)C1CC1 |r|
Cn1cc(F)cc([C@H]2CCCN2c2ccn3ncc(C(=O)NC4(C)CC4)c3n2)c1=O |r|
Cn1cc(F)cc([C@H]2CCCN2c2ccn3ncc(C(=O)NC4CC[C@H](O)CC4)c3n2)c1=O |r,wD:7.6,25.26,(-7.44,5.2,;-5.95,4.81,;-4.86,5.9,;-3.37,5.5,;-2.28,6.59,;-2.97,4.01,;-4.06,2.92,;-3.66,1.43,;-4.57,.19,;-3.66,-1.06,;-2.2,-.58,;-2.2,.96,;-.87,1.73,;-.87,3.27,;.47,4.04,;1.8,3.27,;3.27,3.74,;4.17,2.5,;3.27,1.25,;3.66,-.24,;2.58,-1.33,;5.15,-.64,;5.55,-2.12,;7.04,-2.52,;7.44,-4.01,;6.35,-5.1,;6.75,-6.59,;4.86,-4.7,;4.46,-3.21,;1.8,1.73,;.47,.96,;-5.55,3.32,;-6.64,2.23,)|
Cn1cc(F)cc([C@H]2CCCN2c2ccn3ncc(C(=O)Nc4ccc(F)cn4)c3n2)c1=O |r|
COc1ncc(F)cc1C1CCCN1c1ccn2ncc(C(=O)Nc3cc(C)n[nH]3)c2n1
COc1ncc(F)cc1[C@H]1CCCN1c1ccn2ncc(C(=O)Nc3ccn(C)n3)c2n1 |r|
COc1ncc(F)cc1[C@H]1CCCN1c1ccn2ncc(C(=O)Nc3cc(n[nH]3)C3CC3)c2n1 |r|
CCc1cc(NC(=O)c2cnn3ccc(nc23)N2CCCC2c2cc(F)cnc2OC)[nH]n1
COc1ncc(F)cc1[C@H]1CCCN1c1ccn2ncc(C(=O)Nc3ccn(n3)C(C)C)c2n1 |r|
C[C@@]12[C@@H]([C@@H](C[C@@H](O1)n3c4ccccc4c5c3c6n2c7ccccc7c6c8c5C(=O)NC8)NC)OC
C[C@@H](Cc1c(F)c(F)cc(F)c1F)Nc1cc[nH]c(=O)c1-c1nc2cc3C(=O)N(Cc3cc2[nH]1)C1CCN(C)CC1 |r|
C[C@@H](Cc1c(F)c(F)cc(F)c1F)Nc1cc[nH]c(=O)c1-c1nc2cc3C(=O)N(CCN(C)C)C(=O)c3cc2[nH]1 |r|
C[C@@H](Cc1c(F)c(F)cc(F)c1F)Nc1cc[nH]c(=O)c1-c1nc2cc3C(=O)N(CCN(C)C)Cc3cc2[nH]1 |r|
CC(Cc1cc(F)ccc1F)Nc1cc[nH]c(=O)c1-c1nc2cc3C(=O)N(C4CCN(C)CC4)C(=O)c3cc2[nH]1
C[C@@H](Cc1c(F)c(F)cc(F)c1F)Nc1cc[nH]c(=O)c1-c1nc2cc3C(=O)N(C(=O)c3cc2[nH]1)c1cccnc1 |r|
C[C@@H](Cc1c(F)c(F)cc(F)c1F)Nc1cc[nH]c(=O)c1-c1nc2cc3C(=O)N(C(O)c3cc2[nH]1)c1cccnc1 |r|
COC1N(C(=O)c2cc3nc([nH]c3cc12)-c1c(NC(C)Cc2c(F)c(F)cc(F)c2F)cc[nH]c1=O)c1cccnc1
C[C@@H](Cc1c(F)c(F)cc(F)c1F)Nc1cc[nH]c(=O)c1-c1nc2cc3C(=O)N(C(=O)c3cc2[nH]1)c1ccc(F)nc1 |r|
CC(Cc1cc(F)ccc1F)Nc1cc[nH]c(=O)c1-c1nc2cc3C(=O)N(CCN(C)C)C(=O)c3cc2[nH]1
CC(Cc1cc(F)ccc1F)Nc1cc[nH]c(=O)c1-c1nc2cc3CN(CCN(C)C)C(=O)c3cc2[nH]1
CC(Cc1c(F)c(F)cc(F)c1F)Nc1cc[nH]c(=O)c1-c1nc2cc3CN(C4CCN(C)CC4)C(=O)c3c(C)c2[nH]1
CC(Cc1c(F)c(F)cc(F)c1F)Nc1cc[nH]c(=O)c1-c1nc2c(C)c3CN(C4CCN(C)CC4)C(=O)c3cc2[nH]1
CC(Cc1c(F)c(F)cc(F)c1F)Nc1cc[nH]c(=O)c1-c1nc2c(C)c3C(=O)N(C4CCN(C)CC4)C(=O)c3cc2[nH]1
C[C@H](Nc1nc(Nc2cc([nH]n2)C2CC2)c(Cl)cc1Cl)c1ccc(F)cc1
C[C@H](Nc1nc(Nc2cc([nH]n2)C2CC2)c(F)cc1CNC(=O)C1CCC(=O)N1)c1ccc(F)cc1
C[C@H](Nc1ccc(c(Nc2cc([nH]n2)C2CC2)n1)[N+]([O-])=O)c1ccc(F)cc1
CC(C)n1cc(C(=O)c2cncc(NC(=O)Cc3ccc(F)cc3)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)Cc3cccc(c3)C(F)(F)F)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)Cc3ccc(cc3)C(F)(F)F)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)Cc3ccc(Cl)c(Cl)c3)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)Cc3ccc(Cl)cc3)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)Cc3ccccc3OC3CC3)c2)c2cncnc12
CC(C)n1cc(c2c1ncnc2)C(=O)c3cc(cnc3)NC(=O)Cc4ccc(cc4)C#N
CC(C)n1cc(C(=O)c2cncc(NC(=O)Cc3ccc(C#N)c(c3)C(F)(F)F)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)Cc3ccc(OC4CC4)cc3)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)Cc3cccc(OC4CC4)c3)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)Cc3cccc(CO)c3)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)Cc3ccc(C#N)c(F)c3)c2)c2cncnc12
COc1cc(CC(=O)Nc2cncc(c2)C(=O)c2cn(C(C)C)c3ncncc23)ccc1C#N
CC(C)n1cc(C(=O)c2cncc(NC(=O)CN3Cc4ccc(F)cc4C3=O)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)Cn3ccc(n3)-c3ccccn3)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)Cc3ccc4[nH]cnc4c3)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)Cc3ccc4nccnc4c3)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)Cc3cnc4cccnc4c3)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)Cc3ccc4onc(N)c4c3)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)Cc3ccc4[nH]c(nc4c3)C(F)(F)F)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)Cc3ccn4ccnc4c3)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)Cn3ncc4ncccc34)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)Cc3cccc(c3)S(C)(=O)=O)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)Cn3cc(nn3)C3CC3)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)Cc3ccc4ocnc4c3)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)Cn3ccc(n3)C3CC3)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)Cc3cncc(OC4CC4)c3)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)Cc3ccc4OCCc4c3)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)Cn3cc4ccccc4n3)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)Cn3cc4cc(F)ccc4n3)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)Cn3ncc4cc(F)ccc34)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)Cn3nc(cc3C)C(F)(F)F)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)Cn3ccc(n3)C(F)(F)F)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)Cc3ccc(Cl)cn3)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)Cc3ccc4cn[nH]c4c3)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)Cc3ccc4cccnc4c3)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)Cn3cc4cccc(F)c4n3)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)Cn3ncc4cccnc34)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)Cn3ncc4ccccc34)c2)c2cncnc12
CC(C)c1cc(C)n(CC(=O)Nc2cncc(c2)C(=O)c2cn(C(C)C)c3ncncc23)n1
CC(C)c1cn(CC(=O)Nc2cncc(c2)C(=O)c2cn(C(C)C)c3ncncc23)nn1
CC(C)n1cc(C(=O)c2cncc(NC(=O)Cn3cc(nn3)C(F)(F)F)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)Cn3ncc4cccc(F)c34)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)Cn3nc4ccccc4n3)c2)c2cncnc12
Cn1cc(C(=O)c2cncc(NC(=O)Cc3cccc(Cl)c3)c2)c2cncnc12
Cn1cc(C(=O)c2cncc(NC(=O)CCc3ccccc3Cl)c2)c2cncnc12
CC(C)(C)n1cc(C(=O)c2cncc(NC(=O)Cc3coc(n3)C3CC3)c2)c2cncnc12
CC(C)(C)n1cc(C(=O)c2cncc(NC(=O)Cc3cccc(c3)S(C)(=O)=O)c2)c2cncnc12
Cc1nn(C)cc1CC(=O)Nc1cncc(c1)C(=O)c1cn(c2ncncc12)C(C)(C)C
Cn1cc(CC(=O)Nc2cncc(c2)C(=O)c2cn(c3ncncc23)C(C)(C)C)cn1
Cn1cc(CC(=O)Nc2cncc(c2)C(=O)c2cn(c3ncncc23)C(C)(C)C)c(n1)C1CC1
C[C@@H](CO)n1cc(C(=O)c2cncc(NC(=O)Cc3cccc(c3)C(F)(F)F)c2)c2cncnc12
C[C@H](CO)n1cc(C(=O)c2cncc(NC(=O)Cc3cccc(c3)C(F)(F)F)c2)c2cncnc12
CC(C)c1cn(CC(=O)Nc2cncc(c2)C(=O)c2cn([C@H](C)CO)c3ncncc23)nn1
CC(C)n1ncc(CC(=O)Nc2cncc(c2)C(=O)c2cn([C@H](C)CO)c3ncncc23)c1C(F)(F)F
C[C@H](CO)n1cc(C(=O)c2cncc(NC(=O)Cc3ccc(cc3)C#N)c2)c2cncnc12
C[C@H](CO)n1cc(C(=O)c2cncc(NC(=O)Cc3cccc(c3)S(C)(=O)=O)c2)c2cncnc12
C[C@H](CO)n1cc(C(=O)c2cncc(NC(=O)Cc3ccc4cccnc4c3)c2)c2cncnc12
CC(CO)n1cc(C(=O)c2cncc(NC(=O)Cc3ccc4cccnc4c3)c2)c2cnc(N)nc12
CC(CO)n1cc(C(=O)c2cncc(NC(=O)Cc3ccc(cc3)C#N)c2)c2cnc(N)nc12
CC(CO)n1cc(C(=O)c2cncc(NC(=O)Cc3cccc(c3)C(F)(F)F)c2)c2cnc(N)nc12
Clc1ccc(CC(=O)Nc2cncc(c2)C(=O)c2cn(C3COC3)c3ncncc23)cc1Cl
O=C(Cc1ccc(cc1)C#N)Nc1cncc(c1)C(=O)c1cn(C2COC2)c2ncncc12
Clc1ccc(CC(=O)Nc2cncc(c2)C(=O)c2cn(C3COC3)c3ncncc23)cc1
Clc1cccc(CC(=O)Nc2cncc(c2)C(=O)c2cn(C3COC3)c3ncncc23)c1
O=C(Cc1cccc(c1)C#N)Nc1cncc(c1)C(=O)c1cn(C2COC2)c2ncncc12
O=C(Cc1ccc2cccnc2c1)Nc1cncc(c1)C(=O)c1cn(C2COC2)c2ncncc12
Clc1ccc2nc(CC(=O)Nc3cncc(c3)C(=O)c3cn(C4COC4)c4ncncc34)cn2c1
O=C(CN1Cc2ccccc2C1=O)Nc1cncc(c1)C(=O)c1cn(C2COC2)c2ncncc12
CC(C)(CO)n1cc(C(=O)c2cncc(NC(=O)Cc3ccc(cc3)C#N)c2)c2cncnc12
CC(C)(CO)n1cc(C(=O)c2cncc(NC(=O)Cc3cccc(c3)C(F)(F)F)c2)c2cncnc12
CC(C)c1cn(CC(=O)Nc2cncc(c2)C(=O)c2cn(c3ncncc23)C(C)(C)CO)nn1
CC(C)(CO)n1cc(C(=O)c2cncc(NC(=O)Cc3ccc4cccnc4c3)c2)c2cncnc12
CC(C(N)=O)n1cc(C(=O)c2cncc(NC(=O)Cc3ccc(Cl)cc3)c2)c2cncnc12
CC(C(=O)N(C)C)n1cc(C(=O)c2cncc(NC(=O)Cc3ccc(Cl)cc3)c2)c2cncnc12
CC(CO)(CO)n1cc(C(=O)c2cncc(NC(=O)Cc3ccc(cc3)C#N)c2)c2cncnc12
CC(CO)(CO)n1cc(C(=O)c2cncc(NC(=O)Cc3ccc4cccnc4c3)c2)c2cncnc12
Cc1cc(nn1CC(=O)Nc1cncc(c1)C(=O)c1cn(c2ncncc12)C(C)(CO)CO)C(F)(F)F
CC(CO)(CO)n1cc(C(=O)c2cncc(NC(=O)Cc3ccc(Cl)cc3)c2)c2cncnc12
CC(CO)(CO)n1cc(C(=O)c2cncc(NC(=O)Cc3ccc(cc3)C(F)(F)F)c2)c2cncnc12
CC(CO)(CO)n1cc(C(=O)c2cncc(NC(=O)Cc3ccc(Cl)cn3)c2)c2cncnc12
CC(CO)(CO)n1cc(C(=O)c2cncc(NC(=O)Cc3cccc(c3)C(F)(F)F)c2)c2cncnc12
CC(CO)(CO)n1cc(C(=O)c2cncc(NC(=O)Cn3ccc(n3)C(F)(F)F)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)Cn3cc(nn3)C(F)(F)F)c2)c2cnc(N)nc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)Cc3ccc(cc3)C#N)c2)c2cnc(N)nc12
Cn1cc(C(=O)c2cncc(NC(=O)COc3ccccc3)c2)c2cncnc12
Cn1cc(C(=O)c2cncc(NC(=O)COc3ccc(F)cc3)c2)c2cncnc12
Cn1cc(C(=O)c2cncc(NC(=O)C3(CC3)c3ccccc3)c2)c2cncnc12
Cn1cc(C(=O)c2cncc(NC(=O)C3Cc4ccccc4C3)c2)c2cncnc12
C[C@@H](C(=O)Nc1cncc(c1)C(=O)c1cn(C)c2ncncc12)c1ccccc1
CC(C)n1cc(C(=O)c2cncc(NC(=O)C(CO)c3ccccc3)c2)c2cncnc12
COc1ccc2n(CC(=O)Nc3cncc(c3)C(=O)c3cn(C(C)C)c4ncncc34)ccc2c1
CC(C)n1cc(C(=O)c2cncc(NC(=O)c3cccc(Cl)c3)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)c3ccc(Cl)cc3)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)c3ccc(cc3)C(F)(F)F)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)c3ccc(OC(F)(F)F)cc3)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)COc3ccccc3C#N)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)COc3ccc(OC(F)(F)F)cc3)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)C(N)c3ccc(Cl)cc3)c2)c2cncnc12
CC(C)(CO)n1cc(C(=O)c2cncc(NC(=O)Cc3ccc(cn3)C#N)c2)c2cnc(N)nc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)Cc3cn(nc3C(F)(F)F)C3CC3)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)Cn3cnc(Cl)c3Cl)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)c3nc4nc(C)cc(C(F)F)n4n3)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)Cn3nc(C)nc3C)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)Cn3ccnc3C)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)Cc3cn4ccsc4n3)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)Cc3nnc(O)c4ccccc34)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)Cc3cn4c(C)c(C)sc4n3)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)Cn3cc(nn3)C3(O)CCCC3)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)Cn3nnnc3-c3cccc(C)c3)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)Cn3cnc(c3)-c3ccc(F)cc3)c2)c2cncnc12
CC(C)c1ccnn1CC(=O)Nc1cncc(c1)C(=O)c1cn(C(C)C)c2ncncc12
CCc1nn2cc(CC(=O)Nc3cncc(c3)C(=O)c3cn(C(C)C)c4ncncc34)nc2s1
CC(C)n1cc(C(=O)c2cncc(NC(=O)Cc3cn4cc(C)sc4n3)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)Cn3nc(Cl)nc3C)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)Cn3ccnc3-c3ccccc3)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)Cc3cn4cc(Cl)sc4n3)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)Cn3ccnc3)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)Cc3cn4c(C)csc4n3)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)Cc3ccn(c3)-c3ccc(O)cc3)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)Cc3cnc4ncnn4c3)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)Cc3cnccn3)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)Cn3cc(nn3)-c3cccc(O)c3)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)Cn3nnnc3-c3ccccc3)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)c3nccc4occc34)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)c3cnn4CCCc34)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)c3ncncc3Br)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)c3ccc(nc3)C#N)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)c3cnn4cccnc34)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)c3cnc4[nH]nc(C)c4c3)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)c3cc4cccc(C)n4n3)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)c3ncoc3C)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)c3cc4cscc4cn3)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)c3cc(C)nc(C)n3)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)c3cc(ccn3)C#N)c2)c2cncnc12
COCc1cc(nn1C)C(=O)Nc1cncc(c1)C(=O)c1cn(C(C)C)c2ncncc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)c3nc(Cl)c(Cl)[nH]3)c2)c2cncnc12
COc1cc(nc2c(C)nccc12)C(=O)Nc1cncc(c1)C(=O)c1cn(C(C)C)c2ncncc12
CCc1nc(C)c(o1)C(=O)Nc1cncc(c1)C(=O)c1cn(C(C)C)c2ncncc12
COc1cncc(c1)C(=O)Nc1cncc(c1)C(=O)c1cn(C(C)C)c2ncncc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)c3cnc4[nH]ncc4c3)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)c3cnc4[nH]cnc4c3)c2)c2cncnc12
COc1nccn2cc(nc12)C(=O)Nc1cncc(c1)C(=O)c1cn(C(C)C)c2ncncc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)c3ccncc3)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)c3ncccc3C)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)c3cnc4occc4c3)c2)c2cncnc12
CC(C)c1nnc2ccc(cn12)C(=O)Nc1cncc(c1)C(=O)c1cn(C(C)C)c2ncncc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)c3cocn3)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)c3ncccc3Cl)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)c3cnc4nccn4c3)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)c3cc(on3)C3CC3)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)c3cc(n[nH]3)C3CC3)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)c3nnc4cc(C)nn4c3C)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)c3cnccc3C)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)c3cn(cn3)C3CCC3)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)c3cc4ccccn4n3)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)c3ccc4nnnn4c3)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)c3nnc4CCCCn34)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)c3nc(C)oc3C(F)(F)F)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)c3cnc4cc[nH]c4c3)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)c3ccc4c[nH]nc4n3)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)c3[nH]nc4ccccc34)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)c3cnc4onc(C)c4c3)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)c3ccnnc3)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)c3cc4OCCOc4cn3)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)c3n[nH]c4ncccc34)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)c3n[nH]c4ccc(F)cc34)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)c3cc(C)nn3C)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)c3ccnc4ncsc34)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)Cc3c(C)[nH]c4c(F)cccc34)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)Cc3c(C)[nH]c4ccc(Cl)cc34)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)Cn3ccc4ccccc34)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)Cc3cnn(C(C)C)c3C(F)(F)F)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)Cn3ccc(C)n3)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)Cn3cccn3)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)Cn3nc(C)cc3C)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)Cc3c(C)[nH]c4ccccc34)c2)c2cncnc12
COc1ccc2[nH]cc(CC(=O)Nc3cncc(c3)C(=O)c3cn(C(C)C)c4ncncc34)c2c1
CC(C)n1cc(C(=O)c2cncc(NC(=O)Cc3cccnc3)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)Cn3nnc4cc(Cl)ccc34)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)Cn3ccc(n3)-c3cccs3)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)Cc3cn4ccc(C)nc4n3)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)Cn3cnc4c(C)nc(C)nc34)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)Cn3ncc4ccc(cc34)[N+]([O-])=O)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)Cc3nn(C)c4ccc(Cl)cc34)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)Cc3c(C)[nH]c4ccc(F)cc34)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)Cc3cn4cc(Cl)ccc4n3)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)Cn3c(C)nc4ccccc34)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)Cc3cn4ccccc4n3)c2)c2cncnc12
COc1ccc2n(CC(=O)Nc3cncc(c3)C(=O)c3cn(C(C)C)c4ncncc34)ccc2n1
CC(C)n1cc(C(=O)c2cncc(NC(=O)Cn3nccc3C)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)Cn3cnc4cccc(C)c34)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)Cc3c[nH]c4ccccc34)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)Cn3cnc4ccccc34)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)Cc3cc(C)n[nH]3)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)Cn3nnc4ccccc34)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)Cc3cn(C)c4ccccc34)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)Cc3cc(c[nH]3)-c3ccccc3)c2)c2cncnc12
CCc1nc2cccnc2n1CC(=O)Nc1cncc(c1)C(=O)c1cn(C(C)C)c2ncncc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)Cc3c[nH]c4ccc(Cl)cc34)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)Cc3ccn(c3)-c3ccccc3)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)Cc3c[nH]c4ccc(C)cc34)c2)c2cncnc12
CCc1nc2ccccc2n1CC(=O)Nc1cncc(c1)C(=O)c1cn(C(C)C)c2ncncc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)Cc3cn4cccnc4n3)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)Cc3n[nH]c4ccccc34)c2)c2cncnc12
COc1cc(F)cc2ccn(CC(=O)Nc3cncc(c3)C(=O)c3cn(C(C)C)c4ncncc34)c12
CC(C)n1cc(C(=O)c2cncc(NC(=O)Cc3cn(Cc4ccccc4)nn3)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)Cc3nn(C)c4cc(Cl)ccc34)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)Cc3c[nH]c4c(Cl)cccc34)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)Cn3ncc(c3C)-c3ccccc3)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)Cc3cncc(Br)c3)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)Cc3ccccn3)c2)c2cncnc12
COc1ccc(CC(=O)Nc2cncc(c2)C(=O)c2cn(C(C)C)c3ncncc23)cn1
CC(C)n1cc(C(=O)c2cncc(NC(=O)Cc3ccc(Cl)cn3)c2)c2cnc(N)nc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)Cc3ccc(F)cn3)c2)c2cnc(N)nc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)Cc3ccc(cc3)C(F)(F)F)c2)c2cnc(N)nc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)Cc3cccc(c3)C(F)(F)F)c2)c2cnc(N)nc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)Cc3ccc4ocnc4c3)c2)c2cnc(N)nc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)Cc3cccc(c3)S(C)(=O)=O)c2)c2cnc(N)nc12
CC(C)c1cn(CC(=O)Nc2cncc(c2)C(=O)c2cn(C(C)C)c3nc(N)ncc23)nn1
CC(C)n1cc(C(=O)c2cncc(NC(=O)Cn3cc(nn3)C3CC3)c2)c2cnc(N)nc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)Cc3ccc(Cl)cc3)c2)c2cnc(N)nc12
CC(C)n1ncc(CC(=O)Nc2cncc(c2)C(=O)c2cn(C(C)C)c3nc(N)ncc23)c1C(F)(F)F
CC(C)n1cc(C(=O)c2cncc(NC(=O)Cn3ccc(n3)C(F)(F)F)c2)c2cnc(N)nc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)Cn3ccc(n3)C3CC3)c2)c2cnc(N)nc12
CC(C)n1cc(CC(=O)Nc2cncc(c2)C(=O)c2cn(C(C)C)c3nc(N)ncc23)c(n1)C(F)(F)F
CC(C)(CO)n1cc(C(=O)c2cncc(NC(=O)Cc3cccc(c3)C(F)(F)F)c2)c2cnc(N)nc12
CC(C)(CO)n1cc(C(=O)c2cncc(NC(=O)Cc3ccc4ocnc4c3)c2)c2cnc(N)nc12
CC(C)(CO)n1cc(C(=O)c2cncc(NC(=O)Cc3cccc(c3)S(C)(=O)=O)c2)c2cnc(N)nc12
CC(C)(CO)n1cc(C(=O)c2cncc(NC(=O)Cc3ccc(cc3)C#N)c2)c2cnc(N)nc12
CC(C)n1ncc(CC(=O)Nc2cncc(c2)C(=O)c2cn(c3nc(N)ncc23)C(C)(C)CO)c1C(F)(F)F
CC(CO)(CO)n1cc(C(=O)c2cncc(NC(=O)Cc3ccc(C#N)c(c3)C(F)(F)F)c2)c2cncnc12
CC(CO)(CO)n1cc(C(=O)c2cncc(NC(=O)Cc3ccc(F)c(c3)C(F)(F)F)c2)c2cncnc12
CC(CO)(CO)n1cc(C(=O)c2cncc(NC(=O)c3cccc(c3)C(F)(F)F)c2)c2cncnc12
CC(CO)(CO)n1cc(C(=O)c2cncc(NC(=O)c3ccc(c(F)c3)C(F)(F)F)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)Cc3cccc(CN4CCC4)c3)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)Cc3cccc(CN4CC(F)C4)c3)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)Cc3cccc(CN4CCOCC4)c3)c2)c2cncnc12
OCC(CO)n1cc(C(=O)c2cncc(NC(=O)c3cccc(c3)C(F)(F)F)c2)c2cncnc12
OCC(CO)n1cc(C(=O)c2cncc(NC(=O)Cc3ccc(Cl)cc3)c2)c2cncnc12
OCC(CO)n1cc(C(=O)c2cncc(NC(=O)c3cccc(OC(F)(F)F)c3)c2)c2cncnc12
OCC(CO)n1cc(C(=O)c2cncc(NC(=O)Cc3ccc4cccnc4c3)c2)c2cncnc12
OCC(CO)n1cc(C(=O)c2cncc(NC(=O)Cc3ccc(cc3)C(F)(F)F)c2)c2cncnc12
OCC(CO)n1cc(C(=O)c2cncc(NC(=O)Cc3cccc(c3)C(F)(F)F)c2)c2cncnc12
Cc1ccc2ccc(CC(=O)Nc3cncc(c3)C(=O)c3cn(C(CO)CO)c4ncncc34)cc2n1
OCC(CO)n1cc(C(=O)c2cncc(NC(=O)Cc3ccc(Cl)c(Cl)c3)c2)c2cncnc12
OCC(CO)n1cc(C(=O)c2cncc(NC(=O)Cc3ccc(c(F)c3)C(F)(F)F)c2)c2cncnc12
OCC(CO)n1cc(C(=O)c2cncc(NC(=O)Cc3ccc(Cl)cc3Cl)c2)c2cncnc12
OCC(CO)n1cc(C(=O)c2cncc(NC(=O)Cc3cccc(OC(F)(F)F)c3)c2)c2cncnc12
OCC(CO)n1cc(C(=O)c2cncc(NC(=O)Cc3ccc(OC(F)(F)F)cc3)c2)c2cncnc12
OCC(CO)n1cc(C(=O)c2cncc(NC(=O)c3cc(F)cc(c3)C(F)(F)F)c2)c2cncnc12
OCC(CO)n1cc(C(=O)c2cncc(NC(=O)Cc3ccc(Cl)cn3)c2)c2cncnc12
OCC(CO)n1cc(C(=O)c2cncc(NC(=O)Cn3ccc(n3)C(F)(F)F)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)[C@H](Cc3ccc(cc3)C(=O)c3ccccc3)NC(=O)OC(C)(C)C)c2)c2cncnc12 |r|
CC(C)n1cc(C(=O)c2cncc(NC(=O)[C@H](N)Cc3ccc(cc3)C(=O)c3ccccc3)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)c3nonc3C)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)c3nn(C)c4ccccc34)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)c3cc4ccccc4[nH]3)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)c3sc(C)nc3C(F)(F)F)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)c3ncoc3C3CC3)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)c3cccnn3)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)c3c(C)n[nH]c3C(F)(F)F)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)c3cc(C)ccn3)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)c3c[nH]nc3C3CCC3)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)c3cnco3)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)c3nc(C)c[nH]3)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)c3cc4cc[nH]c4cn3)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)c3cnc(C)cn3)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)c3cn(C)nc3C)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)c3cnc4cn[nH]c4c3)c2)c2cncnc12
CCc1cc(no1)C(=O)Nc1cncc(c1)C(=O)c1cn(C(C)C)c2ncncc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)c3ccnn3C)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)c3cnc4ccccc4c3)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)c3cc4cc(F)cnc4[nH]3)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)c3cc(C)n(C)n3)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)c3coc(n3)C3CC3)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)c3scnc3C(F)(F)F)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)c3ncn4CCCc34)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)c3cc4sccc4cn3)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)c3cn(C)nc3C(F)(F)F)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)c3ccn4cncc4c3)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)c3ccnc4[nH]ccc34)c2)c2cncnc12
CCc1cc(on1)C(=O)Nc1cncc(c1)C(=O)c1cn(C(C)C)c2ncncc12
COc1ccnc(c1)C(=O)Nc1cncc(c1)C(=O)c1cn(C(C)C)c2ncncc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)c3cncnc3)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)c3c[nH]nc3C)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)c3c[nH]c4ncc(C)cc34)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)c3ncncc3C)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)c3cnc4ccsc4c3)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)c3cnc4ccnn4c3)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)c3noc4CCCCc34)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)c3ncc4ccccn34)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)c3ccc4cc[nH]c4n3)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)c3cncnc3N)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)c3c[nH]c4cnccc34)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)c3ccnc(C)c3)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)c3ccc4nccn4c3)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)c3nc[nH]n3)c2)c2cncnc12
COc1ccc(nc1)C(=O)Nc1cncc(c1)C(=O)c1cn(C(C)C)c2ncncc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)CN3CCc4cccnc4C3)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)C(O)c3ccccc3)c2)c2cncnc12
CCOc1ncc(cc1NC(=O)Cn1nc(cc1C)C(F)(F)F)C(=O)c1cn(C(C)C)c2ncncc12
CC(C)(C)n1cc(C(=O)c2cncc(NC(=O)Cc3ccc(cc3)C#N)c2)c2cnc(N)nc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)C(CO)c3ccc(Cl)cc3)c2)c2cncnc12
OCC1(CC1)n1cc(C(=O)c2cncc(NC(=O)Cc3ccc(cc3)C#N)c2)c2cncnc12
OCC1(CC1)n1cc(C(=O)c2cncc(NC(=O)Cc3ccc(Cl)cn3)c2)c2cncnc12
OCC1(CC1)n1cc(C(=O)c2cncc(NC(=O)Cc3ccc(cc3)C(F)(F)F)c2)c2cncnc12
OCC1(CC1)n1cc(C(=O)c2cncc(NC(=O)Cn3ccc(n3)C(F)(F)F)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)Nc3cc(nn3-c3cnn(C)c3)C3CC3)c2)c2cncnc12
CC(C)(C)n1cc(C(=O)c2cncc(NC(=O)Cc3nc4ccccc4[nH]3)c2)c2cnc(N)nc12
CC(C)(C)n1cc(C(=O)c2cncc(NC(=O)Cc3ccc(Br)cn3)c2)c2cnc(N)nc12
CC(C)(C)n1cc(C(=O)c2cncc(NC(=O)Cc3ccc(cn3)C#N)c2)c2cnc(N)nc12
C[C@@H](CO)n1cc(C(=O)c2cncc(NC(=O)Cc3ccc(OC(F)F)cc3)c2)c2cncnc12
C[C@@H](CO)n1cc(C(=O)c2cncc(NC(=O)Cn3cc4ccccc4n3)c2)c2cncnc12
C[C@@H](CO)n1cc(C(=O)c2cncc(NC(=O)Cc3nc4ccccc4[nH]3)c2)c2cncnc12
C[C@@H](CO)n1cc(C(=O)c2cncc(NC(=O)Cc3ccc(OC(F)(F)F)cc3)c2)c2cncnc12
C[C@@H](CO)n1cc(C(=O)c2cncc(NC(=O)Cc3ccc(F)c(F)c3)c2)c2cncnc12
COCC(C)(C)n1cc(C(=O)c2cncc(NC(=O)Cc3ccc(Cl)cn3)c2)c2cncnc12
COCC(C)(C)n1cc(C(=O)c2cncc(NC(=O)Cc3ccc(F)cn3)c2)c2cncnc12
COCC(C)(C)n1cc(C(=O)c2cncc(NC(=O)Cn3ccc(n3)C3CC3)c2)c2cncnc12
COCC(C)(C)n1cc(C(=O)c2cncc(NC(=O)Cc3ccc(F)cc3)c2)c2cncnc12
CN(C(=O)Cc1ccc(F)cc1)c1cncc(c1)C(=O)c1cn(c2ncncc12)C(C)(C)C
CN(C(=O)Cc1ccc(Cl)cn1)c1cncc(c1)C(=O)c1cn(c2ncncc12)C(C)(C)C
CN(C(=O)Cc1ccc(Cl)cc1)c1cncc(c1)C(=O)c1cn(c2ncncc12)C(C)(C)C
CC(C)(C)n1cc(C(=O)c2cncc(NC(=O)Cc3ccc(Cl)cc3)c2)c2cncnc12
CC(C)(C)n1cc(C(=O)c2cncc(NC(=O)Cc3ccc(F)cc3)c2)c2cncnc12
COCC(C)(C)n1cc(C(=O)c2cncc(NC(=O)Cc3ccc(Cl)cn3)c2)c2cnc(N)nc12
COCC(C)(C)n1cc(C(=O)c2cncc(NC(=O)Cc3ccc(F)cn3)c2)c2cnc(N)nc12
COCC(C)(C)n1cc(C(=O)c2cncc(NC(=O)Cn3ccc(n3)C(F)(F)F)c2)c2cnc(N)nc12
COCC(C)(C)n1cc(C(=O)c2cncc(NC(=O)Cn3cc(nn3)C(F)(F)F)c2)c2cnc(N)nc12
COCC(C)(C)n1cc(C(=O)c2cncc(NC(=O)Cn3cc(cn3)C(F)(F)F)c2)c2cnc(N)nc12
COCC(C)(C)n1cc(C(=O)c2cncc(NC(=O)Cn3cc(nn3)C3CC3)c2)c2cnc(N)nc12
CC(C)(CO)n1cc(C(=O)c2cncc(NC(=O)Cn3cc4ccccc4n3)c2)c2cnc(N)nc12
CC(C)(CO)n1cc(C(=O)c2cncc(NC(=O)Cn3cnc4ccccc4c3=O)c2)c2cnc(N)nc12
CC(C)(CO)n1cc(C(=O)c2cncc(NC(=O)Cc3ncc(F)cc3F)c2)c2cnc(N)nc12
Cc1ccc(CC(=O)Nc2cncc(c2)C(=O)c2cn(c3nc(N)ncc23)C(C)(C)CO)nc1
CN(c1ccc(CC(=O)Nc2cncc(c2)C(=O)c2cn(c3nc(N)ncc23)C(C)(C)CO)cc1)S(C)(=O)=O
CC(C)(CO)n1cc(C(=O)c2cncc(NC(=O)Cc3nc4ccccc4[nH]3)c2)c2cnc(N)nc12
CC(C)(CO)n1cc(C(=O)c2cncc(NC(=O)Cn3cc(ccc3=O)C(F)(F)F)c2)c2cnc(N)nc12
CC(C)(CO)n1cc(C(=O)c2cncc(NC(=O)Cc3ncc(Cl)cc3F)c2)c2cnc(N)nc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)Cc3c(C)[nH]c4ccc(C)cc34)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)Cc3ccc(C)nc3)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)Cc3ccc4ccc(C)nc4c3)c2)c2cncnc12
COc1ccc2[nH]c(C)c(CC(=O)Nc3cncc(c3)C(=O)c3cn(C(C)C)c4ncncc34)c2c1
CC(C)n1cc(C(=O)c2cncc(NC(=O)Cc3ccc4nnnn4n3)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)Cc3c[nH]c4ccc(O)cc34)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)Cc3c[nH]c4nccnc34)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)Cn3cnc4cc(C)c(C)cc34)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)Cn3cc(nn3)-c3ccccn3)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)Cn3cc(C)nn3)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)Cc3c(C)[nH]nc3-c3ccccc3)c2)c2cncnc12
CSc1ncc(CC(=O)Nc2cncc(c2)C(=O)c2cn(C(C)C)c3ncncc23)cn1
CC(C)n1cc(C(=O)c2cncc(NC(=O)Cc3ncccn3)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)Cc3ccc(cn3)C#N)c2)c2cncnc12
Cn1cc(C(=O)c2cncc(NC(=O)Cc3cc(F)ccc3C(F)(F)F)c2)c2cncnc12
Cc1cccc(CC(=O)Nc2cncc(c2)C(=O)c2cn(C)c3ncncc23)c1
Cn1cc(C(=O)c2cncc(NC(=O)Cc3ccccc3C(F)(F)F)c2)c2cncnc12
Cn1cc(C(=O)c2cncc(NC(=O)Cc3cc(F)cc(F)c3)c2)c2cncnc12
Cn1cc(C(=O)c2cncc(NC(=O)Cc3c(F)cc(F)cc3F)c2)c2cncnc12
Cn1cc(C(=O)c2cncc(NC(=O)Cc3c(F)ccc(F)c3F)c2)c2cncnc12
Cn1cc(C(=O)c2cncc(NC(=O)Cc3ccc(cc3)S(C)(=O)=O)c2)c2cncnc12
Cn1cc(C(=O)c2cncc(NC(=O)Cc3ccc(c(F)c3)C(F)(F)F)c2)c2cncnc12
COc1cccc(CC(=O)Nc2cncc(c2)C(=O)c2cn(C)c3ncncc23)c1
Cn1cc(C(=O)c2cncc(NC(=O)Cc3cccc(OC(F)(F)F)c3)c2)c2cncnc12
Cn1cc(C(=O)c2cncc(NC(=O)Cc3cc(F)cc(F)c3F)c2)c2cncnc12
Cc1ccc2ccc(CC(=O)Nc3cncc(c3)C(=O)c3cn(C)c4ncncc34)cc2n1
Cn1cc(C(=O)c2cncc(NC(=O)Cc3ccccc3)c2)c2cncnc12
Cn1cc(C(=O)c2cncc(NC(=O)Cc3c(F)cccc3Cl)c2)c2cncnc12
COc1ccc(CC(=O)Nc2cncc(c2)C(=O)c2cn(C)c3ncncc23)cc1
Cn1cc(C(=O)c2cncc(NC(=O)Cc3ccc(SC(F)(F)F)cc3)c2)c2cncnc12
Cn1cc(C(=O)c2cncc(NC(=O)Cc3ccc(cc3)-c3ccccc3)c2)c2cncnc12
Cn1cc(C(=O)c2cncc(NC(=O)Cc3cc(F)c(F)cc3F)c2)c2cncnc12
Cn1cc(C(=O)c2cncc(NC(=O)Cc3cccc(SC(F)(F)F)c3)c2)c2cncnc12
Cc1ccc(CC(=O)Nc2cncc(c2)C(=O)c2cn(C)c3ncncc23)cc1
Cn1cc(C(=O)c2cncc(NC(=O)Cc3cc(F)c(F)c(F)c3)c2)c2cncnc12
Cc1ccc(CC(=O)Nc2cncc(c2)C(=O)c2cn(C)c3ncncc23)c(C)c1
Cn1cc(C(=O)c2cncc(NC(=O)Cc3ccc4OCCc4c3)c2)c2cncnc12
Cn1cc(C(=O)c2cncc(NC(=O)Cc3cc(F)ccc3F)c2)c2cncnc12
Cn1cc(C(=O)c2cncc(NC(=O)Cc3ccc(F)cc3F)c2)c2cncnc12
Cn1cc(C(=O)c2cncc(NC(=O)Cc3cccc(c3F)C(F)(F)F)c2)c2cncnc12
Cn1cc(C(=O)c2cncc(NC(=O)Cc3c(F)cccc3F)c2)c2cncnc12
Cn1cc(C(=O)c2cncc(NC(=O)Cc3cccc(c3)C(F)(F)F)c2)c2cncnc12
Cn1cc(C(=O)c2cncc(NC(=O)Cc3ccc(F)c(F)c3)c2)c2cncnc12
Cn1cc(C(=O)c2cncc(NC(=O)Cc3ccc(OC(F)(F)F)cc3)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)[C@@H](N)Cc3ccc(cc3)C(=O)c3ccccc3)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)Cc3cccc(c3)C(=O)c3ccccc3)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)Cc3ccc(cc3)C(=O)c3ccccc3)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)c3cccc(c3)C3(N=N3)C(F)(F)F)c2)c2cncnc12 |c:24|
CC(C)n1cc(C(=O)c2cncc(NC(=O)c3ccc(cc3)C3(N=N3)C(F)(F)F)c2)c2cncnc12 |c:24|
CC(C)n1cc(C(=O)c2cncc(NC(=O)c3cccc(c3)C(=O)C(F)(F)F)c2)c2cncnc12
Cn1cc(C(=O)c2cncc(NC(=O)Nc3ccc(Cl)cc3)c2)c2cncnc12
Cn1cc(C(=O)c2cncc(NC(=O)Nc3ccc(cc3)C(F)(F)F)c2)c2cncnc12
Cn1cc(C(=O)c2cncc(NC(=O)Nc3cccc(c3)C(F)(F)F)c2)c2cncnc12
Cn1cc(C(=O)c2cncc(NC(=O)Nc3ccc(OC(F)(F)F)cc3)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(c2)N(C)C(=O)Cc2ccc(Cl)cc2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(c2)N(C)C(=O)Cc2ccc(cc2)C#N)c2cncnc12
OCC1(COC1)n1cc(C(=O)c2cncc(NC(=O)Cc3ccc(Cl)cc3)c2)c2cncnc12
OCC1(COC1)n1cc(C(=O)c2cncc(NC(=O)Cc3ccc(cc3)C(F)(F)F)c2)c2cncnc12
OCC1(COC1)n1cc(C(=O)c2cncc(NC(=O)Cc3ccc(Cl)cn3)c2)c2cncnc12
OCC1(COC1)n1cc(C(=O)c2cncc(NC(=O)Cn3ccc(n3)C(F)(F)F)c2)c2cncnc12
NC(=O)Cn1cc(C(=O)c2cncc(NC(=O)Cc3ccc(Cl)cc3)c2)c2cncnc12
CN(C)C(=O)Cn1cc(C(=O)c2cncc(NC(=O)Cc3ccc(Cl)cc3)c2)c2cncnc12
CNC(=O)Cn1cc(C(=O)c2cncc(NC(=O)Cc3ccc(Cl)cc3)c2)c2cncnc12
Clc1ccc(CC(=O)Nc2cncc(c2)C(=O)c2c[nH]c3ncncc23)cc1
CC1(COC1)n1cc(C(=O)c2cncc(NC(=O)Cc3ccc(Cl)cc3)c2)c2cncnc12
CC1(COC1)n1cc(C(=O)c2cncc(NC(=O)Cc3ccc(Cl)cn3)c2)c2cncnc12
CC1(COC1)n1cc(C(=O)c2cncc(NC(=O)Cn3ccc(n3)C(F)(F)F)c2)c2cncnc12
CC1(COC1)n1cc(C(=O)c2cncc(NC(=O)Cn3cc(nn3)C(F)(F)F)c2)c2cncnc12
CS(=O)(=O)Cn1cc(C(=O)c2cncc(NC(=O)Cc3ccc(Cl)cc3)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)Cc3cnn(C4CC4)c3C(F)(F)F)c2)c2cncnc12
Cn1cc(C(=O)c2cncc(NC(=O)Cc3ccc(Cl)cc3)c2)c2cncnc12
Cn1cc(C(=O)c2cncc(NC(=O)CCc3ccc(Cl)cc3)c2)c2cncnc12
Cc1cccc(CCC(=O)Nc2cncc(c2)C(=O)c2cn(C)c3ncncc23)c1
Cn1cc(C(=O)c2cncc(NC(=O)CCc3cccnc3)c2)c2cncnc12
Cn1cc(C(=O)c2cncc(NC(=O)CCc3cccc(Cl)c3)c2)c2cncnc12
Cn1cc(C(=O)c2cncc(NC(=O)CCc3cccc(F)c3)c2)c2cncnc12
Cn1cc(C(=O)c2cncc(NC(=O)COc3ccccc3OC(F)(F)F)c2)c2cncnc12
Cc1ccccc1CCC(=O)Nc1cncc(c1)C(=O)c1cn(C)c2ncncc12
Cn1cc(C(=O)c2cncc(NC(=O)CCc3ccccc3F)c2)c2cncnc12
Cn1cc(C(=O)c2cncc(NC(=O)CCc3ccc(F)cc3)c2)c2cncnc12
Cn1cc(C(=O)c2cncc(NC(=O)CCc3ccccc3)c2)c2cncnc12
Cc1ccc(CCC(=O)Nc2cncc(c2)C(=O)c2cn(C)c3ncncc23)cc1
Cn1cc(C(=O)c2cncc(NC(=O)Cc3ccc(NS(=O)(=O)C(F)(F)F)cc3)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)c3cnnc4ccccc34)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)c3ccn4ncnc4c3)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)c3cc4ncccn4n3)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)c3ccccn3)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)c3cncc(Cl)c3)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)c3cc4occc4[nH]3)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)c3ccn4ccnc4c3)c2)c2cncnc12
CCn1cc(cn1)C(=O)Nc1cncc(c1)C(=O)c1cn(C(C)C)c2ncncc12
CC(C)n1cnc(c1)C(=O)Nc1cncc(c1)C(=O)c1cn(C(C)C)c2ncncc12
COc1nc(cn2ccnc12)C(=O)Nc1cncc(c1)C(=O)c1cn(C(C)C)c2ncncc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)c3cnc4[nH]ccc4c3)c2)c2cncnc12
CCCc1cc(C(=O)Nc2cncc(c2)C(=O)c2cn(C(C)C)c3ncncc23)n(C)n1
CC(C)c1csc(n1)C(=O)Nc1cncc(c1)C(=O)c1cn(C(C)C)c2ncncc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)c3cc4c(C)coc4cn3)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)c3cccc(C)n3)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)c3c(Cl)n(C)nc3C(F)(F)F)c2)c2cncnc12
COc1ccc2[nH]c(nc2c1)C(=O)Nc1cncc(c1)C(=O)c1cn(C(C)C)c2ncncc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)c3nn(C)c(C)c3Cl)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)c3nccc4[nH]ccc34)c2)c2cncnc12
CCc1ccnc(c1)C(=O)Nc1cncc(c1)C(=O)c1cn(C(C)C)c2ncncc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)c3cnc4OCCOc4c3)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)c3ccc4[nH]ccc4n3)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)c3ccn4nccc4c3)c2)c2cncnc12
COc1ccc2ncc(cc2c1)C(=O)Nc1cncc(c1)C(=O)c1cn(C(C)C)c2ncncc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)c3cc(C)nn3CC(F)(F)F)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)c3cnccc3C(F)(F)F)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)c3cnn(CCC#N)c3)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)c3cc4cnccc4o3)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)c3cc4cnccc4[nH]3)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)c3cc4occc4cn3)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)c3oc(C)nc3C)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)c3cn(C)c4cnccc34)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)c3cc4CCCn4n3)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)c3csc(n3)C3CCC3)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)c3ccncc3F)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)c3c(C)nc4ncccn34)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)c3cc(C)on3)c2)c2cncnc12
COc1cc(OC)nc(n1)C(=O)Nc1cncc(c1)C(=O)c1cn(C(C)C)c2ncncc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)c3cncc(C)n3)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)c3cn(C)cn3)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)c3ccc(Cl)cn3)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)c3ccc4cccnc4n3)c2)c2cncnc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)c3nccn3C)c2)c2cncnc12
COCc1cc(no1)C(=O)Nc1cncc(c1)C(=O)c1cn(C(C)C)c2ncncc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)c3nncc4ccccc34)c2)c2cncnc12
CC(C)(CO)n1cc(C(=O)c2cncc(NC(=O)Cc3ccc(cn3)C(F)(F)F)c2)c2cnc(N)nc12
CC(C)(CO)n1cc(C(=O)c2cncc(NC(=O)Cn3cc(cn3)C(F)(F)F)c2)c2cnc(N)nc12
CC(C)(CO)n1cc(C(=O)c2cncc(NC(=O)Cc3ccc(NS(C)(=O)=O)cc3)c2)c2cnc(N)nc12
CC(C)(CO)n1cc(C(=O)c2cncc(NC(=O)Cc3ccc(OC(F)F)cc3)c2)c2cnc(N)nc12
CC(C)(CO)n1cc(C(=O)c2cncc(NC(=O)Cc3ccc(OC(F)(F)F)cc3)c2)c2cnc(N)nc12
CC(C)(CO)n1cc(C(=O)c2cncc(NC(=O)Cc3ccc(F)c(F)c3)c2)c2cnc(N)nc12
CC(C)(CO)n1cc(C(=O)c2cncc(NC(=O)Cc3ncc(Cl)cn3)c2)c2cnc(N)nc12
O=C(Cc1ccc(cc1)C#N)Nc1cncc(c1)C(=O)c1c[nH]c2ncncc12
CC1(COC1)n1cc(C(=O)c2cncc(NC(=O)Cc3ccc(cc3)C(F)(F)F)c2)c2cncnc12
CC1(COC1)n1cc(C(=O)c2cncc(NC(=O)Cc3cccc(c3)C(F)(F)F)c2)c2cncnc12
CC1(COC1)n1cc(C(=O)c2cncc(NC(=O)Cc3ccc(c(F)c3)C(F)(F)F)c2)c2cncnc12
CC1(COC1)n1cc(C(=O)c2cncc(NC(=O)c3cccc(c3)C(F)(F)F)c2)c2cncnc12
CC1(COC1)n1cc(C(=O)c2cncc(NC(=O)c3cccc(OC(F)(F)F)c3)c2)c2cncnc12
CC(C)(CO)n1cc(C(=O)c2cncc(NC(=O)Cn3cc(cn3)C3CC3)c2)c2cnc(N)nc12
CC(C)(C)n1cc(C(=O)c2cncc(NC(=O)Cn3cc(cn3)C3CC3)c2)c2cnc(N)nc12
Nc1ncc2c(cn(c2n1)C12CC(C1)C2)C(=O)c1cncc(NC(=O)Cc2ccc(F)cn2)c1
CC(C)n1cc(C(=O)c2c[nH]c(=O)c(NC(=O)Cc3ccc(cc3)C#N)c2)c2cncnc12
CC(C)n1cc(C(=O)c2c[nH]c(=O)c(NC(=O)COc3ccccc3OC(F)(F)F)c2)c2cncnc12
CC(C)n1cc(C(=O)c2c[nH]c(=O)c(NC(=O)Cc3coc(n3)C3CC3)c2)c2cncnc12
CC(C)n1cc(C(=O)c2c[nH]c(=O)c(NC(=O)Cn3nc(cc3C)C(F)(F)F)c2)c2cncnc12
CC(C)n1cc(C(=O)c2c[nH]c(=O)c(NC(=O)Cc3ccc4cccnc4c3)c2)c2cncnc12
CC(C)n1cc(C(=O)c2c[nH]c(=O)c(NC(=O)Cc3ccc(Cl)cc3)c2)c2cncnc12
CC(C)n1cc(C(=O)c2c[nH]c(=O)c(NC(=O)Cc3ccc(Cl)cn3)c2)c2cncnc12
CC(C)n1cc(C(=O)c2c[nH]c(=O)c(NC(=O)Cn3cc(nn3)C(F)(F)F)c2)c2cncnc12
OC1CN(C1)C(=O)Nc1cnn2ccc(nc12)N1CCC[C@@H]1c1cc(F)ccc1F |r|
CN(C)C(=O)Nc1cnn2ccc(nc12)N1CCC[C@@H]1c1cc(F)ccc1F |r|
CC(C)(C)NC(=O)Nc1cnn2ccc(nc12)N1CCC[C@@H]1c1cc(F)ccc1F |r|
Fc1ccc(F)c(c1)[C@H]1CCCN1c1ccn2ncc(NC(=O)Nc3ccccc3)c2n1 |r|
CC(C)C(=O)Nc1cnn2ccc(nc12)N1CCC[C@@H]1c1cc(F)ccc1F |r|
Cn1nc(ccc1=O)C(=O)Nc1cnn2ccc(nc12)N1CCC[C@@H]1c1cccc(F)c1 |r|
OC1CN(C1)C(=O)Nc1cnn2ccc(nc12)N1CC(F)(F)C[C@@H]1c1cccc(F)c1 |r|
OC1CN(C1)C(=O)Nc1cnn2ccc(nc12)N1CCC[C@@H]1c1cc(F)ccc1Cl |r|
Fc1cccc(c1)[C@H]1CCCN1c1ccn2ncc(NC(=O)N3CCOCC3)c2n1 |r|
CC1(CCCN1c1ccn2ncc(NC(=O)N3CC(O)C3)c2n1)c1cccc(F)c1
OC1CN(C1)C(=O)Nc1cnn2ccc(nc12)N1CCC[C@@H]1c1cc(F)cc(Cl)c1 |r|
OC1CN(C1)C(=O)Nc1cnn2ccc(nc12)N1CCC[C@@H]1c1cc(F)ccc1C(F)F |r|
Fc1ccc(F)c(c1)[C@H]1CCCN1c1ccn2ncc(NC(=O)N3CCOCC3)c2n1 |r|
O[C@H]1CCN(C1)C(=O)Nc1cnn2ccc(nc12)N1CCC[C@@H]1c1cc(F)ccc1F |r|
O[C@@H]1CN(C[C@H]1O)C(=O)Nc1cnn2ccc(nc12)N1CCC[C@@H]1c1cc(F)ccc1F |r|
COC1CN(C1)C(=O)Nc1cnn2ccc(nc12)N1CCC[C@@H]1c1cc(F)ccc1F |r|
CC1(O)CN(C1)C(=O)Nc1cnn2ccc(nc12)N1CCC[C@@H]1c1cc(F)ccc1F |r|
Fc1ccc(NC(=O)Nc2cnn3ccc(nc23)N2CCC[C@@H]2c2cc(F)ccc2F)cc1 |r|
Fc1ccc(F)c(c1)[C@H]1CCCN1c1ccn2ncc(NC(=O)Nc3ccc(Cl)cc3)c2n1 |r|
COc1ccc(NC(=O)Nc2cnn3ccc(nc23)N2CCC[C@@H]2c2cc(F)ccc2F)cc1 |r|
COC1CN(C1)C(=O)Nc1cnn2ccc(nc12)N1CCC[C@@H]1c1cc(F)ccc1Cl |r|
CC1(O)CN(C1)C(=O)Nc1cnn2ccc(nc12)N1CCC[C@@H]1c1cc(F)ccc1Cl |r|
Fc1ccc(Cl)c(c1)[C@H]1CCCN1c1ccn2ncc(NC(=O)N3CCOCC3)c2n1 |r|
C[C@H]1CN(CCN1C(=O)OC(C)(C)C)C(=O)Nc1cnn2ccc(nc12)N1CCC[C@@H]1c1cc(F)ccc1Cl |r|
C[C@H]1CN(CCN1)C(=O)Nc1cnn2ccc(nc12)N1CCC[C@@H]1c1cc(F)ccc1Cl |r|
CC(C)N1CCN(CC1)C(=O)Nc1cnn2ccc(nc12)N1CCC[C@@H]1c1cc(F)ccc1F |r|
CCN1CCN(CC1)C(=O)Nc1cnn2ccc(nc12)N1CCC[C@@H]1c1cc(F)ccc1F |r|
CN1CCN(CC1)C(=O)Nc1cnn2ccc(nc12)N1CCC[C@@H]1c1cc(F)ccc1F |r|
CC1CN(CC(C)N1)C(=O)Nc1cnn2ccc(nc12)N1CCC[C@@H]1c1cc(F)ccc1F |r|
C[C@H]1CN(CCN1C(=O)OC(C)(C)C)C(=O)Nc1cnn2ccc(nc12)N1CCC[C@@H]1c1cc(F)ccc1F |r|
C[C@H]1CN(CCN1)C(=O)Nc1cnn2ccc(nc12)N1CCC[C@@H]1c1cc(F)ccc1F |r|
OC1CN(C1)C(=O)Nc1cnn2ccc(nc12)N1CCC[C@@H]1c1cccc(F)c1 |r|
COC(=O)C1(CC1)C(=O)Nc1cnn2ccc(nc12)N1CCC[C@@H]1c1cc(F)ccc1F |r|
OC(=O)C1(CC1)C(=O)Nc1cnn2ccc(nc12)N1CCC[C@@H]1c1cc(F)ccc1F |r|
O[C@H]1CCN(C1)C(=O)Nc1cnn2ccc(nc12)N1CCC[C@@H]1c1cc(F)cc(Cl)c1 |r|
O[C@@H]1CCN(C1)C(=O)Nc1cnn2ccc(nc12)N1CCC[C@@H]1c1cc(F)ccc1C(F)F |r|
O[C@H]1CCN(C1)C(=O)Nc1cnn2ccc(nc12)N1CCC[C@@H]1c1cc(F)ccc1C(F)F |r|
OC1CCN(CC1)C(=O)Nc1cnn2ccc(nc12)N1CCC[C@@H]1c1cc(F)ccc1C(F)F |r|
O[C@@H]1CCCN(C1)C(=O)Nc1cnn2ccc(nc12)N1CCC[C@@H]1c1cc(F)ccc1C(F)F |r|
O[C@H]1CCCN(C1)C(=O)Nc1cnn2ccc(nc12)N1CCC[C@@H]1c1cc(F)ccc1C(F)F |r|
O[C@@H]1CCN(C1)C(=O)Nc1cnn2ccc(nc12)N1CCC[C@@H]1c1cc(F)ccc1Cl |r|
OC1CCN(CC1)C(=O)Nc1cnn2ccc(nc12)N1CCC[C@@H]1c1cc(F)ccc1Cl |r|
O[C@@H]1CCCN(C1)C(=O)Nc1cnn2ccc(nc12)N1CCC[C@@H]1c1cc(F)ccc1Cl |r|
O[C@H]1CCCN(C1)C(=O)Nc1cnn2ccc(nc12)N1CCC[C@@H]1c1cc(F)ccc1Cl |r|
CC(C)(C)C(=O)Nc1cnn2ccc(nc12)N1CCC[C@@H]1c1cc(F)ccc1F |r|
CC(C)(C)OC(=O)N1CC(C1)C(=O)Nc1cnn2ccc(nc12)N1CCC[C@@H]1c1cc(F)ccc1Cl |r|
Fc1ccc(Cl)c(c1)[C@H]1CCCN1c1ccn2ncc(NC(=O)C3CNC3)c2n1 |r|
CC(C)(C)OC(=O)N1CCC(C)(CC1)C(=O)Nc1cnn2ccc(nc12)N1CCC[C@@H]1c1cc(F)ccc1Cl |r|
CC1(CCNCC1)C(=O)Nc1cnn2ccc(nc12)N1CCC[C@@H]1c1cc(F)ccc1Cl |r|
CC(C)(O)C(=O)Nc1cnn2ccc(nc12)N1CCC[C@@H]1c1cc(F)ccc1F |r|
Fc1ccc(F)c(c1)[C@H]1CCCN1c1ccn2ncc(NC(=O)C3(CC3)C(F)(F)F)c2n1 |r|
Fc1ccc(F)c(c1)[C@H]1CCCN1c1ccn2ncc(NC(=O)C3(CC3)C#N)c2n1 |r|
C[C@@]1(CCCN1)C(=O)Nc1cnn2ccc(nc12)N1CCC[C@@H]1c1cc(F)ccc1F |r|
CC(C)(F)C(=O)Nc1cnn2ccc(nc12)N1CCC[C@@H]1c1cc(F)ccc1F |r|
CC(C)Nc1nc(cs1)C(=O)Nc1cnn2ccc(nc12)N1CCC[C@@H]1c1cc(F)ccc1F |r|
CC(C)(C(=O)Nc1cnn2ccc(nc12)N1CCC[C@@H]1c1cc(F)ccc1F)n1cncn1 |r|
Fc1ccc(F)c(c1)[C@H]1CCCN1c1ccn2ncc(NC(=O)c3cnccn3)c2n1 |r|
Cc1cnc(cn1)C(=O)Nc1cnn2ccc(nc12)N1CCC[C@@H]1c1cc(F)ccc1F |r|
Fc1ccc(F)c(c1)[C@H]1CCCN1c1ccn2ncc(NC(=O)c3ccccn3)c2n1 |r|
Cc1cccc(n1)C(=O)Nc1cnn2ccc(nc12)N1CCC[C@@H]1c1cc(F)ccc1F |r|
Fc1ccc(F)c(c1)[C@H]1CCCN1c1ccn2ncc(NC(=O)c3ccc(Cl)cn3)c2n1 |r|
Fc1ccc(F)c(c1)[C@H]1CCCN1c1ccn2ncc(NC(=O)c3cc(Cl)ccn3)c2n1 |r|
Cc1cccnc1C(=O)Nc1cnn2ccc(nc12)N1CCC[C@@H]1c1cc(F)ccc1F |r|
CC(C)(CO)C(=O)Nc1cnn2ccc(nc12)N1CCC[C@@H]1c1cc(F)ccc1F |r|
OC1(CC1)C(=O)Nc1cnn2ccc(nc12)N1CCC[C@@H]1c1cc(F)ccc1F |r|
CNC(C)(C)C(=O)Nc1cnn2ccc(nc12)N1CCC[C@@H]1c1cc(F)ccc1F |r|
Fc1ccc(F)c(c1)[C@H]1CCCN1c1ccn2ncc(NC(=O)c3ncccn3)c2n1 |r|
Fc1cccc(c1)[C@H]1CCCN1c1ccn2ncc(NC(=O)c3ccccn3)c2n1 |r|
Cc1cccnc1C(=O)Nc1cnn2ccc(nc12)N1CCC[C@@H]1c1cccc(F)c1 |r|
Cn1ccc(cc1=O)C(=O)Nc1cnn2ccc(nc12)N1CCC[C@@H]1c1cccc(F)c1 |r|
Fc1ccc(F)c(c1)[C@H]1CCCN1c1ccn2ncc(NC(=O)c3cccc(Cl)n3)c2n1 |r|
CCS(=O)(=O)Nc1ccc(cc1)C(=O)Nc1cnn2ccc(nc12)N1CCC[C@@H]1c1cccc(F)c1 |r|
Cn1ccc(n1)C(=O)Nc1cnn2ccc(nc12)N1CCC[C@@H]1c1cccc(F)c1 |r|
Fc1cccc(c1)[C@H]1CCCN1c1ccn2ncc(NC(=O)c3cc[nH]n3)c2n1 |r|
COc1cccc(n1)C(=O)Nc1cnn2ccc(nc12)N1CCC[C@@H]1c1cccc(F)c1 |r|
Fc1cccc(c1)[C@H]1CCCN1c1ccn2ncc(NC(=O)c3cccnc3)c2n1 |r|
Fc1cccc(c1)[C@H]1CCCN1c1ccn2ncc(NC(=O)c3ccncc3)c2n1 |r|
Cc1ccc(cn1)C(=O)Nc1cnn2ccc(nc12)N1CCC[C@@H]1c1cccc(F)c1 |r|
COc1ncccc1C(=O)Nc1cnn2ccc(nc12)N1CCC[C@@H]1c1cccc(F)c1 |r|
Cc1cnccc1C(=O)Nc1cnn2ccc(nc12)N1CCC[C@@H]1c1cccc(F)c1 |r|
O[C@H]1CCN(C1)C(=O)Nc1cnn2ccc(nc12)N1CCC[C@@H]1c1cc(F)ccc1Cl |r|
Cc1cnc(cn1)C(=O)Nc1cnn2ccc(nc12)N1CCC[C@@H]1c1cccc(F)c1 |r|
Cn1ccnc1C(=O)Nc1cnn2ccc(nc12)N1CCC[C@@H]1c1cccc(F)c1 |r|
O[C@H]1CCN(C1)C(=O)Nc1cnn2ccc(nc12)N1CCC[C@@H]1c1cc(F)ccc1C(F)(F)F |r|
O[C@@H]1CCN(C1)C(=O)Nc1cnn2ccc(nc12)N1CCC[C@@H]1c1cc(F)ccc1C(F)(F)F |r|
O[C@@H]1CCCN(C1)C(=O)Nc1cnn2ccc(nc12)N1CCC[C@@H]1c1cc(F)ccc1C(F)(F)F |r|
O[C@H]1CCCN(C1)C(=O)Nc1cnn2ccc(nc12)N1CCC[C@@H]1c1cc(F)ccc1C(F)(F)F |r|
O[C@H]1CCN(C1)C(=O)Nc1cnn2ccc(nc12)N1CCC[C@@H]1c1cncc(F)c1 |r|
O[C@@H]1CCN(C1)C(=O)Nc1cnn2ccc(nc12)N1CCC[C@@H]1c1cncc(F)c1 |r|
COc1ccc(F)cc1[C@H]1CCCN1c1ccn2ncc(NC(=O)N3CC[C@H](O)C3)c2n1 |r|
COc1ccc(F)cc1[C@H]1CCCN1c1ccn2ncc(NC(=O)N3CCC[C@H](O)C3)c2n1 |r|
Fc1ccc(F)c(c1)[C@H]1CCCN1c1ccn2ncc(NC(=O)N3C[C@@H]4C[C@H]3CO4)c2n1 |r,THB:21:23:28.29:26|
O[C@@H]1CCN(C1)C(=O)Nc1cnn2ccc(nc12)N1CCC[C@@H]1c1cc(F)ccc1F |r|
O[C@@H]1CC[C@@H](C1)C(=O)Nc1cnn2ccc(nc12)N1CCC[C@@H]1c1cc(F)ccc1F |r|
O[C@H]1CC[C@@H](C1)C(=O)Nc1cnn2ccc(nc12)N1CCC[C@@H]1c1cc(F)ccc1F |r|
OC1CC(C1)C(=O)Nc1cnn2ccc(nc12)N1CCC[C@@H]1c1cc(F)ccc1F |r,wU:21.25,(5.36,-4.88,;4.96,-3.39,;3.62,-2.62,;4.39,-1.28,;5.73,-2.05,;3.99,.2,;5.08,1.29,;2.51,.6,;2.11,2.09,;3.01,3.34,;2.11,4.58,;.64,4.11,;-.69,4.88,;-2.02,4.11,;-2.02,2.57,;-.69,1.8,;.64,2.57,;-3.36,1.8,;-4.82,2.27,;-5.73,1.03,;-4.82,-.22,;-3.36,.26,;-2.27,-.83,;-.78,-.43,;.31,-1.52,;1.8,-1.13,;-.09,-3.01,;-1.58,-3.41,;-2.67,-2.32,;-4.15,-2.72,)|
CN(C)C(=O)C(=O)Nc1cnn2ccc(nc12)N1CCC[C@@H]1c1cc(F)ccc1F |r|
CNC(=O)C(=O)Nc1cnn2ccc(nc12)N1CCC[C@@H]1c1cc(F)ccc1F |r|
NC(=O)C(=O)Nc1cnn2ccc(nc12)N1CCC[C@@H]1c1cc(F)ccc1F |r|
Fc1ccc(F)c(c1)[C@H]1CCCN1c1ccn2ncc(NC(=O)C(=O)NC3CC3)c2n1 |r|
OC1CN(C1)C(=O)C(=O)Nc1cnn2ccc(nc12)N1CCC[C@@H]1c1cc(F)ccc1F |r|
O[C@H]1CCN(C1)C(=O)C(=O)Nc1cnn2ccc(nc12)N1CCC[C@@H]1c1cc(F)ccc1F |r|
Fc1ccc(F)c(c1)[C@H]1CCCN1c1ccn2ncc(NC(=O)C(=O)N3CCOCC3)c2n1 |r|
COC(=O)C(=O)Nc1cnn2ccc(nc12)N1CCC[C@@H]1c1cc(F)ccc1F |r|
OC(=O)C(=O)Nc1cnn2ccc(nc12)N1CCC[C@@H]1c1cc(F)ccc1F |r|
CC(CO)n1cc(C(=O)c2cncc(NC(=O)Cc3ccc(cc3)C#N)c2)c2cnccc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)Cc3cccc(CC(C)(C)O)c3)c2)c2cnccc12
CC(C)c1cc(C)n(CC(=O)Nc2cncc(c2)C(=O)c2cn(C(C)C)c3ccncc23)n1
CC(C)n1cc(C(=O)c2cncc(NC(=O)Cn3nc(cc3C)C(F)(F)F)c2)c2cnccc12
CC(C)c1cn(CC(=O)Nc2cncc(c2)C(=O)c2cn(C(C)C)c3ccncc23)nn1
CC(C)c1ccnn1CC(=O)Nc1cncc(c1)C(=O)c1cn(C(C)C)c2ccncc12
CC(C)n1cc(C(=O)c2ccnc(NC(=O)Cc3ccc(c(F)c3)C(F)(F)F)c2)c2cnccc12
COCc1cn(CC(=O)Nc2cncc(c2)C(=O)c2cn(C(C)C)c3ccncc23)nn1
CC(C)n1cc(C(=O)c2cncc(NC(=O)Cc3nnn[nH]3)c2)c2cnccc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)Cn3cc(nn3)C(C)(C)O)c2)c2cnccc12
COc1ccc(COc2ccc(Cn3c(N)nc4cc(ccc34)-c3cnn(C)c3)cc2OC)cc1
COc1ccc(COc2ccc(Cn3c(N)nc4cc(ccc34)-c3cncnc3)cc2OC)cc1
COc1ccc(COc2ccc(Cn3c(N)nc4cc(ccc34)-c3ccncc3)cc2OC)cc1
COc1ccc(COc2ccc(Cn3c(N)nc4cc(ccc34)-c3cnn(CCN4CCOCC4)c3)cc2OC)cc1
COc1ccc(COc2ccc(Cn3c(N)nc4cc(ccc34)-c3ccc(nc3)P(C)(C)=O)cc2OC)cc1
COc1ccc(COc2ccc(Cn3cnc4cc(ccc34)-c3ccnnc3)cc2OC)cn1
COc1ccc(COc2ccc(Cn3cnc4cc(ccc34)-c3cnn(c3)C3CCNCC3)cc2OC)cn1
COc1ccc(COc2ccc(Cn3cnc4cc(ccc34)-n3cc(nn3)C3CCCNC3)cc2OC)cn1
COc1ccc(COc2ccc(Cn3cnc4cc(ccc34)-c3nnc(o3)C3CCCNC3)cc2OC)cn1
COc1ccc(COc2ccc(Cn3cnc4cc(ccc34)C3CCNCC3)cc2OC)cn1
COc1ccc(COc2ccc(Cn3cnc4cc(ccc34)C3CCOCC3)cc2OC)cn1
COc1ccc(COc2ccc(Cn3cnc4cc(ccc34)N3CCC(CC3)C(C)(C)N)cc2OC)cn1
COc1ccc(COc2ccc(Cn3cnc4cc(ccc34)N3CC4(C3)CCNCC4)cc2OC)cn1
COc1ccc(COc2ccc(Cn3cnc4cc(ccc34)N3CCC(N)CC3)cc2OC)cn1
COc1ccc(COc2ccc(Cn3cnc4cc(ccc34)N3CCN(C)CC3)cc2OC)cn1
COc1ccc(COc2ccc(Cn3c(N)nc4cc(ccc34)N3CCN(C)CC3=O)cc2OC)cn1
COc1ccc(COc2ccc(Cn3c(N)nc4cc(cnc34)-c3cnn(C)c3)cc2OC)cc1
COc1ccc(COc2ccc(Cn3c(N)nc4cc(cnc34)-c3ccc(nc3)P(C)(C)=O)cc2OC)cc1
COc1ccc(COc2ccc(Cn3cnc4cc(cnc34)N3CCN(C)CC3)cc2OC)cn1
COc1ccc(COc2ccc(Cn3cnc4cc(cnc34)N3CCC(CC3)C(C)(C)N)cc2OC)cn1
COc1ccc(COc2ccc(Cn3cnc4cc(cnc34)N3CCOCC3)cc2OC)cn1
COc1ccc(COc2ccc(Cn3cnc4cc(cnc34)N3CCN(CC3)C3CC3)cc2OC)cn1
COc1ccc(COc2ccc(Cn3cnc4cc(cnc34)N3CCN4CCC3CC4)cc2OC)cn1 |(-1.02,-9.85,;-1.79,-8.52,;-1.02,-7.18,;-1.79,-5.85,;-1.02,-4.52,;.52,-4.52,;1.61,-3.43,;1.21,-1.94,;2.3,-.85,;1.53,.48,;2.3,1.82,;3.84,1.82,;4.61,3.15,;3.84,4.48,;4.75,5.73,;3.84,6.97,;2.38,6.5,;1.04,7.27,;-.29,6.5,;-.29,4.96,;1.04,4.19,;2.38,4.96,;-1.62,7.27,;-2.9,6.4,;-4.37,6.86,;-4.93,8.29,;-4.16,9.62,;-2.64,9.85,;-1.51,8.8,;-2.53,9.45,;-3.25,8.29,;4.61,.48,;3.84,-.85,;4.93,-1.94,;4.53,-3.43,;1.29,-5.85,;.52,-7.18,)|
COc1ccc(COc2ccc(Cn3cnc4cc(cnc34)N3CC4(C3)CCNCC4)cc2OC)cn1
COc1ccc(COc2ccc(Cn3cnc4cc(cnc34)N3CCC(N)CC3)cc2OC)cn1
COc1ccc(COc2ccc(Cn3cnc4cc(cnc34)N3CCC[C@H]3C(O)=O)cc2OC)cn1 |r|
COc1ccc(COc2ccc(Cn3cnc4cc(cnc34)-c3cnn(c3)C3CCNCC3)cc2OC)cn1
COc1cc(Cn2cnc3cc(cnc23)-c2cnn(c2)C2CCNCC2)ccc1OCc1ccc(C)nc1
COc1ccc(COc2ccc(Cn3cnc4cc(cnc34)-c3noc(n3)C3CCNCC3)cc2OC)cn1
COc1ccc(COc2ccc(Cn3cnc4cc(ccc34)-c3noc(n3)C3CCNCC3)cc2OC)cn1
COc1ccc(COc2ccc(Cn3cnc4cc(cnc34)-c3nnc(o3)C3CCNCC3)cc2OC)cn1
COc1ccc(COc2ccc(Cn3cnc4cc(cnc34)-n3cc(nn3)C(C)(C)N)cc2OC)cn1
COc1ccc(COc2ccc(Cn3cnc4cc(cnc34)-n3cc(nn3)C3CCCNC3)cc2OC)cn1
COc1ccc(COc2ccc(Cn3c(N)nc4cc(ccc34)N3CCN(C)CC3)cc2OC)cn1
COc1ccc(COc2cc(F)c(Cn3cnc4cc(ccc34)N3CCN(C)CC3)cc2OC)cn1
COc1ccc(COc2ccc(Cn3cnc4cc(ccc34)N3CCN(C)CC3=O)cc2OC)cn1
COc1ccc(COc2ccc(Cn3cnc4cc(cnc34)C3=CC4(C)CN3CCC4)cc2OC)cn1 |t:24|
COc1ccc(COc2ccc(Cn3cnc4cc(ccc34)C3=CC4(C)CN3CCC4)cc2OC)cn1 |t:24|
COc1ccc(COc2ccc(Cn3cnc4cc(cnc34)C3=CC4(O)CN3CCC4)cc2OC)cn1 |t:24|
COc1ccc(COc2ccc(Cn3cnc4cc(ccc34)C3=CC4(O)CN3CCC4)cc2OC)cn1 |t:24|
CCC(Oc1ccc(Cn2c(N)nc3cc(cnc23)-c2cnn(C)c2)cc1OC)c1ccc(OC)nc1
COc1ccc(COc2ccc(Cn3c(N)nc4cc(cnc34)-c3cnn(C)c3)cc2OC)cn1
COc1cc(Cn2c(N)nc3cc(cnc23)-c2cnn(C)c2)ccc1OCc1ccc(nc1)C(F)(F)F
COc1cc(Cn2c(N)nc3cc(cnc23)-c2cnn(C)c2)ccc1OCc1ccc(cc1)C(F)(F)F
COc1cc(Cn2c(N)nc3cc(cnc23)-c2cnn(C)c2)ccc1OCc1ccc(nc1)C1CC1
COc1cc(Cn2c(N)nc3cc(cnc23)-c2cnn(C)c2)ccc1OCc1csc(C)n1
COc1ccc(COc2ccc(Cn3c(N)nc4cc(cnc34)-c3ccccc3)cc2OC)cn1
COc1ccc(COc2ccc(Cn3c(N)nc4cc(cnc34)-c3ccc(F)cc3)cc2OC)cn1
COc1ccc(COc2ccc(Cn3c(N)nc4cc(cnc34)-c3ccn(C)n3)cc2OC)cn1
COc1ccc(COc2ccc(Cn3c(N)nc4cc(cnc34)-c3cncnc3)cc2OC)cn1
COc1ccc(COc2ccc(Cn3c(N)nc4cc(cnc34)-c3c(C)nn(C)c3C)cc2OC)cn1
COc1ccc(COc2ccc(Cn3c(N)nc4cc(cnc34)-c3ccncc3)cc2OC)cn1
COc1ccc(COc2ccc(Cn3c(N)nc4cc(cnc34)-c3cccnc3)cc2OC)cn1
COc1ccc(COc2ccc(Cn3c(N)nc4cc(cnc34)-c3ccccn3)cc2OC)cn1
COc1cc(Cn2c(N)nc3cc(cnc23)-c2cnn(C)c2)ccc1OCc1ccc(cc1)C(F)(F)C(F)(F)F
COc1cc(Cn2c(N)nc3cc(cnc23)-c2cnn(C)c2)ccc1OCc1ccc(OC(F)(F)F)cc1
COc1cc(Cn2c(N)nc3cc(cnc23)-c2cnn(C)c2)ccc1OCc1ccc(SC(F)(F)F)cc1
COc1cc(Cn2c(N)nc3cc(cnc23)-c2cnn(C)c2)ccc1OCc1ccc(nc1)C(C)C
COc1cc(Cn2c(N)nc3cc(cnc23)-c2cnn(C)c2)ccc1OCc1ccc(CC(F)(F)F)cc1
COc1cc(Cn2c(N)nc3cc(cnc23)-c2cnn(C)c2)ccc1OCc1csc(n1)C(F)(F)F
COc1ccc(COc2ccc(Cn3c(N)nc4cc(cnc34)C#CC3CCCCC3)cc2OC)cn1
COc1ccc(COc2ccc(Cn3c(N)nc4cc(cnc34)C#CCCO)cc2OC)cn1
COc1ccc(cn1)C(Oc1ccc(Cn2c(N)nc3cc(cnc23)-c2cnn(C)c2)cc1OC)C1CC1
COc1cc2CCCC(Oc3ccc(Cn4c(N)nc5cc(cnc45)-c4cnn(C)c4)cc3OC)c2cn1
COc1ccc(COc2ccc(cc2OC)C(C)n2c(N)nc3cc(ccc23)-c2cnn(C)c2)cn1
COc1ccc(COc2ccc(cc2OC)C(C)n2c(N)nc3cc(ccc23)-c2ccc(F)cc2)cn1
COc1cc(ccc1OCc1ccc(nc1)C(F)(F)F)C(C)n1cnc2cc(ccc12)-c1ccc(F)cc1
COc1cc(ccc1OCc1ccc(nc1)C(F)(F)F)C(C)n1cnc2cc(ccc12)-c1cnn(C)c1
COc1cc(ccc1OCc1ccc(nc1)C(F)(F)F)C(C)n1cnc2cc(ccc12)C#CCCO
COc1cc(ccc1OCc1ccc(cc1)C(F)(F)F)[C@H](C)n1c(N)nc2cc(cnc12)-c1cnn(C)c1 |r|
COc1cc(ccc1OCc1ccc(cc1)C(F)(F)F)[C@@H](C)n1c(N)nc2cc(cnc12)-c1cnn(C)c1 |r|
COc1cc(ccc1OCc1ccc(nc1)C(F)(F)F)C(C)n1cnc2cc(cnc12)-c1cnn(C)c1
COc1cc(ccc1OCc1ccc(nc1)C(F)(F)F)C(C)n1c(N)nc2cc(cnc12)-c1cnn(C)c1
COc1cc(ccc1OCc1ccc(nc1)C(F)(F)F)C(C)n1c(N)nc2cc(cnc12)C#CCCO
COc1cc(Cn2cnc3cc(cnc23)C#CCCO)ccc1OCc1ccc(nc1)C(F)F
COc1ccc(cn1)C(C)Oc1ccc(Cn2cnc3cc(cnc23)-c2cnn(C)c2)cc1OC
COc1ccc(cn1)C(C)Oc1ccc(Cn2cnc3cc(cnc23)-c2ccnn2C)cc1OC
COc1ccc(cn1)C(C)Oc1ccc(Cn2cnc3cc(cnc23)-c2ccc(OC)nc2)cc1OC
COc1ccc(cn1)C(C)Oc1ccc(Cn2cnc3cc(cnc23)-c2ccnc(F)c2)cc1OC
Cc1cc(nn1CC(=O)Nc1cncc(c1)C(=O)c1cn(c2c(F)cncc12)C(C)(C)CO)C(F)(F)F
CC(C)(CO)n1cc(C(=O)c2cncc(NC(=O)Cn3ccc(n3)C3CC3)c2)c2cncc(F)c12
CC(C)(CO)n1cc(C(=O)c2cncc(NC(=O)Cc3ccc(Cl)cn3)c2)c2cncc(F)c12
CC(C)(CO)n1cc(C(=O)c2cncc(NC(=O)Cn3cc(cn3)C(F)(F)F)c2)c2cncc(F)c12
CC(C)(CO)n1cc(C(=O)c2cncc(NC(=O)Cc3cccc(c3)C(F)(F)F)c2)c2cncc(F)c12
CC(C)(CO)n1cc(C(=O)c2cncc(NC(=O)Cc3ccc(Cl)cc3)c2)c2cncc(F)c12
CC(C)(CO)n1cc(C(=O)c2cncc(NC(=O)Cc3ccc(cc3)C(F)(F)F)c2)c2cncc(F)c12
CC(C)(CO)n1cc(C(=O)c2cncc(NC(=O)Cc3ccc(Cl)cn3)c2)c2cnccc12
CC(C)(CO)n1cc(C(=O)c2cc(NC(=O)Cc3ccc(cc3)C#N)ccn2)c2cnccc12
CC(C)(CO)n1cc(C(=O)c2cc(NC(=O)Cn3ccc(n3)C(F)(F)F)ccn2)c2cnccc12
CC(C)(CO)n1cc(C(=O)c2cc(NC(=O)Cn3cc(nn3)C(F)(F)F)ccn2)c2cnccc12
CC(C)(CO)n1cc(C(=O)c2cncc(NC(=O)Cc3ccc(cc3)C#N)c2)c2cnccc12
CC(C)(CO)n1cc(C(=O)c2cncc(NC(=O)Cn3cc(nn3)C(F)(F)F)c2)c2cnccc12
CC(C)c1cn(CC(=O)Nc2cncc(c2)C(=O)c2cn(c3ccncc23)C(C)(C)CO)nn1
CC(C)(CO)n1cc(C(=O)c2cncc(NC(=O)Cn3cc(nn3)C3CC3)c2)c2cnccc12
CC(C)(CO)n1cc(C(=O)c2cncc(NC(=O)Cc3ccc(F)cn3)c2)c2cnccc12
CC(CO)n1cc(C(=O)c2cc(NC(=O)Cc3ccc(Cl)cn3)ccn2)c2cnccc12
CC(CO)n1cc(C(=O)c2cc(NC(=O)Cc3cccc(c3)C(F)(F)F)ccn2)c2cnccc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)Cc3nc(oc3C)C3CC3)c2)c2cnccc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)Cc3nc(oc3C3CC3)C3CC3)c2)c2cnccc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)Cn3ccc(n3)C(F)(F)F)c2)c2cnccc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)Cc3ccc(Cl)cn3)c2)c2cnccc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)Cc3ccc(F)cn3)c2)c2cnccc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)Cc3nc(C)oc3C3CC3)c2)c2cnccc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)Cn3cc(C)cn3)c2)c2cnccc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)Cn3ccc(n3)C3CC3)c2)c2cnccc12
CC(C)n1cc(C(=O)c2cc(NC(=O)Cn3ccc(n3)C(F)(F)F)ccn2)c2cnccc12
CC(C)n1cc(C(=O)c2cc(NC(=O)Cn3nc(cc3C)C(F)(F)F)ccn2)c2cnccc12
CC(C)n1cc(C(=O)c2cc(NC(=O)Cn3ccc(n3)C3CC3)ccn2)c2cnccc12
CC(C)n1cc(C(=O)c2cc(NC(=O)Cn3cc(cn3)C(F)(F)F)ccn2)c2cnccc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)Cn3cc(cn3)C(F)(F)F)c2)c2cncc(F)c12
CC(C)n1cc(C(=O)c2cncc(NC(=O)Cn3nc(cc3C)C(F)(F)F)c2)c2cncc(F)c12
CC(C)(CO)n1cc(C(=O)c2cncc(NC(=O)Cc3ccc(cc3)C(F)(F)F)c2)c2cnccc12
CC(CO)n1cc(C(=O)c2cncc(NC(=O)Cc3cccc(c3)C(F)(F)F)c2)c2cnccc12
CC(CO)n1cc(C(=O)c2cncc(NC(=O)Cc3ccc(cc3)C(F)(F)F)c2)c2cnccc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)Cc3ccc(C#N)c(c3)C(F)(F)F)c2)c2cnccc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)Cn3cc(nn3)C(F)(F)F)c2)c2cnccc12
COCc1nc(CC(=O)Nc2cncc(c2)C(=O)c2cn(C(C)C)c3ccncc23)c(o1)C1CC1
CC(C)n1cc(C(=O)c2cncc(NC(=O)Cc3nonc3C)c2)c2cnccc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)Cc3cn(C)cn3)c2)c2cnccc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)Cc3nc(nn3C)C(C)(C)C)c2)c2cnccc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)Cc3coc(n3)C3CC3)c2)c2cnccc12
COCCn1nc(nc1CC(=O)Nc1cncc(c1)C(=O)c1cn(C(C)C)c2ccncc12)C(C)(C)C
CC(C)n1cc(C(=O)c2cncc(NC(=O)Cc3cncn3C)c2)c2cnccc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)Cc3nccn3C)c2)c2cnccc12
COc1ncc(cc1NC(=O)Cc1ccc(cc1)C#N)C(=O)c1cn(C(C)C)c2ccncc12
COc1ncc(cc1NC(=O)Cn1nc(cc1C)C(F)(F)F)C(=O)c1cn(C(C)C)c2ccncc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)Cc3ccc(cc3)C#N)c2)c2cnccc12
CC(C)n1cc(CC(=O)Nc2cncc(c2)C(=O)c2cn(C(C)C)c3ccncc23)c(n1)C(F)(F)F
CC(C)n1cc(C(=O)c2cncc(NC(=O)Cn3cc(nn3)C3CC3)c2)c2cnccc12
CC(C)n1cc(C(=O)c2cc(NC(=O)Cn3cc(nn3)C3CC3)ccn2)c2cnccc12
CC(C)n1cc(C(=O)c2cc(NC(=O)Cn3cc(nn3)C(F)(F)F)ccn2)c2cnccc12
CC(C)n1cc(C(=O)c2cc(NC(=O)Cc3ccc(cc3)C#N)ccn2)c2cnccc12
CC(C)n1cc(C(=O)c2cc(NC(=O)Cc3ccc(Cl)cn3)ccn2)c2cnccc12
CC(C)n1cc(C(=O)c2cc(NC(=O)Cc3cnn(C4CC4)c3C(F)(F)F)ccn2)c2cnccc12
CC(C)n1cc(C(=O)c2cc(NC(=O)Cc3cn(nc3C(F)(F)F)C3CC3)ccn2)c2cnccc12
CC(C)n1cc(C(=O)c2cc(NC(=O)Cc3cn(C)nc3C)ccn2)c2cnccc12
CC(CO)n1cc(C(=O)c2cncc(NC(=O)Cn3cc(nn3)C(F)(F)F)c2)c2cnccc12
CC(CO)n1cc(C(=O)c2cncc(NC(=O)Cn3ccc(n3)C(F)(F)F)c2)c2cnccc12
CC(CO)n1cc(C(=O)c2cncc(NC(=O)Cn3cc(nn3)C3CC3)c2)c2cnccc12
CC(C)c1cn(CC(=O)Nc2cncc(c2)C(=O)c2cn(C(C)CO)c3ccncc23)nn1
CC(CO)n1cc(C(=O)c2cncc(NC(=O)Cn3nc(cc3C)C(F)(F)F)c2)c2cnccc12
CC(C)n1ncc(CC(=O)Nc2cncc(c2)C(=O)c2cn(C(C)CO)c3ccncc23)c1C(F)(F)F
CC(CO)n1cc(C(=O)c2cncc(NC(=O)Cc3ccc(Cl)cn3)c2)c2cnccc12
CC(CO)n1cc(C(=O)c2cncc(NC(=O)Cc3ccc(F)cn3)c2)c2cnccc12
CC(C)n1cc(C(=O)c2ccnc(NC(=O)Cc3nc(oc3C)C3CC3)c2)c2cnccc12
CC(C)n1cc(C(=O)c2ccnc(NC(=O)Cc3nc(oc3C3CC3)C3CC3)c2)c2cnccc12
COCc1nc(CC(=O)Nc2cc(ccn2)C(=O)c2cn(C(C)C)c3ccncc23)c(o1)C1CC1
CC(C)n1cc(C(=O)c2ccnc(NC(=O)Cc3ccc(F)cn3)c2)c2cnccc12
CC(C)n1cc(C(=O)c2ccnc(NC(=O)Cc3ccc(Cl)cn3)c2)c2cnccc12
CC(C)n1cc(C(=O)c2cc(NC(=O)Cn3cc(nn3)C(F)(F)F)ccn2)c2cncc(F)c12
CC(CO)n1cc(C(=O)c2cc(NC(=O)Cc3ccc(cc3)C(F)(F)F)ccn2)c2cnccc12
CC(C)n1cc(C(=O)c2cc(NC(=O)Cc3ccc(Cl)cc3)ccn2)c2cncc(F)c12
CC(C)n1cc(C(=O)c2cncc(NC(=O)Cn3cc(nn3)C(F)(F)F)c2)c2cncc(F)c12
CC(C)n1cc(C(=O)c2cncc(NC(=O)Cc3ccc(F)cn3)c2)c2cncc(F)c12
CC(C)n1cc(C(=O)c2cncc(NC(=O)Cn3cc(nn3)C3CC3)c2)c2cncc(F)c12
CC(C)n1cc(C(=O)c2cncc(NC(=O)Cn3ccc(n3)C3CC3)c2)c2cncc(F)c12
CC(C)n1cc(C(=O)c2cncc(NC(=O)Cn3cc(cn3)C3CC3)c2)c2cncc(F)c12
CC(C)(CO)n1cc(C(=O)c2cncc(NC(=O)Cc3ccc(cc3)C#N)c2)c2cncc(F)c12
CC(C)(CO)n1cc(C(=O)c2cncc(NC(=O)Cc3ccc(F)cn3)c2)c2cncc(F)c12
CC(C)(CO)n1cc(C(=O)c2cncc(NC(=O)Cn3cc(nn3)C(F)(F)F)c2)c2cncc(F)c12
CC(C)(CO)n1cc(C(=O)c2cncc(NC(=O)Cn3ccc(n3)C(F)(F)F)c2)c2cncc(F)c12
CC(C)n1cc(C(=O)c2ccnc(NC(=O)Cc3cccc(Cl)c3)c2)c2cnccc12
CC(C)n1cc(C(=O)c2ccnc(NC(=O)Cc3cccc(CC(C)(C)O)c3)c2)c2cnccc12
CC(C)c1cn(CC(=O)Nc2cc(ccn2)C(=O)c2cn(C(C)C)c3ccncc23)nn1
CC(C)n1cc(C(=O)c2ccnc(NC(=O)Cn3cc(Cl)cn3)c2)c2cnccc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)Cc3ccccc3Cl)c2)c2cnccc12
COc1ccc(CC(=O)Nc2cc(ccn2)C(=O)c2cn(C(C)C)c3ccncc23)cc1
CC(C)n1cc(C(=O)c2ccnc(NC(=O)Cn3ccnc3)c2)c2cnccc12
CC(C)n1cc(C(=O)c2ccnc(NC(=O)Cc3ccc(Cl)cc3)c2)c2cnccc12
CC(C)n1cc(C(=O)c2ccnc(NC(=O)Cn3nc(cc3C)C(F)(F)F)c2)c2cnccc12
CC(C)n1cc(C(=O)c2ccnc(NC(=O)Cc3ccccc3Cl)c2)c2cnccc12
CC(C)n1cc(C(=O)c2ccnc(NC(=O)Cc3ccc(F)cc3F)c2)c2cnccc12
CC(C)n1cc(C(=O)c2ccnc(NC(=O)Cc3ccccc3)c2)c2cnccc12
COc1cccc(CC(=O)Nc2cc(ccn2)C(=O)c2cn(C(C)C)c3ccncc23)c1
CC(C)n1cc(C(=O)c2ccnc(NC(=O)Cn3ccc(C)n3)c2)c2cnccc12
CC(C)n1cc(C(=O)c2ccnc(NC(=O)Cc3cnccn3)c2)c2cnccc12
CC(C)c1ccnn1CC(=O)Nc1cc(ccn1)C(=O)c1cn(C(C)C)c2ccncc12
CC(C)n1cc(C(=O)c2ccnc(NC(=O)Cn3nc(C)nc3C)c2)c2cnccc12
CC(C)c1cc(C)n(CC(=O)Nc2cc(ccn2)C(=O)c2cn(C(C)C)c3ccncc23)n1
CC(C)n1cc(C(=O)c2ccnc(NC(=O)Cn3cc(C)nn3)c2)c2cnccc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)Cc3ccc(F)cc3)c2)c2cnccc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)Cc3ccc(Cl)cc3)c2)c2cnccc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)Cn3ccnc3C)c2)c2cnccc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)Cc3ncccn3)c2)c2cnccc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)Cn3cccn3)c2)c2cnccc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)Cc3cccc(Cl)c3)c2)c2cnccc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)Cn3cc(Cl)cn3)c2)c2cnccc12
COc1ccc(CC(=O)Nc2cncc(c2)C(=O)c2cn(C(C)C)c3ccncc23)cc1
COc1cccc(CC(=O)Nc2cncc(c2)C(=O)c2cn(C(C)C)c3ccncc23)c1
CC(C)n1cc(C(=O)c2cncc(NC(=O)Cc3ccccc3)c2)c2cnccc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)Cn3nc(C)cc3C)c2)c2cnccc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)Cn3cc(C)nn3)c2)c2cnccc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)Cc3cnccn3)c2)c2cnccc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)Cn3ccc(C)n3)c2)c2cnccc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)Cn3nccc3C)c2)c2cnccc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)Cc3cc(C)n[nH]3)c2)c2cnccc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)Cn3nc(C)nc3C)c2)c2cnccc12
CC(C)n1cc(C(=O)c2ccnc(NC(=O)Cc3ccc(cn3)C#N)c2)c2cnccc12
CC(C)n1cc(C(=O)c2cncc(NC(=O)Cc3ccc(cn3)C#N)c2)c2cnccc12
CC(C)n1cc(C(=O)c2cc(NC(=O)Cc3ccc(cn3)C#N)ccn2)c2cnccc12
OCCn1cc(C(=O)c2ccnc(NC(=O)Cc3ccc(cc3)C(F)(F)F)c2)c2cnccc12
OCCn1cc(C(=O)c2ccnc(NC(=O)c3cccc(OC(F)(F)F)c3)c2)c2cnccc12
OCCn1cc(C(=O)c2ccnc(NC(=O)Cc3ccccc3OC(F)(F)F)c2)c2cnccc12
OCCn1cc(C(=O)c2ccnc(NC(=O)Cc3ccc(Cl)c(Cl)c3)c2)c2cnccc12
OCCn1cc(C(=O)c2ccnc(NC(=O)Cc3ccc(F)cc3F)c2)c2cnccc12
OCCn1cc(C(=O)c2ccnc(NC(=O)Cc3ccc(Cl)cc3)c2)c2cnccc12
CC(C)c1ccnn1CC(=O)Nc1cc(ccn1)C(=O)c1cn(CCO)c2ccncc12
OCCn1cc(C(=O)c2ccnc(NC(=O)Cc3ccc(F)cc3)c2)c2cnccc12
OCCn1cc(C(=O)c2ccnc(NC(=O)Cc3cccc(Cl)c3)c2)c2cnccc12
Cc1ccn(CC(=O)Nc2cc(ccn2)C(=O)c2cn(CCO)c3ccncc23)n1
CC(C)(O)Cc1cccc(CC(=O)Nc2cc(ccn2)C(=O)c2cn(CCO)c3ccncc23)c1
Cc1cc(C)n(CC(=O)Nc2cc(ccn2)C(=O)c2cn(CCO)c3ccncc23)n1
Cc1cc(nn1CC(=O)Nc1cc(ccn1)C(=O)c1cn(CCO)c2ccncc12)C(F)(F)F
Cn1nc(nc1CC(=O)Nc1cc(ccn1)C(=O)c1cn(CCO)c2ccncc12)C(C)(C)C
Cc1ccnn1CC(=O)Nc1cc(ccn1)C(=O)c1cn(CCO)c2ccncc12
OCCn1cc(C(=O)c2ccnc(NC(=O)Cn3cc(nn3)C(F)(F)F)c2)c2cnccc12
CC(C)n1ncc(CC(=O)Nc2cc(ccn2)C(=O)c2cn(CCO)c3ccncc23)c1C(F)(F)F
OCCn1cc(C(=O)c2ccnc(NC(=O)Cn3nccn3)c2)c2cnccc12
CC(C)c1cn(CC(=O)Nc2cc(ccn2)C(=O)c2cn(CCO)c3ccncc23)nn1
CC(C)n1cc(C(=O)c2ccnc(NC(=O)Cc3c(C)noc3C)c2)c2cnccc12
CC(C)n1cc(C(=O)c2ccnc(NC(=O)Cc3csc(C)n3)c2)c2cnccc12
CC(C)n1cc(C(=O)c2ccnc(NC(=O)Cc3nc(C)sc3C)c2)c2cnccc12
CC(C)n1cc(C(=O)c2ccnc(NC(=O)Cn3cc(nn3)C(F)(F)F)c2)c2cnccc12
CC(C)n1cc(C(=O)c2ccnc(NC(=O)Cn3nc(C)cc3C)c2)c2cnccc12
CC(C)n1cc(C(=O)c2ccnc(NC(=O)Cc3ccc(Cl)c(Cl)c3)c2)c2cnccc12
CC(C)n1cc(C(=O)c2ccnc(NC(=O)Cn3cccn3)c2)c2cnccc12
CC(C)n1cc(C(=O)c2ccnc(NC(=O)Cc3sc(C)nc3C)c2)c2cnccc12
CC(C)n1cc(C(=O)c2ccnc(NC(=O)Cc3ccc(OC(F)(F)F)cc3)c2)c2cnccc12
CC(C)n1cc(C(=O)c2ccnc(NC(=O)Cn3nccc3C)c2)c2cnccc12
CC(C)n1cc(C(=O)c2ccnc(NC(=O)Cn3cnnn3)c2)c2cnccc12
CC(C)n1cc(C(=O)c2ccnc(NC(=O)Cc3nc(nn3C)C(C)(C)C)c2)c2cnccc12
CC(C)n1cc(C(=O)c2ccnc(NC(=O)c3cccc(OC(F)(F)F)c3)c2)c2cnccc12
CC(C)n1cc(C(=O)c2ccnc(NC(=O)Cc3nc(C)oc3C3CC3)c2)c2cnccc12
CC(C)n1cc(C(=O)c2ccnc(NC(=O)Cc3ccc(cc3)C(F)(F)F)c2)c2cnccc12
CC(C)n1cc(C(=O)c2ccnc(NC(=O)Cc3cc(C)n[nH]3)c2)c2cnccc12
CC(C)n1cc(C(=O)c2ccnc(NC(=O)Cc3cnn(C(C)C)c3C(F)(F)F)c2)c2cnccc12
CC(C)n1cc(C(=O)c2ccnc(NC(=O)Cc3nc(C)oc3C)c2)c2cnccc12
CC(C)n1cc(C(=O)c2ccnc(NC(=O)Cc3ccon3)c2)c2cnccc12
CC(C)n1cc(C(=O)c2ccnc(NC(=O)Cc3cscn3)c2)c2cnccc12
CC(C)n1cc(C(=O)c2ccnc(NC(=O)Cc3ccccc3OC(F)(F)F)c2)c2cnccc12
CC(C)n1cc(C(=O)c2ccnc(NC(=O)Cc3ccc(cc3)C#N)c2)c2cnccc12
CC(C)n1cc(C(=O)c2ccnc(NC(=O)Cc3nc(C)n[nH]3)c2)c2cnccc12
CC(C)n1cc(C(=O)c2ccnc(NC(=O)Cc3cncs3)c2)c2cnccc12
CC(C)n1cc(C(=O)c2ccnc(NC(=O)Cc3ccc(F)cc3)c2)c2cnccc12
CC(C)n1cc(C(=O)c2ccnc(NC(=O)Cc3coc(n3)C3CC3)c2)c2cnccc12
CC(C)n1cc(C(=O)c2ccnc(NC(=O)Cn3nccn3)c2)c2cnccc12
CC(C)n1cc(C(=O)c2ccnc(NC(=O)Cc3cccc(OC(F)(F)F)c3)c2)c2cnccc12
CC(C)n1cc(C(=O)c2ccnc(NC(=O)Cc3nnnn3C)c2)c2cnccc12
CC(C)n1cc(C(=O)c2ccnc(NC(=O)Cn3cncn3)c2)c2cnccc12
FC(F)(F)Oc1cccc(CC(=O)Nc2cc(ccn2)C(=O)c2cn(C3COC3)c3ccncc23)c1
O=C(Cc1ccc(cc1)C#N)Nc1cc(ccn1)C(=O)c1cn(C2COC2)c2ccncc12
Fc1ccc(CC(=O)Nc2cc(ccn2)C(=O)c2cn(C3COC3)c3ccncc23)nc1
O=C(Cc1coc(n1)C1CC1)Nc1cc(ccn1)C(=O)c1cn(C2COC2)c2ccncc12
Fc1ccc(CC(=O)Nc2cc(ccn2)C(=O)c2cn(C3COC3)c3ccncc23)c(F)c1
CC(C)c1cn(CC(=O)Nc2cc(ccn2)C(=O)c2cn(C3COC3)c3ccncc23)nn1
Cc1oc(nc1CC(=O)Nc1cc(ccn1)C(=O)c1cn(C2COC2)c2ccncc12)C1CC1
O=C(Cc1nc(oc1C1CC1)C1CC1)Nc1cc(ccn1)C(=O)c1cn(C2COC2)c2ccncc12
Fc1ccc(CC(=O)Nc2cc(ccn2)C(=O)c2cn(C3COC3)c3ccncc23)cc1
FC(F)(F)Oc1cccc(c1)C(=O)Nc1cc(ccn1)C(=O)c1cn(C2COC2)c2ccncc12
CC(CO)n1cc(C(=O)c2cncc(NC(=O)Cc3ccc(Cl)cc3)c2)c2cncc(F)c12
CC(CO)n1cc(C(=O)c2cncc(NC(=O)Cn3cc(nn3)C3CC3)c2)c2cncc(F)c12
CC(CO)n1cc(C(=O)c2cncc(NC(=O)Cn3ccc(n3)C(F)(F)F)c2)c2cncc(F)c12
CC(CO)n1cc(C(=O)c2cncc(NC(=O)Cc3ccc(cc3)C(F)(F)F)c2)c2cncc(F)c12
CC(CO)n1cc(C(=O)c2cncc(NC(=O)Cc3ccc(Cl)cn3)c2)c2cncc(F)c12
CC(CO)n1cc(C(=O)c2cncc(NC(=O)Cc3ccc(F)cn3)c2)c2cncc(F)c12
CC(CO)n1cc(C(=O)c2cncc(NC(=O)Cc3ccc(cc3)C#N)c2)c2cncc(F)c12
CC(CO)n1cc(C(=O)c2cncc(NC(=O)Cn3cc(nn3)C(F)(F)F)c2)c2cncc(F)c12
CC(CO)n1cc(C(=O)c2cncc(NC(=O)Cn3ccc(n3)C3CC3)c2)c2cncc(F)c12
CC(CO)n1cc(C(=O)c2cncc(NC(=O)Cn3nc(cc3C)C(F)(F)F)c2)c2cncc(F)c12
CC(CO)n1cc(C(=O)c2cncc(NC(=O)Cn3cc(cn3)C(F)(F)F)c2)c2cncc(F)c12
FC(F)(F)c1cc(CC(=O)Nc2cc(ccn2)C(=O)c2cn(C3COC3)c3ccncc23)ccc1C#N
CC(CO)n1cc(C(=O)c2cncc(NC(=O)Cc3cccc(c3)C(F)(F)F)c2)c2cncc(F)c12
CC(C)(CO)n1cc(C(=O)c2cc(NC(=O)Cc3ccc(cc3)C(F)(F)F)ccn2)c2cnccc12
CC(C)(CO)n1cc(C(=O)c2cc(NC(=O)Cc3cccc(c3)C(F)(F)F)ccn2)c2cnccc12
CC(C)n1cc(C(=O)c2ccnc(NC(=O)Cc3ccc(C#N)c(c3)C(F)(F)F)c2)c2cnccc12
CC(C)(CO)n1cc(C(=O)c2cc(NC(=O)Cn3ccc(n3)C3CC3)ccn2)c2cnccc12
CC(C)(CO)n1cc(C(=O)c2cncc(NC(=O)Cc3cccc(c3)C(F)(F)F)c2)c2cnccc12
CC(C)(CO)n1cc(C(=O)c2cncc(NC(=O)Cn3ccc(n3)C(F)(F)F)c2)c2cnccc12
CC(C)(CO)n1cc(C(=O)c2cncc(NC(=O)Cn3cc(nn3)C3CC3)c2)c2cncc(F)c12
CC(C)N(Cc1c[nH]c2ncccc12)C(=O)Nc1ccc(SC(F)(F)F)cc1
CC(C)N(Cc1c[nH]c2ncccc12)C(=O)Nc1ccc(OC(F)(F)F)cc1
CC1(C)CCN(C(=O)N1Cc1c[nH]c2ncccc12)c1ccc(SC(F)(F)F)cc1
CC(C)N(Cc1n[nH]c2ncccc12)C(=O)Nc1ccc(SC(F)(F)F)cc1
CC(C#C)N(Cc1cccc(c1)-c1nccs1)C(=O)Nc1ccc(OC(F)(F)F)cc1
CC(C)N(Cc1cccc(c1)-c1nccs1)C(=O)Nc1cnc(nc1)C(C)(C)C
CC(C)N(Cc1cccc(c1)-c1nccs1)C(=O)Nc1ccc(OC(F)(F)F)cc1
CC(C)N(Cc1n[nH]c2ncccc12)C(=O)Nc1ccc(OC(F)(F)F)cc1
CC1(C)CN(C(=O)N1Cc1cccc(c1)-c1nccs1)c1ccc(OC(F)(F)F)cc1
CC(C)N(Cc1cc(ccn1)-c1nccs1)C(=O)Nc1ccc(OC(F)(F)F)cc1
Fc1ccc(F)c(c1)[C@H]1CCCN1c1ccc2ncc(NC(=O)Nc3ccccc3)n2n1 |r|
Fc1ccc(F)c(c1)[C@H]1CCCN1c1ccc2ncc(NC(=O)N3CCOCC3)n2n1 |r|
CC(=O)Nc1cnc2ccc(nn12)N1CCC[C@@H]1c1cc(F)ccc1F |r|
CS(=O)(=O)Nc1ccc(cc1)C(=O)Nc1cnc2ccc(nn12)N1CCC[C@@H]1c1cc(F)ccc1F |r|
Fc1ccc(F)c(c1)[C@H]1CCCN1c1ccc2ncc(NC(=O)Nc3cccc(c3)C#N)n2n1 |r|
Fc1ccc(F)c(c1)[C@H]1CCCN1c1ccc2ncc(NC(=O)Nc3ccc(cc3)C#N)n2n1 |r|
Fc1ccc(F)c(c1)[C@H]1CCCN1c1ccc2ncc(NC(=O)Nc3ccc(Cl)cc3Cl)n2n1 |r|
Fc1ccc(F)c(c1)[C@H]1CCCN1c1ccc2ncc(NC(=O)Nc3cccc(c3)C(F)(F)F)n2n1 |r|
Fc1ccc(F)c(c1)[C@H]1CCCN1c1ccc2ncc(NC(=O)Nc3cc(Cl)cc(Cl)c3)n2n1 |r|
O[C@H]1CCN(C1)C(=O)Nc1cnc2ccc(nn12)N1CCC[C@@H]1c1cc(F)ccc1F |r|
O[C@@H]1CCN(C1)C(=O)Nc1cnc2ccc(nn12)N1CCC[C@@H]1c1cc(F)ccc1F |r|
CC(C)(C)OC(=O)NC1CCN(CC1)C(=O)Nc1cnc2ccc(nn12)N1CCC[C@@H]1c1cc(F)ccc1F |r|
OC1CN(C1)C(=O)Nc1cnc2ccc(nn12)N1CCC[C@@H]1c1cc(F)ccc1F |r|
CC(C)(C)OC(=O)NC1CN(C1)C(=O)Nc1cnc2ccc(nn12)N1CCC[C@@H]1c1cc(F)ccc1F |r|
CC(C)(C)OC(=O)N1CCN(CC1)C(=O)Nc1cnc2ccc(nn12)N1CCC[C@@H]1c1cc(F)ccc1F |r|
CN(C)C(=O)Nc1cnc2ccc(nn12)N1CCC[C@@H]1c1cc(F)ccc1F |r|
CC(C)(C)OC(=O)NC1CCCN(C1)C(=O)Nc1cnc2ccc(nn12)N1CCC[C@@H]1c1cc(F)ccc1F |r|
NC1CCN(CC1)C(=O)Nc1cnc2ccc(nn12)N1CCC[C@@H]1c1cc(F)ccc1F |r|
NC1CN(C1)C(=O)Nc1cnc2ccc(nn12)N1CCC[C@@H]1c1cc(F)ccc1F |r|
Fc1ccc(F)c(c1)[C@H]1CCCN1c1ccc2ncc(NC(=O)N3CCNCC3)n2n1 |r|
NC1CCCN(C1)C(=O)Nc1cnc2ccc(nn12)N1CCC[C@@H]1c1cc(F)ccc1F |r|
Fc1ccc(NC(=O)Nc2cnc3ccc(nn23)N2CCC[C@@H]2c2cc(F)ccc2F)cc1 |r|
CC(C)(C)OC(=O)N1C2CCC1CN(C2)C(=O)Nc1cnc2ccc(nn12)N1CCC[C@@H]1c1cc(F)ccc1F |r|
Fc1ccc(F)c(c1)[C@H]1CCCN1c1ccc2ncc(NC(=O)N3CC4CCC(C3)N4)n2n1 |r|
OC1CCN(CC1)C(=O)Nc1cnc2ccc(nn12)N1CCC[C@@H]1c1cc(F)ccc1F |r|
Fc1ccc(F)c(c1)[C@H]1CCCN1c1ccc2ncc(NC(=O)N3CCCCC3)n2n1 |r|
NC(=O)Nc1cnc2ccc(nn12)N1CCC[C@@H]1c1cc(F)ccc1F |r|
CNC(=O)Nc1cnc2ccc(nn12)N1CCC[C@@H]1c1cc(F)ccc1F |r|
CC(C)(C)NC(=O)Nc1cnc2ccc(nn12)N1CCC[C@@H]1c1cc(F)ccc1F |r|
COc1ccc(NC(=O)Nc2cnc3ccc(nn23)N2CCC[C@@H]2c2cc(F)ccc2F)cc1 |r|
CCOC(=O)C1CCN(CC1)C(=O)Nc1cnc2ccc(nn12)N1CCC[C@@H]1c1cc(F)ccc1F |r|
COc1cc(NC(=O)Nc2cnc3ccc(nn23)N2CCC[C@@H]2c2cc(F)ccc2F)cc(OC)c1OC |r|
Cc1noc(C)c1NC(=O)Nc1cnc2ccc(nn12)N1CCC[C@@H]1c1cc(F)ccc1F |r|
OC(=O)C1CCN(CC1)C(=O)Nc1cnc2ccc(nn12)N1CCC[C@@H]1c1cc(F)ccc1F |r|
CC1CN(CC(C)N1)C(=O)Nc1cnc2ccc(nn12)N1CCC[C@@H]1c1cc(F)ccc1F |r|
C[C@@H]1CN(CCN1C(=O)OC(C)(C)C)C(=O)Nc1cnc2ccc(nn12)N1CCC[C@@H]1c1cc(F)ccc1F |r|
C[C@H]1CN(CCN1C(=O)OC(C)(C)C)C(=O)Nc1cnc2ccc(nn12)N1CCC[C@@H]1c1cc(F)ccc1F |r|
C[C@@H]1CN(CCN1)C(=O)Nc1cnc2ccc(nn12)N1CCC[C@@H]1c1cc(F)ccc1F |r|
C[C@H]1CN(CCN1)C(=O)Nc1cnc2ccc(nn12)N1CCC[C@@H]1c1cc(F)ccc1F |r|
O[C@@H]1CN(C[C@H]1O)C(=O)Nc1cnc2ccc(nn12)N1CCC[C@@H]1c1cc(F)ccc1F |r|
Fc1ccc(F)c(c1)[C@H]1CCCN1c1ccc2ncc(NC(=O)N3CCS(=O)(=O)CC3)n2n1 |r|
Fc1ccc(F)c(c1)[C@H]1CCCN1c1ccc2ncc(NC(=O)N3CCNC(=O)C3)n2n1 |r|
OC1CN(C1)C(=O)Nc1cnc2ccc(nn12)N1CCCCC1c1cccc(F)c1
Fc1ccc(F)c(c1)[C@H]1CCCN1c1ccc2ncc(NC(=O)N3CCC(F)(F)C3)n2n1 |r|
Fc1ccc(F)c(c1)[C@H]1CCCN1c1ccc2ncc(NC(=O)N3CC(F)(F)C3)n2n1 |r|
Fc1ccc(F)c(c1)[C@H]1CCCN1c1ccc2ncc(NC(=O)N3CCC3)n2n1 |r|
CN(CCO)C(=O)Nc1cnc2ccc(nn12)N1CCC[C@@H]1c1cc(F)ccc1F |r|
CC(C)(C)OC(=O)N1CCN(CC1(C)C)C(=O)Nc1cnc2ccc(nn12)N1CCC[C@@H]1c1cc(F)ccc1F |r|
CC(C)[C@H]1CN(CCN1C(=O)OC(C)(C)C)C(=O)Nc1cnc2ccc(nn12)N1CCC[C@@H]1c1cc(F)ccc1F |r|
CC1(C)CN(CCN1)C(=O)Nc1cnc2ccc(nn12)N1CCC[C@@H]1c1cc(F)ccc1F |r|
CC(C)[C@H]1CN(CCN1)C(=O)Nc1cnc2ccc(nn12)N1CCC[C@@H]1c1cc(F)ccc1F |r|
OCC1CN(C1)C(=O)Nc1cnc2ccc(nn12)N1CCC[C@@H]1c1cc(F)ccc1F |r|
COC1CN(C1)C(=O)Nc1cnc2ccc(nn12)N1CCC[C@@H]1c1cc(F)ccc1F |r|
CC1(O)CN(C1)C(=O)Nc1cnc2ccc(nn12)N1CCC[C@@H]1c1cc(F)ccc1F |r|
CC(C)C(=O)OC1CN(C1)C(=O)Nc1cnc2ccc(nn12)N1CCC[C@@H]1c1cc(F)ccc1F |r|
Cn1cc(ccc1=O)C(=O)Nc1cnc2ccc(nn12)N1CCC[C@@H]1c1cc(F)ccc1F |r|
Cn1nc(ccc1=O)C(=O)Nc1cnc2ccc(nn12)N1CCC[C@@H]1c1cc(F)ccc1F |r|
CN1CCN(CC1)C(=O)Nc1cnc2ccc(nn12)N1CCC[C@@H]1c1cc(F)ccc1F |r|
OC1(CCN(CC1)C(=O)Nc1cnc2ccc(nn12)N1CCC[C@@H]1c1cc(F)ccc1F)C(F)(F)F |r|
Fc1ccc(F)c(c1)[C@H]1CCCN1c1ccc2ncc(NC(=O)C(F)(F)F)n2n1 |r|
Nc1ncc(Cl)cc1-c1ccc(Oc2ncc(NC(=O)Nc3cc(ccc3-n3cccn3)C(F)(F)F)cn2)cc1
Cc1cn(nn1)-c1ccc(cc1NC(=O)Nc1cnc(Oc2ccc(cc2)-c2cc(Cl)cnc2N)nc1)C(F)(F)F
Nc1ncc(Cl)cc1-c1ccc(Oc2ncc(NC(=O)Nc3cc(ccc3-n3ccc(n3)C(F)(F)F)C(F)(F)F)cn2)cc1
Nc1ncc(Cl)cc1-c1ccc(Oc2ncc(NC(=O)Nc3cc(ccc3Cl)C(F)(F)F)cn2)cc1
Nc1ncc(Cl)cc1-c1ccc(Oc2ccc(NC(=O)Nc3cc(ccc3-n3cccn3)C(F)(F)F)cn2)cc1
Nc1ncc(Cl)cc1-c1ccc(Oc2ccc(NC(=O)Nc3cc(ccc3-n3ccnn3)C(F)(F)F)cn2)cc1
Nc1ncc(Cl)cc1-c1ccc(Oc2ccc(NC(=O)Nc3cc(ccc3-c3cccnc3)C(F)(F)F)cn2)cc1
Cn1nccc1-c1ccc(cc1NC(=O)Nc1cnc(Oc2ccc(cc2)-c2cc(Cl)cnc2N)nc1)C(F)(F)F
Nc1ncc(F)cc1-c1ccc(Oc2ncc(NC(=O)Nc3cc(ccc3-n3ccnn3)C(F)(F)F)cn2)cc1
Nc1ncc(F)cc1-c1ccc(Oc2ncc(NC(=O)Nc3cc(ccc3-c3cccnc3)C(F)(F)F)cn2)cc1
Nc1ncc(Cl)cc1-c1ccc(Oc2ncc(NC(=O)Nc3ccc(cc3-n3cccn3)C(F)(F)F)cn2)cc1
Nc1ncc(Cl)cc1-c1ccc(Oc2ncc(NC(=O)Nc3ccc(cc3F)C(F)(F)F)cn2)cc1
Nc1ncc(Cl)cc1-c1ccc(Oc2ncc(NC(=O)Nc3ccc(cc3Cl)C(F)(F)F)cn2)cc1
Nc1ncc(cc1-c1ccc(Oc2ncc(NC(=O)Nc3cc(ccc3-n3ccc(n3)C(F)(F)F)C(F)(F)F)cn2)cc1)C(F)(F)F
Nc1ncc(Cl)cc1-c1ccc(Oc2ncc(NC(=O)Nc3cc(ccc3-c3ccccc3)C(F)(F)F)cn2)cc1
Nc1ncc(F)cc1-c1ccc(Oc2ncc(NC(=O)Nc3cc(ccc3-c3ccccc3)C(F)(F)F)cn2)cc1
Nc1ncc(Cl)cc1-c1ccc(Oc2ncc(NC(=O)Nc3cc(ccc3-n3cc(Cl)cn3)C(F)(F)F)cn2)cc1
Nc1ncc(Cl)cc1-c1ccc(Oc2ncc(NC(=O)Nc3cc(Cl)ccc3-n3ccc(n3)C(F)(F)F)cn2)cc1
Nc1ncc(Cl)cc1-c1ccc(Oc2ncc(NC(=O)Nc3ccc(cc3C(F)(F)F)C(F)(F)F)cn2)cc1
Nc1ncc(cc1-c1ccc(Oc2ncc(NC(=O)Nc3cc(ccc3-n3cc(Cl)cn3)C(F)(F)F)cn2)cc1)C(F)(F)F
CS(=O)(=O)c1ccc(cc1NC(=O)Nc1cnc(Oc2ccc(cc2)-c2cc(F)cnc2N)nc1)C(F)(F)F
CS(=O)(=O)c1ccc(cc1NC(=O)Nc1cnc(Oc2ccc(cc2)-c2cc(cnc2N)C(F)(F)F)nc1)C(F)(F)F
CS(=O)(=O)c1ccc(cc1NC(=O)Nc1cnc(Oc2ccc(cc2)-c2cc(Cl)cnc2N)nc1)C(F)(F)F
CN(C)S(=O)(=O)c1ccc(cc1NC(=O)Nc1cnc(Oc2ccc(cc2)-c2cc(cnc2N)C(F)(F)F)nc1)C(F)(F)F
FC(F)(F)c1ccc(c(NC(=O)Nc2cnc(Oc3ccc(cc3)-c3cnn4ccc(nc34)N3CCC3)nc2)c1)-c1cccnc1
Cn1nccc1-c1ccc(cc1NC(=O)Nc1cnc(Oc2ccc(cc2)-c2cnn3ccc(nc23)N2CCC2)nc1)C(F)(F)F
COc1ccn2ncc(-c3ccc(Oc4ncc(NC(=O)Nc5cc(ccc5-c5cccnc5)C(F)(F)F)cn4)cc3)c2n1
FC(F)(F)c1ccc(c(NC(=O)Nc2cnc(Oc3ccc(cc3)-c3cnn4cccnc34)nc2)c1)-c1cccnc1
CN(C)c1ccn2ncc(-c3ccc(Oc4ncc(NC(=O)Nc5cc(ccc5-c5cccnc5)C(F)(F)F)cn4)cc3)c2n1
CN(C)c1ccn2ncc(-c3ccc(Oc4ncc(NC(=O)Nc5cc(ccc5-c5ccnn5C)C(F)(F)F)cn4)cc3)c2n1
Cc1ccn2ncc(-c3ccc(Oc4ncc(NC(=O)Nc5cc(ccc5-c5cccnc5)C(F)(F)F)cn4)cc3)c2n1
CCNc1ccn2ncc(-c3ccc(Oc4ncc(NC(=O)Nc5cc(ccc5-c5cccc(C)c5)C(F)(F)F)cn4)cc3)c2n1
CN(C)c1ccn2ncc(-c3ccc(Oc4ncc(NC(=O)Nc5cc(ccc5-c5ccccc5)C(F)(F)F)cn4)cc3)c2n1
CN(C)c1ccn2ncc(-c3ccc(Oc4ncc(NC(=O)Nc5cc(ccc5-c5cccc(C)c5)C(F)(F)F)cn4)cc3)c2n1
CN(C)c1ccn2ncc(-c3ccc(Oc4ncc(NC(=O)Nc5cc(ccc5-c5ccccc5C)C(F)(F)F)cn4)cc3)c2n1
COc1ccc2ncc(-c3ccc(Oc4ncc(NC(=O)Nc5cc(ccc5-c5cccnc5)C(F)(F)F)cn4)cc3)n2n1
COc1ccc2ncc(-c3ccc(Oc4ncc(NC(=O)Nc5cc(ccc5-n5cccn5)C(F)(F)F)cn4)cc3)n2n1
CCOc1ccc2ncc(-c3ccc(Oc4ncc(NC(=O)Nc5cc(ccc5-c5cccnc5)C(F)(F)F)cn4)cc3)n2n1
FC(F)(F)c1ccc(c(NC(=O)Nc2cnc(Oc3ccc(cc3)-c3cnc4ccccn34)nc2)c1)-n1cccn1
FC(F)(F)c1ccc(c(NC(=O)Nc2cnc(Oc3ccc(cc3)-c3cnc4[nH]ccc4c3)nc2)c1)-c1cccnc1
FC(F)(F)c1ccc(c(NC(=O)Nc2cnc(Oc3ccc(cc3)-c3cnc4cnccn34)nc2)c1)-c1cccnc1
FC(F)(F)c1ccc(c(NC(=O)Nc2cnc(Oc3ccc(cc3)-c3cnn4ccccc34)nc2)c1)-c1cccnc1
FC(F)(F)c1ccc(c(NC(=O)Nc2cnc(Oc3ccc(cc3)-c3cnc4[nH]ncc4c3)nc2)c1)-c1cccnc1
C[C@H]1CN(CCN1)C(=O)Nc1cnn2ccc(nc12)N1CCC[C@@H]1c1cc(F)ccc1Cl
C[C@H]1CN(CCN1)C(=O)Nc1cnn2ccc(nc12)N1CCC[C@@H]1c1cc(F)ccc1F
Fc1ccc(Cl)c(c1)[C@H]1CCCN1c1ccn2ncc(NC(=O)C3CNC3)c2n1
CC1(CCNCC1)C(=O)Nc1cnn2ccc(nc12)N1CCC[C@@H]1c1cc(F)ccc1Cl
Fc1cc2[C@H]3CCCN3c3ccn4ncc(C(=O)NCCCn(c1)c2=O)c4n3 |r|
O=C1NCCCOc2cccc(n2)[C@H]2CCCN2c2ccn3ncc1c3n2 |r|
Fc1cnc2OCCCNC(=O)c3cnn4ccc(nc34)N3CCC[C@@H]3c2c1 |r|
OC1CNC(=O)c2cnn3ccc(nc23)N2CCC[C@@H]2c2cc(F)cnc2OC1 |r|
O[C@H]1CNC(=O)c2cnn3ccc(nc23)N2CCC[C@@H]2c2cc(F)cn(C1)c2=O |r|
O[C@@H]1CNC(=O)c2cnn3ccc(nc23)N2CCC[C@@H]2c2cc(F)cnc2OC1 |r|
O[C@@H]1CNC(=O)c2cnn3ccc(nc23)N2CCC[C@@H]2c2cc(F)cn(C1)c2=O |r|
Fc1cnc2OCCNC(=O)c3cnn4ccc(nc34)N3CCC[C@@H]3c2c1 |r|
Fc1cc2[C@H]3CCCN3c3ccn4ncc(C(=O)NCCCCn(c1)c2=O)c4n3 |r|
Fc1cnc2NCCNC(=O)c3cnn4ccc(nc34)N3CCC[C@@H]3c2c1 |r|
Fc1cnc2NCCCNC(=O)c3cnn4ccc(nc34)N3CCC[C@@H]3c2c1 |r|
Fc1cnc2OCCOC(=O)c3cnn4ccc(nc34)N3CCC[C@@H]3c2c1 |r|
Fc1cc2[C@H]3CCCN3c3ccn4ncc(C(=O)OCCn(c1)c2=O)c4n3 |r|
Fc1cnc2OCCONC(=O)c3cnn4ccc(nc34)N3CCC[C@@H]3c2c1 |r|
F[C@@H]1CNC(=O)c2cnn3ccc(nc23)N2CCC[C@@H]2c2cc(F)cn(C1)c2=O |r|
CN1CCCOc2ncc(F)cc2[C@H]2CCCN2c2ccn3ncc(C1=O)c3n2 |r|
Fc1cnc2OCC(F)(F)CNC(=O)c3cnn4ccc(nc34)N3CCC[C@@H]3c2c1 |r|
Fc1ccc2OCCCNC(=O)c3cnn4ccc(nc34)N3CCC[C@@H]3c2c1 |r|
Fc1ccc2OCCNCc3cnn4ccc(nc34)N3CCC[C@@H]3c2c1 |r|
CC(=O)N1CCOc2ccc(F)cc2[C@H]2CCCN2c2ccn3ncc(C1)c3n2 |r|
OCC(=O)N1CCOc2ccc(F)cc2[C@H]2CCCN2c2ccn3ncc(C1)c3n2 |r|
Fc1ccc2OCCCNCc3cnn4ccc(nc34)N3CCC[C@@H]3c2c1 |r|
CS(=O)(=O)N1CCOc2ccc(F)cc2[C@H]2CCCN2c2ccn3ncc(C1)c3n2 |r|
OC(=O)CN1CCOc2ccc(F)cc2[C@H]2CCCN2c2ccn3ncc(C1)c3n2 |r|
CS(=O)(=O)N1CCCOc2ccc(F)cc2[C@H]2CCCN2c2ccn3ncc(C1)c3n2 |r|
CCNC(=O)N1CCCOc2ccc(F)cc2[C@H]2CCCN2c2ccn3ncc(C1)c3n2 |r|
CCNC(=O)N1CCOc2ccc(F)cc2[C@H]2CCCN2c2ccn3ncc(C1)c3n2 |r|
Fc1cnc2OCCCNC(=O)c3cnn4ccc(nc34)N3[C@H](COC3=O)c2c1 |r|
Fc1cnc2OCCNC(=O)c3cnn4ccc(nc34)N3[C@H](COC3=O)c2c1 |r|
Fc1cnc2CCCNC(=O)c3cnn4ccc(nc34)N3CCC[C@@H]3c2c1 |r|
CC1CCc2ncc(F)cc2[C@H]2CCCN2c2ccn3ncc(C(=O)N1)c3n2 |r|
C[C@@H]1CNC(=O)c2cnn3ccc(nc23)N2CCC[C@@H]2c2cc(F)cn(C1)c2=O |r|
C[C@H]1CNC(=O)c2cnn3ccc(nc23)N2CCC[C@@H]2c2cc(F)cn(C1)c2=O |r|
CC1(C)CNC(=O)c2cnn3ccc(nc23)N2CCC[C@@H]2c2cc(F)cnc2OC1 |r|
CC1(C)CCc2ncc(F)cc2[C@H]2CCCN2c2ccn3ncc(C(=O)N1)c3n2 |r|
Fc1cnc2OCCn3nccc3NC(=O)c3cnn4ccc(nc34)N3CCC[C@@H]3c2c1 |r|
Fc1cnc2OCc3cccnc3NC(=O)c3cnn4ccc(nc34)N3CCC[C@@H]3c2c1 |r|
CC1(C)CNC(=O)c2cnn3ccc(nc23)N2CCC[C@@H]2c2cc(F)cn(C1)c2=O |r|
O[C@@H]1C[C@H]2N(C1)c1ccn3ncc(C(=O)NC[C@H](O)COc4ccc(F)cc24)c3n1 |r|
O[C@@H]1C[C@@H]2N(C1)c1ccn3ncc(C(=O)NC[C@H](O)COc4ccc(F)cc24)c3n1 |r|
O[C@@H]1C[C@H]2N(C1)c1ccn3ncc(C(=O)NCCCOc4ccc(F)cc24)c3n1 |r|
O[C@@H]1C[C@@H]2N(C1)c1ccn3ncc(C(=O)NCCCOc4ccc(F)cc24)c3n1 |r|
O[C@@H]1C[C@H]2N(C1)c1ccn3ncc(C(=O)NCCOc4ccc(F)cc24)c3n1 |r|
O[C@@H]1C[C@@H]2N(C1)c1ccn3ncc(C(=O)NCCOc4ccc(F)cc24)c3n1 |r|
O[C@@H]1C[C@H]2N(C1)c1ccn3ncc(C(=O)NC[C@@H](O)COc4ccc(F)cc24)c3n1 |r|
O[C@@H]1C[C@@H]2N(C1)c1ccn3ncc(C(=O)NC[C@@H](O)COc4ccc(F)cc24)c3n1 |r|
O[C@H]1CNC(=O)c2cnn3ccc(nc23)N2CC(F)(F)CC2c2cc(F)ccc2OC1 |r|
O[C@@H]1CNC(=O)c2cnn3ccc(nc23)N2CC(F)(F)CC2c2cc(F)ccc2OC1 |r|
COc1cc(ccc1OCc1ccc(cc1)C(F)(F)F)C(C)n1c(N)nc2cc(cnc12)-c1cnn(C)c1
COc1cc(ccc1OCc1ccc(cc1)C(F)(F)F)C(C)n1c(N)nc2cc(cnc12)-c1cnn(CCO)c1
COc1cc(ccc1OCc1ccc(cc1)C(F)(F)F)C(C)n1c(N)nc2cc(cnc12)-c1cn[nH]c1
CCC(c1ccc(OCc2ccc(nc2)C(F)(F)F)c(OC)c1)n1c(N)nc2cc(cnc12)-c1cnn(C)c1
COc1cc(ccc1OCc1ccc(nc1)C(F)(F)F)C(C)n1c(N)nc2cc(cnc12)-c1cnn(CCO)c1
Fc1cc2[C@H]3CCCN3c3ccn4ncc(CC(=O)NCCCCn(c1)c2=O)c4n3 |r|
Oc1ccn2ncc(-c3ccc(Oc4ncc(NC(=O)Nc5cc(ccc5-c5cccnc5)C(F)(F)F)cn4)cc3)c2n1
Cn1cc2cc(NC(=O)c3coc4CCNC(=O)c34)ccc2n1
CN1CCc2occ(C(=O)Nc3ccc4nn(C)cc4c3)c2C1=O
O=C(Nc1ccc(cc1)N1CCOCC1)c1coc2CCNC(=O)c12
CN1CCc2occ(C(=O)Nc3ccc(C)cc3)c2C1=O
COc1cc(ccc1NC(=O)c1coc2CCNC(=O)c12)N1CCN(CC1)C(=O)OC(C)(C)C
COc1cc(ccc1NC(=O)c1coc2CCNC(=O)c12)N1CCNCC1
COc1nc(ccc1NC(=O)c1coc2CCCNC(=O)c12)N1CCN(C)CC1
CCOc1nc(ccc1NC(=O)c1coc2CCN(CCOCc3ccccc3)C(=O)c12)N1CCN(CC1)C(C)=O
CCOc1nc(ccc1NC(=O)c1coc2CCN(CCO)C(=O)c12)N1CCN(CC1)C(C)=O
CC(=O)N1CCN(CC1)c1ccc(NC(=O)c2coc3CCNC(=O)c23)cc1
Cn1ncc2cc(NC(=O)c3coc4CCNC(=O)c34)ccc12
O=C(Nc1ccc2[nH]cnc2c1)c1coc2CCNC(=O)c12
NC(=O)c1ccc(NC(=O)c2coc3CCNC(=O)c23)cc1
O=C(Nc1ccc2[nH]ncc2c1)c1coc2CCNC(=O)c12
Cc1nc2ccc(NC(=O)c3coc4CCNC(=O)c34)cc2s1
CN1CCN(CC1)c1ccc(NC(=O)c2coc3CCNC(=O)c23)nc1
CN1CCN(CC1)c1ccc(NC(=O)c2coc3CCNC(=O)c23)cc1
COc1cc(ccc1NC(=O)c1coc2CCNC(=O)c12)N1CCN(CC1)C(C)=O
CCOc1nc(ccc1NC(=O)c1coc2CCNC(=O)c12)N1CCN(CC1)C(C)=O
COCCOc1nc(ccc1NC(=O)c1coc2CCNC(=O)c12)N1CCN(CC1)C(C)=O
CC(=O)N1CCN(CC1)c1ccc(NC(=O)c2coc3CCNC(=O)c23)c(OC2COC2)n1
CN1CCN(CC1)c1ccc(NC(=O)c2coc3CCN(C)C(=O)c23)cc1
CN1CCc2occ(C(=O)Nc3ccc4[nH]ncc4c3)c2C1=O
CN1CCc2occ(C(=O)Nc3ccc4n(C)ncc4c3)c2C1=O
CN1CCc2occ(C(=O)Nc3ccc(cc3)N3CCOCC3)c2C1=O
CN1CCc2occ(C(=O)Nc3ccc(cc3)C(N)=O)c2C1=O
CN1CCc2occ(C(=O)Nc3ccc4[nH]cnc4c3)c2C1=O
CN1CCc2occ(C(=O)Nc3ccc(cc3)N3CCN(CC3)C(C)=O)c2C1=O
CN1CCc2occ(C(=O)Nc3ccc4nc(C)sc4c3)c2C1=O
Cc1ccc(NC(=O)c2coc3CCNC(=O)c23)cc1
Oc1ccc(NC(=O)c2coc3CCNC(=O)c23)cc1
CC(=O)Nc1ccc(NC(=O)c2coc3CCNC(=O)c23)cc1
O=C(Nc1ccc2ncccc2c1)c1coc2CCNC(=O)c12
O=C(Nc1ccc2cn[nH]c2c1)c1coc2CCNC(=O)c12
COc1ccc(NC(=O)c2coc3CCNC(=O)c23)c(OC)n1
O=C(Nc1ccon1)c1coc2CCNC(=O)c12
O=C(Nc1cnccn1)c1coc2CCNC(=O)c12
Cc1cc(NC(=O)c2coc3CCNC(=O)c23)no1
O=C(Nc1ccc(cc1)C#N)c1coc2CCNC(=O)c12
Fc1ccc(NC(=O)c2coc3CCNC(=O)c23)nc1
COc1ccc(NC(=O)c2coc3CCNC(=O)c23)cn1
Clc1ccc(NC(=O)c2coc3CCNC(=O)c23)nc1
O=C(Nc1cccc(c1)C#N)c1coc2CCNC(=O)c12
CCOc1ccc(NC(=O)c2coc3CCNC(=O)c23)cn1
Cc1n[nH]c2ccc(NC(=O)c3coc4CCNC(=O)c34)cc12
Cc1cc2[nH]ncc2cc1NC(=O)c1coc2CCNC(=O)c12
O=C(Nc1nc2ccccc2s1)c1coc2CCNC(=O)c12
COC(=O)c1n[nH]c2ccc(NC(=O)c3coc4CCNC(=O)c34)cc12
CCN(CC)c1ccc(NC(=O)c2coc3CCNC(=O)c23)cc1
CC(O)Cn1ncc2cc(NC(=O)c3coc4CCNC(=O)c34)ccc12
CS(=O)(=O)NCCn1cc2cc(NC(=O)c3coc4CCNC(=O)c34)ccc2n1
CN1CCN(CCn2cc3cc(NC(=O)c4coc5CCNC(=O)c45)ccc3n2)CC1
OCCn1ncc2cc(NC(=O)c3coc4CCNC(=O)c34)ccc12
O=C(Nc1ccc2n(CCN3CCCC3)ncc2c1)c1coc2CCNC(=O)c12
CC(O)Cn1cc2cc(NC(=O)c3coc4CCNC(=O)c34)ccc2n1
O=C(Nc1ccc2n(CCN3CCOCC3)ncc2c1)c1coc2CCNC(=O)c12
CN1CCN(CCn2ncc3cc(NC(=O)c4coc5CCNC(=O)c45)ccc23)CC1
CS(=O)(=O)NCCn1ncc2cc(NC(=O)c3coc4CCNC(=O)c34)ccc12
CN1CCc2occ(C(=O)Nc3ccc(O)cc3)c2C1=O
CN1CCc2occ(C(=O)Nc3ccc(NC(C)=O)cc3)c2C1=O
CN1CCc2occ(C(=O)Nc3ccc(cc3)N3CCCCC3)c2C1=O
CN1CCc2occ(C(=O)Nc3cnc4ccccc4c3)c2C1=O
CN1CCc2occ(C(=O)Nc3ccc4ncccc4c3)c2C1=O
CN1CCc2occ(C(=O)Nc3ccc4cn[nH]c4c3)c2C1=O
COc1ccc(NC(=O)c2coc3CCN(C)C(=O)c23)c(OC)n1
CN1CCc2occ(C(=O)Nc3cc(C)on3)c2C1=O
CN1CCc2occ(C(=O)Nc3ccc(cc3)C#N)c2C1=O
CN1CCc2occ(C(=O)Nc3ccc(F)cn3)c2C1=O
COc1ccc(NC(=O)c2coc3CCN(C)C(=O)c23)cn1
CN1CCc2occ(C(=O)Nc3ccc(Cl)cn3)c2C1=O
CN1CCc2occ(C(=O)Nc3cccc(c3)C#N)c2C1=O
CCOc1ccc(NC(=O)c2coc3CCN(C)C(=O)c23)cn1
CN1CCc2occ(C(=O)Nc3ccc4[nH]nc(C)c4c3)c2C1=O
CN1CCc2occ(C(=O)Nc3cc4cn[nH]c4cc3C)c2C1=O
CN1CCc2occ(C(=O)Nc3nc4ccccc4s3)c2C1=O
CN1CCc2occ(C(=O)Nc3ccc(cn3)C(F)(F)F)c2C1=O
CN1CCc2occ(C(=O)Nc3cc4cn[nH]c4cc3Cl)c2C1=O
CN1CCc2occ(C(=O)Nc3ccc4[nH]c(C)nc4c3)c2C1=O
COc1cc(ccc1NC(=O)c1coc2CCNC(=O)c12)N1CCN(CC1)C(=O)CC(C)(C)C
COc1cc(ccc1NC(=O)c1coc2CCNC(=O)c12)N1CCN(CC1)C(=O)N1CCCC1
COc1cc(ccc1NC(=O)c1coc2CCNC(=O)c12)N1CCN(CC1)S(=O)(=O)N(C)C
COC(=O)c1ccc(Oc2nc(ccc2NC(=O)c2coc3CCCNC(=O)c23)N2CCN(C)CC2)cc1
CN1CCN(CC1)c1ccc(NC(=O)c2coc3CCCNC(=O)c23)c(Oc2ccc(CO)cc2)n1
CCOc1nc(ccc1NC(=O)c1coc2CCN(CCOC)C(=O)c12)N1CCN(CC1)C(C)=O
COCCOc1nc(ccc1NC(=O)c1coc2CCN(CCOCc3ccccc3)C(=O)c12)N1CCN(CC1)C(C)=O
CC(=O)N1CCN(CC1)c1ccc(NC(=O)c2coc3CCN(CCOCc4ccccc4)C(=O)c23)c(OCCOCc2ccccc2)n1
COCCOc1nc(ccc1NC(=O)c1coc2CCN(CCO)C(=O)c12)N1CCN(CC1)C(C)=O
CC(=O)N1CCN(CC1)c1ccc(NC(=O)c2coc3CCN(CCO)C(=O)c23)c(OCCO)n1
CCOc1nc(ccc1NC(=O)c1coc2CCN(CCCO)C(=O)c12)N1CCN(CC1)C(C)=O
CCOc1nc(ccc1NC(=O)c1coc2CCN(CCCCO)C(=O)c12)N1CCN(CC1)C(C)=O
CCOc1nc(ccc1NC(=O)c1coc2CCN(CCOCCO)C(=O)c12)N1CCN(CC1)C(C)=O
CCOc1nc(ccc1NC(=O)c1coc2CCNC(=O)c12)N1CCN(CC1)C(=O)OC(C)(C)C
CCOc1nc(ccc1NC(=O)c1coc2CCNC(=O)c12)N1CCN(CC1)C(NC)=NC#N |w:31.35|
CCOc1nc(ccc1NC(=O)c1coc2CCN(C[C@@H](C)OC(C)=O)C(=O)c12)N1CCN(CC1)C(C)=O
CCOc1nc(ccc1NC(=O)c1coc2CCN(C[C@@H](C)O)C(=O)c12)N1CCN(CC1)C(C)=O
CCOc1nc(ccc1NC(=O)c1coc2CCN(C[C@H](C)OC(C)=O)C(=O)c12)N1CCN(CC1)C(C)=O
CCOc1nc(ccc1NC(=O)c1coc2CCN(C[C@H](C)O)C(=O)c12)N1CCN(CC1)C(C)=O
CCOc1nc(ccc1NC(=O)c1coc2CCN([C@H](C)COC(C)=O)C(=O)c12)N1CCN(CC1)C(C)=O
CCOc1nc(ccc1NC(=O)c1coc2CCN([C@H](C)CO)C(=O)c12)N1CCN(CC1)C(C)=O
CCOc1nc(ccc1NC(=O)c1coc2CCN([C@@H](C)COC(C)=O)C(=O)c12)N1CCN(CC1)C(C)=O
CCOc1nc(ccc1NC(=O)c1coc2CCN([C@@H](C)CO)C(=O)c12)N1CCN(CC1)C(C)=O
CCOc1nc(ccc1NC(=O)c1coc2CCN(C(=O)c12)C(C)(C)CO)N1CCN(CC1)C(C)=O
CCOc1nc(ccc1NC(=O)c1coc2CCN(CC(C)(C)OC(C)=O)C(=O)c12)N1CCN(CC1)C(C)=O
CCOc1nc(ccc1NC(=O)c1coc2CCN(CC(C)(C)O)C(=O)c12)N1CCN(CC1)C(C)=O
CC(=O)N1CCN(CC1)c1ccc(NC(=O)c2coc3CCNC(=O)c23)c(O[C@H]2CCOC2)n1
CCOc1nc(ccc1NC(=O)c1coc2CCNC(=O)c12)N1CCOCC1
CC(C)(O)COc1nc(ccc1NC(=O)c1coc2CCNC(=O)c12)N1CCOCC1
CCOc1nc(CC(=O)OC)ccc1NC(=O)c1coc2CCNC(=O)c12
CCOc1nc(CCO)ccc1NC(=O)c1coc2CCNC(=O)c12
COc1nc(ccc1NC(=O)c1coc2CC3(CCOCC3)CC(=O)c12)N1CCN(CC1)C(C)=O
CCOc1nc(ccc1NC(=O)c1coc2CC3(CCC3)NC(=O)c12)N1CCN(CC1)C(C)=O
CCOc1nc(ccc1NC(=O)c1coc2CC3(CCCCC3)NC(=O)c12)N1CCN(CC1)C(C)=O
CCOc1nc(ccc1NC(=O)c1coc2CC3(CN(C3)C(C)=O)NC(=O)c12)N1CCN(CC1)C(C)=O
CCOc1nc(ccc1NC(=O)c1coc2CC3(COC3)NC(=O)c12)N1CCN(CC1)C(C)=O
CCOc1nc(ccc1NC(=O)c1coc2C[C@@H](NC(=O)c12)[C@@H](C)O)N1CCN(CC1)C(C)=O
CCOc1nc(ccc1NC(=O)c1coc2CC3(CCC3)N(CCO)C(=O)c12)N1CCN(CC1)C(C)=O
CCOc1nc(ccc1NC(=O)c1coc2CC3(CC3)NC(=O)c12)N1CCN(CC1)C(C)=O
CCOc1nc(ccc1NC(=O)c1coc2CC3(CCC3)NC(=O)c12)N1CCN(CC1)C(NC)=NC#N |w:34.39|
CCOc1nc(ccc1NC(=O)c1coc2CC(C)(C)N(CC(O)CO)C(=O)c12)N1CCN(CC1)C(C)=O
COc1cc(ccc1NC(=O)c1coc2CC(C)(C)NC(=O)c12)N1CCNCC1
COc1nc(ccc1NC(=O)c1coc2CC(C)(C)NC(=O)c12)N1CCN(CC1)C(=O)N1CCOCC1
COc1nc(ccc1NC(=O)c1coc2CC(C)(C)NC(=O)c12)N1CCN(CC1)C(C)=O
COc1nc(ccc1NC(=O)c1coc2CC(C)(C)NC(=O)c12)N1CCN(CC1)C(=O)N1CCCC1
COc1cc(ccc1NC(=O)c1coc2CC(C)NC(=O)c12)N1CCNCC1
COc1cc(ccc1NC(=O)c1coc2CC(C)(C)NC(=O)c12)N1CCN(CC1)S(C)(=O)=O
COc1cc(ccc1NC(=O)c1coc2CC(C)(C)NC(=O)c12)N1CCN(CC1)C(C)=O
CCOc1nc(ccc1NC(=O)c1coc2CC(C)(C)NC(=O)c12)N1CCNCC1
CCOc1nc(ccc1NC(=O)c1coc2CC(C)(C)NC(=O)c12)N1CCN(CC1)C(C)=O
CC(C)Oc1nc(ccc1NC(=O)c1coc2CC(C)(C)NC(=O)c12)N1C[C@H]2CCN[C@H]2C1
COc1nc(ccc1NC(=O)c1coc2CC(C)(C)NC(=O)c12)N1CC[C@@H]2CN(C)C[C@H]12
CC(C)Oc1nc(ccc1NC(=O)c1coc2CC(C)(C)NC(=O)c12)N1C[C@@H]2CCN(CCO)[C@@H]2C1
CC(C)Oc1nc(ccc1NC(=O)c1coc2CC(C)(C)NC(=O)c12)N1C[C@H]2CCN([C@H]2C1)C(=O)N1CCN(C)CC1
CC(C)Oc1nc(ccc1NC(=O)c1coc2CC(C)(C)NC(=O)c12)N1CCN([C@H](CO)C1)C(C)=O
CC(C)Oc1nc(ccc1NC(=O)c1coc2CC(C)(C)NC(=O)c12)N1CCN(C[C@H]1CO)C(C)=O
CC(C)Oc1nc(ccc1NC(=O)c1coc2CC(C)(C)NC(=O)c12)N1CCN(C[C@H]1CO)C(=O)N1CCOCC1
CC(C)Oc1nc(ccc1NC(=O)c1coc2CC(C)(C)NC(=O)c12)N1CC[C@@H](C1)N(C)C
CC(C)Oc1nc(ccc1NC(=O)c1coc2CC(C)(C)NC(=O)c12)N1CCC[C@H](CO)C1
CC(C)Oc1nc(ccc1NC(=O)c1coc2CC(C)(C)NC(=O)c12)N1CCN([C@@H](CO)C1)C(C)=O
CC(C)Oc1nc(ccc1NC(=O)c1coc2CC(C)(C)NC(=O)c12)N1CCN(C[C@@H]1CO)C(C)=O
CC(C)Oc1nc(ccc1NC(=O)c1coc2CC(C)(C)NC(=O)c12)N(CCO)CCO
COCCOc1ccc(NC(=O)c2coc3CC(C)(C)NC(=O)c23)c(OCCOC)n1
COC[C@@H]1CN(CCN1C(C)=O)c1ccc(NC(=O)c2coc3CC(C)(C)NC(=O)c23)c(OCC(C)(C)O)n1
CCOc1nc(CCO)ccc1NC(=O)c1coc2CC(C)(C)NC(=O)c12
CCOc1nc(CO)ccc1NC(=O)c1coc2CC(C)(C)NC(=O)c12
CCOc1nc(ccc1NC(=O)c1coc2CC(C)(C)N(CCOC)C(=O)c12)C(O)=O
Cn1ncc2cc(NC(=O)c3coc4CC(C)(C)CC(=O)c34)ccc12
Cn1cc2cc(NC(=O)c3coc4CC(C)(C)CC(=O)c34)ccc2n1
CC(=O)N1CCN(CC1)c1ccc(NC(=O)c2coc3CC(C)(C)CC(=O)c23)cc1
CC1(C)Cc2occ(C(=O)Nc3ccc(nc3)N3CCNCC3)c2C(=O)C1
Cn1cc2cc(NC(=O)c3coc4CC5(CCC5)CC(=O)c34)ccc2n1
CC1(C)Cc2occ(C(=O)Nc3ccc(cn3)N3CCNCC3)c2C(=O)C1
CC1(C)Cc2occ(C(=O)Nc3ccc(cc3)N3CCN(CC3)S(C)(=O)=O)c2C(=O)C1
CC1(C)Cc2occ(C(=O)Nc3ccc4nn(CCO)cc4c3)c2C(=O)C1
CC1(C)Cc2occ(C(=O)Nc3ccc4[nH]c(CO)nc4c3)c2C(=O)C1
CC1(C)Cc2occ(C(=O)Nc3ccc(cn3)N3CCN(CC3)S(C)(=O)=O)c2C(=O)C1
CC(=O)N1CCN(CC1)c1ccc(NC(=O)c2coc3CC(C)(C)CC(=O)c23)nc1
COc1cc(ccc1NC(=O)c1coc2CC(C)(C)CC(=O)c12)N1CCNCC1
COc1cc(ccc1NC(=O)c1coc2CC(C)(C)CC(=O)c12)N1CCN(CC1)C(C)=O
Cn1cc2cc(NC(=O)c3coc4CC5(CC5)CC(=O)c34)ccc2n1
Cn1cc2cc(NC(=O)c3coc4CNCC(=O)c34)ccc2n1
Cn1cc2cc(NC(=O)c3coc4CN(CC(=O)c34)S(C)(=O)=O)ccc2n1
Cn1cc2cc(NC(=O)c3coc4CC(C)(CC(=O)c34)C(N)=O)ccc2n1
COC(=O)C1(C)Cc2occ(C(=O)Nc3ccc4nn(C)cc4c3)c2C(=O)C1
Cn1cc2cc(NC(=O)c3coc4CC(C)(CO)CC(=O)c34)ccc2n1
COc1cc(ccc1NC(=O)c1coc2CC(C)(CO)CC(=O)c12)N1CCN(CC1)C(=O)OC(C)(C)C
COCC1(C)Cc2occ(C(=O)Nc3ccc(cc3OC)N3CCNCC3)c2C(=O)C1
Cn1cc2cc(NC(=O)c3coc4CCC(C)(CO)C(=O)c34)ccc2n1
Cn1cc2cc(NC(=O)c3coc4CCC(C)(C)C(=O)c34)ccc2n1
COc1cc(ccc1NC(=O)c1coc2CCC(C)(CN)C(=O)c12)N1CCN(CC1)C(C)=O
COc1cc(ccc1NC(=O)c1coc2COC3(CCNCC3)C(=O)c12)N1CCN(CC1)C(C)=O
COc1nc(ccc1NC(=O)c1coc2COC(C)(C)C(=O)c12)N1CCN(CC1)C(C)=O
COc1cc(ccc1NC(=O)c1coc2COC3(COC3)C(=O)c12)N1CCN(CC1)C(C)=O
CCOc1nc(ccc1NC(=O)c1coc2CC(C)(C)N(C)C(=O)c12)N1CCN(CC1)C(C)=O
CCOc1nc(ccc1NC(=O)c1coc2CC(C)(C)N(CCO)C(=O)c12)N1CCN(CC1)C(C)=O
CCOc1nc(ccc1NC(=O)c1coc2CC(C)(C)N(CCOC)C(=O)c12)N1CCN(CC1)C(C)=O
CCOc1nc(ccc1NC(=O)c1coc2CC(C)(C)N(CCOCCO)C(=O)c12)N1CCN(CC1)C(C)=O
COCCOc1nc(ccc1NC(=O)c1coc2CC(C)(C)NC(=O)c12)N1CCN(CC1)C(C)=O
CC(=O)N1CCN(CC1)c1ccc(NC(=O)c2coc3CC(C)(C)NC(=O)c23)c(OCC(F)(F)F)n1
CC(=O)N1CCN(CC1)c1ccc(NC(=O)c2coc3CC(C)(C)NC(=O)c23)c(OC2COC2)n1
CC(=O)N1CCN(CC1)c1ccc(NC(=O)c2coc3CC(C)(C)NC(=O)c23)c(OC2CCOCC2)n1
CC(=O)N1CCN(CC1)c1ccc(NC(=O)c2coc3CC(C)(C)NC(=O)c23)c(O[C@H]2CCOC2)n1
COCCOc1nc(ccc1NC(=O)c1coc2CC(C)(C)NC(=O)c12)N1CCN(CC1)C=O
CC(=O)N1CCN(CC1)c1ccc(NC(=O)c2coc3CC(C)(C)NC(=O)c23)c(OC2CS(=O)C2)n1
CCOc1nc(ccc1NC(=O)c1coc2CC(C)(C)NC(=O)c12)C1CCN(CC1)C(C)=O
CCOc1nc(ccc1NC(=O)c1coc2CCC(C(=O)c12)c1cc(F)ccc1F)N1CCN(CC1)C(C)=O
OC(=O)C1CCN(CC1)C(=O)c1cnn2ccc(nc12)N1CCC[C@@H]1c1cc(F)ccc1F |r|
OC(=O)CC1CCN(CC1)C(=O)c1cnn2ccc(nc12)N1CCC[C@@H]1c1cc(F)ccc1F |r|
Fc1ccc(F)c(c1)[C@H]1CCCN1c1ccn2ncc(C(=O)NCCc3c[nH]cn3)c2n1 |r|
OC(=O)[C@H]1CC[C@@H](CC1)NC(=O)c1cnn2ccc(nc12)N1CCC[C@@H]1c1cc(F)ccc1F |r,wU:6.9,wD:25.29,3.2,(4.87,-7.18,;5.96,-6.09,;7.45,-6.49,;5.57,-4.61,;6.64,-3.46,;6.24,-1.98,;4.75,-1.58,;3.66,-2.67,;4.06,-4.15,;4.35,-.09,;2.87,.31,;1.78,-.78,;2.47,1.8,;3.37,3.04,;2.47,4.29,;1,3.81,;-.33,4.58,;-1.66,3.81,;-1.66,2.27,;-.33,1.5,;1,2.27,;-3,1.5,;-3,-.04,;-4.46,-.51,;-5.37,.73,;-4.46,1.98,;-4.86,3.46,;-3.77,4.55,;-4.17,6.04,;-3.08,7.13,;-5.66,6.44,;-6.75,5.35,;-6.35,3.86,;-7.44,2.77,)|
OCc1ccc(F)cc1[C@H]1CCCN1c1ccn2ncc(C(=O)N[C@H]3CC[C@H](O)CC3)c2n1 |r,wU:24.25,wD:9.9,27.29,(-6.68,.7,;-7.08,2.19,;-5.99,3.28,;-6.35,4.81,;-5.26,5.9,;-3.77,5.5,;-2.68,6.59,;-3.37,4.01,;-4.46,2.92,;-4.06,1.43,;-4.97,.19,;-4.06,-1.06,;-2.6,-.58,;-2.6,.96,;-1.26,1.73,;-1.26,3.27,;.07,4.04,;1.4,3.27,;2.87,3.74,;3.77,2.5,;2.87,1.25,;3.27,-.24,;2.18,-1.33,;4.75,-.64,;5.15,-2.12,;6.64,-2.52,;7.04,-4.01,;5.95,-5.1,;6.35,-6.59,;4.46,-4.7,;4.06,-3.21,;1.4,1.73,;.07,.96,)|
CC(C)(NC(=O)c1cnn2ccc(nc12)N1CCC[C@@H]1c1cc(F)ccc1F)C#N |r|
Fc1ccc(F)c(c1)[C@H]1CCCN1c1ccn2ncc(C(=O)NCC#N)c2n1 |r|
CS(=O)(=O)N1CCC(CC1)NC(=O)c1cnn2ccc(nc12)N1CCC[C@@H]1c1cc(F)ccc1F |r|
NS(=O)(=O)N1CCC(CC1)NC(=O)c1cnn2ccc(nc12)N1CCC[C@@H]1c1cc(F)ccc1F |r|
CS(=O)(=O)NCCNC(=O)c1cnn2ccc(nc12)N1CCC[C@@H]1c1cc(F)ccc1F |r|
NS(=O)(=O)CCNC(=O)c1cnn2ccc(nc12)N1CCC[C@@H]1c1cc(F)ccc1F |r|
OCc1ccc(F)cc1[C@H]1CCCN1c1ccn2ncc(C(=O)NC3CC3)c2n1 |r|
CC(C)(O)CNC(=O)c1cnn2ccc(nc12)N1CCC[C@@H]1c1cc(F)ccc1CO |r|
OCc1ccc(F)cc1[C@H]1CCCN1c1ccn2ncc(C(=O)NCCN3CCOCC3)c2n1 |r|
OC[C@@H](O)CNC(=O)c1cnn2ccc(nc12)N1CCC[C@@H]1c1cc(F)ccc1CO |r|
OC[C@H](O)CNC(=O)c1cnn2ccc(nc12)N1CCC[C@@H]1c1cc(F)ccc1CO |r|
CC(C)(CNS(C)(=O)=O)NC(=O)c1cnn2ccc(nc12)N1CCC[C@@H]1c1cc(F)ccc1F |r|
CC(C)(NC(=O)c1cnn2ccc(nc12)N1CCC[C@@H]1c1cncc(F)c1)C#N |r|
CS(=O)(=O)N1CCC(CC1)NC(=O)c1cnn2ccc(nc12)N1CCC[C@@H]1c1cncc(F)c1 |r|
OCc1ncc(F)cc1[C@H]1CCCN1c1ccn2ncc(C(=O)NC3CC3)c2n1 |r|
CC(C)(C)NC(=O)c1cnn2ccc(nc12)N1CCC[C@@H]1c1cc(F)cnc1CO |r|
CC(C)(CF)NC(=O)c1cnn2ccc(nc12)N1CCC[C@@H]1c1cc(F)cnc1CO |r|
NC(=O)c1cnn2ccc(nc12)N1CCC[C@@H]1c1cc(F)cnc1CO |r|
CONC(=O)c1cnn2ccc(nc12)N1CCC[C@@H]1c1cc(F)cnc1CO |r|
OC(=O)C1(CC1)NC(=O)c1cnn2ccc(nc12)N1CCC[C@@H]1c1cc(F)ccc1F |r|
O[C@H]1CCC(CC1)NC(=O)c1cnn2ccc(nc12)N1CCCC1c1cncc(F)c1 |r,wU:1.0,(5.77,-6.12,;5.38,-4.63,;3.89,-4.23,;3.49,-2.74,;4.58,-1.65,;6.07,-2.05,;6.46,-3.54,;4.18,-.17,;5.27,.92,;6.76,.52,;4.87,2.41,;5.77,3.66,;4.87,4.9,;3.41,4.43,;2.07,5.2,;.74,4.43,;.74,2.89,;2.07,2.12,;3.41,2.89,;-.6,2.12,;-.12,.65,;-1.37,-.25,;-2.61,.65,;-2.14,2.12,;-2.91,3.45,;-2.14,4.78,;-2.91,6.12,;-4.45,6.12,;-5.22,4.78,;-6.76,4.78,;-4.45,3.45,)|
Fc1cncc(c1)C1CCCN1c1ccn2ncc(C(=O)NC3CCC3)c2n1
OC1CCCC1NC(=O)c1cnn2ccc(nc12)N1CCCC1c1cncc(F)c1
OC[C@@H]1[C@H](NC(=O)c2cnn3ccc(nc23)N2CCC[C@@H]2c2cncc(F)c2)C2CC[C@@]1(O)C2 |r,TLB:1:2:30.29:33,THB:4:3:30.29:33|
C[C@@H](O)CNC(=O)c1cnn2ccc(nc12)N1CCC[C@@H]1c1cc(F)ccc1F |r|
Cc1ncc(F)cc1[C@H]1CCCN1c1ccn2ncc(C(=O)NC3(CO)CC3)c2n1 |r|
Cc1ncc(F)cc1C1CCCN1c1ccn2ncc(C(=O)NC3CCC[C@H]3O)c2n1 |r|
C[C@@H](NC(=O)c1cnn2ccc(nc12)N1[C@H](CO)CC[C@@H]1c1cncc(F)c1)C(F)(F)F |r|
C[C@H](NC(=O)c1cnn2ccc(nc12)N1[C@H](CO)CC[C@@H]1c1cncc(F)c1)C(F)(F)F |r|
C[C@H](NC(=O)c1cnn2ccc(nc12)N1C[C@@H](O)C[C@@H]1c1cccc(F)c1)C(F)(F)F |r|
C[C@H](NC(=O)c1cnn2ccc(nc12)N1[C@H](CC[C@@]1(C)CO)c1cncc(F)c1)C(F)(F)F |r|
COc1ncc(F)cc1[C@H]1CCCN1c1ccn2ncc(C(=O)Nc3cc(C)n[nH]3)c2n1 |r|
CCc1cc(NC(=O)c2cnn3ccc(nc23)N2CCC[C@@H]2c2cc(F)cnc2OC)[nH]n1 |r|
Fc1ccc(F)c(c1)[C@H]1CCCN1c1ccc2ncc(NC(=O)NN3CCS(=O)(=O)CC3)n2n1
CC1CN(CCN1)C(=O)Nc1cnc2ccc(nn12)N1CCC[C@H]1c1cc(F)ccc1F |r|
Fc1ccc(F)c(c1)[C@@H]1CCCN1c1ccc2ncc(NC(=O)N3CCS(=O)(=O)CC3)n2n1 |r|
CC(C)C(=O)OC1CN(C1)C(=O)Nc1cnc2ccc(nn12)N1CCC[C@H]1c1cc(F)ccc1F
OC[C@H]1[C@H]2CCC(C2)[C@H]1NC(=O)c1cnn2ccc(nc12)N1CCC[C@@H]1c1cncc(F)c1 |r,TLB:1:2:4.5:7,THB:9:8:4.5:7|
COc1ncc(F)cc1C1CCCN1c1ccn2ncc(C(=O)NCCCO)c2n1
OC1CCN(CCNC(=O)c2cnn3ccc(nc23)N2CCCC2c2cc(F)ccc2F)CC1
C[C@@H](O)[C@H](CO)NC(=O)c1cnn2ccc(nc12)N1CCC[C@@H]1c1cc(F)ccc1F |r|
C[C@H](O)[C@H](CO)NC(=O)c1cnn2ccc(nc12)N1CCC[C@@H]1c1cc(F)ccc1F |r|
C[C@H](O)[C@@H](CO)NC(=O)c1cnn2ccc(nc12)N1CCC[C@@H]1c1cc(F)ccc1F |r|
Cc1ncc(F)cc1C1CCCN1c1ccn2ncc(C(=O)NC3CC3)c2n1
CCc1ncc(F)cc1C1CCCN1c1ccn2ncc(C(=O)NC3CC[C@H](O)CC3)c2n1 |r,wD:27.29,(-8.05,3.64,;-6.72,2.87,;-5.38,3.64,;-5.38,5.18,;-4.05,5.95,;-2.72,5.18,;-1.38,5.95,;-2.72,3.64,;-4.05,2.87,;-4.05,1.33,;-5.3,.42,;-4.82,-1.04,;-3.28,-1.04,;-2.8,.42,;-1.47,1.19,;-1.47,2.73,;-.14,3.5,;1.2,2.73,;2.66,3.21,;3.57,1.96,;2.66,.72,;3.43,-.62,;2.66,-1.95,;4.97,-.62,;5.74,-1.95,;7.28,-1.95,;8.05,-3.28,;7.28,-4.62,;8.05,-5.95,;5.74,-4.62,;4.97,-3.28,;1.2,1.19,;-.14,.42,)|
FC(F)(F)c1ccc(C(=O)Nc2cc(cnc2-c2ccccc2)N2CCOCC2)c(Cl)c1
Cc1ncc(NC(=O)c2cc(c(Cl)cc2F)-c2ncccn2)c(n1)-c1ccccc1
Cc1cc(c(NC(=O)c2ccc(OC(F)(F)F)c(c2)-c2ccn(C)n2)cn1)-c1ccccc1
Cc1nc(Cl)c(NC(=O)c2ccc(c(c2)-c2ccn(C)n2)C(F)(F)F)c(n1)-c1ccccc1
Cc1cc(c(NC(=O)c2ccc(c(c2)-c2cc[nH]n2)C(F)(F)F)cn1)-c1ccccc1
Fc1ccc(cc1)-c1ccccc1NC(=O)c1ccc(cc1F)C(F)(F)F
Cc1cc(n[nH]1)-c1ccccc1NC(=O)c1cccc(c1)-c1nccs1
Cc1ncc(NC(=O)c2ccc(C)c(F)c2F)c(n1)-c1ccccc1
Cc1cc(C)n(n1)-c1ccc(Cl)c(c1)C(=O)Nc1cnc(C)nc1-c1ccccc1
FC(F)(F)c1ccc(cc1)C(=O)Nc1cc(cnc1-c1ccccc1)-c1cccnc1
Cc1cc(on1)-c1ccccc1NC(=O)c1cc(ccc1Cl)-n1nc(C)cc1C
Cc1ncc(NC(=O)c2ccc(c(c2)-c2cscn2)C(F)(F)F)c(n1)-c1ccccc1
Cc1cc(C)n(n1)-c1cc(ccc1F)C(=O)Nc1cnc(C)nc1-c1ccccc1
Cc1ncc(NC(=O)c2cccc(c2)-n2nccc2C(F)(F)F)c(n1)-c1ccccc1
Cc1ncc(NC(=O)c2ccc(c(c2)-c2ccn(C)n2)C(F)(F)F)c(n1)-c1ccccc1
Cc1ncc(NC(=O)c2ccc(c(c2)-n2nccn2)C(F)(F)F)c(n1)-c1ccccc1
Cc1ccn(n1)-c1cc(ccc1C(F)(F)F)C(=O)Nc1cnc(C)nc1-c1ccccc1
Cc1csc(n1)-c1cc(ccc1C(F)(F)F)C(=O)Nc1cnc(C)nc1-c1cc(C)n[nH]1
Cc1cnn(c1)-c1ccncc1NC(=O)c1ccc(c(c1)-c1ccn(C)n1)C(F)(F)F
Cc1ncc(NC(=O)c2ccc(c(c2)-c2ncco2)C(F)(F)F)c(n1)-c1ccccc1
Cc1ncc(NC(=O)c2ccc(c(c2)-c2cc[nH]n2)C(F)(F)F)c(n1)-c1ccccc1
Cn1ccc(n1)-c1cc(ccc1C(F)(F)F)C(=O)Nc1ncccc1-c1ccccc1
Cc1ncc(NC(=O)c2cc(-c3ccn(C)n3)c(cc2Cl)C(F)(F)F)c(n1)-c1ccccc1
Cn1ccc(n1)-c1cc(C(=O)Nc2cccnc2-c2ccccc2)c(Cl)cc1C(F)(F)F
Cn1ccc(n1)-c1cc(ccc1C(F)(F)F)C(=O)Nc1nccnc1-c1ccccc1
Cc1nc(C)c(NC(=O)c2cc(-c3ccn(C)n3)c(cc2Cl)C(F)(F)F)c(n1)-c1ccccc1
Cc1ncc(NC(=O)c2cc(-c3ccn(C)n3)c(cc2F)C(F)(F)F)c(n1)-c1ccccc1
Cc1ncc(NC(=O)c2cc(-c3ncccn3)c(cc2F)C(F)(F)F)c(n1)-c1ccccc1
Cc1coc(n1)-c1cc(ccc1C(F)(F)F)C(=O)Nc1cnc(C)nc1-c1ccccc1
Cc1noc(n1)-c1cc(ccc1C(F)(F)F)C(=O)Nc1cnc(C)nc1-c1ccccc1
Cc1ncc(NC(=O)c2ccc(c(c2)-c2ccn(C)n2)C(F)(F)F)c(n1)-c1ccc(F)cc1
Cc1cccc(c1)-c1nc(C)ncc1NC(=O)c1ccc(c(c1)-c1ccn(C)n1)C(F)(F)F
CC1CCC(O1)c1cc(C(=O)Nc2cnc(C)nc2-c2ccccc2)c(F)cc1C(F)(F)F
Cn1ccc(n1)-c1cc(C(=O)Nc2cnc(CC#N)nc2-c2ccccc2)c(F)cc1C(F)(F)F
Cn1ccc(n1)-c1cc(ccc1C(F)(F)F)C(=O)Nc1cnc(CO)nc1-c1ccccc1
OCc1ncc(NC(=O)c2ccc(c(c2)-c2cc[nH]n2)C(F)(F)F)c(n1)-c1ccccc1
Cn1ccc(n1)-c1cc(ccc1C(F)(F)F)C(=O)Nc1cnc(CCO)nc1-c1ccccc1
Cn1ccc(n1)-c1cc(ccc1C(F)(F)F)C(=O)Nc1cnc(CCN2CCOCC2)nc1-c1ccccc1
OCc1ncc(NC(=O)c2ccc(c(c2)-c2ncccn2)C(F)(F)F)c(n1)-c1ccccc1
OCc1ncc(NC(=O)c2cc(-c3ncccn3)c(cc2F)C(F)(F)F)c(n1)-c1ccccc1
Cn1ccc(n1)-c1cc(ccc1C(F)(F)F)C(=O)Nc1cnc(CNC(=O)OC(C)(C)C)nc1-c1ccccc1
Cn1ccc(n1)-c1cc(ccc1C(F)(F)F)C(=O)Nc1cnc(CN)nc1-c1ccccc1
NCc1ncc(NC(=O)c2ccc(c(c2)-c2ccn(n2)C(F)F)C(F)(F)F)c(n1)-c1ccccc1
Cc1ncc(NC(=O)c2ccc(c(c2)-c2ccn(C)n2)C(F)(F)F)c(n1)-c1cccc(CO)c1
CNCc1ncc(NC(=O)c2ccc(c(c2)-c2ccn(C)n2)C(F)(F)F)c(n1)-c1ccccc1
Cc1nc(CO)c(NC(=O)c2ccc(c(c2)-c2ccn(C)n2)C(F)(F)F)c(n1)-c1ccccc1
Cn1ccc(n1)-c1cc(ccc1C(F)(F)F)C(=O)Nc1ccc(nc1-c1ccccc1)C(C)(C)O
C[C@H](O)C(=O)NCc1ncc(NC(=O)c2cc(-c3ccn(C)n3)c(cc2F)C(F)(F)F)c(n1)-c1ccccc1 |r|
CC(=O)NCc1ncc(NC(=O)c2ccc(c(c2)-c2ccn(C)n2)C(F)(F)F)c(n1)-c1ccccc1
Cn1ccc(n1)-c1cc(ccc1C(F)(F)F)C(=O)Nc1cnc(CNC(=O)CO)nc1-c1ccccc1
Cn1ccc(n1)-c1cc(ccc1C(F)(F)F)C(=O)Nc1cnc(CNC(=O)C2CC2)nc1-c1ccccc1
Cn1ccc(n1)-c1cc(C(=O)Nc2cnc(CNC(=O)CO)nc2-c2ccccc2)c(F)cc1C(F)(F)F
Cn1ccc(n1)-c1cc(ccc1C(F)(F)F)C(=O)Nc1ccc(CNC(=O)CO)nc1-c1ccccc1
CC(=O)NCc1ncc(NC(=O)c2cc(-c3cc[nH]n3)c(cc2F)C(F)(F)F)c(n1)-c1ccccc1
Cn1ccc(n1)-c1cc(ccc1C(F)(F)F)C(=O)Nc1cnc(CNC(=O)CO)cc1-c1ccccc1
C[C@H](O)C(=O)NCc1ccc(NC(=O)c2cc(-c3ccn(C)n3)c(cc2F)C(F)(F)F)c(n1)-c1ccccc1 |r|
Cn1ccc(n1)-c1cc(C(=O)Nc2ccc(CNC(=O)[C@@H]3CCC(=O)N3)nc2-c2ccccc2)c(F)cc1C(F)(F)F |r|
COCC(=O)NCc1ccc(NC(=O)c2cc(-c3ccn(C)n3)c(cc2F)C(F)(F)F)c(n1)-c1ccccc1
Cn1ccc(n1)-c1cc(C(=O)Nc2ccc(CNC(=O)CS(C)(=O)=O)nc2-c2ccccc2)c(F)cc1C(F)(F)F
C[C@@H](O)C(=O)NCc1ncc(NC(=O)c2cc(-c3ccn(C)n3)c(cc2F)C(F)(F)F)c(n1)-c1ccccc1 |r|
Cn1ccc(n1)-c1cc(C(=O)Nc2ccc(CNC(=O)C(O)CO)nc2-c2ccccc2)c(F)cc1C(F)(F)F
CN1CCOC(C1)C(=O)NCc1ccc(NC(=O)c2cc(-c3ccn(C)n3)c(cc2F)C(F)(F)F)c(n1)-c1ccccc1
COCC(=O)NCc1ncc(NC(=O)c2cc(-c3ccn(C)n3)c(cc2F)C(F)(F)F)c(n1)-c1ccccc1
Cn1ccc(n1)-c1cc(C(=O)Nc2ncc(CNC(=O)CO)nc2-c2ccccc2)c(F)cc1C(F)(F)F
Cn1ccc(n1)-c1cc(C(=O)Nc2cnc(CNC(=O)C(C)(N)CO)nc2-c2ccccc2)c(F)cc1C(F)(F)F
Cn1ccc(n1)-c1cc(C(=O)Nc2cnc(CNC(=O)CS(C)(=O)=O)nc2-c2ccccc2)c(F)cc1C(F)(F)F
Cn1ccc(n1)-c1cc(C(=O)Nc2cnc(CNC(=O)Cn3cncn3)nc2-c2ccccc2)c(F)cc1C(F)(F)F
Cn1ccc(n1)-c1cc(C(=O)Nc2ncc(CNC(=O)CO)cc2-c2ccccc2)c(F)cc1C(F)(F)F
Cn1ccc(n1)-c1cc(C(=O)Nc2cnc(CNC(=O)CN3CCOC3=O)nc2-c2ccccc2)c(F)cc1C(F)(F)F
C[C@@H](O)C(=O)NCc1cnc(NC(=O)c2cc(-c3ccn(C)n3)c(cc2F)C(F)(F)F)c(n1)-c1ccccc1 |r|
C[C@H](O)C(=O)N(C)Cc1ccc(NC(=O)c2cc(-c3ccn(C)n3)c(cc2F)C(F)(F)F)c(n1)-c1ccccc1 |r|
C[C@@H](N)C(=O)NCc1ncc(NC(=O)c2cc(-c3ccn(C)n3)c(cc2F)C(F)(F)F)c(n1)-c1ccccc1 |r|
Cn1ccc(n1)-c1cc(C(=O)Nc2cnc(CNC(=O)[C@@H]3COCCN3)nc2-c2ccccc2)c(F)cc1C(F)(F)F |r|
Cn1ccc(n1)-c1cc(ccc1C(F)(F)F)C(=O)Nc1cnc(CNS(C)(=O)=O)nc1-c1ccccc1
Cn1ccc(n1)-c1cc(C(=O)Nc2cnc(CNC(N)=O)nc2-c2ccccc2)c(F)cc1C(F)(F)F
Cn1ccc(n1)-c1cc(C(=O)Nc2cnc(CN3CCNC3=O)nc2-c2ccccc2)c(F)cc1C(F)(F)F
CN(Cc1ccc(NC(=O)c2cc(-c3ccn(C)n3)c(cc2F)C(F)(F)F)c(n1)-c1ccccc1)C(N)=O
CN(Cc1ccc(NC(=O)c2cc(-c3ccn(C)n3)c(cc2F)C(F)(F)F)c(n1)-c1ccccc1)C(=O)NCCO
Cn1ccc(n1)-c1cc(C(=O)Nc2cnc(COC(N)=O)nc2-c2ccccc2)c(F)cc1C(F)(F)F
Cn1ccc(n1)-c1cc(C(=O)Nc2cc(cnc2-c2ccccc2)C(O)=O)c(F)cc1C(F)(F)F
CN(C)C(=O)c1cnc(c(NC(=O)c2cc(-c3ccn(C)n3)c(cc2F)C(F)(F)F)c1)-c1ccccc1
CNC(=O)c1cnc(c(NC(=O)c2cc(-c3ccn(C)n3)c(cc2F)C(F)(F)F)c1)-c1ccccc1
C[C@H](O)CNC(=O)c1cnc(c(NC(=O)c2cc(-c3ccn(C)n3)c(cc2F)C(F)(F)F)c1)-c1ccccc1 |r|
C[C@@H](CO)NC(=O)c1cnc(c(NC(=O)c2cc(-c3ccn(C)n3)c(cc2F)C(F)(F)F)c1)-c1ccccc1 |r|
Cc1cnn(c1)-c1ccc(cc1NC(=O)c1ccc(c(c1)-c1ccn(C)n1)C(F)(F)F)C(N)=O
Cn1ccc(n1)-c1cc(ccc1C(F)(F)F)C(=O)Nc1cc(C(N)=O)c(N)cc1-c1ccccc1
FC(F)(F)c1ccc(cc1-c1cc[nH]n1)C(=O)Nc1cnc(nc1-c1ccccc1)C(=O)N1CCOCC1
Cn1ccc(n1)-c1cc(ccc1C(F)(F)F)C(=O)Nc1cc(cnc1-c1ccccc1)C(N)=O
CN1CC(C1)NC(=O)c1cnc(c(NC(=O)c2cc(-c3cc[nH]n3)c(cc2F)C(F)(F)F)c1)-c1ccccc1
NC(=O)c1cnc(c(NC(=O)c2cc(-c3ncccn3)c(cc2F)C(F)(F)F)c1)-c1ccccc1
Fc1cc(c(cc1C(=O)Nc1cc(cnc1-c1ccccc1)C(=O)NCc1cccnc1)-c1ncccn1)C(F)(F)F
NC(=O)c1cnc(c(NC(=O)c2cc(-c3cc[nH]n3)c(cc2F)C(F)(F)F)c1)-c1ccccc1
Cn1ccc(n1)-c1cc(C(=O)Nc2cc(nnc2-c2ccccc2)C(N)=O)c(F)cc1C(F)(F)F
CN1CC(=O)N(Cc2ncc(NC(=O)c3cc(-c4ccn(C)n4)c(cc3F)C(F)(F)F)c(n2)-c2ccccc2)C1=O
Cn1ccc(n1)-c1cc(C(=O)Nc2cnc(CN3C(=O)CNC3=O)nc2-c2ccccc2)c(F)cc1C(F)(F)F
Cn1ccc(n1)-c1cc(C(=O)Nc2cnc(CN3C(=O)COC3=O)nc2-c2ccccc2)c(F)cc1C(F)(F)F
Cn1ccc(n1)-c1cc(C(=O)Nc2ccc(CN3C(=O)CNC3=O)nc2-c2ccccc2)c(F)cc1C(F)(F)F
Cn1ccc(n1)-c1cc(C(=O)Nc2cnc(CC(N)=O)nc2-c2ccccc2)c(F)cc1C(F)(F)F
CN(C)C(=O)Cc1ncc(NC(=O)c2cc(-c3ccn(C)n3)c(cc2F)C(F)(F)F)c(n1)-c1ccccc1
Cn1ccc(n1)-c1cc(C(=O)Nc2cnc(CC(N)=O)cc2-c2ccccc2)c(F)cc1C(F)(F)F
Cn1ccc(n1)-c1cc(C(=O)Nc2ccc(CC(N)=O)nc2-c2ccccc2)c(F)cc1C(F)(F)F
CNC(=O)Cc1ncc(NC(=O)c2ccc(c(c2)-c2ccn(C)n2)C(F)(F)F)c(n1)-c1ccccc1
CNC(=O)Cc1ncc(NC(=O)c2cc(-c3ccn(C)n3)c(cc2F)C(F)(F)F)c(n1)-c1ccccc1
CCNC(=O)Cc1ncc(NC(=O)c2cc(-c3ccn(C)n3)c(cc2F)C(F)(F)F)c(n1)-c1ccccc1
Cn1ccc(n1)-c1cc(C(=O)Nc2cnc(CC(O)=O)nc2-c2ccccc2)c(F)cc1C(F)(F)F
Cn1ccc(n1)-c1cc(C(=O)Nc2cnc(CC(=O)NC[C@@H]3CCCO3)nc2-c2ccccc2)c(F)cc1C(F)(F)F |r|
Cn1ccc(n1)-c1cc(C(=O)Nc2cnc(CC(=O)NCCO)nc2-c2ccccc2)c(F)cc1C(F)(F)F
Cn1ccc(n1)-c1cc(C(=O)Nc2cnc(CC(=O)N[C@@H]3C[C@H](O)C3)nc2-c2ccccc2)c(F)cc1C(F)(F)F |r,wU:20.20,22.23,(6.19,-6.32,;4.65,-6.32,;3.74,-7.57,;2.28,-7.09,;2.28,-5.55,;3.74,-5.07,;.94,-4.78,;.94,-3.24,;-.39,-2.47,;-.39,-.93,;-1.72,-.16,;.94,-.16,;.94,1.38,;-.39,2.15,;-.39,3.69,;.94,4.46,;.94,6,;-.39,6.77,;-.39,8.31,;-1.72,6,;-3.06,6.77,;-3.46,8.26,;-4.94,7.86,;-6.28,8.63,;-4.55,6.37,;2.28,3.69,;2.28,2.15,;3.61,1.38,;3.61,-.16,;4.94,-.93,;6.28,-.16,;6.28,1.38,;4.94,2.15,;-1.72,-3.24,;-3.06,-2.47,;-1.72,-4.78,;-.39,-5.6,;-.39,-7.14,;-.39,-8.68,;1.15,-7.14,;-1.93,-7.14,)|
Cn1ccc(n1)-c1cc(C(=O)Nc2cnc(CC(=O)N[C@H]3CCOC3)nc2-c2ccccc2)c(F)cc1C(F)(F)F |r|
Cn1ccc(n1)-c1cc(C(=O)Nc2cnc(CC(=O)N3CCOCC3)nc2-c2ccccc2)c(F)cc1C(F)(F)F
Cn1ccc(n1)-c1cc(C(=O)Nc2cnc(CC(=O)NCC3CCOC3)nc2-c2ccccc2)c(F)cc1C(F)(F)F
Cn1ccc(n1)-c1cc(C(=O)Nc2cnc(CC(=O)NC3CCC3)nc2-c2ccccc2)c(F)cc1C(F)(F)F
Cn1ccc(n1)-c1cc(C(=O)Nc2cnc(CC(=O)N3CCNCC3)nc2-c2ccccc2)c(F)cc1C(F)(F)F
CCN(C)C(=O)Cc1ncc(NC(=O)c2cc(-c3ccn(C)n3)c(cc2F)C(F)(F)F)c(n1)-c1ccccc1
Cn1ccc(n1)-c1cc(ccc1C(F)(F)F)C(=O)Nc1cnc(CC(N)=O)nc1-c1ccccc1
Cc1ccccc1-c1nc(CC(N)=O)ncc1NC(=O)c1cc(-c2ccn(C)n2)c(cc1F)C(F)(F)F
Cn1ccc(n1)-c1cc(C(=O)Nc2cnc(nc2-c2ccccc2)C(O)C(N)=O)c(F)cc1C(F)(F)F
Cn1ccc(n1)-c1cc(C(=O)Nc2cnc(nc2-c2ccccc2)C2(CC2)C(N)=O)c(F)cc1C(F)(F)F
Cn1ccc(n1)-c1cc(C(=O)Nc2ncc(CC(N)=O)nc2-c2ccccc2)c(F)cc1C(F)(F)F
Cn1ccc(n1)-c1cc(C(=O)Nc2cnc(nc2-c2ccccc2)C(C)(C)C(O)=O)c(F)cc1C(F)(F)F
Cn1ccc(n1)-c1cc(C(=O)Nc2cnc(nc2-c2ccccc2)C(C)(C)C(N)=O)c(F)cc1C(F)(F)F
NC(=O)Cc1ncc(NC(=O)c2cc(-c3ccccn3)c(cc2F)C(F)(F)F)c(n1)-c1ccccc1
NC(=O)Cc1ccc(NC(=O)c2cc(-c3ccccn3)c(cc2F)C(F)(F)F)c(n1)-c1ccccc1
NC(=O)Cc1ncc(NC(=O)c2cc(-c3ncccn3)c(cc2F)C(F)(F)F)c(n1)-c1ccccc1
NC(=O)Cc1ncc(NC(=O)c2cc(-c3cc[nH]n3)c(cc2F)C(F)(F)F)c(n1)-c1ccccc1
NC(=O)Cc1cc(c(NC(=O)c2cc(-c3ccccn3)c(cc2F)C(F)(F)F)cn1)-c1ccccc1
Cn1ccc(n1)-c1cc(C(=O)Nc2cnc(CCC(N)=O)nc2-c2ccccc2)c(F)cc1C(F)(F)F
Cn1ccc(n1)-c1cc(C(=O)Nc2cnc(Cc3nnc[nH]3)nc2-c2ccccc2)c(F)cc1C(F)(F)F
Cn1ccc(n1)-c1cc(C(=O)Nc2cnc(nc2-c2ccccc2)C(N)C(N)=O)c(F)cc1C(F)(F)F
Cn1ccc(n1)-c1cc(C(=O)Nc2cnc(nc2-c2ccccc2)C2NC(=O)NC2=O)c(F)cc1C(F)(F)F
CC(=O)NCc1cccc(c1)-c1nc(C)ncc1NC(=O)c1cc(-c2ccn(C)n2)c(cc1F)C(F)(F)F
CC(=O)Nc1cccc(c1)-c1nc(C)ncc1NC(=O)c1cc(-c2ccn(C)n2)c(cc1F)C(F)(F)F
Cc1ncc(NC(=O)c2cc(-c3ccn(C)n3)c(cc2F)C(F)(F)F)c(n1)-c1ccccc1CCN
CN(C)CCc1ccccc1-c1nc(C)ncc1NC(=O)c1cc(-c2ccn(C)n2)c(cc1F)C(F)(F)F
Cc1ncc(NC(=O)c2cc(-c3ccn(C)n3)c(cc2F)C(F)(F)F)c(n1)-c1ccccc1CO
OC[C@H]1CCCN1c1ncc(cc1NC(=O)c1cc(-c2ncccn2)c(cc1F)C(F)(F)F)-c1csc(n1)C1CC1 |r|
Cn1ccc(n1)-c1cnc(N2CCC[C@@H]2CO)c(NC(=O)c2cc(-c3ncccn3)c(cc2F)C(F)(F)F)c1 |r|
Fc1cc(c(cc1C(=O)Nc1cc2C(=O)NCCc2nc1-c1ccccc1)-c1ncccn1)C(F)(F)F
Cn1ccc(n1)-c1cc(ccc1C(F)(F)F)C(=O)Nc1cc2CN(CC(N)=O)CCc2nc1-c1ccccc1
Cn1ccc(n1)-c1cc(C(=O)Nc2cc3C(=O)NCCc3nc2-c2ccccn2)c(F)cc1C(F)(F)F
Cn1ccc(n1)-c1cc(ccc1C(F)(F)F)C(=O)Nc1cc2CC(=O)NCc2nc1-c1ccccc1
Cn1ccc(n1)-c1cc(ccc1C(F)(F)F)C(=O)Nc1cnc2CN(CCc2c1-c1ccccc1)C(=O)CO
Cn1ccc(n1)-c1cc(C(=O)Nc2cc3CCN(Cc3nc2-c2ccccc2)C(N)=O)c(F)cc1C(F)(F)F
Cn1ccc(n1)-c1cc(C(=O)Nc2cc3CNCCc3nc2-c2ccccc2)c(F)cc1C(F)(F)F
Fc1cc(c(cc1C(=O)Nc1cc2CNCCc2nc1-c1ccccc1)-c1ccccn1)C(F)(F)F
CC(=O)N1CCc2nc(c(NC(=O)c3ccc(c(c3)-c3ncccn3)C(F)(F)F)cc2C1)-c1ccccc1
CC(=O)N1CCc2nc(c(NC(=O)c3cc(-c4ncccn4)c(cc3F)C(F)(F)F)cc2C1)-c1ccccc1
CS(=O)(=O)N1CCc2nc(c(NC(=O)c3cc(-c4ncccn4)c(cc3F)C(F)(F)F)cc2C1)-c1ccccc1
CNC(=O)N1CCc2nc(c(NC(=O)c3cc(-c4ncccn4)c(cc3F)C(F)(F)F)cc2C1)-c1ccccc1
CC(=O)N1CCc2nc(c(NC(=O)c3cc(-c4ccn(C)n4)c(cc3Cl)C(F)(F)F)cc2C1)-c1ccccc1
Cn1ccc(n1)-c1cc(C(=O)Nc2cc3C(=O)NCCc3nc2-c2ccccc2)c(F)cc1C(F)(F)F
Cn1ccc(n1)-c1cc(C(=O)Nc2cc3CNC(=O)Cc3nc2-c2ccccc2)c(F)cc1C(F)(F)F
Cn1ccc(n1)-c1cc(C(=O)Nc2cc3CN(CCc3nc2-c2ccccc2)C(N)=O)c(F)cc1C(F)(F)F
NC(=O)N1CCc2nc(c(NC(=O)c3cc(-c4ncccn4)c(cc3F)C(F)(F)F)cc2C1)-c1ccccc1
Cn1ccc(n1)-c1cc(ccc1C(F)(F)F)C(=O)Nc1cc2CN(CCc2nc1-c1ccccc1)C(=O)CN
Cn1ccc(n1)-c1cc(ccc1C(F)(F)F)C(=O)Nc1cc2CN(CC(O)=O)CCc2nc1-c1ccccc1
Cn1ccc(n1)-c1cc(ccc1C(F)(F)F)C(=O)Nc1cc2CN(CCO)CCc2nc1-c1ccccc1
Cn1ccc(n1)-c1cc(ccc1C(F)(F)F)C(=O)Nc1cnc2C(=O)NCCc2c1-c1ccccc1
Cn1ccc(n1)-c1cc(ccc1C(F)(F)F)C(=O)Nc1cnc2CCN(Cc2c1-c1ccccc1)C(=O)CO
Cn1ccc(n1)-c1cc(C(=O)Nc2cc3C(=O)NCc3nc2-c2ccccc2)c(F)cc1C(F)(F)F
OCC(=O)N1Cc2cc(NC(=O)c3cc(-c4ncccn4)c(cc3F)C(F)(F)F)c(nc2C1)-c1ccccc1
C[C@@H](O)C(=O)N1CCc2nc(c(NC(=O)c3ccc(c(c3)-c3ccn(C)n3)C(F)(F)F)cc2C1)-c1ccccc1 |r|
Cn1ccc(n1)-c1cc(C(=O)Nc2cc(cnc2-c2ccccc2)-c2ccc(cn2)C(N)=O)c(F)cc1C(F)(F)F
NC(=O)c1ccc(cc1)-c1cnc(c(NC(=O)c2cc(-c3cc[nH]n3)c(cc2F)C(F)(F)F)c1)-c1ccccc1
CNC(=O)c1ccc(cc1)-c1cnc(c(NC(=O)c2cc(-c3cc[nH]n3)c(cc2F)C(F)(F)F)c1)-c1ccccc1
Fc1cc(c(cc1C(=O)Nc1cc(Oc2ccccn2)cnc1-c1ccccc1)-c1ncccn1)C(F)(F)F
OCc1ccc(nc1)-c1cnc(c(NC(=O)c2cc(-c3ncccn3)c(cc2F)C(F)(F)F)c1)-c1ccccc1
NC(=O)c1cnc(nc1)-c1cnc(c(NC(=O)c2cc(-c3ncccn3)c(cc2F)C(F)(F)F)c1)-c1ccccc1
CC(=O)NCc1cnc(nc1)-c1cnc(c(NC(=O)c2cc(-c3ncccn3)c(cc2F)C(F)(F)F)c1)-c1ccccc1
Cn1ccc(n1)-c1cc(C(=O)Nc2cc(cnc2-c2ccccc2)-c2ccc(cn2)C(O)=O)c(F)cc1C(F)(F)F
Cn1ccc(n1)-c1cc(C(=O)Nc2cc(cnc2-c2ccccc2)-c2ccc(cn2)C(C)(C)O)c(F)cc1C(F)(F)F
NC(=O)c1ccnc(n1)-c1cnc(c(NC(=O)c2cc(-c3ncccn3)c(cc2F)C(F)(F)F)c1)-c1ccccc1
CNC(=O)c1ccc(nc1)-c1cnc(c(NC(=O)c2cc(-c3ncccn3)c(cc2F)C(F)(F)F)c1)-c1ccccc1
NC(=O)c1ncc(cn1)-c1cnc(c(NC(=O)c2cc(-c3ncccn3)c(cc2F)C(F)(F)F)c1)-c1ccccc1
Fc1cc(c(cc1C(=O)Nc1cc(OCc2ccncc2)cnc1-c1ccccc1)-c1ncccn1)C(F)(F)F
NC(=O)N1CCN(CC1)c1cnc(c(NC(=O)c2cc(-c3ncccn3)c(cc2F)C(F)(F)F)c1)-c1ccccc1
CC(N)c1ccc(nc1)-c1cnc(c(NC(=O)c2cc(-c3ccn(C)n3)c(cc2F)C(F)(F)F)c1)-c1ccccc1
Cn1ccc(n1)-c1cc(C(=O)Nc2cnc(Cc3nnnn3C)nc2-c2ccccc2)c(F)cc1C(F)(F)F
CCn1c(Cc2ncc(NC(=O)c3cc(-c4ccn(C)n4)c(cc3F)C(F)(F)F)c(n2)-c2ccccc2)n[nH]c1=O
Cn1ccc(n1)-c1cc(C(=O)Nc2cc(cnc2-c2ccccc2)C2CCC(=O)N2)c(F)cc1C(F)(F)F
Cn1ccc(n1)-c1cc(C(=O)Nc2cnc(CN3CCN(CC3)S(C)(=O)=O)nc2-c2ccccc2)c(F)cc1C(F)(F)F
Cn1ccc(n1)-c1cc(C(=O)Nc2ccc(CN3CC4(COC4)C3)nc2-c2ccccc2)c(F)cc1C(F)(F)F
Cn1ccc(n1)-c1cc(C(=O)Nc2cnc(CN3C[C@H](O)[C@H](O)C3)nc2-c2ccccc2)c(F)cc1C(F)(F)F |r|
Fc1cc(c(cc1C(=O)Nc1cc2C(=O)NC(=O)c2nc1-c1ccccc1)-c1ncccn1)C(F)(F)F
Cn1ccc(n1)-c1cc(ccc1C(F)(F)F)C(=O)Nc1ccc(nc1-c1ccccc1)C1CCNC1=O
Cn1ccc(n1)-c1cc(C(=O)Nc2cnc(CN3C(=O)CCC3=O)nc2-c2ccccc2)c(F)cc1C(F)(F)F
Cn1ccc(n1)-c1cc(C(=O)Nc2cc3CNCc3nc2-c2ccccc2)c(F)cc1C(F)(F)F
Cn1ccc(n1)-c1cc(ccc1C(F)(F)F)C(=O)Nc1ccc(nc1-c1ccccc1)C1CCC(=O)N1
Cn1ccc(n1)-c1cc(ccc1C(F)(F)F)C(=O)Nc1cnc(CC2NC(=O)NC2=O)nc1-c1ccccc1
Cn1ccc(n1)-c1cc(C(=O)Nc2cnc(CC3CCNC3=O)nc2-c2ccccc2)c(F)cc1C(F)(F)F
Cn1ccc(n1)-c1cc(C(=O)Nc2ccc(nc2-c2ccccc2)C(O)CO)c(F)cc1C(F)(F)F
Cn1ccc(n1)-c1cc(C(=O)Nc2cnc(nc2-c2ccccc2)C2CCCNC2=O)c(F)cc1C(F)(F)F
Cn1ccc(n1)-c1cc(C(=O)Nc2cc(cnc2-c2ccccc2)S(C)(=O)=O)c(F)cc1C(F)(F)F
Cn1ccc(n1)-c1cc(C(=O)Nc2cc(cnc2-c2ccccc2)S(C)(=N)=O)c(F)cc1C(F)(F)F
Cn1ccc(n1)-c1cc(C(=O)Nc2ccc(nc2-c2ccccc2)C2COC(=O)N2)c(F)cc1C(F)(F)F
Cn1ccc(n1)-c1cc(C(=O)Nc2cnc(nc2-c2ccccc2)C2CCNC2=O)c(F)cc1C(F)(F)F
Cn1ccc(n1)-c1cc(C(=O)Nc2ccc(nc2-c2ccccc2)C2CNC(=O)C2)c(F)cc1C(F)(F)F
Cn1ccc(n1)-c1cc(C(=O)Nc2cnc(CS(C)(=O)=O)nc2-c2ccccc2)c(F)cc1C(F)(F)F
CNS(=O)(=O)Cc1ccc(NC(=O)c2cc(-c3ccn(C)n3)c(cc2F)C(F)(F)F)c(n1)-c1ccccc1
Cn1ccc(n1)-c1cc(C(=O)Nc2cnc(CC3CC(=O)NC3=O)nc2-c2ccccc2)c(F)cc1C(F)(F)F
Cn1ccc(n1)-c1cc(C(=O)Nc2cc(CC(N)=O)cnc2-c2ccccc2)c(F)cc1C(F)(F)F
Cn1ccc(n1)-c1cc(ccc1C(F)(F)F)C(=O)Nc1cc(CC(N)=O)cnc1-c1ccccc1
Fc1cc(c(cc1C(=O)Nc1cc(Cc2cnco2)cnc1-c1ccccc1)-c1ncccn1)C(F)(F)F
Cn1ccc(n1)-c1cc(C(=O)Nc2nc(CC(N)=O)ccc2-c2ccccc2)c(F)cc1C(F)(F)F
Cn1ccc(n1)-c1cc(C(=O)Nc2ccc(nc2-c2ccccc2)C2CN(C2)C(=O)CO)c(F)cc1C(F)(F)F
Cn1ccc(n1)-c1cc(C(=O)Nc2ccc(nc2-c2ccccc2)C2CN(C2)C(=O)CN)c(F)cc1C(F)(F)F
CC(=O)N1CC(C1)c1ccc(NC(=O)c2cc(-c3ccn(C)n3)c(cc2F)C(F)(F)F)c(n1)-c1ccccc1
Cn1ccc(n1)-c1cc(C(=O)Nc2cnc(NC(=O)CO)nc2-c2ccccc2)c(F)cc1C(F)(F)F
Cn1ccc(n1)-c1cc(ccc1C(F)(F)F)C(=O)Nc1cnc(NCCO)nc1-c1ccccc1
Cn1ccc(n1)-c1cc(C(=O)Nc2cnc(nc2-c2ccccc2)N2CCNC2=O)c(F)cc1C(F)(F)F
Cn1ccc(n1)-c1cc(C(=O)Nc2cnc(N)nc2-c2ccccc2)c(F)cc1C(F)(F)F
Cn1ccc(n1)-c1cc(C(=O)Nc2cnc(NCC(N)=O)nc2-c2ccccc2)c(F)cc1C(F)(F)F
Cn1ccc(n1)-c1cc(C(=O)Nc2ncc(CN3CCOC3=O)nc2-c2ccccc2)c(F)cc1C(F)(F)F
Cn1ccc(n1)-c1cc(C(=O)Nc2ccc(nc2-c2ccccc2)C2CNC(=O)N2)c(F)cc1C(F)(F)F
Cn1ccc(n1)-c1cc(C(=O)Nc2cnc(OCC(N)=O)nc2-c2ccccc2)c(F)cc1C(F)(F)F
CS(=N)(=O)c1ccc(cc1)-c1cnc(c(NC(=O)c2cc(-c3cc[nH]n3)c(cc2F)C(F)(F)F)c1)-c1ccccc1
Cn1ccc(n1)-c1cc(C(=O)Nc2cnc(CN3CCOC3=O)nc2-c2ccccc2)c(F)cc1C(F)(F)F
Cn1ccc(n1)-c1cc(C(=O)Nc2cnc(CN3CCCC3=O)nc2-c2ccccc2)c(F)cc1C(F)(F)F
Cn1ccc(n1)-c1cc(C(=O)Nc2cnc(CN3CCCCC3=O)nc2-c2ccccc2)c(F)cc1C(F)(F)F
Cn1ccc(n1)-c1cc(C(=O)Nc2cnc(CN3CCCCCC3=O)nc2-c2ccccc2)c(F)cc1C(F)(F)F
Cn1ccc(n1)-c1cc(C(=O)Nc2cnc(CN3CCCOC3=O)nc2-c2ccccc2)c(F)cc1C(F)(F)F
Cn1ccc(n1)-c1cc(C(=O)Nc2cnc(CN3CCOCC3=O)nc2-c2ccccc2)c(F)cc1C(F)(F)F
Cn1ccc(n1)-c1cc(ccc1C(F)(F)F)C(=O)Nc1cnc(Cn2ccnc2)nc1-c1ccccc1
Cn1ccc(n1)-c1cc(C(=O)Nc2cnc(Cn3cccnc3=O)nc2-c2ccccc2)c(F)cc1C(F)(F)F
Cn1ccc(n1)-c1cc(C(=O)Nc2cnc(Cn3ccc(=O)[nH]c3=O)nc2-c2ccccc2)c(F)cc1C(F)(F)F
Cn1ccc(n1)-c1cc(C(=O)Nc2cnc(Cn3cn[nH]c3=O)nc2-c2ccccc2)c(F)cc1C(F)(F)F
Cn1ccc(n1)-c1cc(C(=O)Nc2cnc(CN3CC(CO)OC3=O)nc2-c2ccccc2)c(F)cc1C(F)(F)F
CNC(=O)CC1(O)CCN(C(=O)Nc2cnc3[nH]nc(N4CCC[C@@H]4c4cc(F)ccc4F)c3c2)C1
O=C(Nc1cnc2[nH]nc(N3CCC[C@@H]3c3cc(F)ccc3F)c2c1)N1CC[C@H](O)C1
O=C(Nc1cnc2[nH]nc(N3CCC[C@@H]3c3cc(F)ccc3F)c2c1)c1ccc(N2CC[C@H](O)C2)nc1
NC(=O)c1cnc2[nH]nc(N3CCC[C@@H]3c3cc(F)ccc3F)c2c1
NC(=O)c4cnc3[nH]nc(N1C[C@@H](F)C[C@@H]1c2cc(F)ccc2F)c3c4
O=C(NCCO)c1cnc2[nH]nc(N3CCC[C@@H]3c3cc(F)ccc3F)c2c1
CNC(=O)c1cnc2[nH]nc(N3CCC[C@@H]3c3cc(F)ccc3F)c2c1
COCCNC(=O)c1cnc2[nH]nc(N3CCC[C@@H]3c3cc(F)ccc3F)c2c1
O=C(NCCCO)c1cnc2[nH]nc(N3CCC[C@@H]3c3cc(F)ccc3F)c2c1
CC(C)(O)CNC(=O)c1cnc2[nH]nc(N3CCC[C@@H]3c3cc(F)ccc3F)c2c1
O=C(Nc1cnc2[nH]nc(N3C[C@@H](F)C[C@@H]3c3cc(F)ccc3F)c2c1)c1ccc(N2CC[C@H](O)C2)nc1
O=C(NCCCCO)c1cnc2[nH]nc(N3CCC[C@@H]3c3cc(F)ccc3F)c2c1
COC(=O)c1cnc2[nH]nc(N3C[C@@H](F)C[C@@H]3c3cc(F)ccc3F)c2c1
O=C(N[C@H]1CC[C@@H](O)CC1)c1cnc2[nH]nc(N3CCC[C@@H]3c3cc(F)ccc3F)c2c1
NC(=O)CCNC(=O)c1cnc2[nH]nc(N3CCC[C@@H]3c3cc(F)ccc3F)c2c1
CC1(O)CCN(c2cnc(C(=O)Nc3cnc4[nH]nc(N5C[C@@H](F)C[C@@H]5c5cc(F)ccc5F)c4c3)cn2)C1
O=C(O)c1cnc2[nH]nc(N3C[C@@H](F)C[C@@H]3c3cc(F)ccc3F)c2c1
CN(C)C(=O)c1cnc2[nH]nc(N3C[C@@H](F)C[C@@H]3c3cc(F)ccc3F)c2c1
CC(C)OC(=O)c1cnc2[nH]nc(N3C[C@@H](F)C[C@@H]3c3cc(F)ccc3F)c2c1
Fc1ccc(F)c([C@H]2C[C@H](F)CN2c2n[nH]c3ncc(-c4cn[nH]c4)cc23)c1
Fc1ccc(F)c([C@H]2C[C@H](F)CN2c2n[nH]c3ncc(-c4nn[nH]n4)cc23)c1
Fc1ccc(F)c([C@H]2C[C@H](F)CN2c2n[nH]c3ncc(-c4cnn(C5CCNCC5)c4)cc23)c1
O=C1CC(n2cc(-c3cnc4[nH]nc(N5C[C@@H](F)C[C@@H]5c5cc(F)ccc5F)c4c3)cn2)CCN1
Fc1ccc(F)c([C@H]2C[C@H](F)CN2c2n[nH]c3ncc(-c4cnn([C@@H]5CCNC5)c4)cc23)c1
Fc1ccc(F)c([C@H]2C[C@H](F)CN2c2n[nH]c3ncc(-c4cnn([C@H]5CCNC5)c4)cc23)c1
Fc1ccc(F)c([C@H]2C[C@H](F)CN2c2n[nH]c3ncc(-c4cnn(C5CNC5)c4)cc23)c1
CS(=O)(=O)n1cc(-c2cnc3[nH]nc(N4C[C@@H](F)C[C@@H]4c4cc(F)ccc4F)c3c2)cn1
Fc1ccc(F)c([C@H]2C[C@H](F)CN2c2n[nH]c3ncc(-c4cnn(C5CCOCC5)c4)cc23)c1
CN1CC(n2cc(-c3cnc4[nH]nc(N5C[C@@H](F)C[C@@H]5c5cc(F)ccc5F)c4c3)cn2)C1
Fc1ccc(F)c([C@H]2C[C@H](F)CN2c2n[nH]c3ncc(-c4cnn(CC(F)F)c4)cc23)c1
Fc1ccc(F)c([C@H]2C[C@H](F)CN2c2n[nH]c3ncc(-c4cnn(COCc5ccccc5)c4)cc23)c1
CC(C)(O)Cn1cc(-c2cnc3[nH]nc(N4C[C@@H](F)C[C@@H]4c4cc(F)ccc4F)c3c2)cn1
CN(C)CCn1cc(-c2cnc3[nH]nc(N4C[C@@H](F)C[C@@H]4c4cc(F)ccc4F)c3c2)cn1
Fc1ccc(F)c([C@H]2C[C@H](F)CN2c2n[nH]c3ncc(-c4cnn(CC5CNC5)c4)cc23)c1
Fc1ccc(F)c([C@H]2C[C@H](F)CN2c2n[nH]c3ncc(-c4cnn(CC(F)(F)F)c4)cc23)c1
Fc1ccc(F)c([C@H]2C[C@H](F)CN2c2n[nH]c3ncc(-c4ccn(CC(F)F)n4)cc23)c1
COCC1=NNC(c2cnc3[nH]nc(N4C[C@@H](F)C[C@@H]4c4cc(F)ccc4F)c3c2)O1
COCC1=NNC(c2cnc3c(c2)c(N2C[C@@H](F)C[C@@H]2c2cc(F)ccc2F)nn3COC)O1
NNC(=O)c1cnc2[nH]nc(N3C[C@@H](F)C[C@@H]3c3cc(F)ccc3F)c2c1
Cc1cn(CC(F)F)nc1-c1cnc2[nH]nc(N3C[C@@H](F)C[C@@H]3c3cc(F)ccc3F)c2c1
Fc1ccc(F)c([C@H]2C[C@H](F)CN2c2n[nH]c3ncc(-c4nnc(COC(F)(F)F)o4)cc23)c1
CC(C)OCc1nnc(-c2cnc3[nH]nc(N4C[C@@H](F)C[C@@H]4c4cc(F)ccc4F)c3c2)o1
O=C(c1n[nH]c2nccc(N[C@@H]3CCC[C@H]3O)c12)N1C[C@@H](F)C[C@@H]1c1cc(F)ccc1F
Fc1cc(c(cc1C(=O)Nc1n(nc2cccnc12)-c1ccccc1)-c1ncccn1)C(F)(F)F
Fc1cc(c(cc1C(=O)Nc1n(nc2ccc(=O)[nH]c12)-c1ccccc1)-c1ncccn1)C(F)(F)F
OCc1cccc(c1)-n1nc2cccnc2c1NC(=O)c1cc(-c2ncccn2)c(cc1F)C(F)(F)F
Cn1ccc(n1)-c1cc(ccc1C(F)(F)F)C(=O)Nc1n(nc2ccc(cc12)C#N)-c1ccccc1
Cn1ccc(n1)-c1cc(C(=O)Nc2n(nc3cccnc23)-c2ccccc2)c(F)cc1C(F)(F)F
Cn1ccc(n1)-c1cc(C(=O)Nc2n(nc3ncccc23)-c2ccccc2)c(F)cc1C(F)(F)F
Cn1ccc(n1)-c1cc(C(=O)Nc2n(nc3ccc(cc23)C(F)(F)F)-c2ccccc2)c(F)cc1C(F)(F)F
OCc1ccc2nn(c(NC(=O)c3cc(-c4ncccn4)c(cc3F)C(F)(F)F)c2n1)-c1ccccc1
CC(=O)NCc1cccc(c1)-n1nc2cccnc2c1NC(=O)c1cc(-c2ncccn2)c(cc1F)C(F)(F)F
Cn1ccc(n1)-c1cc(ccc1C(F)(F)F)C(=O)Nc1n(nc2ccc(CO)cc12)-c1ccccc1
OCc1cc2c(NC(=O)c3cc(-c4ncccn4)c(cc3F)C(F)(F)F)n(nc2cn1)-c1ccccc1
OCc1ccc2nn(c(NC(=O)c3cc(-c4ncccn4)c(cc3F)C(F)(F)F)c2c1)-c1ccccc1
OCc1ccc2c(NC(=O)c3cc(-c4ncccn4)c(cc3F)C(F)(F)F)n(nc2c1)-c1ccccc1
OCc1ccc2c(NC(=O)c3cc(-c4cc[nH]n4)c(cc3F)C(F)(F)F)n(nc2c1)-c1ccccc1
Cc1cc(n[nH]1)-n1nc2ccc(CO)cc2c1NC(=O)c1cc(-c2ncccn2)c(cc1F)C(F)(F)F
OCc1ccc2c(NC(=O)c3cc(-c4ncccn4)c(cc3Cl)C(F)(F)F)n(nc2c1)-c1ccccc1
OCc1ccc2nn(c(NC(=O)c3cc(-c4ncccn4)c(cc3Cl)C(F)(F)F)c2n1)-c1ccccc1
Cn1ccc(n1)-c1cc(C(=O)Nc2n(nc3cnc(CO)cc23)-c2ccccc2)c(F)cc1C(F)(F)F
CC(O)c1ccc2c(NC(=O)c3cc(-c4ncccn4)c(cc3F)C(F)(F)F)n(nc2c1)-c1ccccc1
CC(O)c1cnc2c(NC(=O)c3cc(-c4cc[nH]n4)c(cc3F)C(F)(F)F)n(nc2c1)-c1ccccc1
CC(O)c1ccc2nn(c(NC(=O)c3ccc(c(c3)-c3ccn(C)n3)C(F)(F)F)c2c1)-c1ccccc1
CC(O)c1ccc2nn(c(NC(=O)c3cc(-c4ncccn4)c(cc3F)C(F)(F)F)c2c1)-c1ccccc1
CC(O)c1ccc2nn(c(NC(=O)c3cc(-c4ncccn4)c(cc3F)C(F)(F)F)c2n1)-c1ccccc1
CC(O)c1cnc2c(NC(=O)c3cc(-c4ncccn4)c(cc3F)C(F)(F)F)n(nc2c1)-c1ccccc1
CC(O)c1ccc2nn(c(NC(=O)c3cc(-c4cc[nH]n4)c(cc3F)C(F)(F)F)c2n1)-c1ccccc1
CC(O)c1cnc2c(NC(=O)c3cc(-c4ccn(C)n4)c(cc3F)C(F)(F)F)n(nc2c1)-c1ccccc1
CC(O)c1cnc2c(NC(=O)c3cc(-c4ncccn4)c(cc3Cl)C(F)(F)F)n(nc2c1)-c1ccccc1
CC(O)c1ccc2c(NC(=O)c3cc(-c4ncccn4)c(cc3Cl)C(F)(F)F)n(nc2c1)-c1ccccc1
CC(O)c1cc2nn(c(NC(=O)c3cc(-c4ncccn4)c(cc3F)C(F)(F)F)c2cn1)-c1ccccc1
CC(C)(O)c1cnc2c(NC(=O)c3cc(-c4ncccn4)c(cc3F)C(F)(F)F)n(nc2c1)-c1ccccc1
Cn1ccc(n1)-c1cc(C(=O)Nc2n(nc3cc(cnc23)C(C)(C)O)-c2ccccc2)c(F)cc1C(F)(F)F
CC(C)(O)c1ccc2c(NC(=O)c3cc(-c4ncccn4)c(cc3F)C(F)(F)F)n(nc2c1)-c1ccccc1
Cn1ccc(n1)-c1cc(C(=O)Nc2n(nc3cnc(nc23)C(C)(C)O)-c2ccccc2)c(F)cc1C(F)(F)F
CC(C)(O)c1ccc2nn(c(NC(=O)c3cc(-c4ncccn4)c(cc3F)C(F)(F)F)c2c1)-c1ccccc1
CC(C)(O)c1cnc2nn(c(NC(=O)c3cc(-c4ncccn4)c(cc3F)C(F)(F)F)c2c1)-c1ccccc1
CC(C)(O)c1ccc2c(NC(=O)c3cc(-c4ncccn4)c(cc3Cl)C(F)(F)F)n(nc2c1)-c1ccccc1
CC(C)(O)c1cnc2c(NC(=O)c3cc(-c4cc[nH]n4)c(cc3F)C(F)(F)F)n(nc2c1)-c1ccccc1
Cn1ccc(n1)-c1cc(ccc1C(F)(F)F)C(=O)Nc1n(nc2cc(cnc12)C(C)(C)O)-c1ccccc1
OC1(CC1)c1cnc2c(NC(=O)c3cc(-c4ncccn4)c(cc3F)C(F)(F)F)n(nc2c1)-c1ccccc1
Cn1ccc(n1)-c1cc(ccc1C(F)(F)F)C(=O)Nc1n(nc2ccc(cc12)C1(O)CC1)-c1ccccc1
OC(c1ccc2c(NC(=O)c3cc(-c4ncccn4)c(cc3F)C(F)(F)F)n(nc2c1)-c1ccccc1)C(F)(F)F
OC(c1ccc2nn(c(NC(=O)c3cc(-c4ncccn4)c(cc3F)C(F)(F)F)c2c1)-c1ccccc1)C(F)(F)F
OC(C(F)F)c1ccc2c(NC(=O)c3cc(-c4ncccn4)c(cc3F)C(F)(F)F)n(nc2c1)-c1ccccc1
OC(C(F)F)c1ccc2nn(c(NC(=O)c3cc(-c4ncccn4)c(cc3F)C(F)(F)F)c2c1)-c1ccccc1
OCCc1ccc2c(NC(=O)c3cc(-c4ncccn4)c(cc3F)C(F)(F)F)n(nc2c1)-c1ccccc1
OCCc1ccc2nn(c(NC(=O)c3cc(-c4ncccn4)c(cc3F)C(F)(F)F)c2c1)-c1ccccc1
Cn1ccc(n1)-c1cc(ccc1C(F)(F)F)C(=O)Nc1n(nc2cc(ccc12)C(C)(O)CO)-c1ccccc1
OCC(O)c1cnc2c(NC(=O)c3cc(-c4ncccn4)c(cc3Cl)C(F)(F)F)n(nc2c1)-c1ccccc1
NCc1cnc2c(NC(=O)c3cc(-c4ncccn4)c(cc3F)C(F)(F)F)n(nc2c1)-c1ccccc1
CN(C)Cc1ccc2nn(c(NC(=O)c3ccc(c(c3)-c3ccn(C)n3)C(F)(F)F)c2c1)-c1ccccc1
CC(N)c1ccc2c(NC(=O)c3cc(-c4ncccn4)c(cc3F)C(F)(F)F)n(nc2c1)-c1ccccc1
Cn1ccc(n1)-c1cc(C(=O)Nc2n(nc3cc(CN)ccc23)-c2ccccc2)c(F)cc1C(F)(F)F
Cn1ccc(n1)-c1cc(C(=O)Nc2n(nc3cc(CNCCO)ccc23)-c2ccccc2)c(F)cc1C(F)(F)F
NC(=O)c1ccc2c(NC(=O)c3cc(-c4ncccn4)c(cc3F)C(F)(F)F)n(nc2c1)-c1ccccc1
Cn1ccc(n1)-c1cc(C(=O)Nc2n(nc3cc(ccc23)C(N)=O)-c2ccccc2)c(F)cc1C(F)(F)F
NC(=O)c1cnc2c(NC(=O)c3cc(-c4ncccn4)c(cc3F)C(F)(F)F)n(nc2c1)-c1ccccc1
NC(=O)c1cc2nn(c(NC(=O)c3cc(-c4ncccn4)c(cc3F)C(F)(F)F)c2cn1)-c1ccccc1
Cc1ccccc1-n1nc2cc(ccc2c1NC(=O)c1cc(-c2ccn(C)n2)c(cc1F)C(F)(F)F)C(N)=O
NC(=O)c1ccc2c(NC(=O)c3cc(-c4cc[nH]n4)c(cc3F)C(F)(F)F)n(nc2c1)-c1ccccc1
Cn1ccc(n1)-c1cc(ccc1C(F)(F)F)C(=O)Nc1n(nc2ccc(cc12)C(N)=O)-c1ccccc1
NC(=O)c1ccc2nn(c(NC(=O)c3cc(-c4ncccn4)c(cc3F)C(F)(F)F)c2n1)-c1ccccc1
NC(=O)c1ccc2c(NC(=O)c3cc(-c4ccccn4)c(cc3F)C(F)(F)F)n(nc2c1)-c1ccccc1
Cn1ccc(n1)-c1cc(ccc1C(F)(F)F)C(=O)Nc1n(nc2cc(ccc12)C(N)=O)-c1ccccc1
NC(=O)c1ccc2c(NC(=O)c3cc(-c4ccccn4)c(cc3Cl)C(F)(F)F)n(nc2c1)-c1ccccc1
NC(=O)c1cnc2c(NC(=O)c3cc(-c4ccccn4)c(cc3F)C(F)(F)F)n(nc2c1)-c1ccccc1
NC(=O)c1cnc2c(NC(=O)c3cc(-c4ccccn4)c(cc3Cl)C(F)(F)F)n(nc2c1)-c1ccccc1
Cn1ccc(n1)-c1cc(ccc1C(F)(F)F)C(=O)Nc1n(nc2cc(cnc12)C(N)=O)-c1ccccc1
Cn1ccc(n1)-c1cc(C(=O)Nc2n(nc3cc(cnc23)C(N)=O)-c2ccccc2)c(F)cc1C(F)(F)F
NC(=O)c1cnc2c(NC(=O)c3ccc(c(c3)-c3ncccn3)C(F)(F)F)n(nc2c1)-c1ccccc1
NC(=O)c1cccc2c(NC(=O)c3cc(-c4ncccn4)c(cc3F)C(F)(F)F)n(nc12)-c1ccccc1
OCCNC(=O)c1ccc2c(NC(=O)c3cc(-c4ncccn4)c(cc3Cl)C(F)(F)F)n(nc2c1)-c1ccccc1
Cc1ccccc1-n1nc2cc(cnc2c1NC(=O)c1cc(-c2ncccn2)c(cc1F)C(F)(F)F)C(N)=O
OCCNC(=O)c1ccc2c(NC(=O)c3cc(-c4ncccn4)c(cc3F)C(F)(F)F)n(nc2c1)-c1ccccc1
Cc1ccccc1-n1nc2cc(ccc2c1NC(=O)c1cc(-c2ncccn2)c(cc1F)C(F)(F)F)C(N)=O
NC(=O)Cc1ccc2c(NC(=O)c3cc(-c4ncccn4)c(cc3F)C(F)(F)F)n(nc2c1)-c1ccccc1
Cn1ccc(n1)-c1cc(C(=O)Nc2n(nc3c(CC(N)=O)cccc23)-c2ccccc2)c(F)cc1C(F)(F)F
CNC(=O)Cc1ccc2c(NC(=O)c3cc(c(C)cc3F)-c3ncccn3)n(nc2c1)-c1ccccc1
Cc1cc(Cl)c(cc1-c1ncccn1)C(=O)Nc1n(nc2cc(CC(N)=O)cnc12)-c1ccccc1
OCC(=O)NCc1ccc2c(NC(=O)c3cc(-c4ncccn4)c(cc3F)C(F)(F)F)n(nc2c1)-c1ccccc1
Cn1ccc(n1)-c1cc(C(=O)Nc2n(nc3c(CN4C(=O)CNC4=O)ccnc23)-c2ccccc2)c(F)cc1C(F)(F)F
Cn1ccc(n1)-c1cc(ccc1C(F)(F)F)C(=O)Nc1n(nc2cc(ccc12)[C@@H](N)C(F)(F)F)-c1ccccc1 |r|
Cn1ccc(n1)-c1cc(ccc1C(F)(F)F)C(=O)Nc1n(nc2cc(ccc12)[C@H](N)C(F)(F)F)-c1ccccc1 |r|
Fc1cc(c(cc1C(=O)Nc1n(nc2cc(ccc12)C1CCCN1)-c1ccccc1)-c1ncccn1)C(F)(F)F
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2ccc(C)nc2)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2ccnc(C)c2)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cccnc2F)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cccnc2C)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cncc(C)c2)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cncc(OC)c2)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cncc(c2)C#N)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2ccc(OC)nc2)[C@@H](C1)c1ccc(F)c(F)c1 |r|
CCOc1ncc(cn1)-c1nn(c(NC(=O)N[C@@H]2CN(CCOC)C[C@H]2c2ccc(F)c(F)c2)c1C)-c1ccccc1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc(nc2)C2CC2)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc(nc2)C2CC2)[C@@H](C1)c1ccc(F)cc1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc(OC)nc2)[C@@H](C1)c1cc(F)cc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc(C)nc2)[C@@H](C1)c1ccc(F)cc1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc(C)nc2)[C@@H](C1)c1cc(F)cc(F)c1 |r|
CCOc1ncc(cn1)-c1nn(c(NC(=O)N[C@@H]2CN(CCOC)C[C@H]2c2ccc(F)cc2)c1C)-c1ccccc1 |r|
CCOc1ncc(cn1)-c1nn(c(NC(=O)N[C@@H]2CN(CCOC)C[C@H]2c2cc(F)cc(F)c2)c1C)-c1ccccc1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2ccc(=O)n(C)n2)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2ccc(=O)n(C)n2)[C@@H](C1)c1ccc(F)cc1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2ccc(=O)n(C)n2)[C@@H](C1)c1cc(F)cc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc(NC3CC3)nc2)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc(NC3CC3)nc2)[C@@H](C1)c1ccc(F)cc1 |r|
COCCN1CC(NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2ccc(=O)n(C)c2)[C@@H](C1)c1ccc(F)c(Cl)c1 |r|
COCCN1CC(NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2ccc(=O)n(C)c2)[C@@H](C1)c1ccc(Cl)c(F)c1 |r|
COCCN1CC(NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2ccc(=O)n(C)c2)[C@@H](C1)c1cc(F)cc(Cl)c1 |r|
COCCN1CC(NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2ccc(=O)n(C)c2)[C@@H](C1)c1cccc(Cl)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2ccc(=O)n(C)c2)[C@@H](C1)c1cc(F)c(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2ccc(=O)n(C)c2)[C@@H](C1)c1cccc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc(=O)n(C)c2)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cc(C)c(=O)n(C)c2)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)S(C)(=O)=O)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)C(C)=O)[C@@H](C1)c1ccc(F)c(F)c1 |r|
O=C(Nc1c(nc2ccccn12)-c1ccccc1)Nc1c(nc2ccccn12)-c1ccccc1
O=C(Nc1cc(nn1-c1ccccc1)-c1ccccc1)Nc1ccccn1
Cc1cc(NC(=O)Nc2cc(C)nn2-c2ccccc2)n(n1)-c1ccccc1
Cc1cc(NC(=O)Nc2cccc3ccccc23)n(n1)-c1ccccc1
Cc1cc(NC(=O)Nc2cccc(Br)n2)n(n1)-c1ccccc1
Cc1cc(NC(=O)Nc2ccccc2-c2ccccc2)n(n1)-c1ccccc1
Cc1cc(NC(=O)Nc2cccc(C)c2C)n(n1)-c1ccccc1
Cc1cc(NC(=O)Nc2cc(Br)ccn2)n(n1)-c1ccccc1
O=C(Nc1cc(nn1-c1ccccc1)-c1ccncc1)Nc1ccccn1
Cc1cc(NC(=O)Nc2ccccn2)n(n1)-c1ccccc1
COc1ccc(NC(=O)Nc2cc(C)nn2-c2ccccc2)nc1
Cc1ccc(NC(=O)Nc2ccccn2)c(n1)-c1ccccc1
Cc1ncc(NC(=O)Nc2ccccc2-c2ccccc2)c(n1)-c1ccccc1
Cc1onc(c1NC(=O)NCc1ccccc1C(F)(F)F)-c1ccccc1
Cc1ncc(NC(=O)Nc2cccc3ccccc23)c(n1)-c1ccccc1
O=C(Nc1c(nc2sccn12)-c1ccccc1)Nc1cccc2ccccc12
Cc1ncc(NC(=O)Nc2cnc(C)nc2-c2ccccc2)c(n1)-c1ccccc1
CSc1ncc(NC(=O)Nc2cnc(SC)nc2-c2ccccc2)c(n1)-c1ccccc1
Cc1ncc(NC(=O)Nc2c([nH]c3ccccc23)-c2ccccc2)c(n1)-c1ccccc1
Cc1ncc(NC(=O)Nc2ccccn2)c(n1)-c1ccccc1
Cc1ncc(NC(=O)Nc2c(nc3ccccn23)-c2ccccc2)c(n1)-c1ccccc1
FC(F)(F)c1ccc(NC(=O)Nc2c(nc3ccccn23)-c2ccccc2)c(Cl)c1
FC(F)(F)c1ccc(NC(=O)Nc2c(nc3ccccn23)-c2ccccc2)cc1
O=C(Nc1c(nc2ccccn12)-c1ccccc1)Nc1cccnc1-c1ccccc1
Cc1cc(NC(=O)Nc2c(nc3ccccn23)-c2ccccc2)n(n1)-c1ccccc1
Cc1nc(c(NC(=O)Nc2c(nc3ccccn23)-c2ccccc2)s1)-c1ccccc1
Cn1ccnc1-c1cccc(NC(=O)Nc2c(nc3ccccn23)-c2ccccc2)c1
CCOC(=O)c1nc2ccccn2c1NC(=O)Nc1c(nc2ccccn12)-c1ccccc1
O=C(Nc1c(nc2ccccn12)-c1ccccc1)Nc1c(nc2ccccn12)-n1cccn1
O=C(Nc1c(nc2ccccn12)-c1ccccc1)Nc1c(nc2ncccn12)-c1ccccc1
Clc1ccc2nc(c(NC(=O)Nc3c(nc4ccccn34)-c3ccccc3)n2n1)-c1ccccc1
CNC(=O)c1nc2ccccn2c1NC(=O)Nc1c(nc2ccccn12)-c1ccccc1
Cc1nc(c(NC(=O)Nc2c(ncn2C)-c2ccccc2)s1)-c1ccccc1
Cc1nc(c(NC(=O)Nc2c(nc(C)n2C)-c2ccccc2)s1)-c1ccccc1
Cc1nc(c(NC(=O)Nc2sc(C)nc2-c2ccccc2)s1)-c1ccccc1
Cc1nc(c(NC(=O)Nc2cnc(C)nc2-c2ccccc2)s1)-c1ccccc1
Cc1nc(c(NC(=O)Nc2cccnc2-c2ccccc2)s1)-c1ccccc1
Fc1ccc(c(CNC(=O)Nc2ccnn2-c2ccccc2)c1)C(F)(F)F
Fc1ccc(CNC(=O)Nc2ccnn2-c2ccccc2)c(c1)C(F)(F)F
Cc1ncc(NC(=O)NCc2ccccc2SC(F)(F)F)c(n1)-c1ccccc1
C[C@H](NC(=O)Nc1cnc(C)nc1-c1ccccc1)C1CCCCC1 |r|
Cn1ncc(NC(=O)NCc2ccccc2C(F)(F)F)c1-c1ccccc1
Cc1ncc(NC(=O)NCc2cc(F)ccc2C(F)(F)F)c(n1)-c1ccccc1
FC(F)(F)Sc1ccccc1CNC(=O)Nc1ccnn1-c1ccccc1
Cc1onc(c1NC(=O)NCc1ccccc1OC(F)(F)F)-c1ccccc1
Cn1ncc(NC(=O)NCc2ccccc2OC(F)(F)F)c1-c1ccccc1
CC1Oc2ccn3ncc(C(=O)NCCOc4ccc(F)c(Cl)c14)c3n2
CN1Cc2cc(F)ccc2OCCNC(=O)c2cnn3ccc1nc23
CN1Cc2c(Cl)c(F)ccc2OCCNC(=O)c2cnn3ccc1nc23
CC1Oc2ccc3ncc(C(=O)NCCOc4ccc(F)cc14)n3n2
CN1Cc2cc(F)ccc2OCCNC(=O)c2cnc3ccc1nn23
CCN1Cc2cc(F)ccc2OCCNC(=O)c2cnn3ccc1nc23
CC(C)N1Cc2cc(F)ccc2OCCNC(=O)c2cnn3ccc1nc23
CN1Cc2ccccc2OCCNC(=O)c2cnn3ccc1nc23
Fc1ccc2OCCNC(=O)c3cnn4ccc(NCc2c1)nc34
CC1Nc2ccn3ncc(C(=O)NCCOc4ccc(F)cc14)c3n2
C[C@H]1Nc2ccn3ncc(C(=O)NCCOc4ccc(F)cc14)c3n2 |r|
CC1Nc2ccn3ncc(C(=O)NCCOc4ccc(F)c(Cl)c14)c3n2
CN1Cc2cc(F)ccc2OCCCNC(=O)c2cnn3ccc1nc23
CC(C)(CO)CNC(=O)c1cnn2ccc(nc12)N1CCCC1c1cncc(F)c1
Fc1cncc(c1)C1CCCN1c1ccn2ncc(C(=O)N3CCC3)c2n1
C[C@@H](NC(=O)c1cnn2ccc(nc12)N1CCC[C@@H]1c1cncc(F)c1)C(F)(F)F |r|
Fc1cncc(c1)C1CCCN1c1ccn2ncc(C(=O)NCC(F)(F)F)c2n1
CC(C)(CO)NC(=O)c1cnn2ccc(nc12)N1CCCC1c1cncc(F)c1
O[C@@H]1CCC[C@H]1NC(=O)c1cnn2ccc(nc12)N1CCCC1c1cncc(F)c1 |r|
FC(F)CNC(=O)c1cnn2ccc(nc12)N1CCCC1c1cncc(F)c1
O[C@H]1CCC[C@H]1NC(=O)c1cnn2ccc(nc12)N1CCCC1c1cncc(F)c1 |r|
Cc1ncc(F)cc1[C@H]1CCCN1c1ccn2ncc(C(=O)NC3CCC3)c2n1 |r|
Cc1ncc(F)cc1[C@H]1CCCN1c1ccn2ncc(C(=O)NC3(C)CC3)c2n1 |r|
CCc1ncc(F)cc1[C@H]1CCCN1c1ccn2ncc(C(=O)N[C@H]3CC[C@H](O)C3)c2n1 |r|
Cc1nc(c(NC(=O)c2ccc(cc2F)C(F)(F)F)s1)-c1ccccc1
FC(F)(F)c1ccc(C(=O)Nc2cc(nn2-c2ccccc2)C(=O)NC2CC2)c(Cl)c1
Cc1csc(n1)-c1cc(ccc1C(F)(F)F)C(=O)Nc1cc(C)nn1-c1ccccc1
NC(=O)c1ccc(nc1)-c1cc(NC(=O)c2ccc(cc2Cl)C(F)(F)F)n(n1)-c1ccccc1
Cc1csc(n1)-c1cc(ccc1C(F)(F)F)C(=O)Nc1cc(nn1-c1cc(C)[nH]n1)-c1cnn(C)c1
Cc1csc(n1)-c1cc(ccc1C(F)(F)F)C(=O)Nc1cc(nn1-c1cc(C)[nH]n1)-c1ccccn1
CN(C)C(=O)c1cc(NC(=O)c2ccc(c(c2)-c2ccn(C)n2)C(F)(F)F)n(n1)-c1cc(C)n[nH]1
Cc1cc(n[nH]1)-n1nc(cc1NC(=O)c1ccc(c(c1)-c1cccnc1)C(F)(F)F)-c1cnn(C)c1
Cn1ccc(n1)-c1cc(ccc1C(F)(F)F)C(=O)Nc1cc(nn1-c1ccc(F)c(F)c1)-c1ccncc1
FC(F)(F)c1ccc(C(=O)Nc2cc(nn2-c2ccccc2)-c2ccc(=O)[nH]n2)c(Cl)c1
Cn1ccc(n1)-c1cc(ccc1C(F)(F)F)C(=O)Nc1cc(nn1-c1ccccc1)-c1ccc(=O)[nH]n1
Cn1ccc(n1)-c1cc(ccc1C(F)(F)F)C(=O)Nc1c(ncn1C)-c1ccccc1
Cc1nc(c(NC(=O)c2ccc(c(c2)-c2ccn(C)n2)C(F)(F)F)[nH]1)-c1ccccc1
Cc1nc(c(NC(=O)c2ccc(c(c2)-c2ccn(C)n2)C(F)(F)F)n1C)-c1ccccc1
Cc1nc(NC(=O)c2ccc(c(c2)-c2ccn(C)n2)C(F)(F)F)n(n1)-c1ccccc1
Cn1ccc(n1)-c1cc(ccc1C(F)(F)F)C(=O)Nc1cc(nn1-c1ccccc1)-c1n[nH]c(=O)n1C
Cn1ccc(n1)-c1cc(ccc1C(F)(F)F)C(=O)Nc1oncc1-c1ccccc1
Cn1ccc(n1)-c1cc(ccc1C(F)(F)F)C(=O)Nc1cn[nH]c1-c1ccccc1
Cn1ccc(n1)-c1cc(ccc1C(F)(F)F)C(=O)Nc1snnc1-c1ccccc1
Cn1ccc(n1)-c1cc(ccc1C(F)(F)F)C(=O)Nc1cc(nn1C)-c1ccccc1
Cc1csc(n1)-c1cc(ccc1Cl)C(=O)Nc1cc(nn1-c1ccccc1)-c1ccncc1
Cc1cc([nH]n1)-n1nc(CC(=O)Nc2ccccn2)cc1NC(=O)c1ccc(c(c1)-c1ccn(C)n1)C(F)(F)F
Cc1cc(cc(C)c1C)C(=O)Nc1cc(nn1-c1ccccc1)-c1ccncc1
FC(F)(F)c1ccc(cc1-n1cccn1)C(=O)Nc1cc(nn1-c1ccccc1)-c1ccncc1
Cc1cc([nH]n1)-n1nc(cc1NC(=O)c1ccc(c(c1)-c1ccn(C)n1)C(F)(F)F)C(=O)NCc1ccns1
Fc1ccc(cc1)-n1nc(cc1NC(=O)c1ccc(c(c1)-c1ncns1)C(F)(F)F)-c1ccncc1
CN1CC(C1)NC(=O)c1cc(NC(=O)c2ccc(c(c2)-c2ccn(C)n2)C(F)(F)F)n(n1)-c1cc(C)n[nH]1
Cn1ccc(n1)-c1cc(ccc1C(F)(F)F)C(=O)Nc1cc(Cc2ccc(=O)[nH]n2)nn1-c1ccccc1
Cc1cc(no1)-c1cc(ccc1C(F)(F)F)C(=O)Nc1cc(nn1-c1ccc(F)cc1)-c1ccncc1
Cc1cccc(n1)-c1cc(ccc1C(F)(F)F)C(=O)Nc1cc(nn1-c1ccc(F)cc1)-c1ccncc1
Cc1cccnc1-c1cc(ccc1C(F)(F)F)C(=O)Nc1cc(nn1-c1ccc(F)cc1)-c1ccncc1
Cc1nc(c(NC(=O)c2ccc(c(c2)-c2ccn(C)n2)C(F)(F)F)s1)-c1ccccc1
CC(=O)n1cc(NC(=O)c2ccc(c(c2)-c2ccn(C)n2)C(F)(F)F)c(n1)-c1ccccc1
Cn1ccc(n1)-c1cc(ccc1C(F)(F)F)C(=O)Nc1nncn1-c1ccccc1
Fc1ccc(cc1)-n1nc(cc1NC(=O)c1ccc(c(c1)-c1cccnc1)C(F)(F)F)-c1ccncc1
Cn1ccc(n1)-c1cc(C(=O)Nc2cc(nn2-c2ccccc2)-c2ccncc2)c(Cl)cc1C(F)(F)F
Cn1ccc(n1)-c1cc(ccc1C(F)(F)F)C(=O)Nc1cnoc1-c1ccccc1
Cn1ccc(n1)-c1cc(ccc1C(F)(F)F)C(=O)Nc1cc(=O)[nH]n1-c1ccccc1
FC(F)(F)c1cc(Cl)c(cc1-c1cc[nH]n1)C(=O)Nc1cc(nn1-c1ccccc1)-c1ccncc1
Cn1ccc(n1)-c1cc(ccc1Cl)C(=O)Nc1cc(nn1-c1cc(n[nH]1)C(F)(F)F)-c1ccncc1
FC(F)(F)c1cc([nH]n1)-n1nc(cc1NC(=O)c1ccc(Cl)c(c1)-c1cc[nH]n1)-c1ccncc1
Fc1ccc(cc1)-n1nc(cc1NC(=O)c1ccc(Cl)c(c1)-c1cc[nH]n1)-c1ccncc1
Cn1ccc(n1)-c1cc(ccc1C(F)(F)F)C(=O)Nc1cn(C)nc1-c1ccccc1
Cc1c(NC(=O)c2ccc(c(c2)-c2ccn(C)n2)C(F)(F)F)n(nc1-c1cnn(C)c1)-c1ccccc1
Cn1ccc(n1)-c1cc(C(=O)Nc2[nH]ncc2-c2ccccc2)c(Cl)cc1C(F)(F)F
Cc1cnn(c1NC(=O)c1cc(-c2ccn(C)n2)c(cc1Cl)C(F)(F)F)-c1ccccc1
Fc1ccc(cc1)-n1nc(cc1NC(=O)c1ccc(c(c1)-c1cc[nH]c(=O)c1)C(F)(F)F)-c1ccncc1
Cc1cc(NC(=O)c2cc(-c3ccn(C)n3)c(cc2Cl)C(F)(F)F)n(n1)-c1cc(C)[nH]n1
Cn1ccc(n1)-c1cc(C(=O)Nc2cn[nH]c2-c2ccccc2)c(Cl)cc1C(F)(F)F
Cn1ccc(n1)-c1cc(ccc1C(F)(F)F)C(=O)Nc1c(nc(C(N)=O)n1C)-c1ccccc1
Cc1cc([nH]n1)-n1nc(CO)cc1NC(=O)c1ccc(c(c1)-c1ccn(C)n1)C(F)(F)F
Cc1nc(c(NC(=O)c2ccc(c(c2)-c2ccn(C)n2)C(F)(F)F)n1C)-c1ccncc1
Cc1nc(cs1)-c1nc(C)n(C)c1NC(=O)c1ccc(c(c1)-c1ccn(C)n1)C(F)(F)F
Cc1cc(NC(=O)c2cc(ccc2Cl)-c2cc[nH]n2)n(n1)-c1cc(C)[nH]n1
Cn1ccc(n1)-c1cc(C(=O)Nc2cc(nn2-c2ccccc2)-c2ccc(=O)[nH]n2)c(Cl)cc1C(F)(F)F
FC(F)(F)c1ccc(cc1-c1ncccn1)C(=O)Nc1cc(nn1-c1ccccc1)-c1ccc(=O)[nH]n1
Cc1cc(n[nH]1)-n1nc(cc1NC(=O)c1ccc(c(c1)-c1ncccn1)C(F)(F)F)-c1ccc(=O)[nH]n1
Cn1ccc(n1)-c1cc(C(=O)Nc2cc(Cc3nnn(C)n3)nn2-c2ccccc2)c(Cl)cc1C(F)(F)F
Cn1ccc(n1)-c1cc(C(=O)Nc2cc(Cc3nnnn3C)nn2-c2ccccc2)c(Cl)cc1C(F)(F)F
Cn1ccc(n1)-c1cc(ccc1C(F)(F)F)C(=O)Nc1cc(nn1-c1ccc(F)cc1)-c1ncccn1
Cc1coc(n1)-c1cc(ccc1C(F)(F)F)C(=O)Nc1cc(nn1-c1cc(C)[nH]n1)-c1cn[nH]c1
Fc1cc(c(cc1C(=O)Nc1cn[nH]c1-c1ccccc1)-c1cc[nH]n1)C(F)(F)F
CC1C(C)=NC(=C1NC(=O)c1cc(-c2ccn(C)n2)c(cc1F)C(F)(F)F)c1ccccc1 |c:3,5|
Fc1ccc(cc1)-n1nc(cc1NC(=O)c1cc(-c2cc[nH]n2)c(cc1F)C(F)(F)F)-c1ncccn1
Cn1ccc(n1)-c1cc(C(=O)Nc2cn(C)nc2-c2ccccc2)c(F)cc1C(F)(F)F
Cn1ccc(n1)-c1cc(ccc1C(F)(F)F)C(=O)Nc1cc(Cn2cnnn2)nn1-c1ccccc1
Cn1ccc(n1)-c1cc(ccc1C(F)(F)F)C(=O)Nc1cc(Cn2ncnn2)nn1-c1ccccc1
Cc1cc([nH]n1)-n1nc(CNCCO)cc1NC(=O)c1ccc(c(c1)-c1ccn(C)n1)C(F)(F)F
Cc1cc([nH]n1)-n1nc(CN2CCCC2)cc1NC(=O)c1ccc(c(c1)-c1ccn(C)n1)C(F)(F)F
FC(F)(F)Cn1ccc(n1)-c1cc(ccc1C(F)(F)F)C(=O)Nc1cc(nn1-c1ccccc1)-c1ccc(=O)[nH]n1
Cn1ccc(n1)-c1cc(ccc1OC(F)(F)F)C(=O)Nc1cc(nn1-c1ccccc1)-c1ccc(=O)[nH]n1
Cc1nc(NC(=O)c2ccc(c(c2)-c2ccn(C)n2)C(F)(F)F)c(s1)-c1ccccc1
CC1C=CC(=N1)c1cc(ccc1OC(F)(F)F)C(=O)Nc1cc(C)nn1-c1ccc(F)cc1 |c:2,4|
Cc1cc([nH]n1)-c1nn(C)cc1NC(=O)c1ccc(c(c1)-c1ccn(C)n1)C(F)(F)F
CCn1ccc(n1)-c1cc(ccc1C(F)(F)F)C(=O)Nc1cc(C)nn1-c1ccc(F)cc1
Cc1cc([nH]n1)-n1nc(cc1NC(=O)c1cc(-c2ccn(C)n2)c(cc1F)C(F)(F)F)C(=O)NCc1cccnc1
Cn1ccc(n1)-c1cc(ccc1C(F)(F)F)C(=O)Nc1cc(Cc2nnn(CCO)n2)nn1-c1ccc(F)cc1
CNC(=O)Cn1nnc(Cc2cc(NC(=O)c3ccc(c(c3)-c3ccn(C)n3)C(F)(F)F)n(n2)-c2ccc(F)cc2)n1
Cn1ccc(n1)-c1cc(ccc1C(F)(F)F)C(=O)Nc1c(nc2CCCn12)-c1ccccc1
NC(=O)c1ccc(cc1)-c1cc(NC(=O)c2cc(-c3ncccn3)c(cc2F)C(F)(F)F)n(n1)-c1ccc(F)cc1
Cn1ccc(n1)-c1cc(ccc1C(F)(F)F)C(=O)Nc1c2CCCc2nn1-c1ccc(F)cc1
Cc1cc([nH]n1)-n1nc(cc1NC(=O)c1ccc(c(c1)-c1ccn(C)n1)C(F)(F)F)C(=O)NCc1cncnc1
NC(=O)c1ccnc(n1)-c1cc(NC(=O)c2cc(-c3ncccn3)c(cc2F)C(F)(F)F)n(n1)-c1ccc(F)cc1
Cn1ccc(n1)-c1cc(C(=O)Nc2cc(Cc3nnn(C)n3)nn2-c2ccc(F)cc2)c(F)cc1C(F)(F)F
CNC(=O)c1cc(NC(=O)c2cc(-c3ncccn3)c(cc2F)C(F)(F)F)n(n1)-c1ccc(F)cc1
Fc1ccc(cc1)-n1nc(Cn2cccn2)cc1NC(=O)c1cc(-c2ncccn2)c(cc1F)C(F)(F)F
Fc1ccc(cc1)-n1nc(cc1NC(=O)c1cc(-c2ncccn2)c(cc1F)C(F)(F)F)C(=O)N1CCC1
Fc1ccc(cc1)-n1nc(Cc2n[nH]c(=O)s2)cc1NC(=O)c1cc(-c2ncccn2)c(cc1F)C(F)(F)F
Cn1ccc(n1)-c1cc(ccc1C(F)(F)F)C(=O)Nc1cc(Cc2cnn(C)c2)nn1-c1ccc(F)cc1
Cn1ccc(n1)-c1cc(ccc1C(F)(F)F)C(=O)Nc1cc(Cc2cnc(N)nc2)nn1-c1ccc(F)cc1
Cn1ccc(n1)-c1cc(ccc1C(F)(F)F)C(=O)Nc1cc(Cc2nnc(N)o2)nn1-c1ccc(F)cc1
OCCc1cc(NC(=O)c2cc(-c3ncccn3)c(cc2F)C(F)(F)F)n(n1)-c1ccc(F)cc1
Cn1ccc(n1)-c1cc(ccc1C(F)(F)F)C(=O)Nc1cc(Cc2cnc(N)cn2)nn1-c1ccc(F)cc1
Cn1ccc(n1)-c1cc(ccc1C(F)(F)F)C(=O)Nc1cc(Cc2cncnc2)nn1-c1ccc(F)cc1
Cn1ccc(n1)-c1cc(ccc1C(F)(F)F)C(=O)Nc1cc(Cc2cc[nH]n2)nn1-c1ccc(F)cc1
OCc1cc(NC(=O)c2cc(-c3ncccn3)c(cc2F)C(F)(F)F)n(n1)-c1ccc(F)cc1
Cn1ccc(n1)-c1cc(ccc1C(F)(F)F)C(=O)Nc1cc(Cc2ccc[nH]c2=O)nn1-c1ccc(F)cc1
CC(O)c1cc(NC(=O)c2cc(-c3ncccn3)c(cc2F)C(F)(F)F)n(n1)-c1ccc(F)cc1
CC(O)c1ccc(nc1)-c1cc(NC(=O)c2cc(-c3ncccn3)c(cc2F)C(F)(F)F)n(n1)-c1ccc(F)cc1
OCCc1ccc(cc1)-c1cc(NC(=O)c2cc(-c3ncccn3)c(cc2F)C(F)(F)F)n(n1)-c1ccc(F)cc1
Cn1ccc(n1)-c1cc(C(=O)Nc2cc(Cc3nnnn3C)nn2-c2ccc(F)cc2)c(F)cc1C(F)(F)F
NCc1cccc(c1)-c1cc(NC(=O)c2cc(-c3ncccn3)c(cc2F)C(F)(F)F)n(n1)-c1ccc(F)cc1
Cn1nnnc1Cc1cc(NC(=O)c2cc(-c3ncccn3)c(cc2F)C(F)(F)F)n(n1)-c1ccc(F)cc1
Cn1ccc(n1)-c1cc(C(=O)Nc2cc(Cc3ccc(=O)[nH]n3)nn2-c2ccc(F)cc2)c(F)cc1C(F)(F)F
OCCn1cc(cn1)-c1nc(c(NC(=O)c2cc(-c3ncccn3)c(cc2F)C(F)(F)F)s1)-c1ccccc1
CC(O)c1cnc(nc1)-c1cc(NC(=O)c2cc(-c3ccn(C)n3)c(cc2F)C(F)(F)F)n(n1)-c1ccc(F)cc1
Cn1ccc(n1)-c1cc(C(=O)Nc2c3CNC(=O)Cc3nn2-c2ccccc2)c(F)cc1C(F)(F)F
Cn1ccc(n1)-c1cc(C(=O)Nc2cn(CCO)nc2-c2ccccc2)c(F)cc1C(F)(F)F
NC(=O)OCc1cc(NC(=O)c2cc(c(cc2F)C(F)(F)F)-c2ncccn2)n(n1)-c1ccc(F)cc1
Cn1ccc(n1)-c1cc(C(=O)Nc2cc(CC(O)=O)nn2-c2ccc(F)cc2)c(F)cc1C(F)(F)F
Cn1ccc(n1)-c1cc(C(=O)Nc2cc(CN3C(=O)CNC3=O)nn2-c2ccc(F)cc2)c(F)cc1C(F)(F)F
Fc1ccc(cc1)-n1nc(Cc2n[nH]c(=O)o2)cc1NC(=O)c1cc(-c2ncccn2)c(cc1F)C(F)(F)F
CNC(=O)Cc1cc(NC(=O)c2cc(-c3ccn(C)n3)c(cc2F)C(F)(F)F)n(n1)-c1ccc(F)cc1
CCn1nc(C#Cc2cc(ccc2C)C(=O)Nc2ccc(CN3CCN(C)CC3)c(c2)C(F)(F)F)c2c(N)ncnc12
CN1CCN(Cc2ccc(NC(=O)c3ccc(C)c(c3)C#Cc3nn(C(=O)OC(C)(C)C)c4ncnc(N)c34)cc2C(F)(F)F)CC1
CN1CCN(Cc2ccc(NC(=O)c3ccc(C)c(c3)C#Cc3nn(C4CCN(CC4)C(=O)C=C)c4ncnc(N)c34)cc2C(F)(F)F)CC1
COCCN1C[C@@H](NC(=O)Nc2cc(nn2-c2ccccc2)C(C)(C)C)[C@@H](C1)c1ccccc1 |r|
COCCN1C[C@@H](NC(=O)Nc2cc(nn2-c2ccc(C)cc2)C(C)(C)C)[C@@H](C1)c1ccccc1 |r|
COCCN1C[C@@H](NC(=O)Nc2c3CCCc3nn2-c2ccccc2)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2cc(nn2-c2ccccc2)C(C)C)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2cc(nn2C)C(C)(C)C)[C@@H](C1)c1ccccc1 |r|
COCCN1C[C@@H](NC(=O)Nc2cc(C)nn2C)[C@@H](C1)c1ccccc1 |r|
COCCN1C[C@@H](NC(=O)Nc2cc(nn2-c2cccnc2)C(C)(C)C)[C@@H](C1)c1ccccc1 |r|
COCCN1C[C@@H](NC(=O)Nc2cc(nn2-c2ccc(F)cc2)C(C)(C)C)[C@@H](C1)c1ccccc1 |r|
COCCN1C[C@@H](NC(=O)Nc2cc(nn2-c2ccccc2)C2CC2)[C@@H](C1)c1ccccc1 |r|
COCCN1C[C@@H](NC(=O)Nc2cc(nn2-c2ccccc2)-c2ccccc2)[C@@H](C1)c1ccccc1 |r|
COCCN1C[C@@H](NC(=O)Nc2cc(C)nn2-c2ccccc2)[C@@H](C1)c1ccccc1 |r|
COCCN1C[C@@H](NC(=O)Nc2cc(nn2-c2ccccc2)C(C)C)[C@@H](C1)c1ccccc1 |r|
COCCN1C[C@@H](NC(=O)Nc2cc(nn2C)-c2ccccc2)[C@@H](C1)c1ccccc1 |r|
COCCN1C[C@@H](NC(=O)Nc2c3CCCc3nn2-c2ccccc2)[C@@H](C1)c1ccccc1 |r|
COCCN1C[C@@H](NC(=O)Nc2ccnn2-c2ccccc2)[C@@H](C1)c1ccccc1 |r|
COCCN1C[C@@H](NC(=O)Nc2cc(nn2-c2ccccc2F)C(C)(C)C)[C@@H](C1)c1ccccc1 |r|
COCCN1C[C@@H](NC(=O)Nc2cc(nn2-c2cccc(F)c2)C(C)(C)C)[C@@H](C1)c1ccccc1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(C)nn2-c2ccccc2)[C@@H](C1)c1ccccc1 |r|
COCCN1C[C@@H](NC(=O)Nc2c3CCCc3nn2-c2cccnc2)[C@@H](C1)c1ccccc1 |r|
COCCN1C[C@@H](NC(=O)Nc2ccnn2C)[C@@H](C1)c1ccccc1 |r|
COCCN1C[C@@H](NC(=S)Nc2c3CCCc3nn2-c2ccccc2)[C@@H](C1)c1ccccc1 |r|
COCCN1C[C@@H](NC(=O)Nc2c3CCCc3nn2-c2cccc(F)c2)[C@@H](C1)c1ccccc1 |r|
COCCN1C[C@@H](NC(=O)Nc2c3CCCc3nn2-c2ccc(F)cc2)[C@@H](C1)c1ccccc1 |r|
COCCN1C[C@@H](NC(=O)Nc2cc(nn2-c2ccccc2)C2CCCC2)[C@@H](C1)c1ccccc1 |r|
CCn1nc(cc1NC(=O)N[C@@H]1CN(CCOC)C[C@H]1c1ccccc1)-c1ccccc1 |r|
COCCN1C[C@@H](NC(=O)Nc2c3CCCCc3nn2-c2ccccc2)[C@@H](C1)c1ccccc1 |r|
COCCN1C[C@@H](NC(=O)Nc2c3CCCc3nn2C)[C@@H](C1)c1ccccc1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(c(C)nn2C)-c2ccccc2)[C@@H](C1)c1ccccc1 |r|
COCCN1C[C@@H](NC(=O)Nc2cc(nn2-c2ccccc2C)C(C)(C)C)[C@@H](C1)c1ccccc1 |r|
COCCN1C[C@@H](NC(=O)Nc2cc(nn2-c2cccc(C)c2)C(C)(C)C)[C@@H](C1)c1ccccc1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(cnn2C)-c2ccccc2)[C@@H](C1)c1ccccc1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C#N)c(C)nn2-c2ccccc2)[C@@H](C1)c1ccccc1 |r|
COCCN1C[C@@H](NC(=O)Nc2c3CCCc3nn2-c2cnn(C)c2)[C@@H](C1)c1ccccc1 |r|
COCCN1C[C@@H](NC(=O)Nc2cc(nn2C2CCOCC2)C(C)(C)C)[C@@H](C1)c1ccccc1 |r|
COCCN1C[C@@H](NC(=O)Nc2c3CCCc3nn2-c2ccccn2)[C@@H](C1)c1ccccc1 |r|
COCCN1C[C@@H](NC(=O)Nc2c3CCC(C)(C)c3nn2-c2ccccc2)[C@@H](C1)c1ccccc1 |r|
COCCN1C[C@@H](NC(=O)Nc2c3CCCC(C)(C)c3nn2-c2ccccc2)[C@@H](C1)c1ccccc1 |r|
COCCN1C[C@@H](NC(=O)Nc2c3CCCc3nn2-c2ccccc2)[C@@H](C1)c1ccncc1 |r|
COCCN1C[C@@H](NC(=O)Nc2c3CCCc3nn2-c2ccccc2)C(C1)c1cccc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2cc(nn2-c2ccccc2)C(C)C)C(C1)c1cccc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2cc(nn2-c2ccccc2)C(C)C)C(C1)c1ccc(F)cc1 |r|
COCCN1C[C@@H](NC(=O)Nc2cc(nn2-c2ccccc2)C(C)C)C(C1)c1cccc(Cl)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2cc(nn2-c2ccccc2)C(C)C)C(C1)c1ccccc1F |r|
COCCN1C[C@@H](NC(=O)Nc2cc(nn2-c2ccccc2)C(C)C)C(C1)c1cccs1 |r|
COCCN1C[C@@H](NC(=O)Nc2c3CCCc3nn2-c2ccccc2)C(C1)c1sc(C)nc1C |r|
COCCN1C[C@@H](NC(=O)Nc2c3CCCc3nn2-c2ccccc2)C(C1)c1cnco1 |r|
COCCN1C[C@@H](NC(=O)Nc2c3CCCc3nn2-c2ccccc2)C(C1)c1ccno1 |r|
COCCN1CC(NC(=O)Nc2c3CCCc3nn2-c2ccccc2)[C@@H](C1)c1cccc(OC)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c3CCCc3nn2-c2ccccc2)[C@@H](C1)c1nccs1 |r|
COCCN1C[C@@H](NC(=O)Nc2cc(nn2-c2ccccc2)C(F)(F)F)[C@@H](C1)c1ccccc1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2C)-c2ccccc2)[C@@H](C1)c1ccccc1 |r|
COCCN1C[C@@H](NC(=O)Nc2cc(nn2C)C2CC2)[C@@H](C1)c1cc(F)cc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2cc(nn2C)-c2ccccn2)[C@@H](C1)c1cc(F)cc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2cc(nn2C)-c2cccnc2)[C@@H](C1)c1cc(F)cc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2cc(nn2C)-c2cnn(C)c2)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2cc(nn2C)-c2cccc(c2)C#N)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2cc(nn2C)-c2ccc(cc2)C#N)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2cc(nn2C)-c2cccc3nccn23)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(Cl)c(nn2-c2ccccc2)-c2ccccc2)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(Br)c(nn2-c2ccccc2)-c2ccccc2)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(Cl)c(C)nn2-c2ccccc2)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(c(C)nn2C)-c2ccccc2)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C#N)c(C)nn2-c2ccccc2)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(Cl)c(nn2C)-c2ccccc2)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(Br)c(nn2C)-c2ccccc2)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C#N)c(CC#N)nn2-c2ccccc2)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2cc(nn2-c2ccccc2)C(C)(C)C#N)[C@@H](C1)c1ccc(F)c(F)c1 |r|
CCc1nn(c(NC(=O)N[C@@H]2CN(CCOC)C[C@H]2c2ccc(F)c(F)c2)c1C)-c1ccccc1 |r|
COCCN1C[C@@H](NC(=O)Nc2cc(nn2-c2ccccc2)-c2cnn(C)c2)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(OCC3COC3)nn2-c2ccccc2)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(OCC3(C)COC3)nn2-c2ccccc2)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(OC[C@H]3COC(C)(C)O3)nn2-c2ccccc2)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(OC[C@@H]3COC(C)(C)O3)nn2-c2ccccc2)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c3CN(Cc3nn2-c2ccccc2)C(=O)OC(C)(C)C)[C@@H](C1)c1ccccc1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)C(C)C)[C@@H](C1)c1ccccc1 |r|
COCCN1C[C@@H](NC(=O)Nc2c3COCc3nn2-c2ccccc2)[C@@H](C1)c1ccccc1 |r|
COCCN1C[C@@H](NC(=O)Nc2c3CSCc3nn2-c2ccccc2)[C@@H](C1)c1ccccc1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(C)nn2-c2ccccc2)[C@@H](C1)c1cc(F)cc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c3CCCc3nn2-c2ccccc2)[C@@H](C1)c1cc(F)cc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2cc(nn2-c2ccccc2)C(C)C)[C@@H](C1)c1cc(F)cc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2cc(C)nn2-c2ccccc2)[C@@H](C1)c1cc(F)cc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c3COCc3nn2-c2ccccc2)[C@@H](C1)c1cc(F)cc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c3CSCc3nn2-c2ccccc2)[C@@H](C1)c1cc(F)cc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c3COCc3nn2-c2ccccc2)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c3CSCc3nn2-c2ccccc2)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(C)nn2-c2ccccc2)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2cc(nn2C)-c2ccccc2)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2cc(nn2-c2ccccc2)C(C)(C)CO)[C@@H](C1)c1ccccc1 |r|
COCCN1C[C@@H](NC(=O)Nc2c3CS(=O)Cc3nn2-c2ccccc2)[C@@H](C1)c1ccccc1 |r|
COCCN1C[C@@H](NC(=O)Nc2cc(nn2C)-c2ccncc2)[C@@H](C1)c1ccccc1 |r|
COCCN1C[C@@H](NC(=O)Nc2cc(nn2C)-c2ccncc2)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2cc(nn2C)-c2ccccc2)[C@@H](C1)c1cc(F)cc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2cc(nn2C)-c2cccs2)[C@@H](C1)c1cc(F)cc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2cc(COC)nn2-c2ccccc2)[C@@H](C1)c1ccccc1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(COC)nn2-c2ccccc2)[C@@H](C1)c1ccccc1 |r|
COCCN1C[C@@H](NC(=O)Nc2cc(nn2C)-c2ccc(C)cc2)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2cc(nn2C)-c2cccc(C)c2)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2cc(nn2C)-c2ccccc2C)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2cc(nn2C)-c2cccc(OC)c2)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2cc(nn2C)-c2ccccc2OC)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2cc(nn2C)-c2ccc(F)cc2)[C@@H](C1)c1ccccc1 |r|
COCCN1C[C@@H](NC(=O)Nc2cc(nn2C)-c2ccc(OC)cc2)[C@@H](C1)c1ccccc1 |r|
COCCN1C[C@@H](NC(=O)Nc2cc(nn2C)-c2ccccc2)[C@@H](C1)c1cccc(c1)C(F)(F)F |r|
COCCN1C[C@@H](NC(=O)Nc2cc(nn2C)-c2ccccc2)[C@@H](C1)c1cccc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2cc(nn2C)-c2ccccc2)[C@@H](C1)c1ccc(F)cc1F |r|
COCCN1C[C@@H](NC(=O)Nc2cc(nn2C)-c2ccc(F)cc2)[C@@H](C1)c1cccc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2cc(nn2C)-c2ccc(F)cc2)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2cc(nn2C)-c2cccc(F)c2)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2cc(nn2C)-c2ccccc2F)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c3CCCc3nn2-c2ccccc2)[C@@H](C1)c1cccc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)C(C)(C)CO)[C@@H](C1)c1ccccc1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)C(C)(C)CO)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2cc(nn2C)-c2ccc(Cl)cc2)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2cc(nn2C)-c2ccc(F)cc2)[C@@H](C1)c1cc(F)ccc1F |r|
COCCN1C[C@@H](NC(=O)Nc2cc(nn2C)-c2ccc(cc2)C(=O)OC)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2cc(nn2CCO)-c2ccccc2)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(COC)nn2-c2ccccc2)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(COC)nn2-c2ccccc2)[C@@H](C1)c1cc(F)cc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2cc(nn2C)-c2ccc(SC)cc2)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2cc(nn2-c2ccccc2)-c2ccccc2)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCCc1nn(c(NC(=O)N[C@@H]2CN(CCOC)C[C@H]2c2ccc(F)c(F)c2)c1C)-c1ccccc1 |r|
COCCN1C[C@@H](NC(=O)Nc2c3CCCc3nn2-c2ccccc2)[C@@H](C1)c1ccc(F)cc1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(C)nn2-c2ccccc2)[C@@H](C1)c1ccc(F)cc1 |r|
COCCOc1ccc(cc1)-c1cc(NC(=O)N[C@@H]2CN(CCOC)C[C@H]2c2ccc(F)c(F)c2)n(C)n1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(OC)c(C)nn2-c2ccccc2)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(CO)nn2-c2ccccc2)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(CCO)nn2-c2ccccc2)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(CCOC)nn2-c2ccccc2)[C@@H](C1)c1ccc(F)c(F)c1 |r|
CCOc1nn(c(NC(=O)N[C@@H]2CN(CCOC)C[C@H]2c2ccc(F)c(F)c2)c1C)-c1ccccc1 |r|
COCCN1C[C@@H](NC(=O)Nc2cc(OCc3ccccc3)nn2C)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCOc1nn(c(NC(=O)N[C@@H]2CN(CCOC)C[C@H]2c2ccc(F)c(F)c2)c1C)-c1ccccc1 |r|
CCOc1nn(c(NC(=O)N[C@@H]2CN(CCOC)C[C@H]2c2cc(F)cc(F)c2)c1C)-c1ccccc1 |r|
CCOc1nn(c(NC(=O)N[C@@H]2CN(CCOC)C[C@H]2c2ccccc2)c1C)-c1ccccc1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(OC)nn2-c2ccccc2)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(OCC#N)nn2-c2ccccc2)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(OCc3ccc(OC)cc3)nn2-c2ccccc2)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(OC)nn2-c2ccccc2)[C@@H](C1)c1ccc(F)cc1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(OCCF)nn2-c2ccccc2)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(OCC(C)(C)O)nn2-c2ccccc2)[C@@H](C1)c1ccc(F)c(F)c1 |r|
CCOc1cc(NC(=O)N[C@@H]2CN(CCOC)C[C@H]2c2ccc(F)c(F)c2)n(n1)-c1ccccc1 |r|
CCOc1nn(c(NC(=O)N[C@@H]2CN(CCOC)C[C@H]2c2ccc(F)cc2)c1C)-c1ccccc1 |r|
CCOc1nn(c(NC(=O)N[C@@H]2CN(CCOC)C[C@H]2c2cccc(F)c2)c1C)-c1ccccc1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(OCCO)nn2-c2ccccc2)[C@@H](C1)c1cc(F)cc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c3CCCc3nn2C2CCCCC2)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c3CCCc3nn2-c2ccncc2)[C@@H](C1)c1ccccc1 |r|
COCCN1C[C@@H](NC(=O)Nc2cc(nn2C)-c2cnc(C)cn2)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2C)-c2cnc(C)cn2)[C@@H](C1)c1ccc(F)c(F)c1 |r|
CCOC(=O)c1cnn(c1NC(=O)N[C@@H]1CN(CCOC)C[C@H]1c1ccc(F)c(F)c1)-c1ccccc1 |r|
COCCN1C[C@@H](NC(=O)Nc2cc(nn2C)-c2cnccn2)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(c(OC)nn2C)-c2ccccc2)[C@@H](C1)c1ccc(F)c(F)c1 |r|
CCOc1nn(C)c(NC(=O)N[C@@H]2CN(CCOC)C[C@H]2c2ccc(F)c(F)c2)c1-c1ccccc1 |r|
COCCN1C[C@@H](NC(=O)Nc2c3CNCc3nn2-c2ccccc2)[C@@H](C1)c1ccccc1 |r|
COCCN1C[C@@H](NC(=O)Nc2c3CN(Cc3nn2-c2ccccc2)C(C)=O)[C@@H](C1)c1ccccc1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(CO)c(COC)nn2-c2ccccc2)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2cc(nn2C)-c2ccc(cc2)C(O)=O)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2cc(nn2C)-c2ccc(cc2)C(N)=O)[C@@H](C1)c1ccc(F)c(F)c1 |r|
CNC(=O)c1ccc(cc1)-c1cc(NC(=O)N[C@@H]2CN(CCOC)C[C@H]2c2ccc(F)c(F)c2)n(C)n1 |r|
COCCN1C[C@@H](NC(=O)Nc2cc(nn2C)-c2ccc(cc2)C(=O)N(C)C)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2cc(nn2C)-c2ccc(CO)cc2)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2cc(nn2C)-c2ccc(cc2)S(C)(=O)=O)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(F)c(C)nn2-c2ccccc2)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(F)c(nn2C)-c2ccccc2)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(F)c(nn2-c2ccccc2)-c2ccccc2)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCOC(=O)c1ccc(cc1)-c1cc(NC(=O)N[C@@H]2CN(CCOC)C[C@H]2c2ccc(F)c(F)c2)n(C)n1 |r|
COCCN1C[C@@H](NC(=O)Nc2c3CS(=O)(=O)Cc3nn2-c2ccccc2)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c3CS(=O)(=O)Cc3nn2-c2ccccc2)[C@@H](C1)c1ccccc1 |r|
COCCN1C[C@@H](NC(=O)Nc2c3CS(=O)(=O)Cc3nn2-c2ccccc2)[C@@H](C1)c1cc(F)cc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(OCCS(C)(=O)=O)nn2-c2ccccc2)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(CO)cnn2-c2ccccc2)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(OC[C@H](O)CO)nn2-c2ccccc2)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(OC[C@@H](O)CO)nn2-c2ccccc2)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(OCCO)nn2-c2ccccc2)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(OC[C@H](C)O)nn2-c2ccccc2)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c3CCCc3nn2-c2ccccc2)[C@@](O)(C1)c1ccccc1 |r|
COCCN1C[C@@H](NC(=O)Nc2c3CCCc3nn2-c2ccccc2)[C@@](F)(C1)c1ccccc1 |r|
FC(F)(F)OCCN1CC(NC(=O)Nc2c3CCCc3nn2-c2ccccc2)[C@@H](C1)c1ccccc1 |r|
CSCCN1CC(NC(=O)Nc2c3CCCc3nn2-c2ccccc2)[C@@H](C1)c1ccccc1 |r|
CO[C@@H](C)CN1C[C@@H](NC(=O)Nc2c3CCCc3nn2-c2ccccc2)[C@@H](C1)c1ccccc1 |r|
FC(F)(F)CCCN1CC(NC(=O)Nc2c3CCCc3nn2-c2ccccc2)[C@@H](C1)c1ccccc1 |r|
Fc1ccc(cc1F)[C@@H]1CN(CC#N)C[C@H]1NC(=O)Nc1c2CCCc2nn1-c1ccccc1 |r|
COCCOc1nn(c(NC(=O)N[C@@H]2CN(CC#N)C[C@H]2c2ccc(F)c(F)c2)c1C)-c1ccccc1 |r|
O=C(N[C@@H]1CN(CC#N)C[C@H]1c1ccccc1)Nc1c2CCCc2nn1-c1ccccc1 |r|
NC(=O)CN1C[C@@H](NC(=O)Nc2c3CCCc3nn2-c2ccccc2)[C@@H](C1)c1ccccc1 |r|
Cc1nn(c(NC(=O)N[C@@H]2CN(CCO)C[C@H]2c2ccc(F)c(F)c2)c1C)-c1ccccc1 |r|
FC(F)(F)C(F)(F)CCN1C[C@@H](NC(=O)Nc2c3CCCc3nn2-c2ccccc2)[C@@H](C1)c1ccccc1 |r|
CCN1C[C@@H](NC(=O)Nc2c3CCCc3nn2-c2ccccc2)[C@@H](C1)c1ccccc1 |r|
FC(F)(F)CN1C[C@@H](NC(=O)Nc2c3CCCc3nn2-c2ccccc2)[C@@H](C1)c1ccccc1 |r|
Cc1nn(c(NC(=O)N[C@@H]2CN(CC(F)(F)F)C[C@H]2c2ccccc2)c1C)-c1ccccc1 |r|
COCCOc1nn(c(NC(=O)N[C@@H]2CN(CC(F)(F)F)C[C@H]2c2ccccc2)c1C)-c1ccccc1 |r|
Fc1cccc(c1)[C@@H]1CN(CC(F)(F)F)C[C@H]1NC(=O)Nc1c2CCCc2nn1-c1ccccc1 |r|
Cc1nn(c(NC(=O)N[C@@H]2CN(CC(F)(F)F)C[C@H]2c2cccc(F)c2)c1C)-c1ccccc1 |r|
COCCOc1nn(c(NC(=O)N[C@@H]2CN(CC(F)(F)F)C[C@H]2c2cccc(F)c2)c1C)-c1ccccc1 |r|
Cn1nc(cc1NC(=O)N[C@@H]1CN(CC(F)(F)F)C[C@H]1c1cccc(F)c1)-c1ccccc1 |r|
Fc1cccc(c1)[C@H]1CN(CC(F)(F)F)C[C@@H]1NC(=O)Nc1c2CCCc2nn1-c1ccccc1 |r|
CCOc1nn(c(NC(=O)N[C@H]2CN(CC(F)(F)F)C[C@@H]2c2cccc(F)c2)c1C)-c1ccccc1 |r|
FCC(CF)N1C[C@@H](NC(=O)Nc2c3CCCc3nn2-c2ccccc2)C(C1)c1ccccc1 |r|
COc1cccc(c1)C1CN(CC(F)(F)F)C[C@H]1NC(=O)Nc1c2CCCc2nn1-c1ccccc1 |r|
FC(F)(F)CN1C[C@@H](NC(=O)Nc2c3CCCc3nn2-c2ccccc2)C(C1)c1cccc(Cl)c1 |r|
FC(F)(F)CN1C[C@@H](NC(=O)Nc2c3CCCc3nn2-c2ccccc2)C(C1)c1ccccn1 |r|
Fc1ccc(cc1)C1CN(CC(F)(F)F)C[C@H]1NC(=O)Nc1c2CCCc2nn1-c1ccccc1 |r|
FC(F)(F)CN1C[C@@H](NC(=O)Nc2c3CCCc3nn2-c2ccccc2)C(C1)c1ccc(Cl)cc1 |r|
FC(F)(F)CN1C[C@@H](NC(=O)Nc2c3CCCc3nn2-c2ccccc2)C(C1)c1ccccc1Cl |r|
FC(F)(F)CN1C[C@@H](NC(=O)Nc2c3CCCc3nn2-c2ccccc2)C(C1)c1cccnc1 |r|
Fc1ccccc1C1CN(CC(F)(F)F)C[C@H]1NC(=O)Nc1c2CCCc2nn1-c1ccccc1 |r|
FC(F)CN1C[C@@H](NC(=O)Nc2c3CCCc3nn2-c2ccccc2)C(C1)c1ccc(F)cc1 |r|
CCOc1nn(c(NC(=O)N[C@@H]2CN(C[C@H]2c2ccc(F)c(F)c2)c2cn[nH]c2)c1C)-c1ccccc1 |r|
CCOc1nn(c(NC(=O)N[C@@H]2CN(C[C@H]2c2cc(F)cc(F)c2)c2cn[nH]c2)c1C)-c1ccccc1 |r|
CCOc1nn(c(NC(=O)N[C@@H]2CN(C[C@H]2c2cc(F)cc(F)c2)c2cc[nH]n2)c1C)-c1ccccc1 |r|
CCOc1nn(c(NC(=O)N[C@@H]2CN(C[C@H]2c2ccc(F)c(F)c2)c2n[nH]nc2C)c1C)-c1ccccc1 |r|
CCOc1nn(c(NC(=O)N[C@@H]2CN(C[C@H]2c2ccc(F)c(F)c2)c2c[nH]nc2C(F)(F)F)c1C)-c1ccccc1 |r|
C[C@H](O)COc1nn(c(NC(=O)N[C@@H]2CN(C[C@H]2c2ccc(F)c(F)c2)c2cn[nH]c2)c1C)-c1ccccc1 |r|
Cc1c(OC[C@H](O)CO)nn(c1NC(=O)N[C@@H]1CN(C[C@H]1c1ccc(F)c(F)c1)c1cn[nH]c1)-c1ccccc1 |r|
Cc1nn(c(NC(=O)N[C@@H]2CN(C[C@H]2c2cc(F)cc(F)c2)c2cn[nH]c2)c1C)-c1ccccc1 |r|
Cc1nn(c(NC(=O)N[C@@H]2CN(C[C@H]2c2ccc(F)c(F)c2)c2cn[nH]c2)c1C)-c1ccccc1 |r|
COCCCc1nn(c(NC(=O)N[C@@H]2CN(C[C@H]2c2ccc(F)c(F)c2)c2cn[nH]c2)c1C)-c1ccccc1 |r|
COCCOc1nn(c(NC(=O)N[C@@H]2CN(C[C@H]2c2ccc(F)c(F)c2)c2cn[nH]c2)c1C)-c1ccccc1 |r|
Cc1c(OCC(C)(C)O)nn(c1NC(=O)N[C@@H]1CN(C[C@H]1c1ccc(F)c(F)c1)c1cn[nH]c1)-c1ccccc1 |r|
CCOc1nn(c(NC(=O)N[C@@H]2CN(C[C@H]2c2ccccc2)c2ccnn2C)c1C)-c1ccccc1 |r|
CCOc1nn(c(NC(=O)N[C@H]2CN(C[C@@H]2c2ccccc2)c2ccnn2C)c1C)-c1ccccc1 |r|
CCOc1nn(c(NC(=O)N[C@@H]2CN(C[C@H]2c2cc(F)cc(F)c2)c2ccnn2C)c1C)-c1ccccc1 |r|
CCOc1nn(c(NC(=O)N[C@H]2CN(C[C@@H]2c2cc(F)cc(F)c2)c2ccnn2C)c1C)-c1ccccc1 |r|
CCOc1nn(c(NC(=O)N[C@@H]2CN(C[C@H]2c2ccc(F)c(F)c2)c2ccccc2)c1C)-c1ccccc1 |r|
CCOc1nn(c(NC(=O)N[C@@H]2CN(C[C@H]2c2ccc(F)c(F)c2)c2ccccc2OC)c1C)-c1ccccc1 |r|
CCOc1nn(c(NC(=O)N[C@@H]2CN(C[C@H]2c2ccccc2)c2ccccc2F)c1C)-c1ccccc1 |r|
CCOc1nn(c(NC(=O)N[C@@H]2CN(C[C@H]2c2ccccc2)c2ccc(F)cc2)c1C)-c1ccccc1 |r|
CCOc1nn(c(NC(=O)N[C@@H]2CN(C[C@H]2c2ccccc2)c2ccccc2C)c1C)-c1ccccc1 |r|
CCOc1nn(c(NC(=O)N[C@@H]2CN(C[C@H]2c2ccccc2)c2ccccc2OC)c1C)-c1ccccc1 |r|
CCOc1nn(c(NC(=O)N[C@@H]2CN(C[C@H]2c2ccccc2)c2ccccc2Cl)c1C)-c1ccccc1 |r|
CCOc1nn(c(NC(=O)N[C@@H]2CN(C[C@H]2c2ccccc2)c2ccccc2OC(F)(F)F)c1C)-c1ccccc1 |r|
CCOc1nn(c(NC(=O)N[C@@H]2CN(C[C@H]2c2ccccc2)c2c(F)cccc2F)c1C)-c1ccccc1 |r|
CCOc1nn(c(NC(=O)N[C@@H]2CN(C[C@H]2c2ccccc2)c2ccnc(OC)c2)c1C)-c1ccccc1 |r|
CCOc1nn(c(NC(=O)N[C@@H]2CN(C[C@H]2c2ccccc2)c2cccnc2OC)c1C)-c1ccccc1 |r|
CCOc1nn(c(NC(=O)N[C@@H]2CN(C[C@H]2c2ccccc2)c2cccnc2OCC)c1C)-c1ccccc1 |r|
COc1ncccc1N1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnn(C)c2)[C@@H](C1)c1ccccc1 |r|
COc1ncccc1N1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2ccccc2)[C@@H](C1)c1ccccc1 |r|
COc1ncccc1N1C[C@@H](NC(=O)Nc2c(Br)c(nn2-c2ccccc2)-c2cnn(C)c2)[C@@H](C1)c1ccccc1 |r|
COc1ncccc1N1C[C@@H](NC(=O)Nc2c(Br)c(nn2-c2ccccc2)-c2ccccc2)[C@@H](C1)c1ccccc1 |r|
Fc1ccc(cc1F)[C@@H]1CN(Cc2csnn2)C[C@H]1NC(=O)Nc1c2CCCc2nn1-c1ccccc1 |r|
CCOc1nn(c(NC(=O)N[C@@H]2CN(Cc3csnn3)C[C@H]2c2ccc(F)c(F)c2)c1C)-c1ccccc1 |r|
Cc1c(OCC#N)nn(c1NC(=O)N[C@@H]1CN(Cc2csnn2)C[C@H]1c1ccc(F)c(F)c1)-c1ccccc1 |r|
Cc1c(NC(=O)N[C@@H]2CN(Cc3csnn3)C[C@H]2c2ccc(F)c(F)c2)n(nc1-c1cnn(C)c1)-c1ccccc1 |r|
Cc1c(NC(=O)N[C@@H]2CN(Cc3csnn3)C[C@H]2c2ccc(F)c(F)c2)n(nc1-c1cn(C)cn1)-c1ccccc1 |r|
Cn1cc(CN2C[C@@H](NC(=O)Nc3c4CCCc4nn3-c3ccccc3)[C@@H](C2)c2ccc(F)c(F)c2)nn1 |r|
CCOc1nn(c(NC(=O)N[C@@H]2CN(C[C@H]2c2ccc(F)c(F)c2)C(COC)COC)c1C)-c1ccccc1 |r|
CCOc1nn(c(NC(=O)N[C@@H]2CN(C[C@H]2c2ccc(F)c(F)c2)C(C)COC)c1C)-c1ccccc1 |r|
CNCCN1CC(NC(=O)Nc2c3CCCc3nn2-c2ccccc2)[C@@H](C1)c1ccccc1 |r|
O=C(NC1CN(Cc2ncc[nH]2)C[C@H]1c1ccccc1)Nc1c2CCCc2nn1-c1ccccc1 |r|
COCC(N1CC(NC(=O)Nc2c3CCCc3nn2-c2ccccc2)[C@@H](C1)c1ccccc1)C(=O)OC |r|
COCC(N1C[C@@H](NC(=O)Nc2c3CCCc3nn2-c2ccccc2)[C@@H](C1)c1ccc(F)c(F)c1)C(=O)OC |r|
COCC(CO)N1C[C@@H](NC(=O)Nc2c3CCCc3nn2-c2ccccc2)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCC(N1C[C@@H](NC(=O)Nc2c3CCCc3nn2-c2ccccc2)[C@@H](C1)c1ccc(F)c(F)c1)C(C)(C)O |r|
COCC(N1C[C@@H](NC(=O)Nc2c3CCCc3nn2-c2ccccc2)[C@@H](C1)c1ccc(F)c(F)c1)C(O)=O |r|
CCOc1nn(c(NC(=O)N[C@@H]2CN(C[C@H]2c2ccc(F)c(F)c2)C(CO)COC)c1C)-c1ccccc1 |r|
COCC(CO)N1C[C@@H](NC(=O)Nc2c(Cl)c(nn2-c2ccccc2)-c2cnn(C)c2)[C@@H](C1)c1ccc(F)c(F)c1 |r|
Cc1nn(c(NC(=O)N[C@H]2CN(CC(F)(F)F)C[C@@H]2c2ccccc2)c1C)-c1ccccc1 |r|
Cc1c(OCCF)nn(c1NC(=O)N[C@H]1CN(CC(F)(F)F)C[C@@H]1c1ccccc1)-c1ccccc1 |r|
CCOc1nn(c(NC(=O)N[C@H]2CN(CC(F)(F)F)C[C@@H]2c2ccccc2)c1C)-c1ccccc1 |r|
Cc1c(OCC#N)nn(c1NC(=O)N[C@@H]1CN(CC(F)(F)F)C[C@H]1c1ccc(F)c(F)c1)-c1ccccc1 |r|
Cc1c(NC(=O)N[C@H]2CN(CC(F)(F)F)C[C@@H]2c2ccccc2)n(nc1-c1cnn(C)c1)-c1ccccc1 |r|
Cn1cc(cn1)-c1nn(c(NC(=O)N[C@H]2CN(CC(F)(F)F)C[C@@H]2c2ccccc2)c1Cl)-c1ccccc1 |r|
Cc1c(OC[C@H]2COC(C)(C)O2)nn(c1NC(=O)N[C@H]1CN(CC(F)(F)F)C[C@@H]1c1ccccc1)-c1ccccc1 |r|
Cc1c(OC[C@H](O)CO)nn(c1NC(=O)N[C@H]1CN(CC(F)(F)F)C[C@@H]1c1ccccc1)-c1ccccc1 |r|
C[C@@H]1C(NC(=O)Nc2c3CCCc3nn2-c2ccccc2)[C@@H](CN1CC(F)(F)F)c1ccccc1 |r|
C[C@H]1[C@H](C(CN1CC(F)(F)F)NC(=O)Nc1c2CCCc2nn1-c1ccccc1)c1ccccc1 |r|
CCOc1nn(c(NC(=O)N[C@@H]2CN(C[C@H]2c2ccc(F)c(F)c2)[C@@H](CO)C(F)(F)F)c1C)-c1ccccc1 |r|
CCOc1nn(c(NC(=O)N[C@@H]2CN(C[C@H]2c2ccc(F)c(F)c2)[C@@H](COC)C(F)(F)F)c1C)-c1ccccc1 |r|
COC[C@H](N1C[C@@H](NC(=O)Nc2c(C)c(OC[C@H](C)O)nn2-c2ccccc2)[C@@H](C1)c1ccc(F)c(F)c1)C(F)(F)F |r|
COC[C@@H](N1C[C@@H](NC(=O)Nc2c(Cl)c(nn2-c2ccccc2)-c2cnn(C)c2)[C@@H](C1)c1ccc(F)c(F)c1)C(F)(F)F |r|
COC[C@@H](N1C[C@@H](NC(=O)Nc2c(C)c(OC[C@H](C)O)nn2-c2ccccc2)[C@@H](C1)c1ccc(F)c(F)c1)C(F)(F)F |r|
COCCN1C[C@@H](NC(=O)Nc2c(SC)c(C)nn2-c2ccccc2)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCCc1nn(c(NC(=O)N[C@@H]2CN(CCOC)C[C@H]2c2cc(F)cc(F)c2)c1C)-c1ccccc1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)C(F)(F)CO)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)C(F)(F)CO)[C@@H](C1)c1cc(F)cc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)C(F)(F)CO)[C@@H](C1)c1ccc(F)cc1 |r|
COCCN1C[C@@H](NC(=O)Nc2cc(nn2-c2ccccc2)C(F)(F)CO)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(CCO)nn2-c2ccccc2)[C@@H](C1)c1cc(F)cc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(CCO)nn2-c2ccccc2)[C@@H](C1)c1ccc(F)cc1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(CC(C)(C)O)nn2-c2ccccc2)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(C[C@H](C)O)nn2-c2ccccc2)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(C[C@@H](C)O)nn2-c2ccccc2)[C@@H](C1)c1ccc(F)c(F)c1 |r|
CCOC(=O)c1nn(c(NC(=O)N[C@@H]2CN(CCOC)C[C@H]2c2ccc(F)c(F)c2)c1C)-c1ccccc1 |r|
CNC(=O)c1nn(c(NC(=O)N[C@@H]2CN(CCOC)C[C@H]2c2ccc(F)cc2)c1C)-c1ccccc1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnn(C)c2)C(C1)c1ccc(F)c(Cl)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnn(C)c2)C(C1)c1ccc(Cl)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnn(C)c2)C(C1)c1cc(F)cc(Cl)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnn(C)c2)C(C1)c1cccc(Cl)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2nnc(C)o2)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2nc(C)no2)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2nc(no2)C(F)(F)F)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2nc(no2)C(F)(F)F)[C@@H](C1)c1ccc(F)cc1 |r|
CNC(=O)c1nn(c(NC(=O)N[C@@H]2CN(CCOC)CC2c2ccc(F)c(Cl)c2)c1C)-c1ccccc1 |r|
CNC(=O)c1nn(c(NC(=O)N[C@@H]2CN(CCOC)CC2c2ccc(Cl)c(F)c2)c1C)-c1ccccc1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2ccn(C)c(=O)c2)C(C1)c1ccc(Cl)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2ccn(C)c(=O)c2)C(C1)c1ccc(F)c(Cl)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cc(C)n(C)n2)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cc(C)n(C)n2)[C@@H](C1)c1cc(F)cc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cc(C)n(C)n2)[C@@H](C1)c1ccc(F)cc1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cc(C)nn2C)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C3CC3)c(nn2-c2ccccc2)-c2cnn(C)c2)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C(C)C)c(nn2-c2ccccc2)-c2cnn(C)c2)[C@@H](C1)c1ccc(F)c(F)c1 |r|
CCc1c(NC(=O)N[C@@H]2CN(CCOC)C[C@H]2c2ccc(F)c(F)c2)n(nc1-c1cnn(C)c1)-c1ccccc1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccc(F)cc2)-c2cnn(C)c2)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2cccc(F)c2)-c2cnn(C)c2)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2F)-c2cnn(C)c2)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2cccc(Cl)c2)-c2cnn(C)c2)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccc(F)c(Cl)c2)-c2cnn(C)c2)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2cccc(Cl)c2F)-c2cnn(C)c2)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccc(F)cc2)-c2cnn(C)c2)[C@@H](C1)c1ccc(F)cc1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2cccc(F)c2)-c2cnn(C)c2)[C@@H](C1)c1ccc(F)cc1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2F)-c2cnn(C)c2)[C@@H](C1)c1ccc(F)cc1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2cccc(Cl)c2)-c2cnn(C)c2)[C@@H](C1)c1ccc(F)cc1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccc(F)c(Cl)c2)-c2cnn(C)c2)[C@@H](C1)c1ccc(F)cc1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2cccc(Cl)c2F)-c2cnn(C)c2)[C@@H](C1)c1ccc(F)cc1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnn(C)c2)[C@@H](C1)c1ccc(F)cc1F |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnn(C)c2)[C@@H](C1)c1cccc(c1)C#N |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnn(C)c2)[C@@H](C1)c1ccc(cc1)C#N |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnn(C)c2)[C@@H](C1)c1ccc(C)cc1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2ccccc2)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2ccccc2)[C@@H](C1)c1cc(F)cc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2ccccc2)[C@@H](C1)c1cc(F)c(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2ccccc2)[C@@H](C1)c1ccc(F)cc1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(Br)c(C)nn2-c2ccccc2)C(C1)c1cnn(C)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnn(C)c2)C(C1)c1cnn(C)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnn(C)c2)C(C1)c1csnn1 |r|
CCOc1nn(c(NC(=O)N[C@@H]2CN(CCOC)CC2c2cccc(c2)C(F)(F)F)c1C)-c1ccccc1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(C)nn2-c2ccccc2)C(C1)c1cccc(c1)C(F)(F)F |r|
COCCN1C[C@@H](NC(=O)Nc2c3CCCc3nn2-c2ccccc2)[C@@H](C1)c1cncc(F)c1 |r|
COCCN1C[C@H](NC(=O)Nc2c3CCCc3nn2-c2ccccc2)[C@H](C1)c1cncc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(OCCF)nn2-c2ccccc2)[C@@H](C1)c1cncc(F)c1 |r|
COCCN1C[C@H](NC(=O)Nc2c(C)c(OCCF)nn2-c2ccccc2)[C@H](C1)c1cncc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2cc(nn2-c2ccccc2)-c2cnn(C)c2)C(C1)c1cncc(F)c1 |r|
CCOc1nn(c(NC(=O)N[C@@H]2CN(CCOC)CC2c2cncc(Cl)c2)c1C)-c1ccccc1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(C)nn2-c2ccccc2)C(C1)c1cncc(Cl)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2ccccc2)C(C1)c1cncc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnn(C)c2)C(C1)c1ccc(F)cn1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnn(C)c2)C(C1)c1ccncc1F |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2ncn(C)n2)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnn(CCOC)c2)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)C#N)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnn(CCO)c2)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnn(C)n2)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(Br)nn2-c2ccccc2)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c3CN(C)C(=O)c3nn2-c2ccccc2)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c3CN(C)C(=O)c3nn2-c2ccccc2)[C@@H](C1)c1cc(F)cc(F)c1 |r|
CCOc1nn(c(NC(=O)N[C@@H]2CN(CCOC)C[C@H]2c2ccc(F)c(F)c2)c1Cl)-c1ccccc1 |r|
CCOc1nn(c(NC(=O)N[C@@H]2CN(CCOC)C[C@H]2c2ccc(F)c(F)c2)c1F)-c1ccccc1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(Br)c(OCC(C)(C)O)nn2-c2ccccc2)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(Cl)c(OCC(C)(C)O)nn2-c2ccccc2)[C@@H](C1)c1ccc(F)c(F)c1 |r|
CC[C@H](O)COc1nn(c(NC(=O)N[C@@H]2CN(CCOC)C[C@H]2c2ccc(F)c(F)c2)c1C)-c1ccccc1 |r|
CCOC(=O)COc1nn(c(NC(=O)N[C@@H]2CN(CCOC)C[C@H]2c2ccc(F)c(F)c2)c1C)-c1ccccc1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(OCC(C)(C)O)nn2-c2ccccc2)[C@@H](C1)c1ccc(F)cc1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(OCC(C)(C)O)nn2-c2ccccc2)[C@@H](C1)c1cc(F)cc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(OC[C@@H](C)O)nn2-c2ccccc2)[C@@H](C1)c1ccc(F)cc1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(OC[C@@H](C)O)nn2-c2ccccc2)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(OC[C@@H](C)O)nn2-c2ccccc2)[C@@H](C1)c1cc(F)cc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(OC[C@@H](O)C(F)(F)F)nn2-c2ccccc2)[C@@H](C1)c1cc(F)cc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(OC[C@H](C)O)nn2-c2ccccc2)[C@@H](C1)c1ccc(F)cc1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(OC[C@H](O)C(F)(F)F)nn2-c2ccccc2)[C@@H](C1)c1cc(F)cc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(Cl)c(OCC(C)(C)O)nn2-c2ccccc2)[C@@H](C1)c1cc(F)cc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(Cl)c(OCC(C)(C)O)nn2-c2ccccc2)[C@@H](C1)c1ccc(F)cc1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(Cl)c(OC[C@@H](C)O)nn2-c2ccccc2)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(Cl)c(OC[C@@H](C)O)nn2-c2ccccc2)[C@@H](C1)c1cc(F)cc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(Cl)c(OC[C@@H](C)O)nn2-c2ccccc2)[C@@H](C1)c1ccc(F)cc1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(Br)c(OC[C@@H](C)O)nn2-c2ccccc2)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(Br)c(OC[C@@H](C)O)nn2-c2ccccc2)[C@@H](C1)c1cc(F)cc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(Br)c(OC[C@@H](C)O)nn2-c2ccccc2)[C@@H](C1)c1ccc(F)cc1 |r|
CC[C@@H](O)COc1nn(c(NC(=O)N[C@@H]2CN(CCOC)C[C@H]2c2cc(F)cc(F)c2)c1C)-c1ccccc1 |r|
CC[C@@H](O)COc1nn(c(NC(=O)N[C@@H]2CN(CCOC)C[C@H]2c2ccc(F)cc2)c1C)-c1ccccc1 |r|
CC[C@@H](O)COc1nn(c(NC(=O)N[C@@H]2CN(CCOC)C[C@H]2c2ccc(F)c(F)c2)c1C)-c1ccccc1 |r|
CCOC(=O)c1nn(c(NC(=O)N[C@@H]2CN(CCOC)C[C@H]2c2ccc(F)c(F)c2)c1Br)-c1ccccc1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnn(CCOC)c2)[C@@H](C1)c1ccc(F)cc1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnn(CCOC)c2)[C@@H](C1)c1cccc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnn(C)n2)[C@@H](C1)c1cccc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnn(C)n2)[C@@H](C1)c1ccc(F)cc1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(OCCN3CCOCC3)nn2-c2ccccc2)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(OCCN3C(=O)c4ccccc4C3=O)nn2-c2ccccc2)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(OCCN3CCN(CC3)C(=O)OC(C)(C)C)nn2-c2ccccc2)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2n(nc3ccccc23)-c2ccccc2)[C@@H](C1)c1ccccc1 |r|
COCCN1C[C@@H](NC(=O)Nc2n(nc3ccccc23)-c2ccccc2)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(OCc3ncn(C)n3)nn2-c2ccccc2)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(OC[C@@H]3COC(C)(C)O3)nn2-c2ccccc2)[C@@H](C1)c1cc(F)cc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(OC[C@H]3COC(C)(C)O3)nn2-c2ccccc2)[C@@H](C1)c1cc(F)cc(F)c1 |r|
CCOc1nn(c(NC(=O)N[C@@H]2CN(CCOC)C[C@H]2c2ccc(F)c(F)c2)c1C)-c1cnccn1 |r|
COCCN1C[C@@H](NC(=O)Nc2c3CCCc3nn2-c2ccnnc2)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(OC(=O)N(C)C)nn2-c2ccccc2)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(OC(=O)N3CCOCC3)nn2-c2ccccc2)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(OC[C@H]3COC(C)(C)O3)nn2-c2ccccc2)[C@@H](C1)c1cc(F)c(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(OC[C@@H]3COC(C)(C)O3)nn2-c2ccccc2)[C@@H](C1)c1cc(F)c(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(OC[C@H](C)O[Si](C)(C)C(C)(C)C)nn2-c2ccccc2)[C@@H](C1)c1cc(F)c(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(OCC(C)(C)O)nn2-c2ccccc2)[C@@H](C1)c1cc(F)c(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(OC[C@H](COC)O[Si](C)(C)C(C)(C)C)nn2-c2ccccc2)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(Cl)c(COC)nn2-c2ccccc2)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(Br)c(COC)nn2-c2ccccc2)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(Cl)c(COC)nn2-c2ccccc2)[C@@H](C1)c1cc(F)cc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(Br)c(COC)nn2-c2ccccc2)[C@@H](C1)c1cc(F)cc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(Cl)c(COC)nn2-c2ccccc2)[C@@H](C1)c1ccc(F)cc1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(Br)c(COC)nn2-c2ccccc2)[C@@H](C1)c1ccc(F)cc1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(Cl)c(nn2-c2ccccc2)C(F)(F)CO)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(Cl)c(nn2-c2ccccc2)C(F)(F)CO)[C@@H](C1)c1cc(F)cc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(Cl)c(nn2-c2ccccc2)C(F)(F)CO)[C@@H](C1)c1ccc(F)cc1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(Cl)c(C[C@H](C)O)nn2-c2ccccc2)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(Cl)c(C[C@@H](C)O)nn2-c2ccccc2)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(Br)c(C[C@@H](C)O)nn2-c2ccccc2)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(Cl)c(CC(C)(C)O)nn2-c2ccccc2)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(Cl)c(nn2-c2ccccc2)-c2nc(C)no2)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(Br)c(nn2-c2ccccc2)C(C)(C)C#N)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(Cl)c(nn2-c2ccccc2)C(C)(C)C#N)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(Br)c(nn2-c2ccccc2)-c2cnn(C)c2)[C@@H](C1)c1cc(F)cc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(Br)c(nn2-c2ccccc2)-c2cnn(C)c2)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(Br)c(nn2-c2ccccc2)-c2cnn(C)c2)[C@@H](C1)c1ccc(F)cc1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(Cl)c(nn2-c2ccccc2)-c2cnn(C)c2)[C@@H](C1)c1cc(F)cc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(Cl)c(nn2-c2ccccc2)-c2cnn(C)c2)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(Cl)c(nn2-c2ccccc2)-c2cnn(C)c2)[C@@H](C1)c1ccc(F)cc1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(Cl)c(nn2-c2ccccc2)-c2cnn(C)c2)[C@@H](C1)c1ccccc1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(Cl)c(nn2-c2ccccc2)-c2ccccc2)[C@@H](C1)c1cc(F)cc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(Br)c(nn2-c2ccccc2)-c2ccccc2)[C@@H](C1)c1cc(F)cc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(Br)c(nn2-c2ccccc2)-c2ccccc2)[C@@H](C1)c1ccc(F)cc1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(Cl)c(C)nn2-c2ccccc2)[C@@H](C1)c1cc(F)cc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(Br)c(C)nn2-c2ccccc2)[C@@H](C1)c1cc(F)cc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(Cl)c(nn2-c2ccccc2)-c2cnn(C)c2)[C@@H](C1)c1cncc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(F)c(nn2-c2ccccc2)-c2cnn(C)c2)[C@@H](C1)c1cncc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(Br)c(C)nn2-c2ccccc2)[C@@H](C1)c1cncc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(Cl)c(C)nn2-c2ccccc2)[C@@H](C1)c1cncc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(Br)c(nn2-c2ccccc2)-c2ccccc2)[C@@H](C1)c1cncc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(Cl)c(nn2-c2ccccc2)-c2ccccc2)[C@@H](C1)c1cncc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(Br)c(C)nn2-c2ccccc2)[C@@H](C1)c1ccc(F)cn1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(F)c(nn2-c2ccccc2)-c2cnn(C)c2)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(F)c(nn2-c2ccccc2)-c2cnn(C)c2)[C@@H](C1)c1cc(F)cc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(Br)c(nn2-c2ccccc2)-c2cnn(C)c2)[C@@H](C1)c1cncc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnn(C)c2)[C@@H](C1)c1ccc(F)cc1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnn(C)c2)[C@@H](C1)c1cc(F)cc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnn(C)c2)[C@@H](C1)c1cc(F)c(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnn(C)c2)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnn(C)c2)[C@@H](C1)c1ccccc1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnn(Cc3ccc(OC)cc3)c2)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cn[nH]c2)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(Cl)c(CCOC(C)=O)nn2-c2ccccc2)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(Cl)c(CCO)nn2-c2ccccc2)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)[C@@H]2C[C@H](O)C2)[C@@H](C1)c1ccc(F)c(F)c1 |r,wU:28.33,23.24,25.27,wD:6.6,(-6.93,6.86,;-5.6,7.63,;-4.26,6.86,;-2.93,7.63,;-1.6,6.86,;-1.6,5.32,;-.13,4.84,;.27,3.36,;-.82,2.27,;-2.31,2.67,;-.42,.78,;-.82,-.71,;.42,-1.61,;1.76,-.84,;-.05,-3.08,;-1.59,-3.08,;-2.07,-1.61,;-3.56,-1.21,;-3.96,.27,;-5.44,.67,;-6.53,-.42,;-6.13,-1.9,;-4.65,-2.3,;.72,-4.41,;.32,-5.9,;1.81,-6.3,;2.58,-7.63,;2.2,-4.81,;.77,6.09,;-.13,7.34,;2.31,6.09,;3.08,7.42,;4.62,7.42,;5.39,6.09,;6.93,6.09,;4.62,4.76,;5.39,3.42,;3.08,4.76,)|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)[C@H]2C[C@H](O)C2)[C@@H](C1)c1ccc(F)c(F)c1 |r,wU:28.33,23.24,wD:6.6,25.27,(-6.93,6.86,;-5.6,7.63,;-4.26,6.86,;-2.93,7.63,;-1.6,6.86,;-1.6,5.32,;-.13,4.84,;.27,3.36,;-.82,2.27,;-2.31,2.67,;-.42,.78,;-.82,-.71,;.42,-1.61,;1.76,-.84,;-.05,-3.08,;-1.59,-3.08,;-2.07,-1.61,;-3.56,-1.21,;-3.96,.27,;-5.44,.67,;-6.53,-.42,;-6.13,-1.9,;-4.65,-2.3,;.72,-4.41,;2.2,-4.81,;1.81,-6.3,;2.58,-7.63,;.32,-5.9,;.77,6.09,;-.13,7.34,;2.31,6.09,;3.08,7.42,;4.62,7.42,;5.39,6.09,;6.93,6.09,;4.62,4.76,;5.39,3.42,;3.08,4.76,)|
COCCN1C[C@@H](NC(=O)Nc2c(Cl)c(nn2-c2ccccc2)[C@@H]2C[C@H](O)C2)[C@@H](C1)c1ccc(F)c(F)c1 |r,wU:28.33,23.24,25.27,wD:6.6,(-6.93,6.86,;-5.6,7.63,;-4.26,6.86,;-2.93,7.63,;-1.6,6.86,;-1.6,5.32,;-.13,4.84,;.27,3.36,;-.82,2.27,;-2.31,2.67,;-.42,.78,;-.82,-.71,;.42,-1.61,;1.76,-.84,;-.05,-3.08,;-1.59,-3.08,;-2.07,-1.61,;-3.56,-1.21,;-3.96,.27,;-5.44,.67,;-6.53,-.42,;-6.13,-1.9,;-4.65,-2.3,;.72,-4.41,;.32,-5.9,;1.81,-6.3,;2.58,-7.63,;2.2,-4.81,;.77,6.09,;-.13,7.34,;2.31,6.09,;3.08,7.42,;4.62,7.42,;5.39,6.09,;6.93,6.09,;4.62,4.76,;5.39,3.42,;3.08,4.76,)|
COCCN1C[C@@H](NC(=O)Nc2c(Cl)c(nn2-c2ccccc2)[C@H]2C[C@H](O)C2)[C@@H](C1)c1ccc(F)c(F)c1 |r,wU:28.33,23.24,wD:6.6,25.27,(-6.93,6.86,;-5.6,7.63,;-4.26,6.86,;-2.93,7.63,;-1.6,6.86,;-1.6,5.32,;-.13,4.84,;.27,3.36,;-.82,2.27,;-2.31,2.67,;-.42,.78,;-.82,-.71,;.42,-1.61,;1.76,-.84,;-.05,-3.08,;-1.59,-3.08,;-2.07,-1.61,;-3.56,-1.21,;-3.96,.27,;-5.44,.67,;-6.53,-.42,;-6.13,-1.9,;-4.65,-2.3,;.72,-4.41,;2.2,-4.81,;1.81,-6.3,;2.58,-7.63,;.32,-5.9,;.77,6.09,;-.13,7.34,;2.31,6.09,;3.08,7.42,;4.62,7.42,;5.39,6.09,;6.93,6.09,;4.62,4.76,;5.39,3.42,;3.08,4.76,)|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)[C@@H]2C[C@H](O)C2)[C@@H](C1)c1ccc(F)cc1 |r,wU:28.33,23.24,25.27,wD:6.6,(-6.93,6.86,;-5.6,7.63,;-4.26,6.86,;-2.93,7.63,;-1.6,6.86,;-1.6,5.32,;-.13,4.84,;.27,3.36,;-.82,2.27,;-2.31,2.67,;-.42,.78,;-.82,-.71,;.42,-1.61,;1.76,-.84,;-.05,-3.08,;-1.59,-3.08,;-2.07,-1.61,;-3.56,-1.21,;-3.96,.27,;-5.44,.67,;-6.53,-.42,;-6.13,-1.9,;-4.65,-2.3,;.72,-4.41,;.32,-5.9,;1.81,-6.3,;2.58,-7.63,;2.2,-4.81,;.77,6.09,;-.13,7.34,;2.31,6.09,;3.08,7.42,;4.62,7.42,;5.39,6.09,;6.93,6.09,;4.62,4.76,;3.08,4.76,)|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)[C@H]2C[C@H](O)C2)[C@@H](C1)c1ccc(F)cc1 |r,wU:28.33,23.24,wD:6.6,25.27,(-6.93,6.86,;-5.6,7.63,;-4.26,6.86,;-2.93,7.63,;-1.6,6.86,;-1.6,5.32,;-.13,4.84,;.27,3.36,;-.82,2.27,;-2.31,2.67,;-.42,.78,;-.82,-.71,;.42,-1.61,;1.76,-.84,;-.05,-3.08,;-1.59,-3.08,;-2.07,-1.61,;-3.56,-1.21,;-3.96,.27,;-5.44,.67,;-6.53,-.42,;-6.13,-1.9,;-4.65,-2.3,;.72,-4.41,;2.2,-4.81,;1.81,-6.3,;2.58,-7.63,;.32,-5.9,;.77,6.09,;-.13,7.34,;2.31,6.09,;3.08,7.42,;4.62,7.42,;5.39,6.09,;6.93,6.09,;4.62,4.76,;3.08,4.76,)|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)[C@@H]2C[C@H](O)C2)[C@@H](C1)c1cc(F)cc(F)c1 |r,wU:28.33,23.24,25.27,wD:6.6,(-6.16,6.3,;-4.83,7.07,;-3.49,6.3,;-2.16,7.07,;-.83,6.3,;-.83,4.76,;.64,4.28,;1.04,2.79,;-.05,1.7,;-1.54,2.1,;.35,.22,;-.05,-1.27,;1.19,-2.18,;2.53,-1.41,;.72,-3.64,;-.82,-3.64,;-1.3,-2.18,;-2.79,-1.78,;-3.19,-.29,;-4.67,.11,;-5.76,-.98,;-5.36,-2.47,;-3.88,-2.87,;1.49,-4.97,;1.09,-6.46,;2.58,-6.86,;3.35,-8.19,;2.97,-5.37,;1.54,5.53,;.64,6.77,;3.08,5.53,;3.85,4.19,;5.39,4.19,;6.16,2.86,;6.16,5.53,;5.39,6.86,;6.16,8.19,;3.85,6.86,)|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)[C@H]2C[C@H](O)C2)[C@@H](C1)c1cc(F)cc(F)c1 |r,wU:28.33,23.24,wD:6.6,25.27,(-6.16,6.3,;-4.83,7.07,;-3.49,6.3,;-2.16,7.07,;-.83,6.3,;-.83,4.76,;.64,4.28,;1.04,2.79,;-.05,1.7,;-1.54,2.1,;.35,.22,;-.05,-1.27,;1.19,-2.18,;2.53,-1.41,;.72,-3.64,;-.82,-3.64,;-1.3,-2.18,;-2.79,-1.78,;-3.19,-.29,;-4.67,.11,;-5.76,-.98,;-5.36,-2.47,;-3.88,-2.87,;1.49,-4.97,;2.97,-5.37,;2.58,-6.86,;3.35,-8.19,;1.09,-6.46,;1.54,5.53,;.64,6.77,;3.08,5.53,;3.85,4.19,;5.39,4.19,;6.16,2.86,;6.16,5.53,;5.39,6.86,;6.16,8.19,;3.85,6.86,)|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)C(O)=O)[C@@H](C1)c1ccc(F)c(F)c1 |r|
CNC(=O)c1nn(c(NC(=O)N[C@@H]2CN(CCOC)C[C@H]2c2ccc(F)c(F)c2)c1C)-c1ccccc1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)C(=O)N(C)C)[C@@H](C1)c1ccc(F)c(F)c1 |r|
CCNC(=O)c1nn(c(NC(=O)N[C@@H]2CN(CCOC)C[C@H]2c2ccc(F)c(F)c2)c1C)-c1ccccc1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)C(=O)NC(C)C)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)C(N)=O)[C@@H](C1)c1ccc(F)c(F)c1 |r|
CCOc1nn(c(NC(=O)N[C@@H]2CN(CCOC)C[C@H]2c2cc(F)cc(F)c2)c1CO)-c1ccccc1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnn(C)c2)[C@@H](C1)c1ccc(F)c(Cl)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnn(C)c2)[C@@H](C1)c1ccc(Cl)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnn(C)c2)[C@@H](C1)c1cc(F)cc(Cl)c1 |r|
CCOc1nn(c(NC(=O)N[C@@H]2CN(CC(=O)OC)C[C@H]2c2ccc(F)c(F)c2)c1C)-c1ccccc1 |r|
CCOc1nn(c(NC(=O)N[C@@H]2CN(CC(O)C(F)(F)F)C[C@H]2c2ccc(F)c(F)c2)c1C)-c1ccccc1 |r|
CCOc1nn(c(NC(=O)N[C@@H]2CN(CC(C)O)C[C@H]2c2ccc(F)c(F)c2)c1C)-c1ccccc1 |r|
CCOc1nn(c(NC(=O)N[C@@H]2CN(CCC#N)C[C@H]2c2ccc(F)c(F)c2)c1C)-c1ccccc1 |r|
CCOc1nn(c(NC(=O)N[C@@H]2CN(CC(=O)NC)C[C@H]2c2ccc(F)c(F)c2)c1C)-c1ccccc1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(C)nn2C2CCCCC2)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(OCC(CO)CO)nn2-c2ccccc2)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(OCC(F)(F)F)nn2-c2ccccc2)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(OCC(F)(F)F)nn2-c2ccccc2)[C@@H](C1)c1ccc(F)cc1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(OCC(F)(F)F)nn2-c2ccccc2)[C@@H](C1)c1cc(F)cc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(OCC(F)F)nn2-c2ccccc2)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(Cl)c(OCC(F)(F)F)nn2-c2ccccc2)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(Cl)c(nn2-c2ccccc2)-c2ccccn2)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(Cl)c(nn2-c2ccccc2)-c2ccncc2)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(Cl)c(nn2-c2ccccc2)-c2cccnc2)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(Br)c(nn2-c2ccccc2)-c2cccnc2)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(Br)c(nn2-c2ccccc2)-c2ccccn2)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(Cl)c(nn2-c2cccnc2)-c2ccccc2)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cccnc2)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2ccncc2)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2ccccn2)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cncc(F)c2)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2cccnc2)-c2cncc(F)c2)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2ccn(C)n2)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2ccn(C)n2)[C@@H](C1)c1ccc(F)cc1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2ccn(C)n2)[C@@H](C1)c1cc(F)cc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2ccnn2C)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2cncc(F)c2)-c2cnn(C)c2)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2cncc(C)c2)-c2cnn(C)c2)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2cncc(Cl)c2)-c2cnn(C)c2)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnn(c2)C(OCC(F)(F)F)C(F)(F)F)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnn(CC(F)(F)F)c2)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnn(CC3CC3)c2)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnn(c2)C(=O)C2CC2)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnn(c2)S(C)(=O)=O)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnn(c2)C(C)C)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cncnc2)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2ccn(C)c(=O)c2)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2ccc(=O)n(C)c2)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnn(C)c2C)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cn(C)nc2C)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnn(c2)C2CC2)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc(C)s2)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc(C)nc2)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc(N)nc2)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2sc(C)nc2C)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cc(C)nc(C)c2)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2ccc(N)nc2)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(Br)nn2-c2ccccc2)[C@@H](C1)c1ccc(F)cc1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2ccc(=O)n(CC(F)(F)F)c2)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnn(c2)C(C)C)[C@@H](C1)c1ccc(F)cc1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2ccc(=O)n(C)c2)[C@@H](C1)c1ccc(F)cc1 |r|
Cc1c(Br)nn(c1NC(=O)N[C@H]1CN(CC(F)(F)F)C[C@@H]1c1ccccc1)-c1ccccc1 |r|
Cc1c(NC(=O)N[C@H]2CN(CC(F)(F)F)C[C@@H]2c2ccccc2)n(nc1-c1ccc(=O)n(C)c1)-c1ccccc1 |r|
Cc1c(NC(=O)N[C@H]2CN(CC(F)(F)F)C[C@@H]2c2ccccc2)n(nc1-c1cnc(N)nc1)-c1ccccc1 |r|
CCn1cc(cn1)-c1nn(c(NC(=O)N[C@@H]2CN(CCOC)C[C@H]2c2ccc(F)c(F)c2)c1C)-c1ccccc1 |r|
CCn1cc(cn1)-c1nn(c(NC(=O)N[C@@H]2CN(CCOC)C[C@H]2c2ccc(F)cc2)c1C)-c1ccccc1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(OS(=O)(=O)C(F)(F)F)nn2-c2ccccc2)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc(OC)nc2)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc(nc2)N(C)C)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc(OC)nc2)[C@@H](C1)c1ccc(F)cc1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc(nc2)N(C)C)[C@@H](C1)c1ccc(F)cc1 |r|
CCn1cc(cn1)-c1nn(c(NC(=O)N[C@@H]2CN(CCOC)C[C@H]2c2cccc(F)c2)c1C)-c1ccccc1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2ccn(C)c(=O)c2)[C@@H](C1)c1cccc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2ccn(C)c(=O)c2)[C@@H](C1)c1ccc(F)cc1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)C2CC2)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)C2CC2)[C@@H](C1)c1ccc(F)cc1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2ccc(=O)n(c2)C(C)C)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2ccc(=O)n(c2)C(C)C)[C@@H](C1)c1ccc(F)cc1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(OC[C@H](C)O)nn2-c2ccccc2)[C@@H](C1)c1cc(F)cc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(OCCN3CCNCC3)nn2-c2ccccc2)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(Cl)c(OCc3ccccc3)nn2C)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(OCC(O)=O)nn2-c2ccccc2)[C@@H](C1)c1ccc(F)c(F)c1 |r|
CCNC(=O)COc1nn(c(NC(=O)N[C@@H]2CN(CCOC)C[C@H]2c2ccc(F)c(F)c2)c1C)-c1ccccc1 |r|
CCc1c(OCC(C)(C)O)nn(c1NC(=O)N[C@@H]1CN(CCOC)C[C@H]1c1ccc(F)c(F)c1)-c1ccccc1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(OCCN)nn2-c2ccccc2)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(OCCNS(C)(=O)=O)nn2-c2ccccc2)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(OCCNC(C)=O)nn2-c2ccccc2)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(OCCN3CCN(CC3)C(C)=O)nn2-c2ccccc2)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(OCC(N)=O)nn2-c2ccccc2)[C@@H](C1)c1ccc(F)c(F)c1 |r|
CCOc1nn(c(NC(=O)N[C@@H]2CN(CCOC)C[C@H]2c2ccc(F)c(F)c2)c1NC(=O)C(F)(F)F)-c1ccccc1 |r|
CCOc1nn(c(NC(=O)N[C@@H]2CN(CCOC)C[C@H]2c2ccc(F)c(F)c2)c1N)-c1ccccc1 |r|
CCOc1nn(c(NC(=O)N[C@@H]2CN(CCOC)C[C@H]2c2ccc(F)c(F)c2)c1CCO)-c1ccccc1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(OCCN3CCN(C)CC3)nn2-c2ccccc2)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(OCC(=O)N3CCOCC3)nn2-c2ccccc2)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(Br)c(nn2-c2ccccc2)C(O)=O)[C@@H](C1)c1ccc(F)c(F)c1 |r|
CNC(=O)c1nn(c(NC(=O)N[C@@H]2CN(CCOC)C[C@H]2c2ccc(F)c(F)c2)c1Br)-c1ccccc1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(OCc3nnc(C)o3)nn2-c2ccccc2)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(Cl)c(nn2-c2ccccc2)-c2cnn(CCOC)c2)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(OC[C@@H](O)CO)nn2-c2ccccc2)[C@@H](C1)c1cc(F)cc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(OC[C@H](O)CO)nn2-c2ccccc2)[C@@H](C1)c1cc(F)cc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(OC[C@H](O)CO)nn2-c2ccccc2)[C@@H](C1)c1cc(F)c(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(OC[C@@H](O)CO)nn2-c2ccccc2)[C@@H](C1)c1cc(F)c(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(OC[C@H](C)O)nn2-c2ccccc2)[C@@H](C1)c1cc(F)c(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(OC[C@@H](O)COC)nn2-c2ccccc2)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(OC[C@H](O)COC)nn2-c2ccccc2)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(OC[C@@H](O)COC)nn2-c2ccccc2)[C@@H](C1)c1cc(F)c(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(OC[C@H](O)COC)nn2-c2ccccc2)[C@@H](C1)c1cc(F)c(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(Br)c(nn2C)-c2cnn(C)c2)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(Cl)c(nn2C)-c2cnn(C)c2)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(Cl)c(nn2-c2ccccc2)C2CCOCC2)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(Cl)c(nn2-c2ccccc2)C2CCN(CC2)C(=O)OC(C)(C)C)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(Cl)c(nn2-c2ccccc2)C2CCOCC2)[C@@H](C1)c1ccc(F)cc1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(Cl)c(nn2-c2ccccc2)-c2c(C)noc2C)[C@@H](C1)c1ccc(F)c(F)c1 |r,wU:30.35,wD:6.6,(-5.97,6.08,;-4.46,5.76,;-3.43,6.9,;-1.92,6.58,;-1.45,5.12,;-2.35,3.87,;-1.45,2.62,;-1.92,1.16,;-.89,.01,;.61,.34,;-1.37,-1.45,;-.34,-2.59,;1.19,-2.43,;1.96,-1.1,;1.82,-3.84,;.67,-4.87,;-.66,-4.1,;-2.07,-4.73,;-3.31,-3.82,;-4.72,-4.45,;-4.88,-5.98,;-3.63,-6.88,;-2.23,-6.26,;3.33,-4.16,;3.95,-5.57,;3.18,-6.9,;5.48,-5.41,;5.8,-3.9,;4.47,-3.13,;4.31,-1.6,;.02,3.1,;.02,4.64,;1.5,2.7,;1.9,1.21,;3.39,.82,;4.48,1.9,;5.97,1.51,;4.08,3.39,;5.17,4.48,;2.59,3.79,)|
COCCN1C[C@@H](NC(=O)Nc2c(Cl)c(nn2-c2ccccc2)[C@H]2CCCN2C(=O)OC(C)(C)C)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(Cl)c(nn2-c2ccccc2)[C@@H]2CCCN2C(=O)OC(C)(C)C)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(Br)c(nn2-c2ccccc2)C2CCOCC2)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(Br)c(nn2-c2ccccc2)C2CCN(CC2)C(=O)OC(C)(C)C)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(Br)c(nn2-c2ccccc2)C2CCOCC2)[C@@H](C1)c1ccc(F)cc1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(Br)c(nn2-c2ccccc2)-c2c(C)noc2C)[C@@H](C1)c1ccc(F)c(F)c1 |r,wU:30.35,wD:6.6,(-5.97,6.08,;-4.46,5.76,;-3.43,6.9,;-1.92,6.58,;-1.45,5.12,;-2.35,3.87,;-1.45,2.62,;-1.92,1.16,;-.89,.01,;.61,.34,;-1.37,-1.45,;-.34,-2.59,;1.19,-2.43,;1.96,-1.1,;1.82,-3.84,;.67,-4.87,;-.66,-4.1,;-2.07,-4.73,;-3.31,-3.82,;-4.72,-4.45,;-4.88,-5.98,;-3.63,-6.88,;-2.23,-6.26,;3.33,-4.16,;3.95,-5.57,;3.18,-6.9,;5.48,-5.41,;5.8,-3.9,;4.47,-3.13,;4.31,-1.6,;.02,3.1,;.02,4.64,;1.5,2.7,;1.9,1.21,;3.39,.82,;4.48,1.9,;5.97,1.51,;4.08,3.39,;5.17,4.48,;2.59,3.79,)|
COCCN1C[C@@H](NC(=O)Nc2c(Br)c(nn2-c2ccccc2)[C@H]2CCCN2C(=O)OC(C)(C)C)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(Br)c(COC3CCN(CC3)C(=O)OC(C)(C)C)nn2-c2ccccc2)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2cc(nn2-c2ccccc2)C2CCNCC2)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(Cl)c(nn2-c2ccccc2)C2CCNCC2)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(Br)c(nn2-c2ccccc2)C2CCNCC2)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)[C@H]2CCCN2)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)[C@@H]2CCCN2)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(Cl)c(nn2-c2ccccc2)[C@H]2CCCN2)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)[C@@H]2CCCN2)[C@@H](C1)c1cc(F)cc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(Cl)c(nn2-c2ccccc2)[C@@H]2CCCN2)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(Br)c(nn2-c2ccccc2)[C@H]2CCCN2)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2cc(COC3CCNCC3)nn2-c2ccccc2)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(Cl)c(COC3CCNCC3)nn2-c2ccccc2)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(Br)c(COC3CCNCC3)nn2-c2ccccc2)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(Br)c(nn2-c2ccccc2)C2CCN(CC2)S(C)(=O)=O)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(Br)c(nn2-c2ccccc2)C2CCN(CC2)C(C)=O)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(Cl)c(nn2-c2ccccc2)C2CCN(CC2)S(=O)(=O)C(F)(F)F)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)[C@H]2CCCN2S(C)(=O)=O)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)[C@H]2CCCN2C(C)=O)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)[C@H]2CCCN2C)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)[C@@H]2CCCN2C)[C@@H](C1)c1cc(F)cc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(Br)c(COC3CCN(CC3)S(C)(=O)=O)nn2-c2ccccc2)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(Br)c(COC3CCN(CC3)C(C)=O)nn2-c2ccccc2)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2nn(C(C)C)c(=O)o2)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2nn(C)c(=O)o2)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(Oc3cnccn3)nn2-c2ccccc2)[C@@H](C1)c1ccc(F)cc1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(c(OC)nn2-c2ccccc2)C(F)(F)F)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(F)c(OC)nn2-c2ccccc2)[C@@H](C1)c1cc(F)cc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(c(OC)nn2-c2ccccc2)C(F)(F)F)[C@@H](C1)c1ccc(F)cc1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cn(C)cn2)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(=O)[nH]n2-c2ccccc2)C(C1)c1ccc(Cl)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(=O)[nH]n2-c2ccccc2)[C@@H](C1)c1ccc(F)c(Cl)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(=O)[nH]n2-c2ccccc2)[C@@H](C1)c1cc(F)cc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(=O)[nH]n2-c2ccccc2)[C@@H](C1)c1cc(F)c(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(=O)[nH]n2-c2ccccc2)[C@@H](C1)c1cccc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(=O)[nH]n2-c2ccccc2)[C@@H](C1)c1cc(F)cc(Cl)c1 |r|
COCCN1C[C@@H](NC(=O)NC2=C(C#N)C(NN2c2ccccc2)OC)[C@@H](C1)c1ccc(F)c(F)c1 |r,c:11|
CCc1nn(c(NC(=O)N[C@@H]2CN(CCOC)C[C@H]2c2ccc(F)c(F)c2)c1C#N)-c1ccccc1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C#N)c(nn2-c2ccccc2)C(F)(F)F)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C#N)c(=O)[nH]n2-c2ccccc2)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C(N)=O)c(OC)nn2-c2ccccc2)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C(N)=O)c(C)nn2-c2ccccc2)[C@@H](C1)c1ccc(F)c(F)c1 |r|
CCc1nn(c(NC(=O)N[C@@H]2CN(CCOC)C[C@H]2c2ccc(F)c(F)c2)c1C(N)=O)-c1ccccc1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C(N)=O)c(nn2-c2ccccc2)C(F)(F)F)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C(N)=O)c(C)nn2-c2ccccc2)[C@@H](C1)c1ccc(F)c(Cl)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C(N)=O)c(C)nn2-c2ccccc2)[C@@H](C1)c1ccc(Cl)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C(N)=O)c(C)nn2-c2ccccc2)C(C1)c1cc(F)cc(Cl)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C(N)=O)c(C)nn2-c2ccccc2)[C@@H](C1)c1cc(F)cc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(cnn2-c2ccccc2)C(N)=O)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C(N)=O)c(nn2-c2ccccc2)C(F)F)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=N)Nc2c(Br)c(C)nn2-c2ccccc2)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=S)Nc2c(Br)c(C)nn2-c2ccccc2)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=S)Nc2c(C)c(nn2-c2ccccc2)-c2ccc(=O)n(C)c2)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=S)Nc2c(C)c(nn2-c2ccccc2)-c2cnn(C)c2)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=S)Nc2c(C)c(nn2-c2ccccc2)-c2cnn(C)c2)[C@@H](C1)c1ccc(F)cc1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(nn3ccccc23)-c2ccccc2)C(C1)c1ccccc1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(nn3ccccc23)-c2ccccc2)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2cnn3ccccc23)C(C1)c1ccccc1 |r|
COCCN1C[C@@H](NC(=O)Nc2cnn3ccccc23)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)n(nc2-c2ccccc2)-c2cnccn2)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)n(C)nc2-c2ccccc2)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)n(C)nc2-c2ccccc2)[C@@H](C1)c1cc(F)cc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)n(nc2-c2ccccc2)C(C)C)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)n(nc2-c2ccccc2)C(C)C)[C@@H](C1)c1cc(F)cc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)n(CC(F)(F)F)nc2-c2ccccc2)[C@@H](C1)c1ccc(F)c(F)c1 |r|
CCn1nc(c(NC(=O)N[C@@H]2CN(CCOC)C[C@H]2c2ccc(F)c(F)c2)c1C)-c1ccccc1 |r|
CCn1nc(C)c(NC(=O)N[C@@H]2CN(CCOC)C[C@H]2c2ccc(F)c(F)c2)c1-c1ccccc1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(nn(C)c2-c2ccccc2)C(F)(F)F)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(nn(C)c2C(F)(F)F)-c2ccccc2)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2cn(nc2C)-c2ccccc2)[C@@H](C1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2cn(nc2C(F)(F)F)-c2ccccc2)[C@@H](C1)c1ccc(F)c(F)c1 |r|
NC(=O)c1nccnc1C1=C2N=CC=CN2N(C1)N1CCC[C@@H]1c1cc(F)ccc1F |c:10,12,14|
O[C@@H]1CCN(C1)C(=O)C(=O)Nc1cnn2ccc(nc12)N1CCC[C@H]1c1cc(F)ccc1F
C[C@@H]1CN(CCN1)C(=O)Nc1cnc2ccc(nn12)N1CCC[C@H]1c1cc(F)ccc1F
C[C@H]1CN(CCN1)C(=O)Nc1cnc2ccc(nn12)N1CCC[C@H]1c1cc(F)ccc1F
OCC1CN(C1)c1cnc2ccc(nn12)N1CCC[C@@H]1c1cc(F)ccc1F
Fc1ccc(F)c(c1)[C@@H]1CCCN1c1ccc2ncc(NC(=O)C(F)(F)F)n2n1
Cc1c(NC(=O)NC2CCCc3ccccc23)n(nc1-c1cnn(C)c1)-c1ccccc1
Cc1c(NC(=O)N[C@H]2CCCc3ccccc23)n(nc1-c1cnn(C)c1)-c1ccccc1 |r|
O=C(N[C@H]1CCCc2ccccc12)Nc1c2CCCc2nn1-c1ccccc1 |r|
Cc1c(NC(=O)N[C@@H]2CCCc3ccccc23)n(nc1-c1cnn(C)c1)-c1ccccc1 |r|
COc1ccc2C(CCCc2c1)NC(=O)Nc1c(C)c(nn1-c1ccccc1)-c1cnn(C)c1
Cc1c(NC(=O)NC2CCCCc3ccccc23)n(nc1-c1cnn(C)c1)-c1ccccc1
Cc1c(NC(=O)NC2CCOc3ccccc23)n(nc1-c1cnn(C)c1)-c1ccccc1
Cc1c(NC(=O)NC2COCc3ccccc23)n(nc1-c1cnn(C)c1)-c1ccccc1
Cc1c(NC(=O)NC2CC(C)(C)Oc3ccccc23)n(nc1-c1cnn(C)c1)-c1ccccc1
Cc1c(NC(=O)NC2COCc3ccc(Br)cc23)n(nc1-c1cnn(C)c1)-c1ccccc1
Cc1nn(c(NC(=O)N[C@H]2CCCc3ccccc23)c1Br)-c1ccccc1 |r|
Cc1c(NC(=O)NC2CCOc3cc(F)ccc23)n(nc1-c1cnn(C)c1)-c1ccccc1
CCOc1nn(c(NC(=O)NC2CCOc3cc(F)ccc23)c1C)-c1ccccc1
CC1CC(NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnn(C)c2)c2cc(F)ccc2O1
Cc1c(NC(=O)NC2CCCc3ccc(Br)cc23)n(nc1-c1cnn(C)c1)-c1ccccc1
Cc1c(NC(=O)NC2CCC(C)(C)c3ccc(Br)cc23)n(nc1-c1cnn(C)c1)-c1ccccc1
COCCN1CCc2ccccc2C(C1)NC(=O)Nc1c(C)c(nn1-c1ccccc1)-c1cnn(C)c1
Cc1c(NC(=O)NC2CN(CC(F)(F)F)CCc3ccccc23)n(nc1-c1cnn(C)c1)-c1ccccc1
CC(=O)N1CCc2ccccc2C(C1)NC(=O)Nc1c(C)c(nn1-c1ccccc1)-c1cnn(C)c1
CCC(=O)N1CCc2ccccc2C(C1)NC(=O)Nc1c(C)c(nn1-c1ccccc1)-c1cnn(C)c1
CCCN1CCc2ccccc2C(C1)NC(=O)Nc1c(C)c(nn1-c1ccccc1)-c1cnn(C)c1
CCN1CC(NC(=O)Nc2c3CCCc3nn2-c2ccccc2)c2ccccc2C1
COCCN1CC(NC(=O)Nc2c3CCCc3nn2-c2ccccc2)c2ccccc2C1
CC(=O)N1CC(NC(=O)Nc2c3CCCc3nn2-c2ccccc2)c2ccccc2C1
Cc1c(NC(=O)NC2CN(CC(F)(F)F)Cc3ccccc23)n(nc1-c1cnn(C)c1)-c1ccccc1
Cc1c(NC(=O)NC2CN(CC(F)(F)F)Cc3ccccc23)n(nc1-c1ccc(=O)n(C)c1)-c1ccccc1
Cc1c(NC(=O)NC2CN(CC(F)(F)F)Cc3ccccc23)n(nc1-c1cn(C)cn1)-c1ccccc1
FC(F)(F)CN1CC(NC(=O)Nc2c3CCCc3nn2-c2ccccc2)c2ccccc2C1
CNC(=O)c1nn(c(NC(=O)NC2CN(CC(F)(F)F)Cc3ccccc23)c1C)-c1ccccc1
Cc1c(NC(=O)NC2CN(CC(F)(F)F)Cc3ccccc23)n([nH]c1=O)-c1ccccc1
Cc1nn(c(NC(=O)NC2CN(CC(F)(F)F)Cc3ccccc23)c1C(N)=O)-c1ccccc1
COCc1ccc2COCC(NC(=O)Nc3c(C)c(nn3-c3ccccc3)-c3cnn(C)c3)c2c1
Cc1c(NC(=O)NC2CC(Oc3ccc(Br)cc23)C2CC2)n(nc1-c1cnn(C)c1)-c1ccccc1
Cc1c(NC(=O)NC2CC3(CCC3)Oc3ccc(Br)cc23)n(nc1-c1cnn(C)c1)-c1ccccc1
COCc1ccc2OC3(CCC3)CC(NC(=O)Nc3c(C)c(nn3-c3ccccc3)-c3cnn(C)c3)c2c1
Cc1c(NC(=O)NC2CCC(=O)c3ccccc23)n(nc1-c1cnn(C)c1)-c1ccccc1
Cc1c(NC(=O)NC2CCC(C)(O)c3ccccc23)n(nc1-c1cnn(C)c1)-c1ccccc1
Cc1c(NC(=O)Nc2cn(CC(F)(F)F)c(=O)c3ccccc23)n(nc1-c1cnn(C)c1)-c1ccccc1
COc1nn(c(NC(=O)NC2CCN(C)c3ccccc23)c1C)-c1ccccc1
CN1CCC(NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnn(C)c2)c2ccccc12
CN1CCC(NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2ccc(=O)n(C)c2)c2ccccc12
CCN1CCC(NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2ccc(=O)n(C)c2)c2ccccc12
CN1CCC(NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2ccc(=O)n(C)c2)c2cccc(F)c12
CN1CCC(NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2ccc(=O)n(C)c2)c2cc(Cl)cc(F)c12
CCN1CCC(NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2ccc(=O)n(C)c2)c2cc(Cl)ccc12
CCN1CCC(NC(=O)Nc2c(C)c(OC)nn2-c2ccccc2)c2cc(Cl)ccc12
CO[C@H]1Cc2ccccc2[C@@H]1NC(=O)Nc1c2CCCc2nn1-c1ccccc1 |r|
COCCO[C@H]1Cc2ccccc2[C@@H]1NC(=O)Nc1c2CCCc2nn1-c1ccccc1 |r|
CCOc1nn(c(NC(=O)N[C@@H]2[C@H](Cc3ccccc23)OCCOC)c1C)-c1ccccc1 |r|
COCCO[C@@H]1Cc2ccccc2[C@H]1NC(=O)Nc1c2CCCc2nn1-c1ccccc1 |r|
COCCO[C@H]1Cc2ccccc2[C@@H]1NC(=O)Nc1c(C)c(nn1-c1ccccc1)-c1cnn(C)c1 |r|
COCCO[C@H]1Cc2ccccc2[C@@H]1NC(=O)Nc1c(Br)c(C)nn1-c1ccccc1 |r|
CCOc1nn(c(NC(=O)NC2CCc3ccccc23)c1C)-c1ccccc1
CCOc1nn(c(NC(=O)N[C@H]2CCc3ccccc23)c1C)-c1ccccc1 |r|
Cc1c(NC(=O)NC2[C@H](O)C3(CC3)c3ccccc23)n(nc1-c1cnn(C)c1)-c1ccccc1 |r|
Cc1c(NC(=O)NC2[C@H](O)C3(CC3)c3ccccc23)n(nc1-c1cnc(C)nc1)-c1ccccc1 |r|
COc1ncc(cn1)-c1nn(c(NC(=O)NC2[C@H](O)C3(CC3)c3ccccc23)c1C)-c1ccccc1 |r|
Cc1c(NC(=O)NC2[C@H](O)C3(CC3)c3cc(F)c(F)cc23)n(nc1-c1cnn(C)c1)-c1ccccc1 |r|
CNC(=O)c1nn(c(NC(=O)NC2[C@H](O)C3(CC3)c3ccccc23)c1C)-c1ccccc1 |r|
COc1nn(c(NC(=O)NC2[C@H](O)C3(CC3)c3ccccc23)c1C)-c1ccccc1 |r|
CCOc1nn(c(NC(=O)NC2[C@H](O)C3(CC3)c3ccccc23)c1C)-c1ccccc1 |r|
COc1nn(c(NC(=O)NC2[C@H](O)C3(CC3)c3cc(F)c(F)cc23)c1C)-c1ccccc1 |r|
Cc1c(NC(=O)NC2[C@H](O)C3(CC3)c3ccc(F)cc23)n(nc1-c1cnn(C)c1)-c1ccccc1 |r|
Cc1c(NC(=O)NC2[C@H](O)C3(CC3)c3cc(F)ccc23)n(nc1-c1cnn(C)c1)-c1ccccc1 |r|
Cc1c(NC(=O)N[C@H]2[C@H](O)Cc3ccccc23)n(nc1-c1cnn(C)c1)-c1ccccc1 |r|
Cc1c(NC(=O)N[C@H]2[C@H](O)Cc3ccccc23)n(nc1-c1cnc(C)nc1)-c1ccccc1 |r|
CCOc1ncc(cn1)-c1nn(c(NC(=O)N[C@H]2[C@H](O)Cc3ccccc23)c1C)-c1ccccc1 |r|
COc1ncc(cn1)-c1nn(c(NC(=O)N[C@H]2[C@H](O)Cc3ccccc23)c1C)-c1ccccc1 |r|
Cc1c(NC(=O)N[C@H]2[C@H](O)Cc3ccccc23)n(nc1-c1cc(C)c(=O)n(C)c1)-c1ccccc1 |r|
Cc1c(NC(=O)NC2[C@H](O)Cc3ccc(Cl)cc23)n(nc1-c1cnn(C)c1)-c1ccccc1 |r|
Cc1c(NC(=O)NC2[C@H](O)Cc3ccc(Cl)cc23)n(nc1-c1cnc(C)nc1)-c1ccccc1 |r|
Cc1c(NC(=O)NC2[C@H](O)C(C)(C)c3ccccc23)n(nc1-c1cnn(C)c1)-c1ccccc1 |r|
Cc1c(NC(=O)NC2[C@H](O)C(C)(C)c3ccccc23)n(nc1-c1cnc(C)nc1)-c1ccccc1 |r|
CN1CCO[C@@H](COc2nn(c(NC(=O)N[C@H]3[C@H](O)CC(C)(C)c4ccccc34)c2C)-c2ccccc2)C1 |r|
CN1CCO[C@@H](COc2nn(c(NC(=O)N[C@@H]3[C@@H](O)CC(C)(C)c4ccccc34)c2C)-c2ccccc2)C1 |r|
CN1CCO[C@H](COc2nn(c(NC(=O)N[C@H]3[C@H](O)CC(C)(C)c4ccccc34)c2C)-c2ccccc2)C1 |r|
CN1CCO[C@@H](COc2nn(c(NC(=O)NC3[C@H](O)CC(C)(C)c4cc(F)c(F)cc34)c2C)-c2ccccc2)C1 |r|
CN1CCO[C@@H](COc2nn(c(NC(=O)NC3[C@@H](O)C4(CC4)c4ccccc34)c2C)-c2ccccc2)C1 |r|
CNC(=O)c1nn(c(NC(=O)NC2[C@H](O)CC(C)(C)c3cc(F)c(F)cc23)c1C)-c1ccccc1 |r|
Cc1c(NC(=O)N[C@H]2[C@H](O)CC(C)(C)c3cc(F)c(F)cc23)n(nc1-c1cnn(C)c1)-c1ccccc1 |r|
CN1CCC(COc2nn(c(NC(=O)N[C@H]3[C@H](O)CC(C)(C)c4cc(F)c(F)cc34)c2C)-c2ccccc2)CC1 |r|
COc1nn(c(NC(=O)N[C@H]2[C@H](O)CC(C)(C)c3cc(F)c(F)cc23)c1C)-c1ccccc1 |r|
Cc1c(NC(=O)N[C@H]2[C@H](O)CC(C)(C)c3cc(F)c(F)cc23)n(nc1-c1ccc(=O)n(C)c1)-c1ccccc1 |r|
Cc1c(NC(=O)N[C@H]2[C@H](O)CC(C)(C)c3cc(F)c(F)cc23)n(nc1-c1cnc(C)nc1)-c1ccccc1 |r|
CNC(=O)c1nn(c(NC(=O)N[C@H]2[C@H](O)[C@H](OC)C(C)(C)c3ccccc23)c1C)-c1ccccc1 |r|
CO[C@H]1[C@@H](O)[C@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnn(C)c2)c2ccccc2C1(C)C |r|
CO[C@H]1[C@@H](O)[C@H](NC(=O)Nc2c(C)c(OCC3CCN(C)CC3)nn2-c2ccccc2)c2ccccc2C1(C)C |r|
CNC(=O)c1nn(c(NC(=O)N[C@H]2[C@H](O)CC(C)(C)c3cc(F)ccc23)c1C)-c1ccccc1 |r|
Cc1c(NC(=O)N[C@H]2[C@H](O)CC(C)(C)c3cc(F)ccc23)n(nc1-c1cnn(C)c1)-c1ccccc1 |r|
Cc1c(NC(=O)N[C@H]2[C@H](O)CC(C)(C)c3cc(F)ccc23)n(nc1-c1ccc(=O)n(C)c1)-c1ccccc1 |r|
CNC(=O)c1nn(c(NC(=O)N[C@H]2[C@H](O)CC(C)(C)c3ccc(F)cc23)c1C)-c1ccccc1 |r|
Cc1c(NC(=O)N[C@H]2[C@H](O)CC(C)(C)c3ccc(F)cc23)n(nc1-c1cnn(C)c1)-c1ccccc1 |r|
Cc1c(NC(=O)N[C@H]2[C@H](O)CC(C)(C)c3ccc(F)cc23)n(nc1-c1ccc(=O)n(C)c1)-c1ccccc1 |r|
Cc1c(CCO)nn(c1NC(=O)N[C@H]1[C@H](O)CC(C)(C)c2ccccc12)-c1ccccc1 |r|
Cc1c(NC(=O)NC2[C@H](O)CC(C)(C)c3ccccc23)n([nH]c1=O)-c1ccccc1 |r|
COCc1ccc2C(C)N(CC(F)(F)F)CC(NC(=O)Nc3c(C)c(=O)[nH]n3-c3ccccc3)c2c1
COc1nn(c(NC(=O)NC2[C@H](O)CC(C)(C)c3ccccc23)c1C)-c1ccccc1 |r|
Cc1nn(c(NC(=O)NC2[C@H](O)CC(C)(C)c3ccc(cc23)C(N)=O)c1C)-c1ccccc1 |r|
COC(=O)c1ccc2c(c1)C(NC(=O)Nc1c(C)c(C)nn1-c1ccccc1)[C@H](O)CC2(C)C |r|
Cc1nn(c(NC(=O)NC2[C@H](O)CC(C)(C)c3ccc(CO)cc23)c1C)-c1ccccc1 |r|
Cc1c(NC(=O)NC2[C@H](O)CCc3ccccc23)n(nc1-c1cnn(C)c1)-c1ccccc1 |r|
COCc1ccc2c(c1)C(NC(=O)Nc1c(C)c(nn1-c1ccccc1)-c1cnn(C)c1)[C@H](O)CC2(C)C |r|
Cc1c(NC(=O)N[C@H]2CCCc3cc(F)ccc23)n(nc1-c1cnn(C)c1)-c1ccccc1 |r|
Cc1c(NC(=O)NC2[C@H](O)CC(C)(C)c3ccc(Cl)cc23)n(nc1-c1cnn(C)c1)-c1ccccc1 |r|
Cc1c(NC(=O)NC2[C@H](O)CC(C)(C)c3ccccc23)n(nc1-c1cnn(C)c1)-c1ccccc1 |r|
Cc1c(NC(=O)NC2[C@H](O)CC(C)(C)c3ccccc23)n(nc1-c1ccc(=O)n(C)c1)-c1ccccc1 |r|
Cc1c(NC(=O)NC2[C@H](O)CC(C)(C)c3ccccc23)n(nc1-c1ccn(C)c(=O)c1)-c1ccccc1 |r|
CC1(C)C[C@@H](O)C(NC(=O)Nc2c3COCc3nn2-c2ccccc2)c2ccccc12 |r|
COCc1ccc2C(C)N(CC(F)(F)F)CC(NC(=O)Nc3c(C)c(nn3-c3ccccc3)-c3cnn(C)c3)c2c1
COCc1ccc2C(C)N(CC(F)(F)F)CC(NC(=O)Nc3c(C)c(nn3-c3ccccc3)C(N)=O)c2c1
COCc1ccc2C(C)N(CC(F)(F)F)CC(NC(=O)Nc3c(C)c(nn3-c3ccccc3)-c3cn(C)cn3)c2c1
Cc1c(NC(=O)NC2CCSc3ccc(Br)cc23)n(nc1-c1cnn(C)c1)-c1ccccc1
Cc1c(NC(=O)NC2CCS(=O)(=O)c3ccc(Br)cc23)n(nc1-c1cnn(C)c1)-c1ccccc1
Cc1c(NC(=O)NC2CSCc3ccc(Br)cc23)n(nc1-c1cnn(C)c1)-c1ccccc1
Cc1c(NC(=O)NC2CS(=O)(=O)Cc3ccc(Br)cc23)n(nc1-c1cnn(C)c1)-c1ccccc1
Cc1c(NC(=O)NC2CN(CC(F)(F)F)C(=O)c3ccccc23)n(nc1-c1cnn(C)c1)-c1ccccc1
Cc1c(NC(=O)NC2[C@H](O)CC(C)(C)c3ccccc23)n(nc1-c1cnc(C)nc1)-c1ccccc1 |r|
Cc1c(NC(=O)NC2[C@H](O)CCc3ccccc23)n(nc1-c1cnc(C)nc1)-c1ccccc1 |r|
COc1ncc(cn1)-c1nn(c(NC(=O)NC2[C@H](O)CCc3ccccc23)c1C)-c1ccccc1 |r|
CNC(=O)c1nn(c(NC(=O)NC2[C@H](O)CC(C)(C)c3ccc(COC)cc23)c1C)-c1ccccc1 |r|
Cc1nn(c(NC(=O)NC2[C@H](O)CCc3ccccc23)c1C)-c1ccccc1 |r|
CN1CCC(COc2nn(c(NC(=O)NC3[C@H](O)CC(C)(C)c4ccccc34)c2C)-c2ccccc2)CC1 |r|
CN1CCC(COc2nn(c(NC(=O)NC3[C@H](O)CCc4ccccc34)c2C)-c2ccccc2)CC1 |r|
CNC(=O)c1nn(c(NC(=O)NC2[C@H](O)CC(C)(C)c3ccccc23)c1C)-c1ccccc1 |r|
CNC(=O)c1nn(c(NC(=O)NC2[C@H](O)CC(C)(C)c3ccc(Cl)cc23)c1C)-c1ccccc1 |r|
Cc1nn(c(NC(=O)NC2[C@H](O)CCCc3ccccc23)c1C)-c1ccccc1 |r|
Cc1c(NC(=O)NC2[C@H](O)CCCc3ccccc23)n(nc1-c1cnc(C)nc1)-c1ccccc1 |r|
COc1ncc(cn1)-c1nn(c(NC(=O)NC2[C@H](O)CCCc3ccccc23)c1C)-c1ccccc1 |r|
CNC(=O)c1nn(c(NC(=O)NC2CN(CC(F)(F)F)C(C)c3ccc(COC)cc23)c1C)-c1ccccc1
Cc1c(NC(=O)NC2CN(CC(F)(F)F)C(=O)c3ccccc23)n(nc1-c1cnc(C)nc1)-c1ccccc1
Cc1nn(c(NC(=O)NC2CN(CC(F)(F)F)C(=O)c3ccccc23)c1C)-c1ccccc1
Cc1c(OC2CN3CCC2CC3)nn(c1NC(=O)N[C@H]1[C@H](O)CC(C)(C)c2ccccc12)-c1ccccc1 |r,wU:20.23,wD:19.21,TLB:3:4:7.8:10.11,(2.23,-3.74,;.9,-2.97,;-.35,-3.87,;.05,-5.36,;1.39,-6.13,;1.79,-7.62,;3.27,-8.01,;4.36,-6.92,;3.96,-5.44,;2.48,-5.04,;3.56,-6.13,;3.56,-7.13,;-1.59,-2.97,;-1.12,-1.5,;.42,-1.5,;1.51,-.41,;1.12,1.08,;-.37,1.47,;2.2,2.17,;2.2,3.71,;3.29,4.79,;4.78,4.4,;2.89,6.28,;1.41,6.68,;.64,8.01,;2.18,8.01,;.32,5.59,;-1.17,5.99,;-2.26,4.9,;-1.86,3.41,;-.37,3.01,;.72,4.1,;-2.2,-.41,;-1.81,1.08,;-2.89,2.17,;-4.38,1.77,;-4.78,.28,;-3.69,-.81,)|
Cc1c(OCCN2CCOCC2)nn(c1NC(=O)N[C@H]1[C@H](O)CC(C)(C)c2ccccc12)-c1ccccc1 |r|
CN(C)CCOc1nn(c(NC(=O)N[C@H]2[C@H](O)CC(C)(C)c3ccccc23)c1C)-c1ccccc1 |r|
COc1nn(c(NC(=O)N[C@H]2[C@@H](O)CCc3ccccc23)c1C)-c1ccccc1 |r|
Cc1c(NC(=O)NC2CN(CC(F)(F)F)C3(CC3)c3ccccc23)n(nc1-c1cnn(C)c1)-c1ccccc1
Cc1c(NC(=O)N[C@H]2[C@H](O)C3(CC3)c3ccccc23)n(nc1-c1cnn(C)c1)-c1ccccc1 |r|
CC(C)(C)OC(=O)N1CCO[C@@H](COc2nn(c(NC(=O)N[C@H]3[C@H](O)C4(CC4)c4ccccc34)c2Cl)-c2ccccc2)C1 |r|
O[C@H]1[C@H](NC(=O)Nc2c(Cl)c(OC[C@H]3CNCCO3)nn2-c2ccccc2)c2ccccc2C11CC1 |r|
CN1CCO[C@@H](COc2nn(c(NC(=O)N[C@H]3[C@H](O)C4(CC4)c4ccccc34)c2Cl)-c2ccccc2)C1 |r|
Cc1c(NC(=O)N[C@H]2[C@H](O)C3(CCC3)c3ccccc23)n(nc1-c1cnn(C)c1)-c1ccccc1 |r|
Cc1c(OC[C@H]2CN(CCO2)C(=O)OC(C)(C)C)nn(c1NC(=O)NC1[C@H](O)CC(C)(C)c2ccccc12)-c1ccccc1 |r|
COc1nn(c(NC(=O)N[C@H]2[C@H](O)CC(C)(C)c3ccccc23)c1C)-c1ccccc1 |r|
Cn1nc(cc1NC(=O)N[C@H]1[C@H](O)CC(C)(C)c2ccccc12)-c1ccccc1 |r|
CCOc1nn(c(NC(=O)N[C@H]2[C@H](O)CC(C)(C)c3ccccc23)c1C)-c1ccccc1 |r|
COCCOc1nn(c(NC(=O)N[C@H]2[C@H](O)CC(C)(C)c3ccccc23)c1C)-c1ccccc1 |r|
Cc1c(OCCO)nn(c1NC(=O)N[C@H]1[C@H](O)CC(C)(C)c2ccccc12)-c1ccccc1 |r|
Cc1c(OC[C@H]2CNCCO2)nn(c1NC(=O)N[C@H]1[C@H](O)CC(C)(C)c2ccccc12)-c1ccccc1 |r|
CC(C)N1CCO[C@@H](COc2nn(c(NC(=O)N[C@H]3[C@H](O)CC(C)(C)c4ccccc34)c2C)-c2ccccc2)C1 |r|
COc1nn(c(NC(=O)N[C@H]2[C@H](O)CC3(CC3)c3ccccc23)c1C)-c1ccccc1 |r|
CO[C@H]1[C@@H](O)[C@H](NC(=O)Nc2c(C)c(OC)nn2-c2ccccc2)c2ccccc2C1(C)C |r|
CO[C@H]1[C@@H](O)[C@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2ccc(=O)n(C)c2)c2ccccc2C1(C)C |r|
CO[C@H]1[C@@H](O)[C@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc(C)nc2)c2ccccc2C1(C)C |r|
CNC(=O)c1nn(c(NC(=O)N[C@H]2[C@H](O)[C@@H](OC)C(C)(C)c3ccccc23)c1C)-c1ccccc1 |r|
CO[C@@H]1[C@@H](O)[C@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnn(C)c2)c2ccccc2C1(C)C |r|
CO[C@@H]1[C@@H](O)[C@H](NC(=O)Nc2c(C)c(OCC3CCN(C)CC3)nn2-c2ccccc2)c2ccccc2C1(C)C |r|
COc1nn(c(NC(=O)N[C@H]2[C@H](O)C3(CCC3)Oc3ccccc23)c1C)-c1ccccc1 |r|
Cc1c(NC(=O)N[C@H]2[C@H](O)C3(CCC3)Oc3ccccc23)n(nc1-c1cnn(C)c1)-c1ccccc1 |r|
CN1CCN(CC1)c2ccc(c(c2)NC3CCOCC3)C(=O)Nc4c5cc(ccc5[nH]n4)Cc6cc(cc(c6)F)F
CC(C)NC(=O)[C@H]1CC[C@H](CC1)n1c(NC(=O)c2ccc(F)cc2)nc2ccc(CN3CCC(CC3)C(C)(C)O)cc12 |r,wU:9.12,6.5,(21.34,-25.87,;19.83,-25.56,;19.35,-24.09,;18.81,-26.7,;17.3,-26.39,;16.27,-27.53,;16.82,-24.92,;15.31,-24.6,;14.83,-23.15,;15.87,-22,;17.37,-22.31,;17.85,-23.77,;15.38,-20.54,;16.29,-19.28,;17.83,-19.27,;18.59,-17.94,;17.81,-16.61,;20.13,-17.93,;20.9,-19.25,;22.44,-19.25,;23.2,-17.91,;24.74,-17.9,;22.42,-16.57,;20.88,-16.59,;15.37,-18.03,;13.9,-18.52,;12.56,-17.76,;11.23,-18.53,;11.23,-20.07,;9.9,-20.84,;8.56,-20.07,;8.56,-18.53,;7.24,-17.76,;5.9,-18.52,;5.9,-20.06,;7.23,-20.84,;4.56,-17.74,;3.79,-16.41,;5.33,-16.4,;3.23,-18.51,;12.56,-20.84,;13.9,-20.07,)|
C[C@@H](Oc1cc(cnc1N)-c1cnn(c1)C1CCNCC1)c1c(Cl)ccc(F)c1Cl |r|
F[C@H]1C[C@@H](N(C1)c1ccn2ncc(C#N)c2n1)c1cncc(F)c1 |r|
F[C@H]1C[C@@H](N(C1)c1ccn2ncc(C#N)c2n1)c1cc(F)ccc1F |r|
Fc1cncc(c1)[C@H]1CC(F)(F)CN1c1ccn2ncc(C#N)c2n1 |r|
F[C@H]1C[C@@H](N(C1)c1nc2c(cnn2cc1F)C#N)c1cncc(F)c1 |r|
Fc1ccc(F)c(c1)[C@H]1C[C@@H](CN1c1ccn2ncc(C#N)c2n1)C#N |r|
F[C@H]1C[C@@H](N(C1)c1ccn2ncc(C#N)c2n1)c1cc(F)cc(c1)C#N |r|
COc1ncc(F)cc1[C@H]1C[C@H](F)CN1c1ccn2ncc(C#N)c2n1 |r|
Cn1cc(F)cc([C@H]2C[C@H](F)CN2c2ccn3ncc(C#N)c3n2)c1=O |r|
F[C@H]1C[C@@H](N(C1)c1ccn2ncc(C#N)c2n1)c1cc(F)cc(Cl)c1 |r|
F[C@H]1C[C@@H](N(C1)c1ccn2ncc(C#N)c2n1)c1cc(F)cnc1Cl |r|
NC(=O)c1cc(F)cc(c1)[C@H]1C[C@H](F)CN1c1ccn2ncc(C#N)c2n1 |r|
F[C@H]1C[C@@H](N(C1)c1nc2c(cnn2cc1F)C#N)c1cc(F)cc(c1)C#N |r|
COc1c(F)cc(F)cc1[C@H]1C[C@H](F)CN1c1ccn2ncc(C#N)c2n1 |r|
CC(C)(O)c1cc(F)cc(c1)[C@H]1C[C@H](F)CN1c1ccn2ncc(C#N)c2n1 |r|
NC(=O)c1cc(F)cc(c1)[C@H]1C[C@H](F)CN1c1nc2c(cnn2cc1F)C#N |r|
NS(=O)(=O)c1cc(F)cc(c1)[C@H]1C[C@H](F)CN1c1ccn2ncc(C#N)c2n1 |r|
F[C@H]1C[C@@H](N(C1)c1ccn2ncc(C#N)c2n1)c1cc(F)ccc1OC(F)(F)F |r|
OCCNC(=O)c1cc(F)cc(c1)[C@H]1C[C@H](F)CN1c1ccn2ncc(C#N)c2n1 |r|
F[C@H]1C[C@@H](N(C1)c1ccn2ncc(C#N)c2n1)c1cc(F)cc(c1)C(=O)NCC1CC1 |r|
CNC(=O)c1cc(F)cc(c1)[C@H]1C[C@H](F)CN1c1ccn2ncc(C#N)c2n1 |r|
CN(C)C(=O)c1cc(F)cc(c1)[C@H]1C[C@H](F)CN1c1ccn2ncc(C#N)c2n1 |r|
NC(=O)c1ccc(F)cc1[C@H]1C[C@H](F)CN1c1ccn2ncc(C#N)c2n1 |r|
CC1(C)C[C@@H](O)[C@H](NC(=O)Nc2cccnc2-c2ccccc2)c2ccccc12 |r|
Cc1cnc(c(NC(=O)N[C@H]2[C@H](O)CC(C)(C)c3ccccc23)c1)-c1ccccc1 |r|
Cc1ncc(cn1)-c1nc(c(NC(=O)N[C@H]2[C@H](O)CC(C)(C)c3ccccc23)cc1C)-c1ccccc1 |r|
Cc1cc(NC(=O)N[C@H]2[C@H](O)CC(C)(C)c3ccccc23)c(nc1-c1cnn(C)c1)-c1ccccc1 |r|
Cc1cc(NC(=O)N[C@H]2[C@H](O)CC(C)(C)c3ccccc23)c(nc1-c1cn[nH]c1)-c1ccccc1 |r|
Cc1cc(NC(=O)N[C@H]2[C@H](O)CC(C)(C)c3ccccc23)c(nc1-c1ccc(O)nc1)-c1ccccc1 |r|
Cc1cc(NC(=O)N[C@H]2[C@H](O)CC(C)(C)c3ccccc23)c(nc1CO)-c1ccccc1 |r|
Cc1cc(NC(=O)N[C@H]2[C@H](O)CC(C)(C)c3ccccc23)c(nc1-c1cncc(c1)C(F)(F)F)-c1ccccc1 |r|
Cc1ccc(cn1)-c1nc(c(NC(=O)N[C@H]2[C@H](O)CC(C)(C)c3ccccc23)cc1C)-c1ccccc1 |r|
Cc1cc(NC(=O)N[C@H]2[C@H](O)CC(C)(C)c3ccccc23)c(nc1-c1ccc(nc1)C#C)-c1ccccc1 |r|
Cc1cc(NC(=O)N[C@H]2[C@H](O)CC(C)(C)c3ccccc23)c(nc1-c1ccc(nc1)S(C)(=O)=O)-c1ccccc1 |r|
Cc1cc(NC(=O)N[C@H]2[C@H](O)CC(C)(C)c3ccccc23)c(nc1-c1cnc(nc1)C(F)(F)F)-c1ccccc1 |r|
Cc1cc(NC(=O)N[C@H]2[C@H](O)CC(C)(C)c3ccccc23)c(nc1-c1ccc(cc1)C#N)-c1ccccc1 |r|
Cc1cc(NC(=O)N[C@H]2[C@H](O)CC(C)(C)c3ccccc23)c(nc1-c1ccnc(c1)C(F)(F)F)-c1ccccc1 |r|
Cc1cc(NC(=O)N[C@H]2[C@H](O)CC(C)(C)c3ccccc23)c(nc1-c1cnc(O)nc1)-c1ccccc1 |r|
Cc1cc(NC(=O)NC2[C@H](O)CC(C)(C)c3ccccc23)c(nc1-c1ccc(O)nc1)-c1ccccc1 |r|
Cc1cc(NC(=O)N[C@H]2[C@H](O)CC(C)(C)c3ccccc23)c(nc1-c1cnc(nc1)C(C)(C)C)-c1ccccc1 |r|
Cc1cnc(c(NC(=O)N[C@H]2[C@H](O)CC(C)(C)c3cc(Br)ccc23)c1)-c1ccccc1 |r|
Cc1cc(NC(=O)N[C@H]2[C@H](O)CC(C)(C)c3cc(Br)ccc23)c(nc1C(N)=O)-c1ccccc1 |r|
Cc1cc(NC(=O)N[C@H]2[C@H](O)CC(C)(C)c3ccccc23)c(nc1C(N)=O)-c1ccccc1 |r|
Cc1cc(NC(=O)N[C@H]2[C@H](O)CC(C)(C)c3ccccc23)c(nc1C(=O)NCC(C)(C)O)-c1ccccc1 |r|
Cc1cnc(C2CCOCC2)c(NC(=O)N[C@H]2[C@H](O)CC(C)(C)c3ccccc23)c1 |r|
Cc1cc(NC(=O)N[C@H]2[C@H](O)CC(C)(C)c3ccccc23)c(nc1C(N)=O)C1CCOCC1 |r|
Cc1ncc(cn1)-c1nc(C2CCOCC2)c(NC(=O)N[C@H]2[C@H](O)CC(C)(C)c3ccccc23)cc1C |r|
Cc1cc(NC(=O)N[C@H]2[C@H](O)CC(C)(C)c3ccccc23)c(nc1-c1cnn(C)c1)C1CCOCC1 |r|
Cc1cc(NC(=O)N[C@H]2[C@H](O)CC(C)(C)c3ccccc23)c(nc1-c1cn[nH]c1)C1CCOCC1 |r|
Cc1cc(NC(=O)N[C@H]2[C@H](O)CC(C)(C)c3ccccc23)c(nc1-c1ccc(O)nc1)C1CCOCC1 |r|
Cc1cnc(c(NC(=O)N[C@H]2[C@H](O)CC(C)(C)c3ccc(Br)cc23)c1)-c1ccccc1 |r|
COc1ccc2c(c1)[C@@H](NC(=O)Nc1cc(C)cnc1C1CCOCC1)[C@H](O)CC2(C)C |r|
Cc1ncc(cn1)-c1nc(c(NC(=O)N[C@H]2[C@H](O)CC(C)(C)c3ccc(F)cc23)cc1C)-c1ccccc1 |r|
Cc1ncc(cn1)-c1nc(c(NC(=O)N[C@@H]2[C@H](O)CC(C)(C)c3ccc(F)cc23)cc1C)-c1ccccc1 |r|
Cc1ncc(cn1)-c1nc(c(NC(=O)N[C@H]2[C@H](O)CC(C)(C)c3cc(F)ccc23)cc1C)-c1ccccc1 |r|
Cc1ncc(cn1)-c1nc(c(NC(=O)N[C@@H]2[C@H](O)CC(C)(C)c3cc(F)ccc23)cc1C)-c1ccccc1 |r|
CC1(C)C[C@@H](O)[C@H](NC(=O)Nc2cccnc2-c2ccccc2)c2cc(F)c(F)cc12 |r|
Cc1cnc(c(NC(=O)N[C@H]2[C@H](O)CC(C)(C)c3cc(F)c(F)cc23)c1)-c1ccccc1 |r|
Cc1cnc(c(NC(=O)N[C@@H]2[C@H](O)CC(C)(C)c3cc(F)c(F)cc23)c1)-c1ccccc1 |r|
Cc1ccnc(-c2ccccc2)c1NC(=O)N[C@H]1[C@H](O)CC(C)(C)c2cc(F)c(F)cc12 |r|
Cc1ccc(NC(=O)N[C@H]2[C@H](O)CC(C)(C)c3cc(F)c(F)cc23)c(n1)-c1ccccc1 |r|
Cc1cc(NC(=O)NC2[C@H](O)CC(C)(C)c3cc(F)c(F)cc23)c(nc1C(N)=O)-c1ccccc1 |r|
Cc1nnc(CNC(=O)c2nc(c(NC(=O)NC3[C@H](O)CC(C)(C)c4cc(F)c(F)cc34)cc2C)-c2ccccc2)o1 |r|
Cc1nnc(CNC(=O)c2nc(c(NC(=O)N[C@H]3[C@H](O)CC(C)(C)c4cc(F)c(F)cc34)cc2C)-c2ccccc2)o1 |r|
Cc1nnc(CNC(=O)c2nc(c(NC(=O)N[C@@H]3[C@H](O)CC(C)(C)c4cc(F)c(F)cc34)cc2C)-c2ccccc2)o1 |r|
Cc1cc(NC(=O)N[C@H]2[C@H](O)CC(C)(C)c3cc(F)c(F)cc23)c(nc1C(=O)NCC(C)(C)O)-c1ccccc1 |r|
Cc1cc(NC(=O)NC2[C@H](O)CC(C)(C)c3cc(F)c(F)cc23)c(nc1CO)-c1ccccc1 |r|
Cc1ncc(cn1)-c1nc(c(NC(=O)N[C@H]2[C@H](O)CC(C)(C)c3cc(F)c(F)cc23)cc1C)-c1ccccc1 |r|
Cc1cc(NC(=O)N[C@@H]2[C@H](O)CC(C)(C)c3cc(F)c(F)cc23)c(nc1-c1ccc(CO)cc1)-c1ccccc1 |r|
Cc1cc(NC(=O)NC2[C@H](O)CC(C)(C)c3cc(F)c(F)cc23)c(nc1-c1ccc(CO)cc1)-c1ccccc1 |r|
Cc1cc(NC(=O)NC2[C@H](O)CC(C)(C)c3cc(F)c(F)cc23)c(nc1-c1cccc(CO)c1)-c1ccccc1 |r|
Cc1cc(NC(=O)NC2[C@H](O)CC(C)(C)c3cc(F)c(F)cc23)c(nc1-c1cccc(c1)C#N)-c1ccccc1 |r|
Cc1cc(NC(=O)NC2[C@H](O)CC(C)(C)c3cc(F)c(F)cc23)c(nc1-c1ccn(C)n1)-c1ccccc1 |r|
Cc1cc(NC(=O)N[C@H]2[C@H](O)CC(C)(C)c3cc(F)c(F)cc23)c(nc1-c1ccn(C)n1)-c1ccccc1 |r|
Cc1cc(NC(=O)N[C@@H]2[C@H](O)CC(C)(C)c3cc(F)c(F)cc23)c(nc1-c1ccn(C)n1)-c1ccccc1 |r|
Cc1cc(cnn1)-c1nc(c(NC(=O)N[C@H]2[C@H](O)CC(C)(C)c3cc(F)c(F)cc23)cc1C)-c1ccccc1 |r|
Cc1ncc(s1)-c1nc(c(NC(=O)N[C@H]2[C@H](O)CC(C)(C)c3cc(F)c(F)cc23)cc1C)-c1ccccc1 |r|
Cc1cc(NC(=O)N[C@H]2[C@H](O)CC(C)(C)c3cc(F)c(F)cc23)c(nc1-c1cnn(C)c1)-c1ccccc1 |r|
Cc1cc(NC(=O)N[C@H]2[C@H](O)CC(C)(C)c3cc(F)c(F)cc23)c(nc1-c1ccc(cc1)C#N)-c1ccccc1 |r|
Cc1cc(NC(=O)N[C@H]2[C@H](O)CC(C)(C)c3cc(F)c(F)cc23)c(nc1-c1cn[nH]c1)-c1ccccc1 |r|
Cc1cc(NC(=O)N[C@H]2[C@H](O)CC(C)(C)c3cc(F)c(F)cc23)c(nc1-c1cnc(nc1)C(C)(C)O)-c1ccccc1 |r|
Cc1cc(NC(=O)N[C@H]2[C@H](O)CC(C)(C)c3cc(F)c(F)cc23)c(nc1-c1ccc(CO)nc1)C1CCOCC1 |r|
Cc1cc(NC(=O)N[C@H]2[C@H](O)CC(C)(C)c3cc(F)c(F)cc23)c(nc1-c1ccnc(CO)c1)C1CCOCC1 |r|
Cc1cnc(C2CCOCC2)c(NC(=O)N[C@H]2[C@H](O)CC(C)(C)c3cc(F)c(F)cc23)c1 |r|
Cc1cc(NC(=O)N[C@H]2[C@H](O)CC(C)(C)c3cc(F)c(F)cc23)c(nc1C(O)=O)C1CCOCC1 |r|
Cc1ncc(cn1)-c1nc(C2CCOCC2)c(NC(=O)N[C@H]2[C@H](O)CC(C)(C)c3cc(F)c(F)cc23)cc1C |r|
Cc1cc(NC(=O)N[C@H]2[C@H](O)CC(C)(C)c3cc(F)c(F)cc23)c(nc1C(=O)NCC(C)(C)O)C1CCOCC1 |r|
Cc1cc(NC(=O)NC2[C@H](O)CC(C)(C)c3cc(F)c(F)cc23)c(nc1C(=O)NCC(C)(C)O)C1CCOCC1 |r|
Cc1cc(NC(=O)N[C@@H]2[C@H](O)CC(C)(C)c3cc(F)c(F)cc23)c(nc1-c1cnc(O)nc1)C1CCOCC1 |r|
Cc1cc(NC(=O)N[C@H]2[C@H](O)CC(C)(C)c3cc(F)c(F)cc23)c(nc1-c1cn[nH]c1)C1CCOCC1 |r|
Cc1cc(NC(=O)N[C@H]2[C@H](O)CC(C)(C)c3cc(F)c(F)cc23)c(nc1-c1cnc(O)nc1)C1CCOCC1 |r|
Cn1ccc(n1)-c1cc(ccc1C(F)(F)F)C(=O)Nc1c(ccc2nc(cn12)C(C)(C)O)-c1ccccc1
Cn1ccc(n1)-c1cc(ccc1C(F)(F)F)C(=O)Nc1c(ccn2cc(nc12)C(C)(C)O)-c1ccccc1
Cn1ccc(n1)-c1cc(ccc1C(F)(F)F)C(=O)Nc1c(ccc2nc(sc12)C(C)(C)O)-c1ccccc1
Cn1ccc(n1)-c1cc(ccc1C(F)(F)F)C(=O)Nc1c(ccc2sc(nc12)C(C)(C)O)-c1ccccc1
C[C@@H](O)c1nc2c(NC(=O)c3ccc(c(c3)-c3ccn(C)n3)C(F)(F)F)c(ccc2s1)-c1ccccc1
C[C@H](O)c1nc2c(NC(=O)c3ccc(c(c3)-c3ccn(C)n3)C(F)(F)F)c(ccc2s1)-c1ccccc1
NC(=O)c1cnc2c(NC(=O)c3cc(-c4ncccn4)c(cc3F)C(F)(F)F)c(ccn12)-c1ccccc1
CC(O)c1cnc2c(NC(=O)c3cc(-c4ncccn4)c(cc3F)C(F)(F)F)c(ccn12)-c1ccccc1
C[C@@H](O)c1cnc2c(NC(=O)c3cc(-c4ncccn4)c(cc3F)C(F)(F)F)c(ccn12)-c1ccccc1
C[C@H](O)c1cnc2c(NC(=O)c3cc(-c4ncccn4)c(cc3F)C(F)(F)F)c(ccn12)-c1ccccc1
CC(C)(O)c1cnc2c(NC(=O)c3cc(-c4ncccn4)c(cc3F)C(F)(F)F)c(ccn12)-c1ccccc1
Cn1ccc(n1)-c1cc(ccc1C(F)(F)F)C(=O)Nc1c(ccn2c(cnc12)C(N)=O)-c1ccccc1
Cn1ccc(n1)-c1cc(ccc1C(F)(F)F)C(=O)Nc1c(ccn2c(CO)cnc12)-c1ccccc1
CC(O)c1cnc2c(NC(=O)c3ccc(c(c3)-c3ccn(C)n3)C(F)(F)F)c(ccn12)-c1ccccc1
Cn1ccc(n1)-c1cc(C(=O)Nc2c(ccn3c(cnc23)C(C)(C)O)-c2ccccc2)c(F)cc1C(F)(F)F
Cn1ccc(n1)-c1cc(C(=O)Nc2c(ccn3c(cnc23)C(C)(C)O)-c2ccccc2)c(Cl)cc1C(F)(F)F
CC(C)(O)c1cnc2c(NC(=O)c3cc(-c4ccccn4)c(cc3Cl)C(F)(F)F)c(ccn12)-c1ccccc1
CC(C)(O)c1cnc2c(NC(=O)c3cc(-c4ccccn4)c(cc3F)C(F)(F)F)c(ccn12)-c1ccccc1
CC(C)(O)c1cnc2c(NC(=O)c3cc(-c4ncccn4)c(cc3Cl)C(F)(F)F)c(ccn12)-c1ccccc1
NC(=O)c1cnc2c(NC(=O)c3cc(-c4ccccn4)c(cc3F)C(F)(F)F)c(ccn12)-c1ccccc1
Cn1ccc(n1)-c1cc(C(=O)Nc2c(ccn3c(cnc23)C(N)=O)-c2ccccc2)c(F)cc1C(F)(F)F
Cn1ccc(n1)-c1cc(C(=O)Nc2c(ccn3c(CO)cnc23)-c2ccccc2)c(F)cc1C(F)(F)F
OCc1cnc2c(NC(=O)c3cc(-c4ccccn4)c(cc3F)C(F)(F)F)c(ccn12)-c1ccccc1
CC(O)c1cnc2c(NC(=O)c3cc(-c4ccn(C)n4)c(cc3F)C(F)(F)F)c(ccn12)-c1ccccc1
CC(O)c1cnc2c(NC(=O)c3cc(-c4cc[nH]n4)c(cc3F)C(F)(F)F)c(ccn12)-c1ccccc1
CC(O)c1cnc2c(NC(=O)c3cc(-c4ccccn4)c(cc3F)C(F)(F)F)c(ccn12)-c1ccccc1
CC(C)(O)c1cnc2c(NC(=O)c3cc(-c4cc[nH]n4)c(cc3F)C(F)(F)F)c(ccn12)-c1ccccc1
Cn1ccc(n1)-c1cc(ccc1C(F)(F)F)C(=O)Nc1c(ccn2c(cnc12)C(C)(C)O)-c1ccccc1
Cn1ccc(n1)-c1cc(ccc1C(F)(F)F)C(=O)Nc1c(ncn2cnnc12)-c1ccccc1
Cn1ccc(n1)-c1cc(ccc1C(F)(F)F)C(=O)Nc1c(ccn2ccnc12)-c1ccccc1
Cc1cc(c(cc1C(=O)Nc1c(ccn2ccnc12)-c1ccccc1)-c1ncccn1)C(F)(F)F
Cn1ccc(n1)-c1cc(C(=O)Nc2c(ccc3c(cnn23)C(C)(C)O)-c2ccccc2)c(F)cc1C(F)(F)F
Cn1ccc(n1)-c1cc(ccc1C(F)(F)F)C(=O)Nc1c(ccc2c(cnn12)C(C)(C)O)-c1ccccc1
CC(C)(O)c1cnn2c(NC(=O)c3cc(-c4ncccn4)c(cc3F)C(F)(F)F)c(ccc12)-c1ccccc1
Cn1ccc(n1)-c1cc(C(=O)Nc2c(ccc3c(CO)cnn23)-c2ccccc2)c(F)cc1C(F)(F)F
Cn1ccc(n1)-c1cc(ccc1C(F)(F)F)C(=O)Nc1c(ccc2c(CO)cnn12)-c1ccccc1
OCc1cnn2c(NC(=O)c3cc(-c4ncccn4)c(cc3F)C(F)(F)F)c(ccc12)-c1ccccc1
Cn1ccc(n1)-c1cc(ccc1C(F)(F)F)C(=O)Nc1c(ccc2cc([nH]c12)C(C)(C)O)-c1ccccc1
CC(=O)c1c[nH]c2c(NC(=O)c3ccc(c(c3)-c3ccn(C)n3)C(F)(F)F)c(ccc12)-c1ccccc1
CC(C)(O)c1cc2cc(c(NC(=O)c3cc(-c4ncccn4)c(cc3F)C(F)(F)F)cc2[nH]1)-c1ccccc1
CC(C)(O)c1n[nH]c2c(NC(=O)c3cc(-c4ncccn4)c(cc3F)C(F)(F)F)c(ccc12)-c1ccccc1
C[C@@H](O)c1n[nH]c2c(NC(=O)c3cc(-c4ncccn4)c(cc3F)C(F)(F)F)c(ccc12)-c1ccccc1
C[C@H](O)c1n[nH]c2c(NC(=O)c3cc(-c4ncccn4)c(cc3F)C(F)(F)F)c(ccc12)-c1ccccc1
C[C@@H](O)c1n[nH]c2c(NC(=O)c3ccc(cc3-c3ccn(C)n3)C(F)(F)F)c(ccc12)-c1ccccc1
C[C@H](O)c1n[nH]c2c(NC(=O)c3ccc(cc3-c3ccn(C)n3)C(F)(F)F)c(ccc12)-c1ccccc1
NC(=O)Cc1cnc2c(NC(=O)c3cc(-c4ncccn4)c(cc3F)C(F)(F)F)c(ccn12)-c1ccccc1
OCc1cnc2c(NC(=O)c3cc(-c4ncccn4)c(cc3F)C(F)(F)F)c(ccn12)-c1ccc(F)cc1
C[C@H](O)c1cnc2c(NC(=O)c3cc(-c4ncccn4)c(cc3F)C(F)(F)F)c(ccn12)-c1ccc(F)cc1 |r|
C[C@@H](O)c1cnc2c(NC(=O)c3cc(-c4ncccn4)c(cc3F)C(F)(F)F)c(ccn12)-c1ccc(F)cc1 |r|
CC(C)(O)c1cnc2c(NC(=O)c3cc(-c4ncccn4)c(cc3F)C(F)(F)F)c(ccn12)-c1ccc(F)cc1
Cc1ccccc1-c1ccn2c(cnc2c1NC(=O)c1cc(-c2ncccn2)c(cc1F)C(F)(F)F)C(C)(C)O
Cc1ccccc1-c1ccn2c(cnc2c1NC(=O)c1cc(-c2ccn(C)n2)c(cc1F)C(F)(F)F)C(N)=O
CC(C)(O)c1cnc2c(NC(=O)c3cc(-c4ncccn4)c(cc3F)C(F)(F)F)c(ccn12)-c1cccc(CO)c1
OCc1cccc(c1)-c1ccn2ccnc2c1NC(=O)c1cc(-c2ncccn2)c(cc1F)C(F)(F)F
CC(C)(O)c1ncn2c(NC(=O)c3cc(-c4ccccn4)c(cc3F)C(F)(F)F)c(ccc12)-c1ccccc1
Cn1ccc(n1)-c1cc(C(=O)Nc2c(ccc3c(ncn23)C(C)(C)O)-c2ccccc2)c(F)cc1C(F)(F)F
Cn1ccc(n1)-c1cc(C(=O)Nc2cn3c(CO)ncc3nc2-c2ccccc2)c(F)cc1C(F)(F)F
Cc1ncc2nc(c(NC(=O)c3ccc(c(c3)-c3ccn(C)n3)C(F)(F)F)cn12)-c1ccccc1
Cn1ccc(n1)-c1cc(C(=O)Nc2cn3c(ncc3nc2-c2ccccc2)C(O)=O)c(F)cc1C(F)(F)F
Cn1ccc(n1)-c1cc(C(=O)Nc2cn3cncc3nc2-c2ccccc2)c(F)cc1C(F)(F)F
Cn1ccc(n1)-c1cc(C(=O)Nc2cn3c(CO)ncc3cc2-c2ccccc2)c(F)cc1C(F)(F)F
CCOC(=O)c1cnc2c(NC(=O)c3cc(-c4ccn(C)n4)c(s3)C(F)(F)F)c(ccn12)-c1ccccc1
Cn1ccc(n1)-c1cc(sc1C(F)(F)F)C(=O)Nc1c(ccn2c(cnc12)C(N)=O)-c1ccccc1
Cn1ccc(n1)-c1cc(sc1C(F)(F)F)C(=O)Nc1c(ccn2c(CO)cnc12)-c1ccccc1
OCc1cnc2c(NC(=O)c3cc(-c4ncccn4)c(cc3F)C(F)(F)F)c(ncn12)-c1ccccc1
Cn1ccc(n1)-c1cc(ccc1C(F)(F)F)C(=O)Nc1c(ncn2c(CO)cnc12)-c1ccccc1
C[C@@H](O)c1cnc2c(NC(=O)c3cc(-c4ncccn4)c(cc3F)C(F)(F)F)c(ncn12)-c1ccccc1 |r|
C[C@H](O)c1cnc2c(NC(=O)c3cc(-c4ncccn4)c(cc3F)C(F)(F)F)c(ncn12)-c1ccccc1 |r|
CC(C)(O)c1cnc2c(NC(=O)c3cc(-c4ncccn4)c(cc3F)C(F)(F)F)c(ncn12)-c1ccccc1
C[C@@H](O)c1cnc2c(NC(=O)c3cc(-c4ncccn4)c(cc3F)C(F)(F)F)c(ccn12)-c1ccccc1 |r|
C[C@H](O)c1cnc2c(NC(=O)c3cc(-c4ncccn4)c(cc3F)C(F)(F)F)c(ccn12)-c1ccccc1 |r|
CC(C)(C)OC(=O)C1C2CCC1CN(C2)C(=O)Nc1cnc2ccc(nn12)N1CCC[C@@H]1c1cc(F)ccc1F |r|
Cc1c(NC(=O)N[C@@H]2OC(C)(C)O[C@H]2c2ccccc2)n(nc1-c1cnn(C)c1)-c1ccccc1 |r|
CCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnn(C)c2)[C@@H](O1)c1ccccc1 |r|
COCC[C@@H]1O[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnn(C)c2)[C@@H](O1)c1ccccc1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnn(C)c2)[C@@H](N1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2ccc3n(C)ncc3c2)[C@@H](O1)c1ccc(F)c(F)c1 |r|
COCC[C@@H]1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnn(C)c2)[C@@H](O1)c1ccc(F)c(F)c1 |r|
COCC[C@@H]1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc(C)nc2)[C@@H](O1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)C2=CCN(CC2)C(C)=O)[C@@H](O1)c1ccc(F)c(F)c1 |r,t:25|
CCN1CCC(CC1)NC(=O)c1ccc(cc1)-c1nn(c(NC(=O)N[C@@H]2CN(CCOC)O[C@H]2c2ccc(F)c(F)c2)c1C)-c1ccccc1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc3n(C)ncc3c2)[C@@H](O1)c1ccnc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc(C)nc2)[C@@H](O1)c1ccnc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc(OC)nc2)[C@@H](O1)c1cnc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2ccc(N=S(C)(C)=O)nc2)[C@@H](O1)c1ccc(F)c(F)c1 |r|
CNC(=O)c1cc(cnc1OC)-c1nn(c(NC(=O)N[C@@H]2CN(CCOC)O[C@H]2c2cnc(F)c(F)c2)c1C)-c1ccccc1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc3n(C)n(C)c(=O)c3c2)[C@@H](O1)c1cnc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(OCC(C)(C)O)nn2-c2ccccc2)[C@@H](O1)c1cnc(F)c(F)c1 |r|
COCC[C@@H]1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc(C)nc2)[C@@H](O1)c1ccnc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cc(C(=O)NC3CCOCC3)c(=O)n(C)c2)[C@@H](O1)c1ccnc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc(OC)nc2)[C@@H](O1)c1ccnc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc3n(C)c(=O)oc3c2)[C@@H](O1)c1ccnc(F)c1 |r|
CNc1ncc(cn1)-c1nn(c(NC(=O)N[C@@H]2CN(CCOC)O[C@H]2c2cnc(F)c(F)c2)c1C)-c1ccccc1 |r|
COCCN1C[C@H]([C@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnn(C)c2)O1)c1ccnc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2ccc(nc2)-c2nn[nH]n2)[C@@H](O1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2C2CCC2)-c2cnn(C)c2)[C@@H](O1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2ccc3nc(C)nn3c2)[C@@H](O1)c1ccnc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc(C(N)=O)c(C)c2)[C@@H](O1)c1ccnc(F)c1 |r|
CNC(=O)c1ncc(cc1C)-c1nn(c(NC(=O)N[C@@H]2CN(CCOC)O[C@H]2c2ccnc(F)c2)c1C)-c1ccccc1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2ccnc(c2)C(O)=O)[C@@H](O1)c1ccc(F)c(F)c1 |r|
CNC(=O)c1cc(cn(C)c1=O)-c1nn(c(NC(=O)N[C@@H]2CN(C)O[C@H]2c2ccc(F)c(F)c2)c1C)-c1ccccc1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnn(C)c2)[C@@H](O1)c1cc(F)nc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2ccnc(c2)C(=O)NOC)[C@@H](O1)c1ccnc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2ccnc(c2)C(=O)NOC)[C@@H](O1)c1cnc(F)c(F)c1 |r|
COCC[C@@H]1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc3n(C)ncc3c2)[C@@H](O1)c1ccnc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccc(F)cc2)-c2cnc(OC)c(c2)C(=O)NC2CCOCC2)[C@@H](O1)c1ccnc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc3ncn(CC(F)(F)F)c3c2)[C@@H](O1)c1ccnc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)N2Cc3cnn(C)c3C2)[C@@H](O1)c1ccnc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnn(C)c2)[C@@H](O1)c1cnc(F)c(F)c1 |r|
CNC(=O)c1ncc(cc1C)-c1nn(c(NC(=O)N[C@@H]2CN(CCOC)O[C@H]2c2cnc(F)c(F)c2)c1C)-c1ccccc1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc3n(C)c(=O)[nH]c3c2)[C@@H](O1)c1cnc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc(N=S(C)(C)=O)nc2)[C@@H](O1)c1ccc(F)c(F)c1 |r|
COCC[C@@H]1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc(OC)nc2)[C@@H](O1)c1ccnc(F)c1 |r|
COCC[C@@H]1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc3n(C)nnc3c2)[C@@H](O1)c1ccnc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2ccc(nc2)N2CCC(O)CC2)[C@@H](O1)c1ccnc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc3NC(=O)COc3c2)[C@@H](O1)c1ccnc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc(C)nc2)[C@@H](O1)c1cc(F)nc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc3N(C)C(=O)Cc3c2)[C@@H](O1)c1ccnc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc3n(C)nc(N=S(C)(C)=O)c3c2)[C@@H](O1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc3[nH]ncc3c2)[C@@H](O1)c1ccnc(F)c1 |r|
CNC(=O)c1cc(nn(C)c1=O)-c1nn(c(NC(=O)N[C@@H]2CN(CCOC)O[C@H]2c2ccnc(F)c2)c1C)-c1ccccc1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc3N(C)C(=O)Cc3c2)[C@@H](O1)c1cnc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2ccc3nc(cn3c2)C(N)=O)[C@@H](O1)c1cnc(F)c(F)c1 |r|
CNC(=O)c1ncc(cc1F)-c1nn(c(NC(=O)N[C@@H]2CN(CCOC)O[C@H]2c2cnc(F)c(F)c2)c1C)-c1ccccc1 |r|
CNC(=O)c1ncc(cc1NC)-c1nn(c(NC(=O)N[C@@H]2CN(CCOC)O[C@H]2c2ccc(F)c(F)c2)c1C)-c1ccccc1 |r|
CNC(=O)c1cc(cnc1OC)-c1nn(c(NC(=O)N[C@@H]2C[C@@H](CCOC)O[C@H]2c2ccnc(F)c2)c1C)-c1ccccc1 |r|
COCC[C@@H]1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc3N(C)C(=O)Cc3c2)[C@@H](O1)c1ccnc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2ccc(CN=S(C)(C)=O)cc2)[C@@H](O1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)N2CCN(C)C(=O)C2)[C@@H](O1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc3NC(=O)CNc3c2)[C@@H](O1)c1ccnc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2ccc(nc2)N2CCN(C)CC2)[C@@H](O1)c1ccnc(F)c1 |r|
CCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc(OC)c(c2)C(=O)NC)[C@@H](O1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc3n(ncc3c2)C2CCN(C)CC2)[C@@H](O1)c1ccnc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc(OCC3CC3)nc2)[C@@H](O1)c1ccnc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc(OCC(F)F)nc2)[C@@H](O1)c1ccnc(F)c1 |r|
CNC(=O)c1ccc(cn1)-c1nn(c(NC(=O)N[C@@H]2CN(CCOC)O[C@H]2c2ccc(F)c(F)c2)c1C)-c1ccccc1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc(COC)nc2)[C@@H](O1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2ccc(OC)nc2)[C@@H](O1)c1ccnc(F)c1 |r|
COc1ncc(cn1)-c1nn(c(NC(=O)N[C@@H]2CN(CC(F)F)O[C@H]2c2ccc(F)c(F)c2)c1C)-c1ccccc1 |r|
CCN1C[C@@H](NC(=O)Nc2c(C)c(OCC3CCN(C)CC3)nn2-c2ccccc2)[C@@H](O1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(OCCCN(C)C)nn2-c2ccccc2)[C@@H](O1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc(nc2)N2CC(C2)OC)[C@@H](O1)c1ccnc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc(OCF)nc2)[C@@H](O1)c1ccnc(F)c1 |r|
CCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2ccc(OC)nc2)[C@@H](O1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2ccc(CN(C)C)nc2)[C@@H](O1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc(OC)c(CN(C)C)c2)[C@@H](O1)c1ccc(F)c(F)c1 |r|
CCN1C[C@@H](NC(=O)Nc2c(C)c(OCC(N)=O)nn2-c2ccccc2)[C@@H](O1)c1ccc(F)c(F)c1 |r|
CCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)C2=CCN(CC2)C(=O)CO)[C@@H](O1)c1ccc(F)c(F)c1 |r,t:23|
COCCN1C[C@@H](NC(=O)Nc2c(c(C)nn2-c2ccccc2)C(F)(F)F)[C@@H](O1)c1ccnc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc(C)nc2)[C@@H](O1)c1cnc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)C2=CCN(CC2)C(=O)OC(C)(C)C)[C@@H](O1)c1cnc(F)c(F)c1 |r,t:25|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)C2=CCNCC2)[C@@H](O1)c1cnc(F)c(F)c1 |r,t:25|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)C2=CCN(CC2)C(C)=O)[C@@H](O1)c1cnc(F)c(F)c1 |r,t:25|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cccc(c2)C(=O)OC(C)(C)C)[C@@H](O1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cccc(c2)C(O)=O)[C@@H](O1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)C2=CCN(CC2)C(=O)CO)[C@@H](O1)c1ccc(F)c(F)c1 |r,t:25|
COCC[C@@H]1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)C2=CCN(CC2)C(=O)OC(C)(C)C)[C@@H](O1)c1ccc(F)c(F)c1 |r,t:25|
COCC[C@@H]1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)C2=CCNCC2)[C@@H](O1)c1ccc(F)c(F)c1 |r,t:25|
COCC[C@@H]1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)C2=CCN(CC2)C(=O)CO)[C@@H](O1)c1ccc(F)c(F)c1 |r,t:25|
COCC[C@H]1C[C@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)C2=CCN(CC2)C(=O)CO)[C@H](O1)c1ccc(F)c(F)c1 |r,t:25|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2ccc(cc2)C#N)[C@@H](O1)c1cnc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(OCC(C)(C)O)nn2-c2ccccc2)[C@@H](O1)c1ccc(F)c(F)c1 |r|
CCN1CCC(CC1)NC(=O)c1cc(ccn1)-c1nn(c(NC(=O)N[C@@H]2CN(CCOC)O[C@H]2c2ccc(F)c(F)c2)c1C)-c1ccccc1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc3cnn(C)c3c2)[C@@H](O1)c1ccnc(F)c1 |r|
CCN1CCC(CC1)NC(=O)c1cc(ccn1)-c1nn(c(NC(=O)N[C@@H]2C[C@@H](CCOC)O[C@H]2c2ccc(F)c(F)c2)c1C)-c1ccccc1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc3n(C)ncc3c2)[C@@H](O1)c1cnc(F)c(F)c1 |r|
CCOc1ncc(cn1)-c1nn(c(NC(=O)N[C@@H]2CN(CCOC)O[C@H]2c2cnc(F)c(F)c2)c1C)-c1ccccc1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc3n(C)cnc3c2)[C@@H](O1)c1cnc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc(nc2)C2CC2)[C@@H](O1)c1cnc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cc(C)c(=O)n(C)c2)[C@@H](O1)c1cnc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc3n(C)cnc3c2)[C@@H](O1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cc(C(=O)NC3CCOCC3)c(=O)n(C)c2)[C@@H](O1)c1cnc(F)c(F)c1 |r|
CNC(=O)c1cc(cn(C)c1=O)-c1nn(c(NC(=O)N[C@@H]2CN(CCOC)O[C@H]2c2cnc(F)c(F)c2)c1C)-c1ccccc1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2ccnc(c2)C(=O)OCc2ccccc2)[C@@H](O1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2ccnc(c2)N=S(C)(C)=O)[C@@H](O1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc3n(C)c(CO)nc3c2)[C@@H](O1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cc(COC(C)=O)c(=O)n(C)c2)[C@@H](O1)c1cnc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cc(CO)c(=O)n(C)c2)[C@@H](O1)c1cnc(F)c(F)c1 |r|
COCCN1C[C@H](NC(=O)Nc2c(C)c(OCC(C)(C)O)nn2-c2ccccc2)[C@H](O1)c1cnc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc3n(C)nc(CO)c3c2)[C@@H](O1)c1cnc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cncc(c2)N=S(C)(C)=O)[C@@H](O1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccc(F)c(F)c2)-c2cnn(C)c2)[C@@H](O1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccc(F)cc2)-c2cnn(C)c2)[C@@H](O1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2C2CC2)-c2cnn(C)c2)[C@@H](O1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cccc(c2)N=S(C)(C)=O)[C@@H](O1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc3n(C)nnc3c2)[C@@H](O1)c1ccnc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnn(C)c2)[C@@H](O1)c1ccnc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc(N=S(C)(C)=O)c(C)c2)[C@@H](O1)c1ccc(F)c(F)c1 |r|
CNc1ncc(cn1)-c1nn(c(NC(=O)N[C@@H]2CN(CCOC)O[C@H]2c2ccnc(F)c2)c1C)-c1ccccc1 |r|
COCCN1C[C@@H](NC(=O)Nc2cc(nn2C)-c2cnc(OC)c(c2)C(=O)NC2CCOCC2)[C@@H](O1)c1ccnc(F)c1 |r|
CNC(=O)c1cc(cnc1OC)-c1cc(NC(=O)N[C@@H]2CN(CCOC)O[C@H]2c2ccnc(F)c2)n(C)n1 |r|
COCCC1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc3n(C)ncc3c2)[C@@H](O1)c1ccccc1 |r|
COCC[C@@H]1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc3n(C)ncc3c2)[C@@H](O1)c1ccc(F)c(F)c1 |r|
CNC(=O)c1cc(cnc1OC)-c1nn(c(NC(=O)N[C@@H]2CN(CCOC)O[C@H]2c2ccnc(F)c2)c1C)-c1ccccc1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc(OC)c(c2)C(N)=O)[C@@H](O1)c1cnc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc(OC)c(c2)C(N)=O)[C@@H](O1)c1cnc(OC)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc(OC)c(c2)C(=O)NC2CCS(=O)(=O)CC2)[C@@H](O1)c1cnc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc(OC)c(c2)C(=O)NC2CCS(=O)(=O)CC2)[C@@H](O1)c1cnc(OC)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cc(C(N)=O)c(=O)n(C)c2)[C@@H](O1)c1ccnc(F)c1 |r|
CNC(=O)c1cc(cn(C)c1=O)-c1nn(c(NC(=O)N[C@@H]2CN(CCOC)O[C@H]2c2ccnc(F)c2)c1C)-c1ccccc1 |r|
CCNC(=O)c1cc(cn(C)c1=O)-c1nn(c(NC(=O)N[C@@H]2CN(CCOC)O[C@H]2c2ccnc(F)c2)c1C)-c1ccccc1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc(OC)c(c2)C(N)=O)[C@@H](O1)c1ccnc(F)c1 |r|
CCNC(=O)c1cc(cnc1OC)-c1nn(c(NC(=O)N[C@@H]2CN(CCOC)O[C@H]2c2ccnc(F)c2)c1C)-c1ccccc1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc(OC)c(c2)C(=O)NC2CCOCC2)[C@@H](O1)c1ccnc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc(OC)c(c2)C(=O)NC2CCS(=O)(=O)CC2)[C@@H](O1)c1ccnc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc(OC)c(c2)C(=O)N[C@@H]2CCOC2)[C@@H](O1)c1ccnc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc3n(C)nc(C)c3c2)[C@@H](O1)c1ccnc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc(nc2)C2CC2)[C@@H](O1)c1ccnc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnn(C)c2)[C@@H](O1)c1ccc(F)cc1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc(C)nc2)[C@@H](O1)c1ccc(F)cc1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc3n(C)nnc3c2)[C@@H](O1)c1ccc(F)cc1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc(nc2)N(C2CC2)C(=O)OC(C)(C)C)[C@@H](O1)c1ccnc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc3n(C)c(=O)oc3c2)[C@@H](O1)c1cnc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cc(COC(C)=O)c(=O)n(C)c2)[C@@H](O1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cc(CO)c(=O)n(C)c2)[C@@H](O1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc3n(C)nnc3c2)[C@@H](O1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc3n(C)nnc3c2)[C@@H](O1)c1cnc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2ccc(nc2)C#N)[C@@H](O1)c1ccc(F)c(F)c1 |r|
CCOc1ncc(cn1)-c1nn(c(NC(=O)N[C@H]2CN(CCOC)O[C@@H]2c2ccnc(F)c2)c1C)-c1ccccc1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc(NC3CC3)nc2)[C@@H](O1)c1ccnc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc(nc2)N(C)C)[C@@H](O1)c1ccnc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc(nc2)N(C)C)[C@@H](O1)c1cnc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc3nccnc3c2)[C@@H](O1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnn(C)c2)[C@@H](O1)c1cnc(Cl)s1 |r|
CNC(=O)c1cc(cn(C)c1=O)-c1nn(c(NC(=O)N[C@@H]2CN(CCOC)O[C@H]2c2ccc(F)cc2)c1C)-c1ccccc1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnn(C)c2)[C@@H](O1)c1cccc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc(C)nc2)[C@@H](O1)c1cccc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc3n(C)cnc3c2)[C@@H](O1)c1cccc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc3n(C)nnc3c2)[C@@H](O1)c1cccc(F)c1 |r|
CNC(=O)c1cc(cn(C)c1=O)-c1nn(c(NC(=O)N[C@@H]2CN(CCOC)O[C@H]2c2cccc(F)c2)c1C)-c1ccccc1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc(nc2)N2CC(O)C2)[C@@H](O1)c1ccnc(F)c1 |r|
CNC(=O)c1cc(cn(C)c1=O)-c1nn(c(NC(=O)N[C@@H]2CN(CCOC)O[C@H]2c2ccc(F)c(F)c2)c1C)-c1ccccc1 |r|
CCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cc(C(=O)NC)c(=O)n(C)c2)[C@@H](O1)c1ccc(F)c(F)c1 |r|
CNC(=O)c1cc(cn(C)c1=O)-c1nn(c(NC(=O)N[C@@H]2CN(Cc3ccco3)O[C@H]2c2ccc(F)c(F)c2)c1C)-c1ccccc1 |r|
CNC(=O)c1cc(cn(C)c1=O)-c1nn(c(NC(=O)N[C@@H]2CN(Cc3ccc(o3)C#N)O[C@H]2c2ccc(F)c(F)c2)c1C)-c1ccccc1 |r|
CNC(=O)c1cc(cn(C)c1=O)-c1nn(c(NC(=O)N[C@@H]2CN(Cc3csnn3)O[C@H]2c2ccc(F)c(F)c2)c1C)-c1ccccc1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc3cccnc3c2)[C@@H](O1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)C2=CCN(CC2)c2ncc(Cl)cn2)[C@@H](O1)c1ccc(F)c(F)c1 |r,t:25|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc(C)nc2)[C@@H](O1)c1cnc(Cl)s1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2ccn3c(C)nnc3c2)[C@@H](O1)c1ccnc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2ccn3nc(C)nc3c2)[C@@H](O1)c1ccnc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc(OC)nc2)[C@@H](O1)c1cnc(Cl)s1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2ccc3nnc(C)n3c2)[C@@H](O1)c1ccnc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc(C)nc2)[C@@H](O1)c1ccccc1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc3n(C)cnc3c2)[C@@H](O1)c1ccccc1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc3n(C)nnc3c2)[C@@H](O1)c1ccccc1 |r|
CNC(=O)c1cc(cn(C)c1=O)-c1nn(c(NC(=O)N[C@@H]2CN(CCOC)O[C@H]2c2ccccc2)c1C)-c1ccccc1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc3n(C)cnc3c2)[C@@H](O1)c1ccnc(F)c1 |r|
CCNC(=O)c1ncc(cc1C)-c1nn(c(NC(=O)N[C@@H]2CN(CCOC)O[C@H]2c2ccnc(F)c2)c1C)-c1ccccc1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc(C(=O)NCC(F)(F)F)c(C)c2)[C@@H](O1)c1ccnc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc(C(=O)NC3CC3)c(C)c2)[C@@H](O1)c1ccnc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc(C(=O)NCC3CC3)c(C)c2)[C@@H](O1)c1ccnc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc(C(=O)NC3CCOCC3)c(C)c2)[C@@H](O1)c1ccnc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc(C(=O)N[C@@H]3CCOC3)c(C)c2)[C@@H](O1)c1ccnc(F)c1 |r|
COCCNC(=O)c1ncc(cc1C)-c1nn(c(NC(=O)N[C@@H]2CN(CCOC)O[C@H]2c2ccnc(F)c2)c1C)-c1ccccc1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccc(F)cc2)-c2cnc3n(C)ncc3c2)[C@@H](O1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccc(F)c(F)c2)-c2cnc3n(C)ncc3c2)[C@@H](O1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc(C)c(c2)N=S(C)(C)=O)[C@@H](O1)c1ccc(F)c(F)c1 |r|
CNS(=O)(=O)c1cc(cn(C)c1=O)-c1nn(c(NC(=O)N[C@@H]2CN(CCOC)O[C@H]2c2ccc(F)c(F)c2)c1C)-c1ccccc1 |r|
CNS(=O)(=O)c1cc(cn(C)c1=O)-c1nn(c(NC(=O)N[C@@H]2CN(CCOC)O[C@H]2c2ccnc(F)c2)c1C)-c1ccccc1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc(OC)c(c2)C(O)=O)[C@@H](O1)c1cnc(F)c(F)c1 |r|
CNC(=O)c1cc(cnc1OC)-c1nn(c(NC(=O)N[C@@H]2CN(CCOC)O[C@H]2c2ccc(F)c(F)c2)c1C)-c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccc(F)c(F)c2)-c2cnc(OC)c(c2)C(=O)NC2CCOCC2)[C@@H](O1)c1ccc(F)c(F)c1 |r|
CNC(=O)c1cc(cnc1OC)-c1nn(c(NC(=O)N[C@@H]2CN(CCOC)O[C@H]2c2ccc(F)c(F)c2)c1C)-c1ccc(F)cc1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccc(F)cc2)-c2cnc(OC)c(c2)C(=O)NC2CCOCC2)[C@@H](O1)c1ccc(F)c(F)c1 |r|
COCC[C@@H]1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2ccc(N=S(C)(C)=O)nc2)[C@@H](O1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc(OC)nc2)[C@@H](O1)c1cc(F)nc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc3cccnc3c2)[C@@H](O1)c1ccnc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2ccnc(c2)C(=O)OC)[C@@H](O1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2ccnc(c2)C(=O)OC)[C@@H](O1)c1ccnc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2ccnc(c2)C(=O)NO)[C@@H](O1)c1ccc(F)c(F)c1 |r|
CCOc1ncc(cn1)-c1nn(c(NC(=O)N[C@@H]2CN(CCOC)O[C@H]2c2ccnc(F)c2)c1C)-c1ccccc1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2ccnc(c2)C(=O)OC)[C@@H](O1)c1cnc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2ccnc(c2)C(=O)NOC)[C@@H](O1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2ccc(nc2)C(=O)OC)[C@@H](O1)c1ccc(F)c(F)c1 |r|
CCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc3n(C)ncc3c2)[C@@H](O1)c1ccc(F)c(F)c1 |r|
Cc1c(NC(=O)N[C@@H]2CN(CC3CC3)O[C@H]2c2ccc(F)c(F)c2)n(nc1-c1cnc2n(C)ncc2c1)-c1ccccc1 |r|
Cc1c(NC(=O)N[C@@H]2CN(CC3COC3)O[C@H]2c2ccc(F)c(F)c2)n(nc1-c1cnc2n(C)ncc2c1)-c1ccccc1 |r|
Cc1c(NC(=O)N[C@@H]2CN(Cc3ccn[nH]3)O[C@H]2c2ccc(F)c(F)c2)n(nc1-c1cnc2n(C)ncc2c1)-c1ccccc1 |r|
Cc1c(NC(=O)N[C@@H]2CN(Cc3cn[nH]c3)O[C@H]2c2ccc(F)c(F)c2)n(nc1-c1cnc2n(C)ncc2c1)-c1ccccc1 |r|
Cc1c(NC(=O)N[C@@H]2CN(Cc3cnn(C)c3)O[C@H]2c2ccc(F)c(F)c2)n(nc1-c1cnc2n(C)ncc2c1)-c1ccccc1 |r|
CN(C)CC(C)(C)CN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc3n(C)ncc3c2)[C@@H](O1)c1ccc(F)c(F)c1 |r|
CN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc3n(C)ncc3c2)[C@@H](O1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc3n(C)c(=O)[nH]c3c2)[C@@H](O1)c1ccnc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc(nc2)N2CC(O)C2)[C@@H](O1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc(nc2)N2CC(O)C2)[C@@H](O1)c1cnc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2ccnc(c2)C(O)=O)[C@@H](O1)c1ccnc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2ccnc(c2)C(O)=O)[C@@H](O1)c1cnc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2ccc(nc2)C(O)=O)[C@@H](O1)c1ccc(F)c(F)c1 |r|
COCC[C@@H]1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc3n(C)n(C)c(=O)c3c2)[C@@H](O1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc3n(C)n(C)c(=O)c3c2)[C@@H](O1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc3n(C)c(=O)[nH]c3c2)[C@@H](O1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc3n(C)c(nc3c2)C(N)=O)[C@@H](O1)c1ccnc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc3n(C)c(nc3c2)C#N)[C@@H](O1)c1ccnc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc3n(C)c(nc3c2)C(N)=O)[C@@H](O1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc3n(C)c(nc3c2)C#N)[C@@H](O1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccc(F)cc2)-c2cnc3n(C)ncc3c2)[C@@H](O1)c1ccnc(F)c1 |r|
CNC(=O)c1nc2cc(cnc2n1C)-c1nn(c(NC(=O)N[C@@H]2CN(CCOC)O[C@H]2c2ccnc(F)c2)c1C)-c1ccccc1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc3n(C)c(nc3c2)C(=O)NCCO)[C@@H](O1)c1ccnc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc3n(C)c(nc3c2)C(F)(F)F)[C@@H](O1)c1ccnc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2ccc(cc2)N=S(C)(C)=O)[C@@H](O1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc3n(CC(F)(F)F)ncc3c2)[C@@H](O1)c1ccnc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc3n(C)c(=O)ccc3c2)[C@@H](O1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2ccnc(c2)C(=O)NO)[C@@H](O1)c1ccnc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2ccnc(c2)C(=O)NO)[C@@H](O1)c1cnc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2ccc(nc2)C(=O)NOC)[C@@H](O1)c1ccc(F)c(F)c1 |r|
COCC[C@@H]1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnn(C)c2)[C@@H](O1)c1ccnc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccc(F)cc2)-c2cnc(OC)c(c2)C(N)=O)[C@@H](O1)c1ccnc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc3n(CC(F)(F)F)cnc3c2)[C@@H](O1)c1ccnc(F)c1 |r|
COCC[C@@H]1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc(nc2)N2CC(O)C2)[C@@H](O1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc3nn(CC(F)(F)F)cc3c2)[C@@H](O1)c1ccnc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc3n(C)c(=O)ccc3c2)[C@@H](O1)c1ccnc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc(OC)nc2)[C@@H](O1)c1ccc(F)cc1 |r|
COCC[C@@H]1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc(Cl)nc2)[C@@H](O1)c1ccnc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc(Cl)nc2)[C@@H](O1)c1ccnc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc(SC)nc2)[C@@H](O1)c1ccnc(F)c1 |r|
COCC[C@@H]1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cc(C(=O)OC)c(=O)n(C)c2)[C@@H](O1)c1ccnc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc(C(N)=O)c(C)c2)[C@@H](O1)c1cnc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc(C(=O)NC3CC3)c(C)c2)[C@@H](O1)c1cnc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc(C(N)=O)c(F)c2)[C@@H](O1)c1ccnc(F)c1 |r|
CNC(=O)c1ncc(cc1F)-c1nn(c(NC(=O)N[C@@H]2CN(CCOC)O[C@H]2c2ccnc(F)c2)c1C)-c1ccccc1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc(C(=O)NC3CC3)c(F)c2)[C@@H](O1)c1ccnc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc3C(=O)OCc3c2)[C@@H](O1)c1ccnc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc(OC)c(c2)C(=O)NOC)[C@@H](O1)c1ccnc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc(OC)c(c2)C(=O)NOCCF)[C@@H](O1)c1ccnc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2ccc3N(C)S(=O)(=O)Cc3c2)[C@@H](O1)c1ccnc(F)c1 |r|
COCCN1C[C@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc(OC)nc2)[C@H](O1)c1cnc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc3n(C)nc(c3c2)C(F)(F)F)[C@@H](O1)c1ccnc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc(nc2)N2CC(O)C2)[C@@H](O1)c1ccc(F)cc1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc(nc2)N2CCC2)[C@@H](O1)c1ccnc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2ccc3nnc(C)n3c2)[C@@H](O1)c1ccc(F)cc1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc3n(C)oc(=O)c3c2)[C@@H](O1)c1ccnc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc(nc2)S(C)(=O)=O)[C@@H](O1)c1ccnc(F)c1 |r|
CNC(=O)c1cc(cn(C)c1=O)-c1nn(c(NC(=O)N[C@@H]2C[C@@H](CCOC)O[C@H]2c2ccnc(F)c2)c1C)-c1ccccc1 |r|
COCC[C@@H]1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cc(C(=O)NC3CCOCC3)c(=O)n(C)c2)[C@@H](O1)c1ccnc(F)c1 |r|
COCC[C@@H]1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc3n(C)nc(C)c3c2)[C@@H](O1)c1ccnc(F)c1 |r|
COCC[C@@H]1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc3n(C)cnc3c2)[C@@H](O1)c1ccnc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cc(-c3cn(Cc4ccc(OC)cc4)nn3)c(=O)n(C)c2)[C@@H](O1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc3N(CCOc3c2)C(=O)OC(C)(C)C)[C@@H](O1)c1ccnc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc3NCCOc3c2)[C@@H](O1)c1ccnc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2ccc3nc(cn3c2)C(N)=O)[C@@H](O1)c1ccnc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2ccc(nc2)N2CCCC2)[C@@H](O1)c1ccnc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2ccn3c(C)nnc3c2)[C@@H](O1)c1ccc(F)cc1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc(nc2)N2CC(C2)OC(=O)c2ccccc2)[C@@H](O1)c1cc(F)nc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc(C)s2)[C@@H](O1)c1ccnc(F)c1 |r|
COCC[C@@H]1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cc(C)c(=O)n(C)c2)[C@@H](O1)c1ccnc(F)c1 |r|
COCC[C@@H]1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc(nc2)N(C)C(=O)OC(C)(C)C)[C@@H](O1)c1ccnc(F)c1 |r|
COCC[C@@H]1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc(nc2)N(C2CC2)C(=O)OC(C)(C)C)[C@@H](O1)c1ccnc(F)c1 |r|
CNc1ncc(cn1)-c1nn(c(NC(=O)N[C@@H]2C[C@@H](CCOC)O[C@H]2c2ccnc(F)c2)c1C)-c1ccccc1 |r|
COCC[C@@H]1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc(NC3CC3)nc2)[C@@H](O1)c1ccnc(F)c1 |r|
COCCC1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc(COC(=O)C(C)(C)C)nc2)[C@@H](O1)c1ccccc1 |r|
COCCC1C[C@@H](NC(=O)Nc2c(C)c(OCC(C)(C)O)nn2-c2ccccc2)[C@@H](O1)c1ccccc1 |r|
COCCC1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc(CO)nc2)[C@@H](O1)c1ccccc1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-n2cnc(C)c2)[C@@H](O1)c1cnc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc(F)nc2)[C@@H](O1)c1ccnc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cc(C(N)=O)c(=O)n(C)n2)[C@@H](O1)c1ccnc(F)c1 |r|
Cc1c(NC(=O)N[C@@H]2CN(CC(F)(F)F)O[C@H]2c2ccc(F)c(F)c2)n(nc1-c1cnn(C)c1)-c1ccccc1 |r|
Cc1c(NC(=O)N[C@@H]2CN(CC(F)(F)F)O[C@H]2c2ccc(F)c(F)c2)n(nc1-c1cnc2n(C)ncc2c1)-c1ccccc1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc3OCCNc3c2)[C@@H](O1)c1ccnc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc(OC)c(c2)C#N)[C@@H](O1)c1ccnc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc(OC)c(c2)C(C)(C)O)[C@@H](O1)c1ccnc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2ccc3nc(cn3c2)C(N)=O)[C@@H](O1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc(C(N)=O)c(F)c2)[C@@H](O1)c1cnc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc(C(N)=O)c(F)c2)[C@@H](O1)c1ccc(F)c(F)c1 |r|
CNC(=O)c1ncc(cc1F)-c1nn(c(NC(=O)N[C@@H]2CN(CCOC)O[C@H]2c2ccc(F)c(F)c2)c1C)-c1ccccc1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc(C(N)=O)c(Cl)c2)[C@@H](O1)c1ccnc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc(C(N)=O)c(OC)c2)[C@@H](O1)c1ccnc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc(OC)c(c2)C(=O)NOCC(C)(C)O)[C@@H](O1)c1cnc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc3n(C)cnc3c2)[C@@H](O1)c1cc(F)nc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc(nc2)N2CC(O)C2)[C@@H](O1)c1cc(F)nc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc(nc2)N2CCOCC2)[C@@H](O1)c1ccnc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc3OCC4COC(=O)N4c3c2)[C@@H](O1)c1ccnc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2ccc(C)nc2)[C@@H](O1)c1ccnc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc(OC(F)F)nc2)[C@@H](O1)c1ccnc(F)c1 |r|
COCC[C@@H]1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc3n(C)n(C)c(=O)c3c2)[C@@H](O1)c1ccnc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc3nn(cc3c2)C(F)F)[C@@H](O1)c1ccnc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cccc(CN=S(C)(C)=O)c2)[C@@H](O1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2ccc(N=S(C)(C)=O)nc2)[C@@H](O1)c1ccc(F)cc1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)N2CC(C2)c2ccc(F)cc2)[C@@H](O1)c1ccnc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)N2CC(C2)c2ccc(F)cc2)[C@@H](O1)c1cnc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc3NC(=O)COc3c2)[C@@H](O1)c1cnc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc3OCC(CO)N(C)c3c2)[C@@H](O1)c1ccnc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc(C(=O)NC3CC3)c(OC)c2)[C@@H](O1)c1ccnc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc3OCCN(C)c3c2)[C@@H](O1)c1ccnc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc3OCCN(C(C)=O)c3c2)[C@@H](O1)c1ccnc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc3C(=O)N(C)Cc3c2)[C@@H](O1)c1ccnc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)N2CCN(C)C(=O)C2)[C@@H](O1)c1ccc(F)cc1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-n2cnc(C)c2)[C@@H](O1)c1ccnc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2ccc3nc(CO)cn3c2)[C@@H](O1)c1ccnc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cc(C)c3nccn3c2)[C@@H](O1)c1ccnc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2ccc(nc2)N2CCC(C2)NC(C)=O)[C@@H](O1)c1ccnc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2ccc(C)nc2F)[C@@H](O1)c1ccnc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc3NCCc3c2)[C@@H](O1)c1ccnc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc(OC)cn2)[C@@H](O1)c1ccnc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc3C(O)CCc3c2)[C@@H](O1)c1ccnc(F)c1 |r|
CCC(O)(CC)c1cc(cnc1OC)-c1nn(c(NC(=O)N[C@@H]2CN(CCOC)O[C@H]2c2ccnc(F)c2)c1C)-c1ccccc1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc(OC)c(c2)C2(O)CC2)[C@@H](O1)c1ccnc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc3NCC(=O)Nc3c2)[C@@H](O1)c1ccnc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc(nc2)C2(O)COC2)[C@@H](O1)c1ccnc(F)c1 |r|
COCCN1C[C@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc(C)nc2)[C@H](O1)c1cc(F)nc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2ccc3nc(C)nn3c2)[C@@H](O1)c1cnc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2ccc3OCC(=O)Nc3c2)[C@@H](O1)c1ccnc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2ccc3OCC(=O)N(C)c3c2)[C@@H](O1)c1ccnc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc(OC)c(OC)c2)[C@@H](O1)c1ccnc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc(OC)c(F)c2)[C@@H](O1)c1ccnc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc(nc2)-c2cnn(C)c2)[C@@H](O1)c1ccnc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc3n(C)nc(C(=O)OC)c3c2)[C@@H](O1)c1ccnc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc(nc2)N2CCN(CC2)C(=O)OCc2ccccc2)[C@@H](O1)c1cc(F)nc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc(nc2)N2CCN(CC2)C(=O)OCc2ccccc2)[C@@H](O1)c1ccnc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2ccc(nc2)N2CCN(CC2)C(=O)OC(C)(C)C)[C@@H](O1)c1ccnc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc(nc2)N2CC3(COC3)C2)[C@@H](O1)c1ccnc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2ccc(nc2)N2CCNCC2)[C@@H](O1)c1ccnc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2ccc(nc2)N2CCN(CC#N)CC2)[C@@H](O1)c1ccnc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc3n(C)nc(C(=O)NC4CCN(C)CC4)c3c2)[C@@H](O1)c1ccnc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc3n(C)nc(C(=O)N4CCN(C)CC4)c3c2)[C@@H](O1)c1ccnc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc(nc2)N2CCCC2)[C@@H](O1)c1ccnc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc(nc2)N2CCN(C)CC2)[C@@H](O1)c1ccnc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc(nc2)N2CCN(C)CC2)[C@@H](O1)c1cc(F)nc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc(OC3CCN(C)CC3)nc2)[C@@H](O1)c1ccnc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2ccc3OCCNc3c2)[C@@H](O1)c1ccnc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cc(F)c3OCCNc3c2)[C@@H](O1)c1ccnc(F)c1 |r|
CNC(=O)c1nn(c(NC(=O)N[C@@H]2CN(CCOC)O[C@H]2c2ccnc(F)c2)c1C)-c1ccccc1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)C(=O)NCC(C)(C)O)[C@@H](O1)c1ccnc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)C(=O)NCc2cncnc2)[C@@H](O1)c1ccnc(F)c1 |r|
CNC(=O)c1cc(NC(=O)N[C@@H]2CN(CCOC)O[C@H]2c2ccnc(F)c2)n(n1)-c1ccccc1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cc(C(=O)NC(C)(C)C)c(=O)n(C)c2)[C@@H](O1)c1ccnc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cc(C(=O)NC(C)(C)C(F)(F)F)c(=O)n(C)c2)[C@@H](O1)c1ccnc(F)c1 |r|
CNC(=O)c1cc(cnc1OC)-c1nn(c(NC(=O)N[C@@H]2CN(CCOC)O[C@H]2c2ccc(F)c(F)c2)c1C)-c1ccccc1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2ccc(nc2)N2C[C@@H]3COC[C@H](C2)N3C(=O)OC(C)(C)C)[C@@H](O1)c1ccnc(F)c1 |r,THB:38:37:29.30.36:32.34.33|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2ccc(nc2)N2C[C@@H]3COC[C@H](C2)N3)[C@@H](O1)c1ccnc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc(nc2)N2C[C@@H]3C[C@H](C2)N3)[C@@H](O1)c1ccnc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2ccc(nc2)N2C[C@@H]3COC[C@H](C2)N3C)[C@@H](O1)c1ccnc(F)c1 |r,THB:38:37:29.30.36:32.34.33|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)C2=CC(=O)N(C)C(C)(C)C2)[C@@H](O1)c1ccnc(F)c1 |r,t:25|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc3n(C)c(nc3c2)N2CCCC2)[C@@H](O1)c1ccnc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc3n(C)c(nc3c2)N2CCN(C)CC2)[C@@H](O1)c1ccnc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc3n(CC(=O)N4CCN(C)CC4)cnc3c2)[C@@H](O1)c1ccnc(F)c1 |r|
CNC(=O)Cn1cnc2cc(cnc12)-c1nn(c(NC(=O)N[C@@H]2CN(CCOC)O[C@H]2c2ccnc(F)c2)c1C)-c1ccccc1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc3n(CC(=O)N(C)C)cnc3c2)[C@@H](O1)c1ccnc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc3n(C)c(nc3c2)C(=O)N2CCN(C)CC2)[C@@H](O1)c1ccnc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc3n(C)c(nc3c2)C(=O)NC2CCN(C)CC2)[C@@H](O1)c1ccnc(F)c1 |r|
CCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc(OC)nc2)[C@@H](O1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc(OC)nc2)[C@@H](O1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc(nc2)N2CC3(C2)CCOCC3)[C@@H](O1)c1ccnc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc(OCCN(C)C)nc2)[C@@H](O1)c1ccnc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc3C(=O)N(C)Cc3c2)[C@@H](O1)c1cnc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc3C(=O)N(C)Cc3c2)[C@@H](O1)c1ccc(F)cc1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc3n(C)nc(CN4CCCC4)c3c2)[C@@H](O1)c1ccnc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc(nc2)N2CCNCC2)[C@@H](O1)c1ccnc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc(nc2)N2CCNCC2)[C@@H](O1)c1cc(F)nc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc(nc2)N2CCN(CC#N)CC2)[C@@H](O1)c1ccnc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc(OC3CCN(C)CC3)nc2)[C@@H](O1)c1cc(F)nc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc(nc2)N2CCN(CC#N)CC2)[C@@H](O1)c1cc(F)nc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc(nc2)N2C[C@@H]3C[C@H](C2)N3C)[C@@H](O1)c1ccnc(F)c1 |r,THB:36:35:29.30.34:32|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc(nc2)N2C[C@@H]3COC[C@H](C2)N3)[C@@H](O1)c1ccnc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc(nc2)N2C[C@@H]3COC[C@H](C2)N3C)[C@@H](O1)c1ccnc(F)c1 |r,THB:38:37:29.30.36:32.34.33|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc3n(C)nc(CN4CCC(F)(F)C4)c3c2)[C@@H](O1)c1ccnc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc3n(C)nc(CO[Si](C)(C)C(C)(C)C)c3c2)[C@@H](O1)c1ccnc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc(OC3CC3)nc2)[C@@H](O1)c1ccnc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc3n(cnc3c2)C2CCN(C)CC2)[C@@H](O1)c1ccnc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc3OCCOc3c2)[C@@H](O1)c1ccnc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc3CCN(Cc4ccccc4)Cc3c2)[C@@H](O1)c1ccnc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc(OC)c(OC)c2)[C@@H](O1)c1cnc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc(nc2)N2CC3(COC3)C2)[C@@H](O1)c1cnc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc3n(C)ncc3n2)[C@@H](O1)c1ccnc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc(Br)nc2)[C@@H](O1)c1ccnc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc3n(C)nc(CO)c3c2)[C@@H](O1)c1ccnc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc(C(=O)OC)c(CF)c2)[C@@H](O1)c1ccnc(F)c1 |r|
CNC(=O)c1ncc(cc1CF)-c1nn(c(NC(=O)N[C@@H]2CN(CCOC)O[C@H]2c2ccnc(F)c2)c1C)-c1ccccc1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc(nc2)C2[C@H]3CC[C@@H]2COC3)[C@@H](O1)c1ccnc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc3CCN(Cc3c2)C(C)=O)[C@@H](O1)c1ccnc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc3CCN(C)Cc3c2)[C@@H](O1)c1ccnc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(Oc3ccnc(c3)C(F)(F)F)nn2-c2ccccc2)[C@@H](O1)c1ccnc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(Oc3ccnc(F)c3)nn2-c2ccccc2)[C@@H](O1)c1ccnc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc(OC3CCOCC3)nc2)[C@@H](O1)c1ccnc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc(COC)nc2)[C@@H](O1)c1ccnc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc(nc2)C2=CCN(C)CC2)[C@@H](O1)c1ccnc(F)c1 |r,t:32|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc3n(CC(=O)OC)ncc3c2)[C@@H](O1)c1ccnc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccn2)-c2cnn(C)c2)[C@@H](O1)c1ccc(F)c(F)c1 |r|
COCC[C@@H]1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccn2)-c2cnn(C)c2)[C@@H](O1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cccnc2)[C@@H](O1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cccc(c2)N(C)C)[C@@H](O1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2ccc3nc(CO)cn3c2)[C@@H](O1)c1ccc(F)c(F)c1 |r|
CNC(=O)c1ccc(cn1)-c1nn(c(NC(=O)N[C@@H]2CN(CCOC)O[C@H]2c2ccnc(F)c2)c1C)-c1ccccc1 |r|
CNC(=O)c1ccc(cn1)-c1nn(c(NC(=O)N[C@@H]2CN(CCOC)O[C@H]2c2cnc(F)c(F)c2)c1C)-c1ccccc1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(OCc3ccccn3)nn2-c2ccccc2)[C@@H](O1)c1ccnc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(OCc3cccnc3)nn2-c2ccccc2)[C@@H](O1)c1ccnc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(OCc3ccncc3)nn2-c2ccccc2)[C@@H](O1)c1ccnc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(OCc3ccon3)nn2-c2ccccc2)[C@@H](O1)c1ccnc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc(c(F)c2)C(C)(C)O)[C@@H](O1)c1ccnc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2ccc3nccn3c2)[C@@H](O1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2ccn3ccnc3c2)[C@@H](O1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc3OCCOc3c2)[C@@H](O1)c1cnc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc3OCCOc3c2)[C@@H](O1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc(OC3CCN(C)CC3)nc2)[C@@H](O1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc(OC3COC3)nc2)[C@@H](O1)c1ccnc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2ccncc2)[C@@H](O1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc3n(CC(=O)N4CCN(C)CC4)ncc3c2)[C@@H](O1)c1ccnc(F)c1 |r|
COc1ncc(cn1)-c1nn(c(NC(=O)N[C@@H]2CN(C)O[C@H]2c2ccc(F)c(F)c2)c1C)-c1ccccc1 |r|
CNC(=O)c1cc(cnc1OC)-c1nn(c(NC(=O)N[C@@H]2CN(C)O[C@H]2c2ccc(F)c(F)c2)c1C)-c1ccccc1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2ccc3nccn3c2)[C@@H](O1)c1ccnc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2ccn3ccnc3c2)[C@@H](O1)c1ccnc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(OCc3cnn(C)c3)nn2-c2ccccc2)[C@@H](O1)c1ccnc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc3n(C)ncc3c2)[C@@H](O1)c1ccc(F)c(F)c1 |r|
CNC(=O)c1cc(cnc1OC)-c1nn(c(NC(=O)N[C@@H]2CNO[C@H]2c2ccc(F)c(F)c2)c1C)-c1ccccc1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc(nc2)N2CCN(CC2)C(=O)OCc2ccccc2)[C@@H](O1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc(nc2)-c2cnoc2)[C@@H](O1)c1ccnc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc(OC(C)C)nc2)[C@@H](O1)c1ccnc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc(OC(CF)CF)nc2)[C@@H](O1)c1ccnc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc(nc2)N2CC(C)(O)C2)[C@@H](O1)c1ccnc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc(nc2)N2CC(F)C2)[C@@H](O1)c1ccnc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc(nc2)N2CC(F)(F)C2)[C@@H](O1)c1ccnc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc(nc2)N2CCC3(COC3)C2)[C@@H](O1)c1ccnc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc(nc2)N2CC3(C2)CCOC3)[C@@H](O1)c1ccnc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc(nc2)N2CCC3(COC3)CC2)[C@@H](O1)c1ccnc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc(nc2)N2CC3(CCC3)C2)[C@@H](O1)c1ccnc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc(nc2)N2C[C@@H]3CC[C@H](C2)O3)[C@@H](O1)c1ccnc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc(nc2)N2C[C@@H]3C[C@H](C2)O3)[C@@H](O1)c1ccnc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc(nc2)N2CCN(C)C(=O)C2)[C@@H](O1)c1ccnc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc3n(C)nc(N4CCN(C)CC4)c3c2)[C@@H](O1)c1ccnc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc3n(C)nc(N4CCCC4)c3c2)[C@@H](O1)c1ccnc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2Cc2ccccc2)-c2cnn(C)c2)[C@@H](O1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2CCO)-c2cnn(C)c2)[C@@H](O1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2CCN(C)C)-c2cnn(C)c2)[C@@H](O1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2ccn(C)c(=O)c2)[C@@H](O1)c1ccnc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2ccc(=O)n(C)c2)[C@@H](O1)c1ccnc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2ccn(C)c(=O)c2)[C@@H](O1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2ccc(=O)n(C)c2)[C@@H](O1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(OCC3CN(CCO3)C(=O)OC(C)(C)C)nn2-c2ccccc2)[C@@H](O1)c1ccnc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(OCC3CNCCO3)nn2-c2ccccc2)[C@@H](O1)c1ccnc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(OCc3cc(OC)ccn3)nn2-c2ccccc2)[C@@H](O1)c1ccnc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(OCC3CC3)nn2-c2ccccc2)[C@@H](O1)c1ccnc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(OCC3COC3)nn2-c2ccccc2)[C@@H](O1)c1ccnc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(OCC3CN(CCO3)C(C)=O)nn2-c2ccccc2)[C@@H](O1)c1ccnc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(OCC3CN(C)CCO3)nn2-c2ccccc2)[C@@H](O1)c1ccnc(F)c1 |r|
CCc1ncc(COc2nn(c(NC(=O)N[C@@H]3CN(CCOC)O[C@H]3c3ccnc(F)c3)c2C)-c2ccccc2)cn1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc(nc2)N2CCNOCC2)[C@@H](O1)c1ccnc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2cccc(F)c2)-c2cnn(C)c2)[C@@H](O1)c1ccc(F)c(F)c1 |r|
COCCOc1ncc(cn1)-c1nn(c(NC(=O)N[C@@H]2CN(CCOC)O[C@H]2c2ccnc(F)c2)c1C)-c1ccccc1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc(COC)nc2)[C@@H](O1)c1cnc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc(nc2)C2CCOCC2)[C@@H](O1)c1ccnc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc(nc2)N2CC3CC(C2)O3)[C@@H](O1)c1cnc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnnc(OC)c2)[C@@H](O1)c1ccnc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2ccc(OC)nc2)[C@@H](O1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc3occc3c2)[C@@H](O1)c1ccnc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(C)nn2-c2ccccc2)[C@@H](O1)c1ccc(F)c(F)c1 |r|
CCOc1nn(c(NC(=O)N[C@@H]2CN(CCOC)O[C@H]2c2ccc(F)c(F)c2)c1C)-c1ccccc1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(C)nn2-c2ccccc2)[C@@H](O1)c1cnc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(C)nn2-c2ccccc2)[C@@H](O1)c1ccnc(F)c1 |r|
CCOc1nn(c(NC(=O)N[C@@H]2CN(CCOC)O[C@H]2c2ccnc(F)c2)c1C)-c1ccccc1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc(NCC(F)(F)F)nc2)[C@@H](O1)c1ccnc(F)c1 |r|
COc1ncc(cn1)-c1nn(c(NC(=O)N[C@@H]2CN(CCF)O[C@H]2c2ccc(F)c(F)c2)c1C)-c1ccccc1 |r|
COc1ncc(cn1)-c1nn(c(NC(=O)N[C@@H]2CN(O[C@H]2c2ccc(F)c(F)c2)C(C)C)c1C)-c1ccccc1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc(CN(C)C)nc2)[C@@H](O1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2ccnc(C)c2)[C@@H](O1)c1ccnc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc3OCCc3c2)[C@@H](O1)c1ccnc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2ccc(COC(C)=O)nc2)[C@@H](O1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc(nc2)N2CCC(CC2)N(C)C)[C@@H](O1)c1ccnc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2ccc(CO)nc2)[C@@H](O1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)C(F)(F)F)[C@@H](O1)c1ccnc(F)c1 |r|
CCN1C[C@H](NC(=O)Nc2c(C)c(OCC3CCN(C)CC3)nn2-c2ccccc2)[C@H](O1)c1ccc(F)c(F)c1 |r|
CCN1C[C@@H](NC(=O)Nc2c(C)c(OCC3CNCCO3)nn2-c2ccccc2)[C@@H](O1)c1ccc(F)c(F)c1 |r|
CCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc3n(C)c(=O)oc3c2)[C@@H](O1)c1ccc(F)c(F)c1 |r|
CCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc(nc2)N2CCN(C)CC2)[C@@H](O1)c1ccc(F)c(F)c1 |r|
CCOc1nn(c(NC(=O)N[C@@H]2CN(CC)O[C@H]2c2ccc(F)cc2)c1C)-c1ccccc1 |r|
CCOc1nn(c(NC(=O)N[C@@H]2CN(CC)O[C@H]2c2ccc(F)c(F)c2)c1C)-c1ccccc1 |r|
CCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2ccn(C)c(=O)c2)[C@@H](O1)c1ccc(F)c(F)c1 |r|
CCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2ccc(=O)n(C)c2)[C@@H](O1)c1ccc(F)c(F)c1 |r|
CCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc(OC)c(c2)C(=O)NC2CCOCC2)[C@@H](O1)c1ccc(F)c(F)c1 |r|
CCN1C[C@@H](NC(=O)Nc2c(C)c(OCC3CN(CCO3)C(C)=O)nn2-c2ccccc2)[C@@H](O1)c1ccc(F)c(F)c1 |r|
CCN1C[C@@H](NC(=O)Nc2c(C)c(OCC3CN(C)CCO3)nn2-c2ccccc2)[C@@H](O1)c1ccc(F)c(F)c1 |r|
CNC(=O)c1cc(cnc1OC)-c1nn(c(NC(=O)N[C@@H]2CN(CCF)O[C@H]2c2ccc(F)c(F)c2)c1C)-c1ccccc1 |r|
CNC(=O)c1cc(cnc1OC)-c1nn(c(NC(=O)N[C@@H]2CN(CC(F)F)O[C@H]2c2ccc(F)c(F)c2)c1C)-c1ccccc1 |r|
COCC[C@@H]1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc(nc2)N2CC(C2)OC)[C@@H](O1)c1ccnc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2ccc(OC)cc2)[C@@H](O1)c1ccnc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2ccc(C)nc2)[C@@H](O1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2ccc(nc2)N2CC(C2)OC)[C@@H](O1)c1ccc(F)c(F)c1 |r|
CCN1C[C@@H](NC(=O)Nc2c(C)c(OCC3CCNCC3)nn2-c2ccccc2)[C@@H](O1)c1ccc(F)c(F)c1 |r|
Cc1c(OCC2CCNCC2)nn(c1NC(=O)N[C@@H]1CN(CCF)O[C@H]1c1ccc(F)c(F)c1)-c1ccccc1 |r|
Cc1c(OCC2CCNCC2)nn(c1NC(=O)N[C@@H]1CN(CC(F)F)O[C@H]1c1ccc(F)c(F)c1)-c1ccccc1 |r|
CCN1C[C@@H](NC(=O)Nc2c(C)c(OCC3CCNCC3)nn2-c2ccccc2)[C@@H](O1)c1ccc(F)cc1 |r|
CCN1C[C@@H](NC(=O)Nc2c(C)c(OCC3CCN(CC3)C(C)=O)nn2-c2ccccc2)[C@@H](O1)c1ccc(F)c(F)c1 |r|
CC(=O)N1CCC(COc2nn(c(NC(=O)N[C@@H]3CN(CCF)O[C@H]3c3ccc(F)c(F)c3)c2C)-c2ccccc2)CC1 |r|
CC(=O)N1CCC(COc2nn(c(NC(=O)N[C@@H]3CN(CC(F)F)O[C@H]3c3ccc(F)c(F)c3)c2C)-c2ccccc2)CC1 |r|
CCN1C[C@@H](NC(=O)Nc2c(C)c(OCC3CCN(CC3)C(C)=O)nn2-c2ccccc2)[C@@H](O1)c1ccc(F)cc1 |r|
CN1CCC(COc2nn(c(NC(=O)N[C@@H]3CN(CCF)O[C@H]3c3ccc(F)c(F)c3)c2C)-c2ccccc2)CC1 |r|
CN1CCC(COc2nn(c(NC(=O)N[C@@H]3CN(CC(F)F)O[C@H]3c3ccc(F)c(F)c3)c2C)-c2ccccc2)CC1 |r|
CCN1C[C@@H](NC(=O)Nc2c(C)c(OCC3CCN(C)CC3)nn2-c2ccccc2)[C@@H](O1)c1ccc(F)cc1 |r|
CCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc(OC)c(c2)C(=O)NC)[C@@H](O1)c1ccc(F)cc1 |r|
CNC(=O)c1cc(cnc1OC)-c1nn(c(NC(=O)N[C@@H]2CN(CC(F)(F)F)O[C@H]2c2ccc(F)c(F)c2)c1C)-c1ccccc1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(OCCN(C)C)nn2-c2ccccc2)[C@@H](O1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(OC3CN(C3)C(=O)OC(C)(C)C)nn2-c2ccccc2)[C@@H](O1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(OC3CNC3)nn2-c2ccccc2)[C@@H](O1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(OCC3CNCCO3)nn2-c2ccccc2)[C@@H](O1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(OCC3CN(CCO3)C(C)=O)nn2-c2ccccc2)[C@@H](O1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(OCC3CN(C)CCO3)nn2-c2ccccc2)[C@@H](O1)c1ccc(F)c(F)c1 |r|
COCCN1CC(NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc(nc2)N2CC3(CCO3)C2)C(O1)c1ccnc(F)c1
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc(nc2)N2CC(C2)N(C)C)[C@@H](O1)c1ccnc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc(nc2)N2CC(C2)N2CCOCC2)[C@@H](O1)c1ccnc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc(nc2)N2CC[C@@H](C2)OC)[C@@H](O1)c1ccnc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc(nc2)N2CC[C@H](C2)OC)[C@@H](O1)c1ccnc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc(nc2)N2CC[C@@H](C2)N(C)C)[C@@H](O1)c1ccnc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc(nc2)N2CC[C@H](C2)N(C)C)[C@@H](O1)c1ccnc(F)c1 |r|
COCCN(C)c1ncc(cn1)-c1nn(c(NC(=O)N[C@@H]2CN(CCOC)O[C@H]2c2ccnc(F)c2)c1C)-c1ccccc1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc(nc2)N(C)CCCN(C)C)[C@@H](O1)c1ccnc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc(nc2)N2C[C@H]3C[C@@H]2CO3)[C@@H](O1)c1ccnc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc(nc2)N2C[C@@H]3C[C@H]2CO3)[C@@H](O1)c1ccnc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc(nc2)N2CCN(C)[C@H](C)C2)[C@@H](O1)c1ccnc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc(nc2)N2CCN(C)[C@@H](C)C2)[C@@H](O1)c1ccnc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc(nc2)N2CCN(C)C[C@H]2C)[C@@H](O1)c1ccnc(F)c1 |r|
CNC(=O)c1cc(ccn1)-c1nn(c(NC(=O)N[C@@H]2CN(CCOC)O[C@H]2c2ccc(F)c(F)c2)c1C)-c1ccccc1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc3oc(C)nc3c2)[C@@H](O1)c1ccnc(F)c1 |r|
CCN1C[C@@H](NC(=O)Nc2c(C)c(OCCC3CCN(C3)C(=O)OC(C)(C)C)nn2-c2ccccc2)[C@@H](O1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc(nc2)N2CCN(C)CC2)[C@@H](O1)c1ccc(F)c(F)c1 |r|
CCN1C[C@@H](NC(=O)Nc2c(C)c(OCCC3CCNC3)nn2-c2ccccc2)[C@@H](O1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(OC3CN(C)C3)nn2-c2ccccc2)[C@@H](O1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(OC3CCN(CC3)C(=O)OC(C)(C)C)nn2-c2ccccc2)[C@@H](O1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(OC3CCNCC3)nn2-c2ccccc2)[C@@H](O1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(OC3CCN(C)CC3)nn2-c2ccccc2)[C@@H](O1)c1ccc(F)c(F)c1 |r|
CCN1CCC(CC1)Oc1nn(c(NC(=O)N[C@@H]2CN(CCOC)O[C@H]2c2ccc(F)c(F)c2)c1C)-c1ccccc1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(CO[Si](C)(C)C(C)(C)C)nn2-c2ccccc2)[C@@H](O1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc3OCOc3c2)[C@@H](O1)c1ccnc(F)c1 |r|
CCN1C[C@@H](NC(=O)Nc2c(C)c(OCC3CCN(CC3)C(=O)CO)nn2-c2ccccc2)[C@@H](O1)c1ccc(F)c(F)c1 |r|
CCN1C[C@@H](NC(=O)Nc2c(C)c(OCC3CCN(CC3)C(=O)COC)nn2-c2ccccc2)[C@@H](O1)c1ccc(F)c(F)c1 |r|
CCN1C[C@@H](NC(=O)Nc2c(C)c(OCC3CCN(CC)CC3)nn2-c2ccccc2)[C@@H](O1)c1ccc(F)c(F)c1 |r|
CCN1C[C@@H](NC(=O)Nc2c(C)c(OCCCN(C)C)nn2-c2ccccc2)[C@@H](O1)c1ccc(F)c(F)c1 |r|
CCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2ccc3nc(cn3c2)C(N)=O)[C@@H](O1)c1ccc(F)c(F)c1 |r|
CCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc(C(N)=O)c(F)c2)[C@@H](O1)c1ccc(F)c(F)c1 |r|
CCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc(C(=O)NC)c(F)c2)[C@@H](O1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(OCC3COC(C)(C)O3)nn2-c2ccccc2)[C@@H](O1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(OCC(O)CO)nn2-c2ccccc2)[C@@H](O1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc3nc(C)oc3c2)[C@@H](O1)c1ccnc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2ccnc(CO)c2)[C@@H](O1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2ccnc(CN(C)C)c2)[C@@H](O1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(CO)nn2-c2ccccc2)[C@@H](O1)c1ccc(F)c(F)c1 |r|
COc1ncc(cn1)-c1nn(c(NC(=O)N[C@@H]2CN(CCC(F)(F)F)O[C@H]2c2ccc(F)c(F)c2)c1C)-c1ccccc1 |r|
Cc1c(NC(=O)N[C@@H]2CN(CCC(F)(F)F)O[C@H]2c2ccc(F)c(F)c2)n(nc1-c1cnc2n(C)ncc2c1)-c1ccccc1 |r|
CNC(=O)c1cc(cnc1OC)-c1nn(c(NC(=O)N[C@@H]2CN(CCC(F)(F)F)O[C@H]2c2ccc(F)c(F)c2)c1C)-c1ccccc1 |r|
CCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2ccc3nccn3c2)[C@@H](O1)c1ccc(F)c(F)c1 |r|
CCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2ccn3ccnc3c2)[C@@H](O1)c1ccc(F)c(F)c1 |r|
CCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc3OCCOc3c2)[C@@H](O1)c1ccc(F)c(F)c1 |r|
CCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc(nc2)N2CC(C2)OC)[C@@H](O1)c1ccc(F)c(F)c1 |r|
Cc1c(NC(=O)N[C@@H]2CN(CC(F)F)O[C@H]2c2ccc(F)c(F)c2)n(nc1-c1cccnc1)-c1ccccc1 |r|
Cc1c(NC(=O)N[C@@H]2CN(CC(F)F)O[C@H]2c2ccc(F)c(F)c2)n(nc1-c1ccncc1)-c1ccccc1 |r|
CCN1C[C@@H](NC(=O)Nc2c(C)c(OC3CCN(C)CC3)nn2-c2ccccc2)[C@@H](O1)c1ccc(F)c(F)c1 |r|
CCN1C[C@@H](NC(=O)Nc2c(C)c(OC3CN(C)C3)nn2-c2ccccc2)[C@@H](O1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(OCC(N)=O)nn2-c2ccccc2)[C@@H](O1)c1ccnc(F)c1 |r|
CNC(=O)COc1nn(c(NC(=O)N[C@@H]2CN(CCOC)O[C@H]2c2ccnc(F)c2)c1C)-c1ccccc1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(OCC(=O)NC3CC3)nn2-c2ccccc2)[C@@H](O1)c1ccnc(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc(OC)c(COC(C)=O)c2)[C@@H](O1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc(OC)c(CO)c2)[C@@H](O1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(CN(C)C)nn2-c2ccccc2)[C@@H](O1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(CCN(C)C)nn2-c2ccccc2)[C@@H](O1)c1ccc(F)c(F)c1 |r|
CCN1C[C@@H](NC(=O)Nc2c(C)c(CCN(C)C)nn2-c2ccccc2)[C@@H](O1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2ccnc(CCN(C)C)c2)[C@@H](O1)c1ccc(F)c(F)c1 |r|
CCN1C[C@@H](NC(=O)Nc2c(C)c(OCc3cc(=O)ccn3C)nn2-c2ccccc2)[C@@H](O1)c1ccc(F)c(F)c1 |r|
CCN1C[C@@H](NC(=O)Nc2c(C)c(OCC(=O)NC)nn2-c2ccccc2)[C@@H](O1)c1ccc(F)c(F)c1 |r|
CCN1C[C@@H](NC(=O)Nc2c(C)c(OCC(=O)N(C)C)nn2-c2ccccc2)[C@@H](O1)c1ccc(F)c(F)c1 |r|
CCN1C[C@@H](NC(=O)Nc2c(C)c(OCC(=O)NC3CC3)nn2-c2ccccc2)[C@@H](O1)c1ccc(F)c(F)c1 |r|
CCN1C[C@@H](NC(=O)Nc2c(C)c(OCC(=O)N3CCN(C)CC3)nn2-c2ccccc2)[C@@H](O1)c1ccc(F)c(F)c1 |r|
CCN1C[C@@H](NC(=O)Nc2c(C)c(OCC(=O)NCCN(C)C)nn2-c2ccccc2)[C@@H](O1)c1ccc(F)c(F)c1 |r|
CCN1C[C@@H](NC(=O)Nc2c(C)c(OCC(=O)NCCO)nn2-c2ccccc2)[C@@H](O1)c1ccc(F)c(F)c1 |r|
CCN1C[C@@H](NC(=O)Nc2c(C)c(OCC(=O)NCC(C)(C)O)nn2-c2ccccc2)[C@@H](O1)c1ccc(F)c(F)c1 |r|
CN1CCC(COc2nn(c(NC(=O)N[C@@H]3CN(CC4CC4)O[C@H]3c3ccc(F)c(F)c3)c2C)-c2ccccc2)CC1 |r|
CCCN1C[C@@H](NC(=O)Nc2c(C)c(OCC3CCN(C)CC3)nn2-c2ccccc2)[C@@H](O1)c1ccc(F)c(F)c1 |r|
CCN1C[C@@H](NC(=O)Nc2c(C)c(OCC(C)(C)O)nn2-c2ccccc2)[C@@H](O1)c1ccc(F)c(F)c1 |r|
CCN1C[C@@H](NC(=O)Nc2c(C)c(OCC3CNC3)nn2-c2ccccc2)[C@@H](O1)c1ccc(F)c(F)c1 |r|
CCN1C[C@@H](NC(=O)Nc2c(C)c(OCC3CN(C)C3)nn2-c2ccccc2)[C@@H](O1)c1ccc(F)c(F)c1 |r|
CCN1C[C@@H](NC(=O)Nc2c(C)c(OCCCC(=O)NC)nn2-c2ccccc2)[C@@H](O1)c1ccc(F)c(F)c1 |r|
CCN1C[C@@H](NC(=O)Nc2c(C)c(OCCCN3CCCC3)nn2-c2ccccc2)[C@@H](O1)c1ccc(F)c(F)c1 |r|
CCN1C[C@@H](NC(=O)Nc2c(C)c(OCCCCN(C)C)nn2-c2ccccc2)[C@@H](O1)c1ccc(F)c(F)c1 |r|
CCN1C[C@@H](NC(=O)Nc2c(C)c(OCCCC(N)=O)nn2-c2ccccc2)[C@@H](O1)c1ccc(F)c(F)c1 |r|
CCN1C[C@@H](NC(=O)Nc2c(C)c(OCCCC(=O)N(C)C)nn2-c2ccccc2)[C@@H](O1)c1ccc(F)c(F)c1 |r|
CCN1C[C@@H](NC(=O)Nc2c(C)c(OCCCC(=O)NC3CC3)nn2-c2ccccc2)[C@@H](O1)c1ccc(F)c(F)c1 |r|
CCN1C[C@@H](NC(=O)Nc2c(C)c(OCCCC(=O)N3CCN(C)CC3)nn2-c2ccccc2)[C@@H](O1)c1ccc(F)c(F)c1 |r|
CCN1C[C@@H](NC(=O)Nc2c(C)c(OCCCC(=O)NCCN(C)C)nn2-c2ccccc2)[C@@H](O1)c1ccc(F)c(F)c1 |r|
CCN1C[C@@H](NC(=O)Nc2c(C)c(OCCCC(=O)NCCO)nn2-c2ccccc2)[C@@H](O1)c1ccc(F)c(F)c1 |r|
CCN1C[C@@H](NC(=O)Nc2c(C)c(OCCCC(=O)NCC(C)(C)O)nn2-c2ccccc2)[C@@H](O1)c1ccc(F)c(F)c1 |r|
CCN1C[C@@H](NC(=O)Nc2c(C)c(OCCCCO)nn2-c2ccccc2)[C@@H](O1)c1ccc(F)c(F)c1 |r|
CCN1C[C@@H](NC(=O)Nc2c(C)c(OCCC3CCNCC3)nn2-c2ccccc2)[C@@H](O1)c1ccc(F)c(F)c1 |r|
CCN1C[C@@H](NC(=O)Nc2c(C)c(OCCC3CCN(C)CC3)nn2-c2ccccc2)[C@@H](O1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C(F)F)c(C)nn2-c2ccccc2)[C@@H](O1)c1ccnc(F)c1 |r|
CCN1C[C@@H](NC(=O)Nc2c(C)c(OCC3CNC(=O)O3)nn2-c2ccccc2)[C@@H](O1)c1ccc(F)c(F)c1 |r|
CCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc(OC)nc2)[C@@H](O1)c1ccc(F)c(F)c1 |r|
CCCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc(OC)nc2)[C@@H](O1)c1ccc(F)c(F)c1 |r|
COc1ncc(cn1)-c1nn(c(NC(=O)N[C@@H]2CN(CCCO)O[C@H]2c2ccc(F)c(F)c2)c1C)-c1ccccc1 |r|
CCN1C[C@@H](NC(=O)Nc2c(C)c(OC(C)C3CCN(C)CC3)nn2-c2ccccc2)[C@@H](O1)c1ccc(F)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(Br)c(nn2-c2ccccc2)-c2cnc(OC)nc2)[C@@H](O1)c1ccnc(F)c1 |r|
Cc1cc(NC(=O)NC2[C@H](O)CC(C)(C)c3ccccc23)c(nc1-c1cncc(c1)C(F)(F)F)-c1ccccc1 |r|
Cc1cc(NC(=O)NC2[C@H](O)CC(C)(C)c3ccccc23)c(nc1-c1ccc(nc1)S(C)(=O)=O)-c1ccccc1 |r|
Cc1cc(NC(=O)NC2[C@H](O)CC(C)(C)c3ccccc23)c(nc1-c1ccc(nc1)C#N)-c1ccccc1 |r|
Cc1cc(NC(=O)NC2[C@H](O)CC(C)(C)c3ccccc23)c(nc1-c1cnc(nc1)S(F)(F)F)-c1ccccc1 |r|
Cc1cc(NC(=O)N[C@H]2[C@H](O)CC(C)(C)c3ccccc23)c(nc1-c1cnc(nc1)C(C)(C)O)-c1ccccc1 |r|
Cc1cnc(c(NC(=O)NC2[C@H](O)CC(C)(C)c3ccc(Br)cc23)c1)-c1ccccc1 |r|
Cc1cnc(C2CCOCC2)c(NC(=O)N[C@H]2[C@H](O)CC(C)(C)c3ccc(CO)cc23)c1 |r|
Cc1cnc(c(NC(=O)NC2[C@H](O)CC(C)(C)c3cc(F)c(F)cc23)c1)-c1ccccc1 |r|
Cc1cc(NC(=O)N[C@H]2[C@H](O)CC(C)(C)c3cc(F)c(F)cc23)c(nc1CO)-c1ccccc1 |r|
Cc1ncc(cn1)-c1nc(c(NC(=O)NC2[C@H](O)CC(C)(C)c3cc(F)c(F)cc23)cc1C)-c1ccccc1 |r|
Cc1ncc(cn1)-c1nc(c(NC(=O)N[C@@H]2[C@H](O)CC(C)(C)c3cc(F)c(F)cc23)cc1C)-c1ccccc1 |r|
Cc1cc(NC(=O)N[C@H]2[C@H](O)CC(C)(C)c3cc(F)c(F)cc23)c(nc1-c1ccc(CO)cc1)-c1ccccc1 |r|
Cc1cc(cnn1)-c1nc(c(NC(=O)NC2[C@H](O)CC(C)(C)c3cc(F)c(F)cc23)cc1C)-c1ccccc1 |r|
Cc1ncc(s1)-c1nc(c(NC(=O)N[C@@H]2[C@H](O)CC(C)(C)c3cc(F)c(F)cc23)cc1C)-c1ccccc1 |r|
Cc1cc(NC(=O)NC2[C@H](O)CC(C)(C)c3cc(F)c(F)cc23)c(nc1-c1cnc(nc1)C(C)(C)O)-c1ccccc1 |r|
Cc1cc(NC(=O)N[C@H]2[C@H](O)CC(C)(C)c3cc(F)c(F)cc23)c(nc1-c1ccc(CO)nc1)-c1ccccc1 |r|
Cc1cc(NC(=O)N[C@H]2[C@H](O)CC(C)(C)c3cc(F)c(F)cc23)c(nc1-c1ccnc(CO)c1)-c1ccccc1 |r|
Cc1cc(NC(=O)N[C@H]2[C@H](O)CC(C)(C)c3cc(F)c(F)cc23)c(nc1C(N)=O)C1CCOCC1 |r|
Cc1cc(NC(=O)NC2[C@H](O)CC(C)(C)c3cc(F)c(F)cc23)c(nc1-c1cn[nH]c1)C1CCOCC1 |r|
Cc1cc(NC(=O)N[C@@H]2[C@H](O)CC(C)(C)c3cc(F)c(F)cc23)c(nc1-c1cn[nH]c1)C1CCOCC1 |r|
Cc1cc(NC(=O)NC2[C@H](O)CC(C)(C)c3cc(F)c(F)cc23)c(nc1-c1cnc(O)nc1)C1CCOCC1 |r|
OC(F)CNC(=O)c1cnn2ccc(nc12)N1CCC[C@@H]1c1cncc(F)c1 |r|
COc1ncc(F)cc1[C@H]1CCCN1c1ccn2ncc(C(=O)NC3CCC(CC3)S(C)(=O)=O)c2n1 |r,wD:9.9,(-8.31,3.61,;-6.84,3.14,;-5.7,4.17,;-6.02,5.67,;-4.87,6.7,;-3.41,6.23,;-2.27,7.26,;-3.09,4.72,;-4.23,3.69,;-3.91,2.18,;-4.94,1.04,;-4.17,-.29,;-2.67,.03,;-2.51,1.56,;-1.17,2.33,;-1.17,3.87,;.16,4.64,;1.49,3.87,;2.96,4.34,;3.86,3.1,;2.96,1.85,;3.43,.39,;2.4,-.76,;4.94,.07,;5.42,-1.4,;4.39,-2.54,;4.86,-4.01,;6.37,-4.33,;7.4,-3.18,;6.92,-1.72,;6.84,-5.79,;5.38,-6.27,;7.32,-7.26,;8.31,-5.32,;1.49,2.33,;.16,1.56,)|
Cn1cc(F)cc([C@H]2CCCN2c2ccn3ncc(C(=O)Nc4ccc(O)cn4)c3n2)c1=O |r|
COc1ccc(F)cc1[C@H]1CCCN1c1ccn2ncc(NC(=O)N3CCCC(O)C3)c2n1 |r|
C[C@H]1Nc2ccn3ncc(c3n2)C(=O)NCC2Cc3cc(F)cc1c3O2
C[C@H]1Nc2ccn3ncc(c3n2)C(=O)NCC[C@H]2Cc3cc(F)cc1c3O2
C[C@H]1Nc2ccn3ncc(c3n2)C(=O)NCC2(C)Cc3cc(F)cc1c3O2
C[C@H]1Nc2ccn3ncc(c3n2)C(=O)NCCc2cc3cc(F)cc1c3o2
C[C@H]1Nc2ccn3ncc(c3n2)C(=O)NC[C@@H]2COc3cc(F)cc1c3O2
C[C@H]1Nc2ccn3ncc(c3n2)C(=O)NC[C@@]2(C)Cc3cc(F)cc1c3O2
C[C@H]1Nc2ccn3ncc(c3n2)C(=O)NC[C@]2(C)Cc3cc(F)c(F)c1c3O2
COC[C@@]12CNC(=O)c3cnn4ccc(nc34)N[C@H](C)c3cc(F)cc(c3O1)C2
C[C@H]1Nc2ccn3ncc(c3n2)C(=O)NCC2(CF)Cc3cc(F)cc1c3O2
CCOC(=O)c1c(N)nn2ccc(nc12)N1CCC[C@@H]1c1cc(F)ccc1F |r|
Nc1nn2ccc(nc2c1C(O)=O)N1CCC[C@@H]1c1cc(F)ccc1F |r|
CNC(=O)c1c(N)nn2ccc(nc12)N1CCC[C@@H]1c1cc(F)ccc1F |r|
NC(=O)c1c(N)nn2ccc(nc12)N1CCC[C@@H]1c1cc(F)ccc1F |r|
CCOC(=O)c1c(N)nn2ccc(nc12)N1CCCC1c1cc(F)ccc1F
NC(=O)c1c(N)nn2ccc(nc12)N1CCCC1c1cc(F)ccc1F
CCOC(=O)c1c(NC(=O)NC)nn2ccc(nc12)N1CCCC1c1cc(F)ccc1F
CCOC(=O)c1c(NC(C)=O)nn2ccc(nc12)N1CCC[C@@H]1c1cc(F)ccc1F |r|
Nc1nn2ccc(nc2c1C(=O)N1CCC(O)C1)N1CCC[C@@H]1c1cc(F)ccc1F |r|
Nc1nn2ccc(nc2c1C(=O)NC1CCC(O)CC1)N1CCC[C@@H]1c1cc(F)ccc1F |r,wD:24.28,(2.64,3.82,;1.3,3.05,;-.11,3.68,;-1.14,2.53,;-2.68,2.53,;-3.45,1.2,;-2.68,-.13,;-1.14,-.13,;-.37,1.2,;1.14,1.52,;2.29,.49,;1.97,-1.02,;3.75,.97,;4.89,-.07,;4.57,-1.57,;5.72,-2.6,;7.18,-2.13,;8.33,-3.16,;7.5,-.62,;6.36,.41,;-3.45,-1.47,;-2.97,-2.93,;-4.22,-3.84,;-5.46,-2.93,;-4.99,-1.47,;-5.89,-.22,;-5.26,1.18,;-6.17,2.43,;-5.54,3.84,;-7.7,2.27,;-8.33,.86,;-7.42,-.38,;-8.05,-1.79,)|
Nc1nn2ccc(nc2c1C(=O)N[C@H]1CC[C@H](O)CC1)N1CCC[C@@H]1c1cc(F)ccc1F |r,wU:13.14,wD:24.28,16.18,(3.91,3.31,;2.44,2.83,;1.2,3.74,;-.05,2.83,;-1.56,3.15,;-2.59,2.01,;-2.11,.54,;-.6,.22,;.43,1.37,;1.97,1.37,;2.87,.12,;2.24,-1.29,;4.4,.28,;5.31,-.96,;6.84,-.8,;7.74,-2.05,;7.12,-3.46,;8.02,-4.7,;5.59,-3.62,;4.68,-2.37,;-3.14,-.6,;-2.67,-2.07,;-3.91,-2.97,;-5.16,-2.07,;-4.68,-.6,;-5.59,.64,;-4.96,2.05,;-5.87,3.3,;-5.24,4.7,;-7.4,3.13,;-8.02,1.73,;-7.12,.48,;-7.74,-.92,)|
Nc1nn2ccc(nc2c1C(=O)NCCO)N1CCC[C@@H]1c1cc(F)ccc1F |r|
Nc1nn2ccc(nc2c1C(=O)Nc1ccc(F)cc1)N1CCC[C@@H]1c1cc(F)ccc1F |r|
CN(C)C(=O)c1c(N)nn2ccc(nc12)N1CCC[C@@H]1c1cc(F)ccc1F |r|
CC(C)(CO)ONC(=O)c1c(N)nn2ccc(nc12)N1CCC[C@@H]1c1cc(F)ccc1F |r|
CC1(C)OCC(CONC(=O)c2c(N)nn3ccc(nc23)N2CCC[C@@H]2c2cc(F)ccc2F)O1 |r|
CC(C)(C)ONC(=O)c1c(N)nn2ccc(nc12)N1CCC[C@@H]1c1cc(F)ccc1F |r|
CN(C)CCNC(=O)c1c(N)nn2ccc(nc12)N1CCC[C@@H]1c1cc(F)ccc1F |r|
CCOC(=O)c1c(NC)nn2ccc(nc12)N1CCC[C@@H]1c1cc(F)ccc1F |r|
CNc1nn2ccc(nc2c1C(N)=O)N1CCC[C@@H]1c1cc(F)ccc1F |r|
CCNc1nn2ccc(nc2c1C(=O)OCC)N1CCC[C@@H]1c1cc(F)ccc1F |r|
CCOC(=O)c1c(NCCN2CCOCC2)nn2ccc(nc12)N1CCC[C@@H]1c1cc(F)ccc1F |r|
Nc1cc2nc(ccn2n1)N1CCCC1c1cc(F)ccc1F
Nc1cc2nc(ccn2n1)N1CCC[C@@H]1c1cc(F)ccc1F |r|
CCOC(=O)c1coc(n1)-c1c(NCc2ccc(OC)cc2)nn2ccc(nc12)N1CCCC1c1cc(F)ccc1F
Cc1coc(n1)-c1c(N)nn2ccc(nc12)N1CCCC1c1cc(F)ccc1F
Cc1csc(n1)-c1c(N)nn2ccc(nc12)N1CCCC1c1cc(F)ccc1F
CCOC(=O)c1csc(n1)-c1c(N)nn2ccc(nc12)N1CCCC1c1cc(F)ccc1F
Nc1nn2ccc(nc2c1-c1nc(cs1)C(=O)N1CC[C@H](O)C1)N1CCCC1c1cc(F)ccc1F |r|
NC(=S)c1c(N)nn2ccc(nc12)N1CCCC1c1cc(F)ccc1F
Nc1nn2ccc(nc2c1Br)N1CCC[C@@H]1c1cc(F)ccc1F |r|
Nc1nn2ccc(nc2c1-c1cccc(c1)N1CCOCC1)N1CCCC1c1cc(F)ccc1F
Cn1cc(cn1)-c1c(N)nn2ccc(nc12)N1CCC[C@@H]1c1cc(F)ccc1F |r|
CCOC(=O)c1c(N)nn2ccc(nc12)N1C[C@@H](F)C[C@@H]1c1cc(F)ccc1F |r|
NC(=O)c1c(N)nn2ccc(nc12)N1C[C@@H](F)C[C@@H]1c1cc(F)ccc1F |r|
CCOC(=O)c1c(N)nn2ccc(nc12)N1C[C@@H](F)C[C@H]1c1cc(F)ccc1F |r|
CCOC(=O)c1c(N)nn2ccc(nc12)N1CC(F)(F)CC1c1cc(F)ccc1F
CNC(=O)c1c(N)nn2ccc(nc12)N1C[C@@H](F)C[C@@H]1c1cc(F)ccc1F |r|
Nc1nn2ccc(nc2c1C(=O)NOCCO)N1CCC[C@@H]1c1cc(F)ccc1F |r|
Nc1nn2ccc(nc2c1C#N)N1C[C@@H](F)C[C@@H]1c1cc(F)ccc1F |r|
CCOC(=O)c1c(N)nn2ccc(nc12)N1C[C@H](O)CC1c1cc(F)ccc1F |r|
CCOC(=O)c1c(N)nn2ccc(nc12)N1CC(=O)CC1c1cc(F)ccc1F
Nc1nn2ccc(nc2c1C#N)N1C[C@@H](O)C[C@@H]1c1cc(F)ccc1F |r|
NC(=O)c1c(N)nn2ccc(nc12)N1C[C@@H](O)C[C@@H]1c1cc(F)ccc1F |r|
NC(=O)c1c(N)nn2ccc(nc12)N1C[C@@H](O)C[C@H]1c1cc(F)ccc1F |r|
CCOC(=O)c1c(N)nn2ccc(nc12)N1C[C@@H](O)CC1c1cc(F)ccc1F |r|
Nc1nn2ccc(nc2c1C(=O)NCCO)N1C[C@@H](F)C[C@@H]1c1cc(F)ccc1F |r|
Nc1nn2ccc(nc2c1C(=O)NOCCO)N1C[C@@H](F)C[C@@H]1c1cc(F)ccc1F |r|
Nc1nn2ccc(nc2c1C(=O)NC1CC1)N1C[C@@H](F)C[C@@H]1c1cc(F)ccc1F |r|
Nc1nn2ccc(nc2c1C(=O)NC1(CO)CC1)N1C[C@@H](F)C[C@@H]1c1cc(F)ccc1F |r|
C[C@H]1Nc2ccn3ncc(c3n2)C(=O)NCC2(CO)Cc3cc(F)cc1c3O2
C[C@H]1Nc2ccn3ncc(c3n2)C(=O)NCC[C@@]2(C)Cc3cc(F)cc1c3O2
C[C@H]1Nc2ccn3ncc(c3n2)C(=O)NCC[C@]2(C)Cc3cc(F)cc1c3O2
C[C@H]1Nc2ccn3ncc(c3n2)C(=O)NCC2(C)Cc3cc(Cl)cc1c3O2
C[C@H]1Nc2ccn3ncc(c3n2)C(=O)NC[C@]2(C)COc3cc(F)cc1c3O2
C[C@H]1Nc2ccn3nc(N)c(c3n2)C(=O)NC[C@@]2(C)Cc3cc(F)cc1c3O2
C[C@H]1Nc2ccc3ncc(n3n2)C(=O)NC[C@@]2(C)Cc3cc(F)cc1c3O2
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2ccc(=O)n(C)c2)[C@@H](C1)c1ccc(F)c(Cl)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2ccc(=O)n(C)c2)[C@@H](C1)c1ccc(Cl)c(F)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2ccc(=O)n(C)c2)[C@@H](C1)c1cc(F)cc(Cl)c1 |r|
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2ccc(=O)n(C)c2)[C@@H](C1)c1cccc(Cl)c1 |r|
Cc1c(NC(=O)NC2CC3(CCC3)Oc3ccccc23)n(nc1-c1cnn(C)c1)-c1ccccc1
Cc1c(NC(=O)N[C@H]2[C@H](O)C3(CC3)c3ccccc23)n(nc1-c1cnc(C)nc1)-c1ccccc1 |r|
COc1ncc(cn1)-c1nn(c(NC(=O)N[C@H]2[C@H](O)C3(CC3)c3ccccc23)c1C)-c1ccccc1 |r|
Cc1c(NC(=O)N[C@H]2[C@H](O)C3(CC3)c3cc(F)c(F)cc23)n(nc1-c1cnn(C)c1)-c1ccccc1 |r|
CNC(=O)c1nn(c(NC(=O)N[C@H]2[C@H](O)C3(CC3)c3ccccc23)c1C)-c1ccccc1 |r|
COc1nn(c(NC(=O)N[C@H]2[C@H](O)C3(CC3)c3ccccc23)c1C)-c1ccccc1 |r|
CCOc1nn(c(NC(=O)N[C@H]2[C@H](O)C3(CC3)c3ccccc23)c1C)-c1ccccc1 |r|
COc1nn(c(NC(=O)N[C@H]2[C@H](O)C3(CC3)c3cc(F)c(F)cc23)c1C)-c1ccccc1 |r|
Cc1c(NC(=O)N[C@H]2[C@H](O)C3(CC3)c3ccc(F)cc23)n(nc1-c1cnn(C)c1)-c1ccccc1 |r|
Cc1c(NC(=O)N[C@H]2[C@H](O)C3(CC3)c3cc(F)ccc23)n(nc1-c1cnn(C)c1)-c1ccccc1 |r|
Cc1c(NC(=O)N[C@H]2[C@H](O)Cc3ccc(Cl)cc23)n(nc1-c1cnn(C)c1)-c1ccccc1 |r|
Cc1c(NC(=O)N[C@H]2[C@H](O)Cc3ccc(Cl)cc23)n(nc1-c1cnc(C)nc1)-c1ccccc1 |r|
Cc1c(NC(=O)N[C@H]2[C@H](O)C(C)(C)c3ccccc23)n(nc1-c1cnn(C)c1)-c1ccccc1 |r|
Cc1c(NC(=O)N[C@H]2[C@H](O)C(C)(C)c3ccccc23)n(nc1-c1cnc(C)nc1)-c1ccccc1 |r|
CNC(=O)c1nn(c(NC(=O)N[C@H]2[C@H](O)CC(C)(C)c3cc(F)c(F)cc23)c1C)-c1ccccc1 |r|
Cc1c(NC(=O)N[C@H]2[C@H](O)CC(C)(C)c3ccccc23)n([nH]c1=O)-c1ccccc1 |r|
Cc1nn(c(NC(=O)N[C@H]2[C@H](O)CC(C)(C)c3ccc(cc23)C(N)=O)c1C)-c1ccccc1 |r|
COC(=O)c1ccc2c(c1)[C@@H](NC(=O)Nc1c(C)c(C)nn1-c1ccccc1)[C@H](O)CC2(C)C |r|
Cc1nn(c(NC(=O)N[C@H]2[C@H](O)CC(C)(C)c3ccc(CO)cc23)c1C)-c1ccccc1 |r|
Cc1c(NC(=O)N[C@H]2[C@H](O)CC(C)(C)c3ccccc23)n(nc1-c1cnc(C)nc1)-c1ccccc1 |r|
CN1CCC(CCc2nn(c(NC(=O)NC3[C@H](O)CCc4ccccc34)c2C)-c2ccccc2)CC1 |r|
Cc1c(OC[C@H]2CN(CCO2)C(=O)OC(C)(C)C)nn(c1NC(=O)N[C@H]1[C@H](O)CC(C)(C)c2ccccc12)-c1ccccc1 |r|
CO[C@H]1[C@@H](O)[C@H](NC(=O)Nc2c(C)c(O)nn2-c2ccccc2)c2ccccc2C1(C)C |r|
Cc1cc(NC(=O)N[C@H]2[C@H](O)CC(C)(C)c3ccccc23)c(nc1-c1ccc(nc1)C#N)-c1ccccc1
Cc1cc(NC(=O)N[C@H]2CCC(C)(C)c3ccccc23)c(nc1-c1cnc(nc1)C(C)(C)O)-c1ccccc1
COCc1ccc2c(c1)[C@@H](NC(=O)Nc1cc(C)cnc1C1CCOCC1)[C@H](O)CC2(C)C
Cc1ncc(cn1)-c1nc(c(NC(=O)N[C@H]2[C@@H](O)CC(C)(C)c3ccc(F)cc23)cc1C)-c1ccccc1
Cc1ncc(cn1)-c1nc(c(NC(=O)N[C@H]2[C@@H](O)CC(C)(C)c3cc(F)ccc23)cc1C)-c1ccccc1
Cc1cnc(c(NC(=O)NC2C(O)CC(C)(C)c3cc(F)c(F)cc23)c1)-c1ccccc1
Cc1cnc(c(NC(=O)N[C@H]2[C@@H](O)CC(C)(C)c3cc(F)c(F)cc23)c1)-c1ccccc1
Cc1cc(NC(=O)N[C@H]2[C@H](O)CC(C)(C)c3cc(F)c(F)cc23)c(nc1C(N)=O)-c1ccccc1
Cc1nnc(CNC(=O)c2nc(c(NC(=O)NC3C(O)CC(C)(C)c4cc(F)c(F)cc34)cc2C)-c2ccccc2)o1
Cc1nnc(CNC(=O)c2nc(c(NC(=O)N[C@H]3[C@@H](O)CC(C)(C)c4cc(F)c(F)cc34)cc2C)-c2ccccc2)o1
Cc1ncc(cn1)-c1nc(c(NC(=O)NC2C(O)CC(C)(C)c3cc(F)c(F)cc23)cc1C)-c1ccccc1
Cc1ncc(cn1)-c1nc(c(NC(=O)N[C@H]2[C@@H](O)CC(C)(C)c3cc(F)c(F)cc23)cc1C)-c1ccccc1
Cc1cc(NC(=O)N[C@H]2[C@H](O)CC(C)(C)c3cc(F)c(F)cc23)c(nc1-c1cccc(CO)c1)-c1ccccc1
Cc1cc(NC(=O)N[C@H]2[C@H](O)CC(C)(C)c3cc(F)c(F)cc23)c(nc1-c1cccc(c1)C#N)-c1ccccc1
Cc1cc(NC(=O)NC2C(O)CC(C)(C)c3cc(F)c(F)cc23)c(nc1-c1ccn(C)n1)-c1ccccc1
Cc1cc(NC(=O)N[C@H]2[C@@H](O)CC(C)(C)c3cc(F)c(F)cc23)c(nc1-c1ccn(C)n1)-c1ccccc1
Cc1cnc(C2CCOCC2)c(NC(=O)N[C@H]2[C@H](O)CC(C)(C)c3ccc(F)cc23)c1
Cc1cc(NC(=O)N[C@H]2[C@H](O)CC(C)(C)c3ccc(F)cc23)c(nc1C(N)=O)C1CCOCC1
Cc1cc(NC(=O)NC2C(O)CC(C)(C)c3cc(F)c(F)cc23)c(nc1-c1cn[nH]c1)C1CCOCC1
Cc1cc(NC(=O)N[C@H]2[C@@H](O)CC(C)(C)c3cc(F)c(F)cc23)c(nc1-c1cn[nH]c1)C1CCOCC1
CC(C)NC(=O)C1CCC(CC1)n1c(NC(=O)c2ccc(F)cc2)nc2ccc(CN3CCC(CC3)C(C)(C)O)cc12 |(-.59,-12.16,;-1.62,-11.02,;-3.12,-11.34,;-1.14,-9.55,;-2.17,-8.41,;-3.68,-8.73,;-1.7,-6.94,;-2.73,-5.8,;-2.25,-4.33,;-.74,-4.01,;.29,-5.16,;-.19,-6.62,;-.27,-2.55,;-1.17,-1.3,;-2.71,-1.3,;-3.48,.03,;-5.02,.03,;-2.71,1.36,;-3.48,2.7,;-2.71,4.03,;-1.17,4.03,;-.4,5.37,;-.4,2.7,;-1.17,1.36,;-.27,-.06,;1.2,-.53,;2.53,.24,;3.86,-.53,;3.86,-2.07,;5.2,-2.84,;6.53,-2.07,;6.53,-.53,;7.87,.24,;9.2,-.53,;9.2,-2.07,;7.87,-2.84,;10.53,.24,;11.87,1.01,;11.3,-1.1,;9.76,1.57,;2.53,-2.84,;1.2,-2.07,)|
NC(=O)c1cc(F)cc(c1)[C@H]1C[C@H](F)CN1Cc1nc2c(cnn2cc1F)C#N |r|
C[C@@H]1CCc2ncc(F)cc2N2CCCN2c2ccn3ncc(C(=O)N1)c3n2 |r|
C[C@@H]1CCc2ccccc2N2CCCN2c2ccn3ncc(C(=O)N1)c3n2 |r|
C[C@@H]1CCn2cc(F)cc(N3CCCN3c3ccn4ncc(C(=O)N1)c4n3)c2=O |r|
C[C@@H]1CCOc2ncc(F)cc2N2CCCN2c2ccn3ncc(C(=O)N1)c3n2 |r|
C[C@@H]1CCc2ncc(F)cc2N2CCC(=O)N2c2ccn3ncc(C(=O)N1)c3n2 |r|
C[C@@H]1CCc2ncc(F)cc2N2CC3(CC3)CN2c2ccn3ncc(C(=O)N1)c3n2 |r|
C[C@@H]1CCc2ncc(F)cc2[C@H]2CCCN2c2ccc3ncc(C(=O)N1)n3n2 |r|
C[C@@H]1CCc2ncc(F)cc2[C@@H]2CCCN2c2ccc3ncc(C(=O)N1)n3n2 |r|
CC1(C)CCc2ncc(F)cc2C2CCCN2c2ccn3ncc(NC1=O)c3n2
C[C@@H]3/C=C\c1ncc(F)cc1[C@H]2CCCN2c5ccn4ncc(C(=O)N3)c4n5
C[C@H]1NC(=O)c2cnn3ccc(nc23)N2CCC[C@@H]2c2cc(F)cnc2\C=C/1 |r,c:30|
C[C@H]1NC(=O)c2cnn3ccc(nc23)N2CCC[C@H]2c2cc(F)cnc2\C=C/1 |r,c:30|
C[C@H]1NC(=O)c2cnn3ccc(nc23)N2CCC[C@@H]2c2cc(F)cnc2C1=C |r|
C[C@H]1NC(=O)c2cnn3ccc(nc23)N2CCC[C@H]2c2cc(F)cnc2C1=C |r|
C[C@H]1NC(=O)c2cnn3ccc(nc23)N2CCC[C@@H]2c2cc(F)cnc2C1C |r|
C[C@@H]1CCc2cnc(F)cc2C2CCCN2c2ccc3ncc(C(=O)N1)n3n2 |r|
C[C@@H]1CCc2ncncc2[C@H]2CCCN2c2ccc3ncc(C(=O)N1)n3n2 |r|
C[C@@H]1CCc2ncncc2[C@@H]2CCCN2c2ccc3ncc(C(=O)N1)n3n2 |r|
C[C@@H]1CCn2cc(nn2)[C@H]2CCCN2c2ccn3ncc(C(=O)N1)c3n2 |r|
C[C@@H]1CCn2cc(nn2)[C@@H]2CCCN2c2ccn3ncc(C(=O)N1)c3n2 |r|
C[C@@H]1CCn2nncc2[C@H]2CCCN2c2ccn3ncc(C(=O)N1)c3n2 |r|
C[C@@H]1CCc2ncc(F)cc2N2CCC[C@H]2c2ccn3ncc(C(=O)N1)c3n2 |r|
C[C@@H]1CCc2ncc(F)cc2N2CCC[C@@H]2c2ccn3ncc(C(=O)N1)c3n2 |r|
C[C@@H]1CCc2ncc(F)cc2[C@H]2[C@@H]3[C@H](CN2c2ccn4ncc(C(=O)N1)c4n2)C3(C)C |r|
C[C@@H]1CCc2ncc(F)cc2[C@@H]2[C@H]3[C@@H](CN2c2ccn4ncc(C(=O)N1)c4n2)C3(C)C |r|
C[C@@H]1CCc2ncc(F)cc2[C@H]2[C@@H]3C[C@@H]3CN2c2ccn3ncc(C(=O)N1)c3n2 |r|
C[C@@H]1CCc2ncc(F)cc2[C@@H]2[C@H]3C[C@H]3CN2c2ccn3ncc(C(=O)N1)c3n2 |r|
Fc1cnc2CCC3(CC3)NC(=O)c3cnn4ccc(nc34)N3C[C@H]4C[C@H]4[C@@H]3c2c1 |r|
Fc1cnc2CCC3(CC3)NC(=O)c3cnn4ccc(nc34)N3C[C@@H]4C[C@@H]4[C@H]3c2c1 |r|
Fc1cnc2CC[C@H](NC(=O)c3cnn4ccc(nc34)N3C[C@H]4C[C@H]4[C@@H]3c2c1)C1CC1 |r|
Fc1cnc2CC[C@H](NC(=O)c3cnn4ccc(nc34)N3C[C@@H]4C[C@@H]4[C@H]3c2c1)C1CC1 |r|
C[C@H]1NC(=O)c2cnn3ccc(nc23)N2C[C@H]3C[C@H]3[C@@H]2c2cc(F)cnc2C1=C |r|
C[C@H]1NC(=O)c2cnn3ccc(nc23)N2C[C@@H]3C[C@@H]3[C@H]2c2cc(F)cnc2C1=C |r|
C[C@H]1CNC(=O)c2cnn3ccc(nc23)N2C[C@H]3C[C@H]3[C@@H]2c2cc(F)cnc2O1 |r|
C[C@H]1CNC(=O)c2cnn3ccc(nc23)N2C[C@@H]3C[C@@H]3[C@H]2c2cc(F)cnc2O1 |r|
C[C@H]1CNC(=O)c2cnn3ccc(nc23)N2C[C@H]3C[C@H]3[C@@H]2c2cc(F)cn1c2=O |r|
C[C@H]1CNC(=O)c2cnn3ccc(nc23)N2C[C@@H]3C[C@@H]3[C@H]2c2cc(F)cn1c2=O |r|
C[C@@H]1CCc2ncc(F)cc2[C@H]2[C@H]3[C@@H](CN2c2ccn4ncc(C(=O)N1)c4n2)C3(C)C |r|
C[C@@H]1CCc2ncc(F)cc2[C@@H]2[C@@H]3[C@H](CN2c2ccn4ncc(C(=O)N1)c4n2)C3(C)C |r|
Nc1nn2ccc3nc2c1C(=O)NCCOc1ncc(F)cc1C1CCCN31
Nc1nn2ccc3nc2c1C(=O)NCCCOc1ncc(F)cc1C1CCCN31
Nc1nn2ccc3nc2c1C(=O)NCCCCc1cccc(n1)C1CCCN31
Nc1nn2ccc3nc2c1C(=O)NCCOc1ncccc1[C@H]1CCCN31 |r|
Nc1nn2ccc3nc2c1C(=O)NCCCOc1ncccc1[C@H]1CCCN31 |r|
Nc1nn2ccc3nc2c1C(=O)NCCOc1ccc(F)cc1[C@H]1CCCN31 |r|
Nc1nn2ccc3nc2c1C(=O)NCCOc1ncc(F)cc1[C@H]1C[C@@H](O)CN31 |r|
Nc1nn2ccc3nc2c1C(=O)NCCCOc1ccc(F)cc1[C@H]1CCCN31 |r|
Nc1nn2ccc3nc2c1C(=O)NCCOc1ncccc1C1CCCN31
Nc1nn2ccc3nc2c1C(=O)NCCCOc1ncc(F)cc1[C@H]1C[C@H](F)CN31 |r|
Nc1nn2ccc3nc2c1C(=O)NCCCOc1ncc(F)cc1C1C[C@@H](F)CN31 |r|
Nc1nn2ccc3nc2c1C(=O)NCCOc1ncc(F)cc1[C@H]1C[C@H](F)CN31 |r|
C[C@H]1CNC(=O)c2c(N)nn3ccc(nc23)N2C[C@@H](F)C[C@@H]2c2cc(F)cnc2O1 |r|
Nc1nn2ccc3nc2c1C(=O)NCCCCOc1ncc(F)cc1[C@H]1C[C@H](F)CN31 |r|
CN1CCCOc2ncc(F)cc2[C@H]2C[C@H](F)CN2c2ccn3nc(N)c(C1=O)c3n2 |r|
Nc1nn2ccc3nc2c1C(=O)NCCOc1ccc(F)cc1[C@@H]1CCCN31 |r|
Nc1nn2ccc3nc2c1C(=O)NCCCOc1ncc(F)cc1[C@H]1CCCN31 |r|
Nc1nn2ccc3nc2c1C(=O)NCCCn1cc(F)cc([C@H]2CCCN32)c1=O |r|
Nc1nn2ccc3nc2c1C(=O)NCCCn1cc(F)cc([C@H]2C[C@H](F)CN32)c1=O |r|
Nc1nn2ccc3nc2c1C(=O)NCCCn1cc(F)cc(C2CCCN32)c1=O
C[C@@H]1CCc2ncc(F)cc2[C@H]2C[C@H](F)CN2c2ccn3nc(N)c(C(=O)N1)c3n2 |r|
Nc1nn2ccc3nc2c1C(=O)NCCCc1ncc(F)cc1[C@H]1C[C@H](F)CN31 |r|
C[C@@H]1CCc2ncc(F)cc2[C@H]2CCCN2c2ccn3nc(N)c(C(=O)N1)c3n2 |r|
C[C@H]1CCc2ncc(F)cc2[C@H]2C[C@H](F)CN2c2ccn3nc(N)c(C(=O)N1)c3n2 |r|
COc1nn(C)cc1-c1[nH]c2ncc3c(c2c1-c1ccc2c(cnn2C)c1)n(C1CCOCC1)c(=O)n3C
[2H]C([2H])([2H])n1ncc2cc(-c3c(-c4cn(C)nc4OC)[nH]c4ncc5c(c34)n(C3CCOCC3)c(=O)n5C)ccc21
Cn1cc(-c2[nH]c3ncc4c(c3c2-c2ccc3c(cnn3C)c2)n([C@H]2CC[C@@H](CC#N)CC2)c(=O)n4C)cn1
COc1nn(C)cc1c3[nH]c2ncc7c(c2c3c5ccc4c(cnn4C)c5)n([C@H]6CC[C@@H](CC#N)CC6)c(=O)n7C
CN(C)C(=O)c1ccc(-c2[nH]c3ncc4c(c3c2-c2ccc3c(cnn3C)c2)n(C2CCCC2)c(=O)n4C)cc1
Cn1c(=O)n(C2CCCC2)c2c3c(-c4ccccc4)c(-c4ccc(CN5CCC(S(C)(=O)=O)CC5)cc4)[nH]c3ncc21
Cn1ncc2cc(-c3c(-c4ccc(CN5CCC(S(C)(=O)=O)CC5)cc4)[nH]c4ncc5c(c34)n(C3CCCC3)c(=O)n5C)ccc21
COC(=O)N[C@@H]1CC[C@@H](n2c(=O)n(C)c3cnc4[nH]c(-c5ccc(C(=O)N6C7CCC6COC7)c(OC)c5)c(-c5cccc(F)c5)c4c32)C1
CCNC(=O)c1ccc(-c2[nH]c3ncc4c(c3c2-c2ccc3c(cnn3C(C)C)c2)n([C@@H]2CC[C@@H](NC(=O)OC)C2)c(=O)n4C)cc1F
COC(=O)N[C@@H]1CC[C@@H](n2c(=O)n(C)c3cnc4[nH]c(-c5ccc(C(=O)NCCCNc6ccccc6)c(F)c5)c(-c5ccc6c(cnn6C(C)C)c5)c4c32)C1
COC(=O)N[C@@H]1CC[C@@H](n2c(=O)n(C)c3cnc4[nH]c(-c5ccc(C(=O)NC6CC6)c(F)c5)c(-c5ccc6c(cnn6C(C)C)c5)c4c32)C1
COC(=O)N[C@@H]1CC[C@@H](n2c(=O)n(C)c3cnc4[nH]c(-c5ccc(C(=O)NC6CC6(F)F)c(F)c5)c(-c5ccc6c(cnn6C(C)C)c5)c4c32)C1
COC(=O)N[C@@H]1CC[C@@H](n2c(=O)n(C)c3cnc4[nH]c(-c5ccc(C(=O)NC6CC6C(F)(F)F)c(F)c5)c(-c5ccc6c(cnn6C(C)C)c5)c4c32)C1
COC(=O)N[C@@H]1CC[C@@H](n2c(=O)n(C)c3cnc4[nH]c(-c5ccc(C(=O)NCC(F)(F)F)c(F)c5)c(-c5ccc6c(cnn6C(C)C)c5)c4c32)C1
CNC(=O)c1ccc(-c2[nH]c3ncc4c(c3c2-c2ccc3c(cnn3C(C)C)c2)n([C@@H]2CC[C@@H](NC(=O)OC)C2)c(=O)n4C)cc1F
COC(=O)N[C@@H]1CC[C@@H](n2c(=O)n(C)c3cnc4[nH]c(-c5ccc(C(=O)NC6(C(F)(F)F)CC6)c(F)c5)c(-c5ccc6c(cnn6C(C)C)c5)c4c32)C1
COCCNC(=O)c1ccc(-c2[nH]c3ncc4c(c3c2-c2ccc3c(cnn3C(C)C)c2)n([C@@H]2CC[C@@H](NC(=O)OC)C2)c(=O)n4C)cc1F
COCCN(C)C(=O)c1ccc(-c2[nH]c3ncc4c(c3c2-c2ccc3c(cnn3C(C)C)c2)n([C@@H]2CC[C@@H](NC(=O)OC)C2)c(=O)n4C)cc1F
COC(=O)N[C@@H]1CC[C@@H](n2c(=O)n(C)c3cnc4[nH]c(-c5ccc(C(=O)N6CCOCC6)c(F)c5)c(-c5ccc6c(cnn6C(C)C)c5)c4c32)C1
CCNC(=O)c1ccc(-c2[nH]c3ncc4c(c3c2-c2ccc3c(cnn3C(C)C)c2)n([C@@H]2CC[C@@H](NC(=O)OC)C2)c(=O)n4C)cc1OC
COCCNC(=O)c1ccc(-c2[nH]c3ncc4c(c3c2-c2ccc3c(cnn3C(C)C)c2)n([C@@H]2CC[C@@H](NC(=O)OC)C2)c(=O)n4C)cc1
COC(=O)N[C@@H]1CC[C@@H](n2c(=O)n(C)c3cnc4[nH]c(-c5ccc(C(=O)N6CCOCC6)cc5)c(-c5ccc6c(cnn6C(C)C)c5)c4c32)C1
CNC(=O)c1ccc(-c2[nH]c3ncc4c(c3c2-c2ccc3c(cnn3C(C)C)c2)n([C@@H]2CC[C@@H](NC(=O)OC)C2)c(=O)n4C)cc1
COC(=O)N[C@@H]1CC[C@@H](n2c(=O)n(C)c3cnc4[nH]c(-c5ccc(C(=O)N(C)C)cc5)c(-c5ccc6c(cnn6C(C)C)c5)c4c32)C1
CCNC(=O)c1ccc(-c2[nH]c3ncc4c(c3c2-c2ccc3c(cnn3C(C)C)c2)n([C@@H]2CC[C@@H](NC(=O)OC)C2)c(=O)n4C)cc1
COC(=O)N[C@@H]1CC[C@@H](n2c(=O)n(C)c3cnc4[nH]c(-c5ccc(C(=O)N6CCC(F)(F)CC6)c(F)c5)c(-c5ccc6c(cnn6C(C)C)c5)c4c32)C1
[2H]C([2H])([2H])N(Cc7ccc(c2[nH]c1ncc6c(c1c2c4ccc3OC(C)(C)Cc3c4)n([C@@H]5CC[C@@H](NC(=O)OC)C5)c(=O)n6C([2H])([2H])[2H])cc7)C([2H])([2H])[2H]
[2H]C([2H])([2H])n1c(=O)n([C@@H]2CC[C@@H](NC(=O)OC)C2)c2c3c(-c4ccc5c(cnn5C(C)C)c4)c(-c4ccc(CN(C)C)cc4)[nH]c3ncc21
[2H]C([2H])([2H])N(Cc1ccc(-c2[nH]c3ncc4c(c3c2-c2ccc(OCCOC)cc2)n([C@@H]2CC[C@@H](NC(=O)OC)C2)c(=O)n4C([2H])([2H])[2H])cc1)C([2H])([2H])[2H]
COC(=O)N[C@@H]1CC[C@@H](n2c(=O)n(C)c3cnc4[nH]c(-c5ccc(CN(C)C)cc5)c(-c5ccc(F)cc5)c4c32)C1
[2H]C([2H])([2H])N(Cc1ccc(-c2[nH]c3ncc4c(c3c2-c2ccc3c(c2)COC3(C)C)n([C@@H]2CC[C@@H](NC(=O)OC)C2)c(=O)n4C([2H])([2H])[2H])cc1)C([2H])([2H])[2H]
[2H]C([2H])([2H])n1c(=O)n([C@@H]2CC[C@@H](NC(=O)OC)C2)c2c3c(-c4ccc5c(c4)COC5(C)C)c(-c4ccc(C(=O)N(C)C)cc4)[nH]c3ncc21
CN1CCN(Cc2ccc(cc2)C(=O)Nc2cnn3ccc(nc23)N2CCC[C@@H]2c2cc(F)ccc2F)CC1 |r|
CCS(=O)(=O)NCc1ccc(cc1)C(=O)Nc1cnn2ccc(nc12)N1CCC[C@@H]1c1cc(F)ccc1F |r|
C[C@@H]1CCc2ncc(F)cc2C2CCCN2c2nc3c(cnn3cc2F)C(=O)N1
C[C@@H]1CCc2ncc(F)cc2[C@H]2CCCN2c2ccn3ncc(C(=O)N1)c3n2
O=C1N[C@H]2C[C@H](C2)Oc2ncc(F)cc2[C@H]2CCCN2c2nc3c1cnn3cc2F
O=C1N[C@H]2C[C@H](C2)Oc2ncc(F)cc2C2CCCN2c2ccn3ncc1c3n2
C[C@H]1Nc2nc3c(cnn3cc2F)C(=O)N[C@H]2C[C@H](C2)Oc2ncc(F)cc21
C[C@H]1Nc2ccn3ncc(c3n2)C(=O)N[C@H]2C[C@H](C2)Oc2ncc(F)cc21
C[C@H]1Nc2ccn3ncc(c3n2)C(=O)N[C@H]2C[C@H](C2)Oc2ncccc21
C[C@H]1Nc2nc3c(cnn3cc2F)C(=O)NC2CC(C2)Oc2ncccc21
C[C@H]1Nc2ccn3nc(F)c(c3n2)C(=O)N[C@H]2C[C@H](C2)Oc2ncc(F)cc21
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc(nc2)C2(F)COC2)[C@@H](C1)n1ccc(F)c1
[2H]C([2H])([2H])Oc1ccc(F)cc1[C@@H](C)Nc1ccn2ncc(C3=NOC(C)(C)N3)c2n1
C[C@@H](Nc1ccn2ncc(C3=NOC(C)(C)N3)c2n1)c1cc(F)ccc1F
COc1ccc(F)cc1[C@@H](C)Nc1ccn2ncc(NC3=NC(C)(C)CO3)c2n1 |r,t:21|
C[C@@H](Nc1ccn2ncc(NC3=NC(C)(C)CO3)c2n1)c1cc(F)cc(F)c1F |r,t:11|
C[C@@H](Nc1ccn2ncc(C3=NOCCN3)c2n1)c1cc(F)cc(F)c1F |r,t:10|
C[C@@H](Nc1ccn2ncc(C3=NOCC(C)(C)N3)c2n1)c1cc(F)cc(F)c1F |r,t:10|
C[C@@H](Nc1ccn2ncc(C3=NN=CC(C)(C)N3)c2n1)c1cc(F)cc(F)c1F |r,c:12,t:10|
C[C@@H](Nc1ccn2ncc(C3=NC(=O)C(C)(C)N3)c2n1)c1cc(F)ccc1OC(F)F |r,t:10|
COc1ccc(F)cc1[C@@H](C)Nc1ccn2ncc(C3=NC(=O)C(C)(C)N3)c2n1 |r,t:20|
C[C@@H](Nc1ccn2ncc(C3=NC(=O)C(C)(C)N3)c2n1)c1cc(F)cc(F)c1F |r,t:10|
C[C@@H](Nc1ccn2ncc(C3=NOCCN3)c2n1)c1cc(F)ccc1OC(F)F |r,t:10|
COc1ncc(F)cc1[C@@H](C)Nc1ccn2ncc(C3=NC(=O)C(C)(C)N3)c2n1 |r,t:20|
CCCOC(=O)\N=C(/N)c1cnn2ccc(N[C@H](C)c3cc(F)cc(F)c3F)nc12 |r|
COc1ccc(F)cc1[C@@H](C)Nc1ccn2ncc(NC3=NC(C)(C)CN3)c2n1 |r,t:21|
C[C@@H](Nc1ccn2ncc(C(=O)NOCCO)c2n1)c1cc(F)cc(F)c1F |r|
COc1ccc(F)cc1[C@@H](C)Nc1ccn2ncc(OC3=NC(C)(C)CN3)c2n1 |r,t:21|
C[C@@H](Nc1ccn2ncc(OC3=NCC(C)(C)N3)c2n1)c1cc(F)cc(F)c1F |r,t:11|
C[C@@H](Nc1ccn2ncc(C3=NOCC(C)(C)N3)c2n1)c1cc(F)ccc1OC(F)F |r,t:10|
C[C@@H](Nc1ccn2ncc(NC3=NCC(C)(C)N3)c2n1)c1cc(F)cc(F)c1F |r,t:11|
COc1c(F)cc(F)cc1[C@@H](C)Nc1ccn2ncc(NC3=NC(C)(C)CO3)c2n1 |r,t:22|
C[C@@H](Nc1ccn2ncc(C3=NOCCN3)c2n1)c1cc(F)cc(c1F)C(F)(F)F |r,t:10|
COc1c(F)cc(F)cc1[C@@H](C)Nc1ccn2ncc(C3=NC(=O)C(C)(C)N3)c2n1 |r,t:21|
C[C@@H](Nc1ccn2ncc(C3=NC(=O)C(C)(C)N3)c2n1)c1cc(F)ccc1OC(F)(F)F |r,t:10|
CCOc1ncc(F)cc1[C@@H](C)Nc1ccn2ncc(C3=NOCCN3)c2n1 |r,t:21|
C[C@@H](Nc1ccn2ncc(C3=NC(=O)C(C)(C)N3)c2n1)c1cc(F)cnc1OCC(F)(F)F |r,t:10|
CONC(=O)c1cnn2ccc(N[C@H](C)c3cc(F)cc(F)c3F)nc12 |r|
C[C@@H](Nc1ccn2ncc(C3=NC(=O)C(C)(C)N3)c2n1)c1cc(F)cnc1OC(F)(F)F |r,t:10|
C[C@@H](Nc1ccn2ncc(C3=NOCCN3)c2n1)c1cc(F)ccc1OC(F)(F)F |r,t:10|
C[C@@H](Nc1ccn2ncc(C3=NOCCN3)c2n1)c1cc(F)ccc1C(F)(F)F |r,t:10|
C[C@@H](Nc1ccn2ncc(C3=NOCCN3)c2n1)c1cc(F)ccc1C(F)F |r,t:10|
CN[C@@H]1CC2OC([C@@H]1OC)n1c3ccccc3c3c4CNC(=O)c4c4c5ccccc5n2c4c13 |r|
C[C@@H](Oc1ccn2ncc(C3=NOC(C)(C)N3)c2n1)c1c(Cl)ccc(F)c1Cl
COc1ccc(F)cc1[C@@H](C)Nc1ccn2ncc(C3=NOC(C)(C)N3)c2n1
C[C@@H](Nc1ccn2ncc(C3=NOC(C)(C)N3)c2n1)c1c(Cl)ccc(F)c1Cl
C[C@@H](Nc1ccn2ncc(C3=NOC(C)(C)N3)c2n1)c1cc(F)ccc1Br
C[C@H](Nc1ccn2ncc(C3=NOC(C)(C)N3)c2n1)c1cc(F)ccc1Br
C[C@@H](Nc1ccn2ncc(C3=NOC(C)(C)N3)c2n1)c1ccc(F)cc1
C[C@@H](Nc1ccn2ncc(C3=NOC(C)(C)N3)c2n1)c1ccc(F)cc1
C[C@@H](Nc1ccn2ncc(C3=NOC(C)(C)N3)c2n1)c1ccccc1Cl
C[C@@H](Nc1ccn2ncc(C3=NOC(C)(C)N3)c2n1)c1cc(F)cc(F)c1
COc1ncc(F)cc1[C@@H](C)Nc1ccn2ncc(C3=NOC(C)(C)N3)c2n1
COc1ccc(F)cc1[C@H](C)Nc1ccn2ncc(C3=NOC(C)(C)N3)c2n1
Cc1ccc(F)cc1[C@@H](C)Nc1ccn2ncc(C3=NOC(C)(C)N3)c2n1
Cc1ccc(F)cc1[C@H](C)Nc1ccn2ncc(C3=NOC(C)(C)N3)c2n1
CCOc1ccc(F)cc1[C@@H](C)Nc1ccn2ncc(C3=NOC(C)(C)N3)c2n1
CC(C)Oc1ccc(F)cc1[C@@H](C)Nc1ccn2ncc(C3=NOC(C)(C)N3)c2n1
CCc1ccc(F)cc1[C@@H](C)Nc1ccn2ncc(C3=NOC(C)(C)N3)c2n1
COC(=O)N1CCC2(CC1)NC(c1cnn3ccc(N[C@H](C)c4cc(F)ccc4OC)nc13)=NO2
C[C@H](Nc1ccn2ncc(C3=NOC(C)(C)N3)c2n1)c1cc(F)cc2ccccc12
COc1ccc(F)cc1[C@@H](C)Nc1ccn2ncc(C3=NOC4(CCN(S(C)(=O)=O)CC4)N3)c2n1
C[C@@H](Nc1ccn2ncc(C3=NCC(C)(C)N3)c2n1)c1cc(F)ccc1F
CCOCC1(C)NC(c2cnn3ccc(N[C@H](C)c4cc(F)ccc4O)nc23)=NO1
Cc1nc(-c2cnn3ccc(N[C@H](C)c4cc(F)ccc4O)nc23)no1
C[C@@H](Nc1ccn2ncc(C3=NOC(C)(C)N3)c2n1)c1cc(F)ccc1O
CCCCC1NC(c2cnn3ccc(N[C@H](C)c4cc(F)ccc4O)nc23)=NO1
COc1ccc(F)cc1[C@@H](C)Oc1ccn2ncc(C3=NOC(C)(C)N3)c2n1
Cc1cc(c(cc1C2CCNCC2)OC(C)C)Nc3ncc(c(n3)Nc4ccccc4S(=O)(=O)C(C)C)Cl
CCc1cc2C(=O)c3c([nH]c4cc(ccc34)C#N)C(C)(C)c2cc1N1CCC(CC1)N1CCOCC1
C[C@H]1Oc2cc(cnc2N)-c2c(CN(C)C(=O)c3ccc(F)cc13)nn(C)c2C#N |r|
C[C@H]1CNC(=O)c2cnn3c2nc(cc3)N[C@@H](c4cc(ccc4O1)F)C
C[C@H]1COC(=O)c2cnn3ccc(N[C@H](C)c4cc(F)ccc4O1)nc23 |r|
C[C@H]1Nc2ccn3ncc(c3n2)C(=O)OCCOc2ccc(F)cc21
C[C@@H]1COc2ccc(F)cc2[C@@H](C)Nc2ccn3ncc(c3n2)C(=O)O1
C[C@@H]1c2cc(F)ccc2OCCOC(=O)c2cnn3ccc(nc23)N1C
C[C@H]1Nc2ccn3ncc(c3n2)C(=O)OCC(F)(F)Oc2ccc(F)cc21
C[C@H]1COC(=O)c2cnn3ccc(nc23)N[C@H](C)c2cc(F)ccc2S1
C[C@H]1Nc2ccn3ncc(c3n2)C(=O)OCCSc2ccc(F)cc21
COc1cc2ncnc(Oc3ccc(NC(=O)c4cccn(-c5ccc(F)cc5)c4=O)cc3F)c2c2c1OCCO2
COc1cc2ncnc(Oc3ccc(NC(=O)c4c(OC)ccn(-c5ccc(F)cc5)c4=O)cc3F)c2c2c1OCCO2
CCOc1ccn(-c2ccc(F)cc2)c(=O)c1C(=O)Nc1ccc(Oc2ncnc3cc(OC)c4c(c23)OCCO4)c(F)c1
O=C(Nc1ccc(Oc2ncnc3cc(OCCCN4CCOCC4)c4c(c23)OCCO4)c(F)c1)c1cccn(-c2ccc(F)cc2)c1=O
COc1ccn(-c2ccc(F)cc2)c(=O)c1C(=O)Nc1ccc(Oc2ncnc3cc(OCCCN4CCOCC4)c4c(c23)OCCO4)c(F)c1
CCOc1ccn(-c2ccc(F)cc2)c(=O)c1C(=O)Nc1ccc(Oc2ncnc3cc(OCCCN4CCOCC4)c4c(c23)OCCO4)c(F)c1
COc1cc2nccc(Oc3ccc(NC(=O)c4cn(C)c(=O)n(-c5ccc(F)cc5)c4=O)cc3F)c2c2c1OCCO2
COc1cc2nccc(Oc3ccc(NC(=O)c4cn(C(C)C)c(=O)n(-c5ccc(F)cc5)c4=O)cc3F)c2c2c1OCCO2
Cn1cc(C(=O)Nc2ccc(Oc3ccnc4cc(OCCCN5CCOCC5)c5c(c34)OCCO5)c(F)c2)c(=O)n(-c2ccc(F)cc2)c1=O
CC(C)n1cc(C(=O)Nc2ccc(Oc3ccnc4cc(OCCCN5CCOCC5)c5c(c34)OCCO5)c(F)c2)c(=O)n(-c2ccc(F)cc2)c1=O
COc1cc2nccc(Oc3ccc(NC(=O)c4cccn(-c5ccc(F)cc5)c4=O)cc3F)c2c2c1OCCO2
COc1cc2nccc(Oc3ccc(NC(=O)c4c(OC)ccn(-c5ccc(F)cc5)c4=O)cc3F)c2c2c1OCCO2
CCOc1ccn(-c2ccc(F)cc2)c(=O)c1C(=O)Nc1ccc(OC2=CC=NC3=CC(OC)=C4OCCOC4C32)c(F)c1
O=C(Nc1ccc(OC2=CC=NC3=CC(OCCCN4CCOCC4)=C4OCCOC4C32)c(F)c1)c1cccn(-c2ccc(F)cc2)c1=O
COc1ccn(-c2ccc(F)cc2)c(=O)c1C(=O)Nc1ccc(Oc2ccnc3cc(OCCCN4CCOCC4)c4c(c23)OCCO4)c(F)c1
CCOc1ccn(-c2ccc(F)cc2)c(=O)c1C(=O)Nc1ccc(Oc2ccnc3cc(OCCCN4CCOCC4)c4c(c23)OCCO4)c(F)c1
COc1cc2nccc(Oc3ccc(NC(=O)c4ccn(-c5ccc(F)cc5C)n4)cc3F)c2c2c1OCCO2
COc1cn(-c2ccc(F)cc2C)nc1C(=O)Nc1ccc(Oc2ccnc3cc(OC)c4c(c23)OCCO4)c(F)c1
CCOc1cn(-c2ccc(F)cc2C)nc1C(=O)Nc1ccc(Oc2ccnc3cc(OC)c4c(c23)OCCO4)c(F)c1
Cc1cc(F)ccc1-n1ccc(C(=O)Nc2ccc(Oc3ccnc4cc(OCCCN5CCOCC5)c5c(c34)OCCO5)c(F)c2)n1
COc1cn(-c2ccc(F)cc2C)nc1C(=O)Nc1ccc(Oc2ccnc3cc(OCCCN4CCOCC4)c4c(c23)OCCO4)c(F)c1
CCOc1cn(-c2ccc(F)cc2C)nc1C(=O)Nc1ccc(Oc2ccnc3cc(OCCCN4CCOCC4)c4c(c23)OCCO4)c(F)c1
COc1cc2ncnc(Oc3ccc(NC(=O)c4cn(C)c(=O)n(-c5ccc(F)cc5)c4=O)cc3F)c2c2c1OCCO2
Cn1cc(C(=O)Nc2ccc(Oc3ncnc4cc(OCCCN5CCOCC5)c5c(c34)OCCO5)c(F)c2)c(=O)n(-c2ccc(F)cc2)c1=O
O=C(Nc1ccc(Oc2ccnc3cc(OCCCN4CCOCC4)c4c(c23)OCCO4)c(F)c1)c1cccn(-c2ccc(F)cc2)c1=O
COc1ccn(-c2ccc(F)cc2)c(=O)c1C(=O)Nc1ccc(Oc2ccnc3cc(OCCCN4CCOCC4)c4c(c23)OCCO4)c(F)c1
CCOc1ccn(-c2ccc(F)cc2)c(=O)c1C(=O)Nc1ccc(Oc2ccnc3cc(OCCCN4CCOCC4)c4c(c23)OCCO4)c(F)c1
COCCOc1cc2nccc(Oc3ccc(NC(=O)c4cccn(-c5ccc(F)cc5)c4=O)cc3F)c2c2c1OCCO2
COCCOc1cc2nccc(Oc3ccc(NC(=O)c4c(OC)ccn(-c5ccc(F)cc5)c4=O)cc3F)c2c2c1OCCO2
CCOc1ccn(-c2ccc(F)cc2)c(=O)c1C(=O)Nc1ccc(Oc2ccnc3cc(OCCOC)c4c(c23)OCCO4)c(F)c1
CCn1cc(C(=O)Nc2ccc(Oc3ccnc4cc(OC)c5c(c34)OCCO5)c(F)c2)c(=O)n(-c2ccc(F)cc2)c1=O
CCn7cc(C(=O)Nc5ccc(Oc3ccnc4cc(OCCCN1CCOCC1)c2OCCOc2c34)c(F)c5)c(=O)n(c6ccc(F)cc6)c7=O
Cn1cc(C(=O)Nc2ccc(Oc3ccnc4cc(OCCCN5CCOCC5)c5c(c34)OCCO5)c(F)c2)c(=O)n(-c2ccc(F)cc2)c1=O
CC(C)n1cc(C(=O)Nc2ccc(Oc3ccnc4cc(OCCCN5CCOCC5)c5c(c34)OCCO5)c(F)c2)c(=O)n(-c2ccc(F)cc2)c1=O
CCn1cc(C(=O)Nc2ccc(Oc3ccnc4cc(OCCCN5CCCCC5)c5c(c34)OCCO5)c(F)c2)c(=O)n(-c2ccc(F)cc2)c1=O
COCCOc1cc2nccc(Oc3ccc(NC(=O)c4cn(C)c(=O)n(-c5ccc(F)cc5)c4=O)cc3F)c2c2c1OCCO2
COCCOc1cc2nccc(Oc3ccc(NC(=O)c4cn(C(C)C)c(=O)n(-c5ccc(F)cc5)c4=O)cc3F)c2c2c1OCCO2
CCn1cc(C(=O)Nc2ccc(Oc3ccnc4cc(OCCOC)c5c(c34)OCCO5)c(F)c2)c(=O)n(-c2ccc(F)cc2)c1=O
COc1cc2nccc(Oc3ccc(NC(=O)c4cn(CCO)c(=O)n(-c5ccc(F)cc5)c4=O)cc3F)c2c2c1OCCO2
COCCn1cc(C(=O)Nc2ccc(Oc3ccnc4cc(OC)c5c(c34)OCCO5)c(F)c2)c(=O)n(-c2ccc(F)cc2)c1=O
COc1cc2nccc(Oc3ccc(NC(=O)c4cn(CC(C)C)c(=O)n(-c5ccc(F)cc5)c4=O)cc3F)c2c2c1OCCO2
COc1cc2nccc(Oc3ccc(NC(=O)c4cn(CC5CC5)c(=O)n(-c5ccc(F)cc5)c4=O)cc3F)c2c2c1OCCO2
CCOc1ccn(-c2ccc(F)cc2)c(=O)c1C(=O)Nc1ccc(Oc2ccnc3cc(OCCCN4CCN(C)CC4)c4c(c23)OCCO4)c(F)c1
CCOc1ccn(-c2ccc(F)cc2)c(=O)c1C(=O)Nc1ccc(Oc2ccnc3cc(OCCCN4CCN(C(C)=O)CC4)c4c(c23)OCCO4)c(F)c1
CCOc1ccn(-c2ccc(F)cc2)c(=O)c1C(=O)Nc1ccc(Oc2ccnc3cc(OCCCN4CCS(=O)(=O)CC4)c4c(c23)OCCO4)c(F)c1
CCOc1ccn(-c2ccc(F)cc2)c(=O)c1C(=O)Nc1ccc(Oc2ccnc3cc(OCCCN4CCCC4)c4c(c23)OCCO4)c(F)c1
CCOc1ccn(-c2ccc(F)cc2)c(=O)c1C(=O)Nc1ccc(Oc2ccnc3cc(OCCO)c4c(c23)OCCO4)c(F)c1
CCOc1ccn(-c2ccc(F)cc2)c(=O)c1C(=O)Nc1ccc(Oc2ccnc3cc(OCCCO)c4c(c23)OCCO4)c(F)c1
CCOc1ccn(-c2ccc(F)cc2)c(=O)c1C(=O)Nc1ccc(Oc2ccnc3cc(OCCCOC)c4c(c23)OCCO4)c(F)c1
CCOc1ccn(-c2ccc(F)cc2)c(=O)c1C(=O)Nc1ccc(Oc2ccnc3cc(OCC#N)c4c(c23)OCCO4)c(F)c1
CCOc1ccn(-c2ccc(F)cc2)c(=O)c1C(=O)Nc1ccc(Oc2ccnc3cc(OCCCC#N)c4c(c23)OCCO4)c(F)c1
CCOc1ccn(-c2ccc(F)cc2)c(=O)c1C(=O)Nc1ccc(Oc2ccnc3cc(OCC(C)C)c4c(c23)OCCO4)c(F)c1
CCOc1ccn(-c2ccc(F)cc2)c(=O)c1C(=O)Nc1ccc(Oc2ccnc3cc(OCC4CC4)c4c(c23)OCCO4)c(F)c1
CCOc1ccn(-c2ccc(F)cc2)c(=O)c1C(=O)Nc1ccc(Oc2ccnc3cc(OCCCCCCN(C)C)c4c(c23)OCCO4)c(F)c1
CCOc1ccn(-c2ccc(F)cc2)c(=O)c1C(=O)Nc1ccc(Oc2ccnc3cc(OCCCN(C)C)c4c(c23)OCCO4)c(F)c1
CCOc1cc2nccc(Oc3ccc(NC(=O)c4c(OCC)ccn(-c5ccc(F)cc5)c4=O)cc3F)c2c2c1OCCO2
CCOc1ccn(-c2ccc(F)cc2)c(=O)c1C(=O)Nc1ccc(Oc2ccnc3cc(OC(C)C)c4c(c23)OCCO4)c(F)c1
CCOc1ccn(-c2ccc(F)cc2)c(=O)c1C(=O)Nc1ccc(Oc2ccnc3cc(OC4COC4)c4c(c23)OCCO4)c(F)c1
CCOc1ccn(-c2ccc(F)cc2)c(=O)c1C(=O)Nc1ccc(Oc2ccnc3cc(OC4CCOC4)c4c(c23)OCCO4)c(F)c1
CCOc1ccn(-c2ccc(F)cc2)c(=O)c1C(=O)Nc1ccc(Oc2ccnc3cc(OC4CCOCC4)c4c(c23)OCCO4)c(F)c1
CCOc1ccn(-c2ccc(F)cc2)c(=O)c1C(=O)Nc1ccc(Oc2ccnc3cc(OCCCN4CCC(C)(C)CC4)c4c(c23)OCCO4)c(F)c1
CCOc1ccn(-c2ccc(F)cc2)c(=O)c1C(=O)Nc1ccc(Oc2ccnc3cc(OCCCN4CCC(C)(N)CC4)c4c(c23)OCCO4)c(F)c1
CCOc1ccn(-c2ccc(F)cc2)c(=O)c1C(=O)Nc1ccc(Oc2ccnc3cc(OCCCN4CCC(C)(O)CC4)c4c(c23)OCCO4)c(F)c1
CCOc1ccn(-c2ccc(F)cc2)c(=O)c1C(=O)Nc1ccc(Oc2ccnc3cc(OCCCN(C)CCOC)c4c(c23)OCCO4)c(F)c1
CCOc1ccn(-c2ccc(F)cc2)c(=O)c1C(=O)Nc1ccc(Oc2ccnc3cc(OCCCN(C)C4CCC4)c4c(c23)OCCO4)c(F)c1
CCOc1ccn(-c2ccc(F)cc2)c(=O)c1C(=O)Nc1ccc(Oc2ccnc3cc(OCCCN4CCOCC4)c4c(c23)OCCO4)c(Cl)c1
CCOc1ccn(-c2ccc(F)cc2)c(=O)c1C(=O)Nc1ccc(Oc2ccnc3cc(OCCCN4CCOCC4)c4c(c23)OCCO4)cc1Cl
CN1CCN(CCCOc2cc3nccc(Oc4ccc(NC(=O)c5cn(C)c(=O)n(-c6ccc(F)cc6)c5=O)cc4F)c3c3c2OCCO3)CC1
CC(=O)N1CCN(CCCOc2cc3nccc(Oc4ccc(NC(=O)c5cn(C(C)C)c(=O)n(-c6ccc(F)cc6)c5=O)cc4F)c3c3c2OCCO3)CC1
CC(C)n1cc(C(=O)Nc2ccc(Oc3ccnc4cc(OCCCN5CCS(=O)(=O)CC5)c5c(c34)OCCO5)c(F)c2)c(=O)n(-c2ccc(F)cc2)c1=O
CC(C)n1cc(C(=O)Nc2ccc(Oc3ccnc4cc(OCCCN5CCCC5)c5c(c34)OCCO5)c(F)c2)c(=O)n(-c2ccc(F)cc2)c1=O
CC(C)n1cc(C(=O)Nc2ccc(Oc3ccnc4cc(OCCO)c5c(c34)OCCO5)c(F)c2)c(=O)n(-c2ccc(F)cc2)c1=O
CC(C)n1cc(C(=O)Nc2ccc(Oc3ccnc4cc(OCCCO)c5c(c34)OCCO5)c(F)c2)c(=O)n(-c2ccc(F)cc2)c1=O
COCCCOc1cc2nccc(Oc3ccc(NC(=O)c4cn(C)c(=O)n(-c5ccc(F)cc5)c4=O)cc3F)c2c2c1OCCO2
CC(C)n1cc(C(=O)Nc2ccc(Oc3ccnc4cc(OCC#N)c5c(c34)OCCO5)c(F)c2)c(=O)n(-c2ccc(F)cc2)c1=O
CC(C)n1cc(C(=O)Nc2ccc(Oc3ccnc4cc(OCCCC#N)c5c(c34)OCCO5)c(F)c2)c(=O)n(-c2ccc(F)cc2)c1=O
CC(C)COc1cc2nccc(Oc3ccc(NC(=O)c4cn(C)c(=O)n(-c5ccc(F)cc5)c4=O)cc3F)c2c2c1OCCO2
Cn1cc(C(=O)Nc2ccc(Oc3ccnc4cc(OCC5CC5)c5c(c34)OCCO5)c(F)c2)c(=O)n(-c2ccc(F)cc2)c1=O
CC(C)n1cc(C(=O)Nc2ccc(Oc3ccnc4cc(OCCCCCCN(C)C)c5c(c34)OCCO5)c(F)c2)c(=O)n(-c2ccc(F)cc2)c1=O
CN(C)CCCOc1cc2nccc(Oc3ccc(NC(=O)c4cn(C)c(=O)n(-c5ccc(F)cc5)c4=O)cc3F)c2c2c1OCCO2
CCOc1cc2nccc(Oc3ccc(NC(=O)c4cn(C(C)C)c(=O)n(-c5ccc(F)cc5)c4=O)cc3F)c2c2c1OCCO2
CC(C)Oc1cc2nccc(Oc3ccc(NC(=O)c4cn(C)c(=O)n(-c5ccc(F)cc5)c4=O)cc3F)c2c2c1OCCO2
CC(C)n1cc(C(=O)Nc2ccc(Oc3ccnc4cc(OC5COC5)c5c(c34)OCCO5)c(F)c2)c(=O)n(-c2ccc(F)cc2)c1=O
Cn1cc(C(=O)Nc2ccc(Oc3ccnc4cc(OC5CCOC5)c5c(c34)OCCO5)c(F)c2)c(=O)n(-c2ccc(F)cc2)c1=O
Cn1cc(C(=O)Nc2ccc(Oc3ccnc4cc(OC5CCOCC5)c5c(c34)OCCO5)c(F)c2)c(=O)n(-c2ccc(F)cc2)c1=O
CC(C)n1cc(C(=O)Nc2ccc(Oc3ccnc4cc(OCCCN5CCC(C)(C)CC5)c5c(c34)OCCO5)c(F)c2)c(=O)n(-c2ccc(F)cc2)c1=O
CC(C)n1cc(C(=O)Nc2ccc(Oc3ccnc4cc(OCCCN5CCC(C)(N)CC5)c5c(c34)OCCO5)c(F)c2)c(=O)n(-c2ccc(F)cc2)c1=O
CC(C)n1cc(C(=O)Nc2ccc(Oc3ccnc4cc(OCCCN5CCC(C)(O)CC5)c5c(c34)OCCO5)c(F)c2)c(=O)n(-c2ccc(F)cc2)c1=O
COCCN(C)CCCOc1cc2nccc(Oc3ccc(NC(=O)c4cn(C(C)C)c(=O)n(-c5ccc(F)cc5)c4=O)cc3F)c2c2c1OCCO2
CC(C)n1cc(C(=O)Nc2ccc(Oc3ccnc4cc(OCCCN(C)C5CCC5)c5c(c34)OCCO5)c(F)c2)c(=O)n(-c2ccc(F)cc2)c1=O
CC(C)n1cc(C(=O)Nc2ccc(Oc3ccnc4cc(OCCCN5CCOCC5)c5c(c34)OCCO5)c(Cl)c2)c(=O)n(-c2ccc(F)cc2)c1=O
Cn1cc(C(=O)Nc2ccc(Oc3ccnc4cc(OCCCN5CCOCC5)c5c(c34)OCCO5)cc2Cl)c(=O)n(-c2ccc(F)cc2)c1=O
COc1cc2nccc(Oc3ccc(NC(=O)c4cn(CCCO)c(=O)n(-c5ccc(F)cc5)c4=O)cc3F)c2c2c1OCCO2
C=CCn1cc(C(=O)Nc2ccc(Oc3ccnc4cc(OC)c5c(c34)OCCO5)c(F)c2)c(=O)n(-c2ccc(F)cc2)c1=O
COc1cc2nccc(Oc3ccc(NC(=O)c4cn(CCF)c(=O)n(-c5ccc(F)cc5)c4=O)cc3F)c2c2c1OCCO2
COc1cc2nccc(Oc3ccc(NC(=O)c4cn(CCCN5CCOCC5)c(=O)n(-c5ccc(F)cc5)c4=O)cc3F)c2c2c1OCCO2
COc1cc2nccc(Oc3ccc(NC(=O)c4cn(CC(=O)O)c(=O)n(-c5ccc(F)cc5)c4=O)cc3F)c2c2c1OCCO2
CCOc1ccn(-c2ccc(F)cc2)c(=O)c1C(=O)Nc1ccc(Oc2ccnc3cc(OCC4(N)CC4)c4c(c23)OCCO4)c(F)c1
CC(C)n1cc(C(=O)Nc2ccc(Oc3ccnc4cc(OCC5(N)CC5)c5c(c34)OCCO5)c(F)c2)c(=O)n(-c2ccc(F)cc2)c1=O
COc1cc2nccc(Oc3ccc(NC(=O)c4cn(C(C)C)c(=O)n(-c5ccc(C)cc5)c4=O)cc3F)c2c2c1OCCO2
COc1cc2nccc(Oc3ccc(NC(=O)c4cn(C(C)C)c(=O)n(-c5ccc(Cl)cc5)c4=O)cc3F)c2c2c1OCCO2
COc1cc2nccc(Oc3ccc(NC(=O)c4cn(C(C)C)c(=O)n(-c5cccc(F)c5)c4=O)cc3F)c2c2c1OCCO2
COc1cc2nccc(Oc3ccc(NC(=O)c4cn(C(C)C)c(=O)n(-c5ccccc5F)c4=O)cc3F)c2c2c1OCCO2
COc1cc2nccc(Oc3ccc(NC(=O)c4cn(C(C)C)c(=O)n(Cc5ccc(F)cc5)c4=O)cc3F)c2c2c1OCCO2
CCOc1ccn(-c2ccc(C)cc2)c(=O)c1C(=O)Nc1ccc(Oc2ccnc3cc(OC)c4c(c23)OCCO4)c(F)c1
CCOc1ccn(-c2ccc(Cl)cc2)c(=O)c1C(=O)Nc1ccc(Oc2ccnc3cc(OC)c4c(c23)OCCO4)c(F)c1
CCOc1ccn(-c2cccc(F)c2)c(=O)c1C(=O)Nc1ccc(Oc2ccnc3cc(OC)c4c(c23)OCCO4)c(F)c1
CCOc1ccn(-c2ccc(F)cc2)c(=O)c1C(=O)Nc1cc(F)c(Oc2ccnc3cc(OC)c4c(c23)OCCO4)cc1Cl
COc1cc2nccc(Oc3cc(Cl)c(NC(=O)c4cn(C)c(=O)n(-c5ccc(F)cc5)c4=O)cc3F)c2c2c1OCCO2
CCOc1ccn(Cc2ccccc2)c(=O)c1C(=O)Nc1ccc(Oc2ccnc3cc(OC)c4c(c23)OCCO4)c(F)c1
COc1cc2nccc(Oc3cc(Cl)c(NC(=O)c4cn(C(C)C)c(=O)n(-c5ccc(F)cc5)c4=O)cc3F)c2c2c1OCCO2
CCOc1ccn(C2CCCCC2)c(=O)c1C(=O)Nc1ccc(Oc2ccnc3cc(OC)c4c(c23)OCCO4)c(F)c1
CCOc1ccn(-c2ccc(F)cc2)c(=O)c1C(=O)Nc1ccc(Oc2ccnc3cc(OCC(C)(C)O)c4c(c23)OCCO4)c(F)c1
Cn1cc(C(=O)Nc2ccc(Oc3ccnc4cc(OCC(C)(C)O)c5c(c34)OCCO5)c(F)c2)c(=O)n(-c2ccc(F)cc2)c1=O
CC(C)n1cc(C(=O)Nc2ccc(Oc3ccnc4cc(OCC(C)(C)O)c5c(c34)OCCO5)c(F)c2)c(=O)n(-c2ccc(F)cc2)c1=O
COc1cc2nccc(Oc3ccc(NC(=O)c4cccn(-c5ccc(F)cc5)c4=O)c(Cl)c3)c2c2c1OCCO2
COc1cc2nccc(Oc3ccc(NC(=O)c4c(OC)ccn(-c5ccc(C)cc5)c4=O)c(Cl)c3)c2c2c1OCCO2
COc1cc2nccc(Oc3ccc(NC(=O)c4cn(C)c(=O)n(-c5ccc(F)cc5)c4=O)c(Cl)c3)c2c2c1OCCO2
CCOc1ccn(-c2ccc(C)cc2)c(=O)c1C(=O)Nc1ccc(Oc2ccnc3cc(OC)c4c(c23)OCCO4)cc1Cl
CCOc1cc2nccc(Oc3ccc(NC(=O)c4cccn(-c5ccc(F)cc5)c4=O)c(Cl)c3)c2c2c1OCCO2
CCOc1cc2nccc(Oc3ccc(NC(=O)c4c(OC)ccn(-c5ccc(F)cc5)c4=O)c(Cl)c3)c2c2c1OCCO2
CCOc1cc2nccc(Oc3ccc(NC(=O)c4cn(C)c(=O)n(-c5ccc(F)cc5)c4=O)c(Cl)c3)c2c2c1OCCO2
CCOc1cc2nccc(Oc3ccc(NC(=O)c4c(OCC)ccn(-c5ccc(F)cc5)c4=O)c(Cl)c3)c2c2c1OCCO2
N#CCCCOc1cc2nccc(Oc3ccc(NC(=O)c4cccn(-c5ccc(F)cc5)c4=O)c(Cl)c3)c2c2c1OCCO2
COc1ccn(-c2ccc(F)cc2)c(=O)c1C(=O)Nc1ccc(Oc2ccnc3cc(OCCCC#N)c4c(c23)OCCO4)cc1Cl
Cn1cc(C(=O)Nc2ccc(Oc3ccnc4cc(OCCCC#N)c5c(c34)OCCO5)cc2Cl)c(=O)n(-c2ccc(F)cc2)c1=O
CCOc1ccn(-c2ccc(F)cc2)c(=O)c1C(=O)Nc1ccc(Oc2ccnc3cc(OCCCC#N)c4c(c23)OCCO4)cc1Cl
O=C(Nc1ccc(Oc2ccnc3cc(OCCCN4CCCCC4)c4c(c23)OCCO4)cc1Cl)c1cccn(-c2ccc(F)cc2)c1=O
COc1ccn(-c2ccc(F)cc2)c(=O)c1C(=O)Nc1ccc(Oc2ccnc3cc(OCCCN4CCCCC4)c4c(c23)OCCO4)cc1Cl
Cn1cc(C(=O)Nc2ccc(Oc3ccnc4cc(OCCCN5CCCCC5)c5c(c34)OCCO5)cc2Cl)c(=O)n(-c2ccc(F)cc2)c1=O
CCOc1ccn(-c2ccc(F)cc2)c(=O)c1C(=O)Nc1ccc(Oc2ccnc3cc(OCCCN4CCCCC4)c4c(c23)OCCO4)cc1Cl
CC(C)(O)COc1cc2nccc(Oc3ccc(NC(=O)c4cccn(-c5ccc(F)cc5)c4=O)c(Cl)c3)c2c2c1OCCO2
COc1ccn(-c2ccc(F)cc2)c(=O)c1C(=O)Nc1ccc(Oc2ccnc3cc(OCC(C)(C)O)c4c(c23)OCCO4)cc1Cl
Cn1cc(C(=O)Nc2ccc(Oc3ccnc4cc(OCC(C)(C)O)c5c(c34)OCCC5)cc2Cl)c(=O)n(-c2ccc(F)cc2)c1=O
CCOc1ccn(-c2ccc(F)cc2)c(=O)c1C(=O)Nc1ccc(Oc2ccnc3cc(OCC(C)(C)O)c4c(c23)OCCO4)cc1Cl
O=C(Nc1ccc(Oc2ccnc3cc(OCCCN4CCOCC4)c4c(c23)OCCO4)cc1Cl)c1cccn(-c2ccc(F)cc2)c1=O
COc1ccn(-c2ccc(F)cc2)c(=O)c1C(=O)Nc1ccc(Oc2ccnc3cc(OCCCN4CCOCC4)c4c(c23)OCCO4)cc1Cl
COc1cc2nccc(Oc3ccc(NC(=O)c4cn(C)c(=O)n(-c5ccc(F)cc5)c4=O)cc3)c2c2c1OCCO2
CCn1cc(C(=O)Nc2ccc(Oc3ccnc4cc(OC)c5c(c34)OCCO5)cc2)c(=O)n(-c2ccc(F)cc2)c1=O
COCCOc1cc2nccc(Oc3ccc(NC(=O)c4cn(C)c(=O)n(-c5ccc(F)cc5)c4=O)cc3)c2c2c1OCCO2
CCn1cc(C(=O)Nc2ccc(Oc3ccnc4cc(OCCOC)c5c(c34)OCCO5)cc2)c(=O)n(-c2ccc(F)cc2)c1=O
Cn1cc(C(=O)Nc2ccc(Oc3ccnc4cc(OCC(C)(C)O)c5c(c34)OCCO5)cc2)c(=O)n(-c2ccc(F)cc2)c1=O
CCn1cc(C(=O)Nc2ccc(Oc3ccnc4cc(OCC(C)(C)O)c5c(c34)OCCO5)cc2)c(=O)n(-c2ccc(F)cc2)c1=O
Cn1cc(C(=O)Nc2ccc(Oc3ccnc4cc(OC5CC5)c5c(c34)OCCO5)cc2)c(=O)n(-c2ccc(F)cc2)c1=O
CCn1cc(C(=O)Nc2ccc(Oc3ccnc4cc(OC5CC5)c5c(c34)OCCO5)cc2)c(=O)n(-c2ccc(F)cc2)c1=O
COc1cc2nccc(Oc3ccc(NC(=O)c4cn(C)c(=O)n(-c5ccc(F)cc5)c4=O)c(F)c3)c2c2c1OCCO2
CCn1cc(C(=O)Nc2ccc(Oc3ccnc4cc(OC)c5c(c34)OCCO5)cc2F)c(=O)n(-c2ccc(F)cc2)c1=O
COCCOc1cc2nccc(Oc3ccc(NC(=O)c4cn(C)c(=O)n(-c5ccc(F)cc5)c4=O)c(F)c3)c2c2c1OCCO2
CCn1cc(C(=O)Nc2ccc(Oc3ccnc4cc(OCCOC)c5c(c34)OCCO5)cc2F)c(=O)n(-c2ccc(F)cc2)c1=O
COc1cc2nccc(Oc3ccc(NC(=O)c4cn(C(C)C)c(=O)n(C5CCCCC5)c4=O)cc3F)c2c2c1OCCO2
Cn1cc(C(=O)Nc2ccc(Oc3ccnc4ccc5c(c34)OCCO5)cc2)c(=O)n(-c2ccc(F)cc2)c1=O
CCn1cc(C(=O)Nc2ccc(Oc3ccnc4ccc5c(c34)OCCO5)cc2)c(=O)n(-c2ccc(F)cc2)c1=O
Cn1cc(C(=O)Nc2ccc(Oc3ccnc4ccc5c(c34)OCCO5)c(F)c2)c(=O)n(-c2ccc(F)cc2)c1=O
CCn1cc(C(=O)Nc2ccc(Oc3ccnc4ccc5c(c34)OCCO5)c(F)c2)c(=O)n(-c2ccc(F)cc2)c1=O
Cn1cc(C(=O)Nc2ccc(Oc3ccnc4ccc5c(c34)OCCO5)cc2F)c(=O)n(-c2ccc(F)cc2)c1=O
CCn1cc(C(=O)Nc2ccc(Oc3ccnc4ccc5c(c34)OCCO5)cc2F)c(=O)n(-c2ccc(F)cc2)c1=O
CCOc1ccn(-c2ccc(F)cc2)c(=O)c1C(=O)Nc1ccc(Oc2ccnc3ccc4c(c23)OCCO4)cc1
O=C(Nc1ccc(Oc2ccnc3ccc4c(c23)OCCO4)cc1)c1cccn(-c2ccc(F)cc2)c1=O
COc1ccn(-c2ccc(F)cc2)c(=O)c1C(=O)Nc1ccc(Oc2ccnc3ccc4c(c23)OCCO4)cc1
COc1ccn(-c2ccc(F)cc2)c(=O)c1C(=O)Nc1ccc(Oc2ccnc3ccc4c(c23)OCCO4)c(F)c1
CCOc1ccn(-c2ccc(F)cc2)c(=O)c1C(=O)Nc1ccc(Oc2ccnc3ccc4c(c23)OCCO4)c(F)c1
O=C(Nc1ccc(Oc2ccnc3ccc4c(c23)OCCO4)c(F)c1)c1cccn(-c2ccc(F)cc2)c1=O
O=C(Nc1ccc(Oc2ccnc3ccc4c(c23)OCCO4)cc1F)c1cccn(-c2ccc(F)cc2)c1=O
CCOc1ccn(-c2ccc(F)cc2)c(=O)c1C(=O)Nc1ccc(Oc2ccnc3ccc4c(c23)OCCO4)cc1F
COc1ccn(-c2ccc(F)cc2)c(=O)c1C(=O)Nc1ccc(Oc2ccnc3ccc4c(c23)OCCO4)cc1F
Cn1cc(C(=O)Nc2cc(F)c(Oc3ccnc4ccc5c(c34)OCCO5)cc2Cl)c(=O)n(-c2ccc(F)cc2)c1=O
CCn1cc(C(=O)Nc2cc(F)c(Oc3ccnc4ccc5c(c34)OCCO5)cc2Cl)c(=O)n(-c2ccc(F)cc2)c1=O
Cc1cc(Oc2ccnc3ccc4c(c23)OCCO4)c(F)cc1NC(=O)c1cn(C)c(=O)n(-c2ccc(F)cc2)c1=O
CCn1cc(C(=O)Nc2cc(F)c(Oc3ccnc4ccc5c(c34)OCCO5)cc2C)c(=O)n(-c2ccc(F)cc2)c1=O
COc1cc2nccc(Oc3cc(C)c(NC(=O)c4cn(C)c(=O)n(-c5ccc(F)cc5)c4=O)cc3F)c2c2c1OCCO2
CCn1cc(C(=O)Nc2cc(F)c(Oc3ccnc4cc(OC)c5c(c34)OCCO5)cc2C)c(=O)n(-c2ccc(F)cc2)c1=O
COCCOc1cc2nccc(Oc3cc(C)c(NC(=O)c4cn(C)c(=O)n(-c5ccc(F)cc5)c4=O)cc3F)c2c2c1OCCO2
CCn1cc(C(=O)Nc2cc(F)c(Oc3ccnc4cc(OCCOC)c5c(c34)OCCO5)cc2C)c(=O)n(-c2ccc(F)cc2)c1=O
CCc1cc(Oc2ccnc3cc(OCCOC)c4c(c23)OCCO4)c(F)cc1NC(=O)c1cn(C)c(=O)n(-c2ccc(F)cc2)c1=O
CCc1cc(Oc2ccnc3cc(OCCOC)c4c(c23)OCCO4)c(F)cc1NC(=O)c1cn(CC)c(=O)n(-c2ccc(F)cc2)c1=O
COCCOc1cc2nccc(Oc3cc(C(C)C)c(NC(=O)c4cn(C)c(=O)n(-c5ccc(F)cc5)c4=O)cc3F)c2c2c1OCCO2
CCc1cc(Oc2ccnc3cc(OCCOC)c4c(c23)OCCO4)c(F)cc1NC(=O)c1cn(CC)c(=O)n(-c2ccc(F)cc2)c1=O
COC(=O)[C@]1(O)C[C@H]2O[C@]1(C)n1c3ccccc3c3c4CNC(=O)c4c4c5ccccc5n2c4c13
COC(=O)[C@@]1(O)C[C@H]2O[C@]1(C)n1c3ccccc3c3c4CNC(=O)c4c4c5ccccc5n2c4c13 |r|
Fc1cccc(CNc2ccn3ncc(C(=O)NC4CCOCC4)c3n2)c1
O[C@H]1CC[C@@H](CC1)NC(=O)c1cnn2ccc(NCc3cccc(F)c3)nc12 |r,wU:4.7,wD:1.0,(9.18,2.41,;8.09,1.32,;6.6,1.72,;5.52,.63,;5.91,-.86,;7.4,-1.26,;8.49,-.17,;4.83,-1.95,;3.34,-1.55,;2.25,-2.64,;2.94,-.06,;3.85,1.18,;2.97,2.39,;1.48,1.92,;.15,2.69,;-1.18,1.93,;-1.18,.39,;-2.52,-.38,;-3.85,.39,;-5.19,-.38,;-5.19,-1.92,;-6.51,-2.69,;-7.85,-1.93,;-7.85,-.38,;-9.18,.39,;-6.51,.38,;.16,-.39,;1.48,.39,)|
CO[C@H]1CC[C@@H](CC1)NC(=O)c1cnn2ccc(NCc3cccc(F)c3)nc12 |r,wU:5.8,wD:2.1,(8.78,3.29,;9.18,1.81,;8.09,.72,;6.6,1.11,;5.52,.03,;5.91,-1.46,;7.4,-1.86,;8.49,-.77,;4.83,-2.55,;3.34,-2.15,;2.25,-3.24,;2.94,-.66,;3.85,.58,;2.97,1.79,;1.48,1.32,;.15,2.09,;-1.18,1.33,;-1.18,-.21,;-2.52,-.98,;-3.85,-.21,;-5.19,-.98,;-5.19,-2.52,;-6.51,-3.29,;-7.85,-2.53,;-7.85,-.99,;-9.18,-.22,;-6.51,-.22,;.16,-.99,;1.48,-.21,)|
CC(Nc1ccn2ncc(C(=O)NC3CCOCC3)c2n1)c1cccc(F)c1
CC(Nc1ccn2ncc(C(=O)N[C@H]3CC[C@H](O)CC3)c2n1)c1cccc(F)c1 |r,wU:13.12,wD:16.16,(-3.85,1.93,;-3.85,.39,;-2.52,-.38,;-1.18,.39,;-1.18,1.93,;.15,2.69,;1.48,1.92,;2.97,2.39,;3.85,1.18,;2.94,-.06,;3.34,-1.55,;2.25,-2.64,;4.82,-1.95,;5.91,-.86,;5.52,.63,;6.6,1.72,;8.09,1.32,;9.18,2.41,;8.49,-.17,;7.4,-1.26,;1.48,.39,;.16,-.39,;-5.19,-.38,;-5.19,-1.92,;-6.51,-2.69,;-7.85,-1.93,;-7.85,-.38,;-9.18,.39,;-6.51,.38,)|
CN(Cc1cccc(F)c1)c1ccn2ncc(C(=O)NC3CCOCC3)c2n1
CN(Cc1cccc(F)c1)c1ccn2ncc(C(=O)N[C@H]3CC[C@H](O)CC3)c2n1 |r,wU:20.20,wD:23.24,(-2.52,-1.92,;-2.52,-.38,;-3.85,.39,;-5.19,-.38,;-5.19,-1.92,;-6.51,-2.69,;-7.85,-1.93,;-7.85,-.38,;-9.18,.39,;-6.51,.38,;-1.18,.39,;-1.18,1.93,;.15,2.69,;1.48,1.92,;2.97,2.39,;3.85,1.18,;2.94,-.06,;3.34,-1.55,;2.25,-2.64,;4.83,-1.95,;5.91,-.86,;5.52,.63,;6.6,1.72,;8.09,1.32,;9.18,2.41,;8.49,-.17,;7.4,-1.26,;1.48,.39,;.16,-.39,)|
CO[C@H]1CC[C@@H](CC1)NC(=O)c1cnn2ccc(nc12)N(C)Cc1cccc(F)c1 |r,wU:5.8,wD:2.1,(8.78,3.29,;9.18,1.81,;8.09,.72,;6.6,1.11,;5.52,.03,;5.91,-1.46,;7.4,-1.86,;8.49,-.77,;4.83,-2.55,;3.34,-2.15,;2.25,-3.24,;2.94,-.66,;3.85,.58,;2.97,1.79,;1.48,1.32,;.15,2.09,;-1.18,1.33,;-1.18,-.21,;.16,-.99,;1.48,-.21,;-2.52,-.98,;-2.52,-2.52,;-3.85,-.21,;-5.19,-.98,;-5.19,-2.52,;-6.51,-3.29,;-7.85,-2.53,;-7.85,-.99,;-9.18,-.22,;-6.51,-.22,)|
Fc1cccc(CNc2ccc3ncc(C(=O)NC4CCOCC4)n3n2)c1
O[C@H]1CC[C@@H](CC1)NC(=O)c1cnc2ccc(NCc3cccc(F)c3)nn12 |r,wU:4.7,wD:1.0,(9.18,2.41,;8.09,1.32,;6.6,1.72,;5.52,.63,;5.91,-.86,;7.4,-1.26,;8.49,-.17,;4.83,-1.95,;3.34,-1.55,;2.25,-2.64,;2.94,-.06,;3.85,1.18,;2.97,2.39,;1.48,1.92,;.15,2.69,;-1.18,1.93,;-1.18,.39,;-2.52,-.38,;-3.85,.39,;-5.19,-.38,;-5.19,-1.92,;-6.51,-2.69,;-7.85,-1.93,;-7.85,-.38,;-9.18,.38,;-6.51,.38,;.16,-.39,;1.48,.39,)|
CO[C@H]1CC[C@@H](CC1)NC(=O)c1cnc2ccc(NCc3cccc(F)c3)nn12 |r,wU:5.8,wD:2.1,(8.78,3.29,;9.18,1.81,;8.09,.72,;6.6,1.11,;5.52,.03,;5.91,-1.46,;7.4,-1.86,;8.49,-.77,;4.83,-2.55,;3.34,-2.15,;2.25,-3.24,;2.94,-.66,;3.85,.58,;2.97,1.79,;1.48,1.32,;.15,2.09,;-1.18,1.33,;-1.18,-.21,;-2.52,-.98,;-3.85,-.21,;-5.19,-.98,;-5.19,-2.52,;-6.51,-3.29,;-7.85,-2.53,;-7.85,-.99,;-9.18,-.22,;-6.51,-.22,;.16,-.99,;1.48,-.21,)|
OCCNN1C(=O)c2cccc3cc(cc(C1=O)c23)[N+]([O-])=O
CSc1ccccc1Nc1nc(nc2c(NCC3CC3)ncnc12)N1CCN(CC1)C1CCNCC1
CCCSCc1ccc2n3C4C[C@](O)(C(=O)OC)[C@](C)(O4)n4c5ccc(CSCCC)cc5c5c6CNC(=O)c6c(c2c1)c3c45
CCCCSCc1ccc2n3C4C[C@](O)(C(=O)OC)[C@](C)(O4)n4c5ccc(CSCCCC)cc5c5c6CNC(=O)c6c(c2c1)c3c45
CCSCc1ccc2n3C4C[C@](O)(C(=O)OC)[C@](C)(O4)n4c5ccc(CSCC)cc5c5c6CNC(=O)c6c(c2c1)c3c45
COCc1ccc2n3C4C[C@](O)(C(=O)OC)[C@](C)(O4)n4c5ccc(COC)cc5c5c6CNC(=O)c6c(c2c1)c3c45
COC(=O)[C@@]1(O)CC2O[C@]1(C)n1c3ccc(CSC(C)C)cc3c3c4CNC(=O)c4c4c5cc(CSC(C)C)ccc5n2c4c13
COC(=O)[C@@]1(O)CC2O[C@]1(C)n1c3ccc(CSCC=C)cc3c3c4CNC(=O)c4c4c5cc(CSCC=C)ccc5n2c4c13
CCOCc1ccc2n3C4C[C@](O)(C(=O)OC)[C@](C)(O4)n4c5ccc(COCC)cc5c5c6CNC(=O)c6c(c2c1)c3c45
CC(C)(C)CNC(=O)CC1CNC(=O)c2cc(cn12)-c1ccsc1
CN1CCN(C[C@@H](NC(=O)C[C@H]2CNC(=O)c3cc(cn23)-c2cccc(Cl)c2)C2CCCCC2)CC1 |r|
c1cc(cnc1)CNc2ccc3c(n2)c(ncn3)Nc4ccc(cc4)N5CCOCC5
CN1CCN(CC1)c1ccc(Nc2ncnc3ccc(NCc4cccc(Cl)c4)nc23)cc1
Cc1cn2cc(CNc3ncnc4ccc(nc34)N3CCC[C@@H]3c3cc(F)ccc3F)nc2s1 |r|
COc1cc(ccc1-n1cnc(C)c1)-c1cn(CC(=O)Nc2cc(nn2-c2ccccc2)C2CC2)nn1
Cc1cn(cn1)-c1ccc(cc1)-c1cn(CC(=O)Nc2cc(nn2-c2ccccc2)C2CC2)nn1
CC(C)(C)c1cc(NC(=O)Cn2cc(nn2)-c2ccc(nc2)-n2ccnc2)n(n1)-c1cccnc1
FC(F)(F)Oc1ccc(NC(=O)N(Cc2cccc(c2)-c2nccs2)C2CC2)cc1
FC(F)(F)Oc1ccc(NC(=O)NCc2cccc(c2)-c2nccs2)cc1
CCOc1cccc(c1)-c1nccc2n(CCOc3ccc(OC(F)(F)F)cc3)c(cc12)C(O)=O
OC(=O)c1cc2cnccc2n1CCOc1ccc(OC(F)(F)F)cc1
OC(=O)c1cc2cc(ccc2n1CCOc1ccc(OC(F)(F)F)cc1)C#N
OC(=O)c1cc2cc(ccc2n1CCOc1ccc(OC(F)(F)F)cc1)-c1cc[nH]n1
OC(=O)c1cc2c(nccc2n1Cc1noc(n1)-c1ccccc1)-c1cccc2ccccc12
CCOc1cccc(c1)-c1nccc2n(CCOc3ccc(Cl)cc3)c(cc12)C(O)=O
CCOc1cccc(c1)-c1nccc2n(CCOc3ccccc3)c(cc12)C(O)=O
C[C@@]12[C@@H]([C@@H](C[C@@H](O1)n3c4ccccc4c5c3c6n2c7ccccc7c6c8c5C(=O)NC8)NC)OC
C[C@@]12[C@](C[C@@H](O1)n3c4ccccc4c5c3c6n2c7ccccc7c6c8c5C(=O)NC8)(CO)O
C[C@@]12[C@@H]([C@@H](C[C@@H](O1)n3c4ccccc4c5c3c6n2c7ccccc7c6c8c5C(=O)NC8)N(C)C(=O)c9ccccc9)OC
CN1CCN(CC1)CC(=O)N(C)c2ccc(cc2)N/C(=C\3/c4ccc(cc4NC3=O)C(=O)OC)/c5ccccc5
CCSCc1ccc2n3[C@H]4C[C@](O)(C(=O)OC)[C@](C)(O4)n4c5ccccc5c5c6CNC(=O)c6c(c2c1)c3c45
COCc1ccc2n3[C@H]4C[C@](O)(C(=O)OC)[C@](C)(O4)n4c5ccc(COC)cc5c5c6CNC(=O)c6c(c2c1)c3c45
CCSCc1ccc2n3[C@H]4C[C@](O)(C(=O)OC)[C@](C)(O4)n4c5ccc(CSCC)cc5c5c6CNC(=O)c6c(c2c1)c3c45 |r|
COC(=O)[C@@]1(O)C[C@H]2O[C@]1(C)n1c3ccc(CSC(C)C)cc3c3c4CNC(=O)c4c4c5cc(CSC(C)C)ccc5n2c4c13
CCSCc1ccc2n3c4c(c5CNC(=O)c5c5c6ccccc6n([C@H]6C[C@](O)(C(=O)OC)[C@]3(C)O6)c45)c2c1
CCOCc1ccc2n3[C@H]4C[C@](O)(C(=O)OC)[C@](C)(O4)n4c5ccc(COCC)cc5c5c6CNC(=O)c6c(c2c1)c3c45
COC(=O)[C@@]1(O)C[C@H]2O[C@]1(C)n1c3ccc(CSCC=C)cc3c3c4CNC(=O)c4c4c5cc(CSCC=C)ccc5n2c4c13
CCCSCc1ccc2n3[C@H]4C[C@](O)(C(=O)OC)[C@](C)(O4)n4c5ccc(CSCCC)cc5c5c6CNC(=O)c6c(c2c1)c3c45
CCCCSCc1ccc2n3[C@H]4C[C@](O)(C(=O)OC)[C@](C)(O4)n4c5ccc(CSCCCC)cc5c5c6CNC(=O)c6c(c2c1)c3c45
COC(=O)[C@@]1(O)C[C@H]2O[C@]1(C)n1c3ccc(CSCCN(C)C)cc3c3c4CNC(=O)c4c4c5cc(CSCCN(C)C)ccc5n2c4c13
NC(=O)c1cc([nH]c1-c1ccccc1)-c1ccnc(N)n1
CC(C)OCc1ccc2n(CCCO)c3c4Cc5ccccc5-c4c4C(=O)NCc4c3c2c1
c1cc2c(c(c1)F)c3nc(nn3c(n2)Cc4ccc5c(c4)OCO5)N
Nc1nc2c3ccc(N)cc3nc(Cc3ccc4OCOc4c3)n2n1
OCCCNc1ccc2c3ncnn3c(nc2c1)-c1ccc2OCOc2c1
c1cc2c(cc1Cc3nc4cc(ccc4c5n3nc(n5)N)NCCO)OCO2
CN1CCN(CC1)c1cc(F)c2c3nc(N)nn3c(Cc3ccc4OCOc4c3)nc2c1
CCNC(=O)Nc1ccc2ncc(cc2n1)-c1ccc(OC)cc1
CCNC(=O)Nc1ccc2ncc(cc2n1)-c1ccc(OC)c(OC)c1
COc1ccc(cc1OC)-c1cnc2ccc(NC(=O)NC(C)(C)C)nc2c1
COc1cc(ccc1O)-c1cnc2ccc(NC(=O)NC(C)(C)C)nc2c1
Cn1cc(cn1)-c1cnc2ccc(NC(=O)NC(C)(C)C)nc2c1
Cn1cc(cn1)-c1cnc2ccc(NC(=O)Nc3ccccc3)nc2c1
Cn1cc(cn1)-c1cnc2ccc(NC(=O)NCc3ccccc3)nc2c1
Cn1cc(cn1)-c1cnc2ccc(NC(=O)NCCc3ccccc3)nc2c1
CCCCNc1ncc2c(cn([C@H]3CC[C@H](O)CC3)c2n1)-c1ccc(CN2CCN(C)CC2)cc1 |r,wU:12.11,wD:15.15,(14.5,-10.38,;14.49,-11.92,;15.83,-12.69,;17.16,-11.92,;18.49,-12.69,;19.83,-11.92,;19.83,-10.38,;21.16,-9.61,;22.49,-10.37,;23.97,-9.89,;24.88,-11.15,;23.97,-12.4,;24.44,-13.87,;25.95,-14.19,;26.42,-15.66,;25.39,-16.8,;25.86,-18.27,;23.88,-16.47,;23.41,-15.02,;22.49,-11.92,;21.16,-12.69,;24.45,-8.43,;25.96,-8.11,;26.43,-6.65,;25.41,-5.5,;25.89,-4.03,;27.4,-3.74,;28.41,-4.9,;29.91,-4.6,;30.41,-3.14,;31.92,-2.84,;29.4,-1.99,;27.88,-2.28,;23.9,-5.82,;23.42,-7.29,)|
[#6]-[#7](-[#6])-[#6]-[#6]\[#6]=[#6]-1/c2ccccc2-[#6]-[#6]-c2ccccc-12
CC1(C)O[C@H](C[C@]1(O)CO)n1c2ccccc2c2c3C(=O)NCc3c3c4ccccc4[nH]c3c12
CC1(C)O[C@H](C[C@@]1(O)CO)n1c2ccccc2c2c3C(=O)NCc3c3c4ccccc4[nH]c3c12
COc1ccc2NC(=O)[C@@]3(C[C@H]3c3ccc4c(\C=C\c5ccc(CN6C[C@H](C)O[C@H](C)C6)cc5)n[nH]c4c3)c2c1 |r|
NS(=O)(=O)c1ccc(cc1)-c1cnc2ccc(NCc3cccc(F)c3)nn12
Fc1cccc(CNc2ccc3ncc(-c4ccc(NC(=O)C5CCOCC5)cc4)n3n2)c1
OCc1ccc(cc1)-c1cnc2ccc(NCc3cccc(F)c3)nn12
COc1ccccc1CNc1ccc2ncc(-c3ccc(cc3)C#N)n2n1
Fc1cccc(CNc2ccc3ncc(-c4ccc(cc4)C#N)n3n2)c1
N#Cc1cccc(c1)-c1cnc2ccc(NCc3ccccc3)nn12
N#Cc1ccc(cc1)-c1cnc2ccc(NCc3ccccc3)nn12
OC1CCN(CC1)c1cc(ccn1)-c1cnc2ccc(nn12)N1CCC[C@@H]1c1cccc(F)c1 |r|
OC(=O)CN1CCN(CC1)c1cc(ccn1)-c1cnc2ccc(nn12)N1CCC[C@@H]1c1cccc(F)c1 |r|
Fc1cccc(c1)[C@@H]1CCCN1c1ccc2ncc(-c3ccc(cc3)C#N)n2n1 |r|
Fc1cccc(c1)C1CCCN1c1ccc2ncc(-c3ccc(cc3)C#N)n2n1
Fc1cccc(c1)C1COCCN1c1ccc2ncc(-c3ccc(cc3)C#N)n2n1
Fc1cccc(c1)C1CCCCN1c1ccc2ncc(-c3ccc(cc3)C#N)n2n1
CN(Cc1ccccc1)c1ccc2ncc(-c3ccc(cc3)C#N)n2n1
OC1CCN(CC1)c1cccc(n1)-c1cnc2ccc(nn12)N1CCC[C@@H]1c1cccc(F)c1 |r|
Fc1cccc(c1)[C@H]1CCCN1c1ccc2ncc(-c3ccccn3)n2n1 |r|
Fc1cccc(c1)[C@H]1CCCN1c1ccc2ncc(-c3ccc(cc3)C#N)n2n1 |r|
COc1cc(cnc1Cl)N1CCc2nc(NC(=O)NCCc3cn(CC(F)F)cn3)sc2C1
COc1cncc(n1)N1CCc2nc(NC(=O)NCCc3cn(CC(F)F)cn3)sc2C1
NC(=O)c1cnc2[nH]ccc2c1N[C@@H]1CCN(C[C@@H]1F)c1ccc(cn1)C#N |r|
CCOc1cccc2n(C)cc(C=c3c(=O)[nH][nH]\c3=c3/snnc3=C)c12 |w:12.11|
c1c(cc(c2c1CN(C2=O)C3CCN(CC3)C4CCC(CC4)(F)F)C(=O)N)F
Cc1ccc(Sc2cnc(Nc3ccccn3)s2)cc1C(=O)NCCO
C[C@@H](N)C(=O)N1CCN(CC1)C(=O)c1cc(Sc2cnc(Nc3cccc(Br)n3)s2)ccc1C
Cc1ccc(Sc2cnc(Nc3ccccn3)s2)cc1C(N)=O
Cc1ccc(Sc2cnc(Nc3ccccn3)s2)cc1C(=O)NCc1ccccc1
CC(=O)N1CCN(CC1)C(=O)c1cc(Sc2cnc(Nc3cccc(Br)n3)s2)ccc1C
Cc1ccc(Sc2cnc(Nc3cccc(Br)n3)s2)cc1C(=O)N1CCN(CC(N)=O)CC1
CC(=O)N1CCN(CC1)C(=O)c1cccc(Sc2cnc(Nc3cccc(C)n3)s2)c1
Cc1ccc(Sc2cnc(Nc3ccccn3)s2)cc1C(=O)NCC#C
CC(=O)N1CCN(CC1)C(=O)c1cccc(Sc2cnc(Nc3ccc(Br)cn3)s2)c1
CC(=O)N1CCCN(CC1)C(=O)c1cc(Sc2cnc(Nc3ccccn3)s2)ccc1C
C[C@H](N)C(=O)N1CCN(CC1)C(=O)c1cc(Sc2cnc(Nc3cccc(Br)n3)s2)ccc1C
COC(=O)N1CCN(CC1)C(=O)c1cc(Sc2cnc(Nc3ccccn3)s2)ccc1C
CC(=O)Nc1ncc(Sc2ccc(C)c(c2)C(=O)N2CCN(CC2)C(C)=O)s1
Cc1ccc(Sc2cnc(Nc3ccccn3)s2)cc1C(=O)NCC#N
CC(=O)N1CCN(CC1)C(=O)c1cc(Sc2cnc(N)s2)ccc1C
CCNC(=O)c1cc(Sc2cnc(Nc3ccccn3)s2)ccc1C
CC(=O)N1CCN(Cc2cc(Sc3cnc(Nc4ccccn4)s3)ccc2C)CC1
CC(=O)N1CCN(CC1)C(=O)c1ccccc1Sc1cnc(Nc2cccc(Br)n2)s1
Cc1ccc(Sc2cnc(Nc3ccccn3)s2)cc1C(=O)N1CCN(CC1)S(C)(=O)=O
CC(=O)N1CCN(CC1)C(=O)c1cc(Sc2cnc(Nc3ccccn3)s2)ccc1C
CN(CC#N)C(=O)c1cc(Sc2cnc(Nc3cccc(Br)n3)s2)ccc1C
CN(CCC#N)C(=O)c1cc(Sc2cnc(Nc3cccc(Br)n3)s2)ccc1C
CC(C)NC(=O)c1cc(Sc2cnc(Nc3ccccn3)s2)ccc1C
Cc1ccc(Sc2cnc(Nc3ccccn3)s2)cc1NC(=O)CC#N
Cc1ccc(Sc2cnc(Nc3ccccn3)s2)cc1C(=O)NCCC#N
CC(=O)N1CCN(CC1)C(=O)c1cccc(Sc2cnc(Nc3ccccn3)s2)c1
CC(=O)NCCNC(=O)c1cc(Sc2cnc(Nc3ccccn3)s2)ccc1C
CC(=O)N1CCN(CC1)C(=O)c1ccc(Sc2cnc(Nc3cccc(Br)n3)s2)cc1
CC(=O)N1CCN(CC1)C(=O)c1cccc(Sc2cnc(Nc3cccc(Br)n3)s2)c1
CNCCN(C)C(=O)c1cc(Sc2cnc(Nc3cccc(Br)n3)s2)ccc1C
Cc1ccc(Sc2cnc(Nc3ccccn3)s2)cc1C(=O)N1CCNCC1
Cc1ccc(Sc2cnc(Nc3cccc(Br)n3)s2)cc1C(=O)NCCC#N
CCC(=O)N1CCN(CC1)C(=O)c1cc(Sc2cnc(Nc3cccc(Br)n3)s2)ccc1C
Cc1ccc(Sc2cnc(Nc3cccc(Br)n3)s2)cc1C(=O)N1CCN(CC1)C(=O)CN
CNCCNC(=O)c1cc(Sc2cnc(Nc3ccccn3)s2)ccc1C
CCN1CCN(CC1)C(=O)c1cc(Sc2cnc(Nc3cccc(Br)n3)s2)ccc1C
CC1CCN(CC1)c1cc(ccc1NC(=O)c1cc(c[nH]1)C#N)N1CCN(C)CC1
c1cc(ccc1CC(=O)NC(=O)Nc2ccc(c(c2)F)Oc3c4c(ccn4ncn3)CN5CCC(CC5)N)F
c1cnc(cc1C#N)Nc2cc(n(n2)C3CCCC3)C4CCN(CC4)C5COC5
O=C1c2ccccc2-c2c1oc1ccccc1c2=O
COc1ccc-2c(c1)C(=O)c1c-2c(=O)c2ccccc2n1Cc1ccccc1
CCOC(=O)n1c2C(=O)c3ccccc3-c2c(=O)c2ccccc12
O=C1c2ccccc2-c2c1n(Cc1ccccc1)c1ccccc1c2=O
COc1cccc2C(=O)c3c(-c12)c(=O)c1ccccc1n3C
COc1ccc2C(=O)c3c(-c2c1)c(=O)c1ccccc1n3C
COc1ccc-2c(c1)C(=O)c1c-2c(=O)c2ccccc2n1C
Cn1c2C(=O)c3c(cccc3O)-c2c(=O)c2ccccc12
Cc1ccc-2c(c1)C(=O)c1c-2c(=O)c2ccccc2n1C
Cc1cccc-2c1C(=O)c1c-2c(=O)c2ccccc2n1C
Cn1c2C(=O)c3ccccc3-c2c(=O)c2ccc(Cl)cc12
Cn1c2C(=O)c3ccccc3-c2c(=O)c2ccccc12
Cn1c2C(=O)c3ccccc3-c2c(=O)c2ccc(cc12)C(F)(F)F
Cn1c2nc(Nc3ccc4[nH]ccc4c3)ncc2cc(c1=O)S(=O)(=O)c1ccc(F)cc1F
O=C(CCc1ccco1)Nc1nc(cs1)-c1ccccc1
C[C@@H]1C[C@H]1C(=O)N1CCN(C[C@H]1C)c1cnc(C#N)c(n1)-c1cnn(C)c1 |r|
O=C(Nc1ccc(CN2CCN(CC2)c2ccccc2)cc1)c1n[nH]c2ccccc12
C[C@@H](N1c2cc(ccc2C(=O)NC1(C)C)-n1c2cccnc2[nH]c1=O)c1ccccc1 |r|
CN1C(=O)COc2c1cnc1ccc(Sc3nnc4c(F)cc(cn34)-c3cnn(C)c3)cc21
c1cc(ccc1NC(=O)C2(CC2)C(=O)Nc3cc(c(cc3F)Oc4ccnc(c4)NC(=O)C5CC5)F)F
COCc1ccc2cccc(NC(=O)Nc3c(C)c(nn3-c3ccccc3)-c3cnn(C)c3)c2c1
Cc1c(NC(=O)Nc2sc(nc2-c2ccccc2)C(F)(F)F)n(nc1-c1cnn(C)c1)-c1ccccc1
Cc1c(NC(=O)Nc2cc(nn2-c2ccccc2)C(F)(F)F)n(nc1-c1cnn(C)c1)-c1ccccc1
Cn1c2cc(nn2c(=O)c2cc(NC(=O)c3ccccc3)ccc12)C(O)=O
Cc1cc2nc3c(nc(=O)[nH]c3=O)n(C)c2cc1C=O
OC(=O)c1ccc(Nc2cc(N3CCN(CC3)C3CCCCC3)c3noc4-c5ccccc5C(=O)c2c34)cc1
COCCCc1cc(Cl)c(Cl)cc1NC(=O)Nc1c(C)c(nn1-c1ccccc1)-c1cnn(C)c1
Cc1ccc(Cl)cc1N1CCN(CCCNC(=O)c2ccc3N4CCCCC4C(=O)Nc3c2)CC1
Oc1ccc(\C=N\NC(=O)c2ccccc2O)c(O)c1O
Cn1cc(\C=C2/C(=O)Nc3cccnc23)c2ccccc12
COc1ccccc1\C=C\C(=O)Nc1nc(N)n(n1)-c1ccccc1
CC1(C)C[C@@H](N(C1)c1ccn2ncc(NC(=O)c3cnccn3)c2n1)c1cc(F)ccc1F |r|
COc1ncc(cc1NC(=O)Nc1cc(Cl)cc(Cl)c1)C(=O)C1CC(C(C)C)c2ncncc12
Oc1ccc(\C=N\NC(=O)c2ccccc2O)c(O)c1
Oc1ccc(Nc2nc(nc3ccccc23)-c2ccccc2O)cc1
Oc1ccc(\C=N\NC(=O)c2ccccc2O)cc1O
Nc1ccc(Cc2cccc(NC(=O)N3CCN(C3=O)c3ccccc3)c2)cn1
CCc1ncc(cc1NC(=O)Cc1ccc(cc1)C(F)(F)F)C(=O)C1CC([C@@H](C)CO)c2ncncc12 |r|
C[C@H](Nc1nc(Nc2cc(C)n[nH]2)cnc1C#N)c1ncc(F)cn1 |r|
C[C@H](Nc1nc(Nc2cc(C)n[nH]2)c(C)nc1C#N)c1ncc(F)cn1 |r|
C[C@H](Nc1nc(Nc2cc(C)n[nH]2)c(C)nc1C#N)c1ccc(F)cn1 |r|
C[C@H](Nc1nc(Nc2cc(C)n[nH]2)cnc1C#N)c1ccc(F)cn1 |r|
NCCn1cc(-c2cc(-c3cc4ccccc4s3)c3[nH]ncc3c2)c2nc(N)ncc12
CC1(C)C(=O)N([C@H]2CCc3c2cccc3O)c2nc(Nc3ccccc3)ncc12 |r|
Cn1nc(C(N)=O)c2CCc3cnc(NC4CCN(CC4)C(=O)c4ccccc4)nc3-c12
CNC(=O)c1nn(C)c-2c1CCc1cnc(NC3CCN(CC3)C(=O)C3CCN(CC3)S(C)(=O)=O)nc-21
CC(=O)N1CCC(CC1)Nc1ncc2CCc3c(nn(C)c3-c2n1)C(N)=O
O=C(Cc1ccccc1)Nc1cccc(c1)-c1nc2sccn2c1-c1ccnc(Nc2cccc(c2)N2CCOCC2)n1
Oc1ccc2[nH]c(c(N=[OH+])c2c1)-[c-]1c2cc(ccc2[nH]c1=O)[N+]([O-])=O |(-8.68,.59,;-7.35,-.18,;-7.35,-1.72,;-6.01,-2.49,;-4.68,-1.72,;-3.21,-2.2,;-2.29,-.95,;-3.21,.31,;-2.73,1.77,;-1.22,2.09,;-4.68,-.17,;-6.02,.59,;-.75,-.95,;.15,.3,;-.18,1.8,;.96,2.83,;2.43,2.36,;2.75,.85,;1.61,-.18,;1.61,-1.72,;.15,-2.19,;-.33,-3.66,;.63,4.33,;1.77,5.37,;-.84,4.8,)|
Fc1ccc(NC(=O)c2cccnc2Nc2ccc(Oc3ccnc4[nH]ccc34)c(F)c2)c(F)c1
COc1ccc(cc1Nc1ncc2CCc3c(nn(C)c3-c2n1)C(N)=O)N1CCN(C)CC1
[O-][N+](=O)c1ccc(NC(=O)CCc2cn(Cc3ccc(Cl)cc3)c3ccccc23)cc1
Clc1ccc(Cn2cc(CCC(=O)Nc3ccncc3)c3ccccc23)cc1
CN1CCN(CC1)CCCOc2cc3c(cc2OC)c(c(cn3)C#N)Nc4cc(c(cc4Cl)Cl)OC
CC(C)(C)c1cc(NC(=O)Nc2ccc(cc2)-c2cn3c(n2)sc2cc(OCCN4CCOCC4)ccc32)no1
CO[C@@H]1[C@@H](C[C@H]2O[C@]1(C)n1c3ccccc3c3c4[C@H](O)NC(=O)c4c4c5ccccc5n2c4c13)N(C)C(=O)c1ccccc1 |r|
O=C(N[C@H](CN1CCCC1)c1ccccc1)c1cc2n[nH]c(NC(=O)c3ccc(cc3)N3CCOCC3)c2s1 |r|
CN1CCN(CC1)c1ccc(OC(F)(F)F)c(Nc2ncc3CCc4c(nn(CCO)c4-c3n2)C(N)=O)c1
C[C@H](Nc1nc(Nc2cc(C)n[nH]2)c(F)cc1C#N)c1ccc(F)cn1 |r|
Cc1cnc2c(NCCN)nc3ccc(C)cc3n12
CC(C)S(=O)(=O)c1ccccc1Nc2c(cnc(n2)Nc3ccc(cc3OC)N4CCC(CC4)N5CCN(CC5)C)Cl
COc1cc(Oc2ccnc3cc(OC)c(OC)cc23)ccc1NC(=O)NC(C)c1nccs1
Cc1n[nH]c2ccc(cc12)-c1cncc(OC[C@@H](N)Cc2ccccc2)c1 |r|
CN(c1ccc2c(C)n(C)nc2c1)c1ccnc(Nc2ccc(C)c(c2)S(N)(=O)=O)n1
COc1ccc(c(c1C(=O)c2cnc(nc2N)NC3CCN(CC3)S(=O)(=O)C)F)F
Cn1cnc2c1cc(c(c2F)Nc3ccc(cc3Cl)Br)C(=O)NOCCO
Cc1cn(cn1)-c1cc(NC(=O)c2ccc(C)c(Nc3nccc(n3)-c3cccnc3)c2)cc(c1)C(F)(F)F
Oc1cccc(c1)-c1nc(N2CCOCC2)c2oc3ncccc3c2n1
CCCS(=O)(=O)Nc1ccc(F)c(C(=O)c2c[nH]c3ncc(Cl)cc23)c1F
COc1cc2c(Oc3ccc4[nH]c(C)cc4c3F)ncnc2cc1OCCCN1CCCC1
COc1cc2c(cc1OCCCN3CCOCC3)c(ncn2)Nc4ccc(c(c4)Cl)F
OCCn1cc(c(n1)-c1ccncc1)-c1ccc2C(CCc2c1)N=O
CN(C)C/C=C/C(=O)Nc1cc2c(cc1O[C@H]3CCOC3)ncnc2Nc4ccc(c(c4)Cl)F
C=CC(=O)Nc1cc2c(cc1OCCCN3CCOCC3)ncnc2Nc4ccc(c(c4)Cl)F
CS(=O)(=O)N1CCN(Cc2cc3nc(nc(N4CCOCC4)c3s2)-c2cccc3[nH]ncc23)CC1
Cn1cc(cn1)-c1ccc2nnc(Sc3ccc4ncccc4c3)n2n1
Cn1c(Nc2ccc(cc2)C(F)(F)F)nc2cc(Oc3ccnc(c3)-c3ncc([nH]3)C(F)(F)F)ccc12
c1c[nH]c2c1c(ncn2)c3cnn(c3)[C@H](CC#N)C4CCCC4
Cn1cc(C2=C(C(=O)NC2=O)c2cn(C3CCN(Cc4ccccn4)CC3)c3ccccc23)c2ccccc12 |t:4|
CN(C)C[C@@H]1CCn2cc(C3=C(C(=O)NC3=O)c3cn(CCO1)c1ccccc31)c1ccccc21 |r,t:10|
C[C@@H](Oc1cc(sc1C(N)=O)-n1cnc2ccc(CN3CCN(C)CC3)cc12)c1ccccc1C(F)(F)F |r|
CC1(CNc2c1ccc(c2)NC(=O)c3cccnc3NCc4ccncc4)C
CC(C)n1nc(-c2cc3cc(O)ccc3[nH]2)c2c(N)ncnc12
COc1c(Cl)cc2c3ccncc3[nH]c2c1NC(=O)c1cccnc1C
CC(C)(C)c1cnc(o1)CSc2cnc(s2)NC(=O)C3CCNCC3
CCOc1cc2ncc(C#N)c(Nc3ccc(OCc4ccccn4)c(Cl)c3)c2cc1NC(=O)\C=C\CN(C)C
CN1c2c(cnc(n2)Nc3cccc(c3)SC)C=C(C1=O)c4c(cccc4Cl)Cl
Cc1cccc(c1NC(=O)c2cnc(s2)Nc3cc(nc(n3)C)N4CCN(CC4)CCO)Cl
Nc1nc(N)c2nc(-c3cccc(O)c3)c(nc2n1)-c1cccc(O)c1
COCCOc1cc2c(cc1OCCOC)ncnc2Nc3cccc(c3)C#C
Cc1cnc(nc1Nc2cccc(c2)S(=O)(=O)NC(C)(C)C)Nc3ccc(cc3)OCCN4CCCC4
CN(C)CC(=O)N1CCC(CC1)c1ccc(NC(=O)c2ncc([nH]2)C#N)c(c1)C1=CCCCC1 |t:31|
C[C@@H](O)COc1cn2ncnc(Oc3ccc4[nH]c(C)cc4c3F)c2c1C
CS(=O)c1ccc(cc1)-c1nc(c([nH]1)-c1ccc(F)cc1)-c1ccncc1
O=C(N1CCNCC1)c1ccc(\C=C\c2n[nH]c3ccccc23)cc1
CCn1c(nc2c(ncc(OC[C@H]3CCCNC3)c12)C#CC(C)(C)O)-c1nonc1N |r|
OC(=O)c1ccc(Nc2ncc3CN=C(c4cc(Cl)ccc4-c3n2)c2c(F)cccc2F)cc1 |c:13|
C[C@@H](c1ccc(cn1)F)Nc2ncc(c(n2)Nc3cc(n[nH]3)OC(C)C)Cl
c1cc(c(c(c1)Cl)C2=C3C=CC(=NN3C=NC2=O)Sc4ccc(cc4F)F)Cl
CC1(C(=O)Nc2c(ccc(n2)Nc3c(cnc(n3)Nc4cc(c(c(c4)OC)OC)OC)F)O1)C
CNC(=O)c1c(F)cccc1Nc1nc(Nc2cc3N(CCc3cc2OC)C(=O)CN(C)C)nc2[nH]ccc12
CN1CCN(Cc2ccc(cc2)C(=O)Nc2ccc(C)c(Nc3nccc(n3)-c3cccnc3)c2)CC1
Clc1ccc(Nc2nnc(Cc3ccncc3)c3ccccc23)cc1
CN1CCC(CC1)COc2cc3c(cc2OC)c(ncn3)Nc4ccc(cc4F)Br
C[C@@H]1CCN(C[C@@H]1N(C)c1ncnc2[nH]ccc12)C(=O)CC#N |r|
CS(=O)(=O)CCNCc1ccc(o1)-c1ccc2ncnc(Nc3ccc(OCc4cccc(F)c4)c(Cl)c3)c2c1
CN1CC[C@@H]([C@H](O)C1)c1c(O)cc(O)c2c1oc(cc2=O)-c1ccccc1Cl |r|
Clc1cccc(Cl)c1C(=O)Nc1cn[nH]c1C(=O)NC1CCNCC1
COc1cc2c(Oc3ccc(NC(=O)C4(CC4)C(=O)NC4=CCC(F)C=C4)cc3F)ccnc2cc1OCCCN1CCOCC1 |c:26,t:21|
CC[C@H]1N(C2CCCC2)c2nc(Nc3ccc(cc3OC)C(=O)NC3CCN(C)CC3)ncc2N(C)C1=O |r|
CNC(=O)c1ccccc1Sc2ccc3c(c2)[nH]nc3/C=C/c4ccccn4
CCN(CCCOc1ccc2c(c1)ncnc2Nc3cc(n[nH]3)CC(=O)Nc4cccc(c4)F)CCO
Cc1ccc(cc1Nc2nc(cs2)c3cccnc3)NC(=O)c4ccc(cc4)CN5CCN(CC5)C
Fc1ccc(C(=O)NOCC2CC2)c(Nc2ccc(I)cc2Cl)c1F
Cc1[nH]c(\C=C2/C(=O)Nc3ccc(cc23)S(=O)(=O)Cc2c(Cl)cccc2Cl)c(C)c1C(=O)N1CCC[C@@H]1CN1CCCC1 |r|
Cc1nnc([nH]1)-c1ccc(C)c(c1)-c1ccc2c(NC(=O)C22CCOCC2)c1
Cn1cc(cn1)-c1ccc2nnc(Cc3cccc4c3cc[nH]c4=O)n2n1
O=c1[nH]ccc2c(Cc3nnc4ccc(nn34)-c3ccccc3)cccc12
CC(C)(C)c1cc(c(s1)NC(=O)Nc2cccc(c2Cl)Cl)C(=O)N3CCC(=O)N(CC3)CCN(C)C
C[C@@H]1CCC(CN1)N1CC[C@@]2(C1)CN(C(=O)c1cc3ccc(F)cc3[nH]1)c1ccccc21 |r|
CN1CCN(CC1)c1ccc(OC(F)(F)F)c(Nc2nccc(n2)-c2cc3c(CCNC3=O)n2C)c1
CN1CCN(CC1)c1ccc(OC(F)(F)F)c(Nc2nccc(n2)-c2cc(cn2C)C(N)=O)c1
CC(C)n1cc(C(=O)c2cncc(N[C@@H]3CCN(C=O)[C@@H]3c3ccc(F)cc3)n2)c2c(N)ncnc12 |r|
CC(C)n1cc(C(=O)c2cncc(N[C@@H]3CCN([C@@H]3c3ccc(F)cc3)C(C)=O)n2)c2c(N)ncnc12 |r|
CC(C)n1cc(C(=O)c2cncc(N[C@@H]3CCN([C@@H]3c3ccccc3)C(C)=O)n2)c2c(N)ncnc12 |r|
CC1(C)OCC(=O)Nc2cc(Nc3nc(NCC(F)(F)F)c4occc4n3)ccc12
FC(F)(F)CNc1nc(Nc2ccc3cn[nH]c3c2)nc2ccoc12
CCCNC(=O)c1ccc(Nc2nc(NCC(F)(F)F)c3cc[nH]c3n2)cc1
FC(F)(F)CNc1nc(Nc2ccc(N3CCOCC3)c(Cl)c2)nc2ccoc12
Cc1c2ccc(cc2[nH]n1)Nc3nc4ccoc4c(n3)NC5CC5
Oc1ccc2\C(CCc2c1)=C1/C(=O)Nc2ccccc12
O=C1Nc2ccc3ncsc3c2C1C=Nc1ccc(cc1)S(=O)(=O)Nc1ccccn1 |w:13.15|
NS(=O)(=O)c1cccc(c1)N=CC1C(=O)Nc2ccccc12 |w:10.10|
COc1ccccc1-c1cc(\C=C2/C(=O)Nc3ncc(Br)cc23)cc(Br)c1O
O=C1Nc2ccccc2C1C=Nc1ccc2[nH]c(=O)[nH]c2c1 |w:10.11|
OC1Nc2ccc(I)cc2C1=Cc1cc(Br)c(O)c(Br)c1
Brc1cnc2NC(=O)\C(=C/c3cccc(Oc4ccccc4)c3)c2c1
Cn1cc(\C=C2/C(=O)Nc3ncccc23)c2ccccc12
CS(=O)(=O)Nc1ccc(cc1)N=CC1C(=O)Nc2ccccc12 |w:11.11|
O=C1Nc2ccccc2C1C=Nc1ccc(cc1)-n1cncn1 |w:10.11|
O=C(Cn1c(cc2ccccc12)-c1ncco1)NCc1ccccn1
Fc1ccc2cc(-c3ccccc3)n(CC(=O)NCc3ccccn3)c2c1
O=C(Cn1c(cc2ccccc12)-c1cccs1)NCc1c[nH]cn1
O=C(Cn1c(cc2ccccc12)-c1cccs1)NCc1ccccc1
O=C(Cn1c(cc2ccccc12)-c1cccs1)Nc1ccccn1
Fc1cccc2n(CC(=O)NCc3ccccn3)c(cc12)-c1ccccc1
O=C(Cn1c(cc2ccccc12)-c1cccs1)NCc1ncc[nH]1
O=C(Cn1c(cc2ccccc12)-c1cncs1)NCc1ccccn1
O=C(Cn1c(cc2ccccc12)-c1nccs1)NCc1ccccn1
O=C(Cn1c(cc2ccccc12)-c1ccsn1)NCc1ccccn1
O=C(Cn1c(cc2ccccc12)-c1cccs1)NCc1cnccn1
O=C(Cn1c(cc2ccccc12)-c1ccccc1)NCc1ccccn1
O=C(Cn1c(cc2ccncc12)-c1ccccc1)NCc1ccccn1
O=C(NCCc1ccccn1)n1c(cc2ccccc12)-c1cccs1
O=C(NCCn1c(cc2ccccc12)-c1cccs1)c1ccccn1
Cn1ccnc1CNC(=O)Cn1c(cc2ccccc12)-c1cccs1
O=C(Cn1c(cc2ccccc12)-c1ccns1)NCc1ccccn1
Fc1ccc2n(CC(=O)NCc3ccccn3)c(cc2c1)-c1ccccc1
O=C(Cn1c(cc2ccccc12)-c1cccs1)NCc1nc2ccccc2[nH]1
O=C(Cn1c(cc2ccccc12)-c1cccs1)NCc1cn2ccccc2n1
O=S(=O)(NCCn1c(cc2ccccc12)-c1cccs1)c1ccccn1
O=C(Cn1c(cc2ccccc12)-c1cccs1)NCc1ncco1
Fc1cccc2cc(-c3ccccc3)n(CC(=O)NCc3ccccn3)c12
O=C(Cn1c(cc2ccccc12)-c1cccs1)NCc1cccnc1
Cc1ccc(o1)-c1cc2ccccc2n1CC(=O)NCc1ccccn1
O=C(Cn1c(cc2ccccc12)-c1cccs1)NCc1ccncc1
O=C(Cn1c(cc2ncccc12)-c1ccccc1)NCc1ccccn1
O=C(Cn1c(cc2ccccc12)-c1cccs1)NCc1nccs1
O=C(Cn1c(cc2ccccc12)-c1cccs1)NCc1ncccn1
O=C(Cn1c(cc2ccccc12)-c1cccs1)NCc1c[nH]c(n1)-c1ccccc1
O=C(Cn1c(cc2cnccc12)-c1ccccc1)NCc1ccccn1
O=C(Cn1c(cc2ccccc12)-c1cccnc1)NCc1ccccn1
CN(Cc1ccccn1)C(=O)Cn1c(cc2ccccc12)-c1cccs1
O=C(NCc1ccccn1)n1c(cc2ccccc12)-c1cccs1
O=C(Cn1c(cc2ccccc12)-c1ccccn1)NCc1ccccn1
O=C(Cn1c(cc2ccccc12)-c1ccncc1)NCc1ccccn1
Fc1ccc2n(CC(=O)NCc3nc4ccccc4[nH]3)c(cc2c1)-c1ncco1
C(Cn1c(cc2ccccc12)-c1cccs1)NCc1ccccn1
c1ccc2c(c1)cc(n2CC(=O)NCc3ccccn3)c4cccs4
O=C(Cn1c(cc2ccccc12)-c1ncco1)NCc1nc2ccccc2[nH]1
Cc1ccc(s1)-c1cc2ccccc2n1CC(=O)NCc1ccccn1
O=C(Cn1c(cc2cccnc12)-c1ccccc1)NCc1ccccn1
O=C(Cn1c(cc2ccccc12)-c1cccs1)NCc1ncc([nH]1)-c1ccccc1
CN(C)C(=O)c1cc2cnc(Nc3ccc(NC(=O)CCCCCCC(=O)NO)cc3)nc2n1C1CCCC1
Clc1cc2NC(=O)Nc3cnc(C#N)c(OCCCCOc2cc1NCc1cncs1)n3
CN1CCN(CC1)c1ccc(Nc2ncc3c(n2)n(cc(C(N)=O)c3=O)-c2ccc3CCCc3c2)cc1
CN1CCN(Cc2ccc(Nc3ncc4c(n3)n(cc(C(N)=O)c4=O)-c3ccc4CCCc4c3)cc2)CC1
CCNC(=O)O[C@@H](C)[C@H]1c2ccccc2-c2c1c1[nH]c3ccccc3c1c1CNC(=O)c21
C[C@@H](OC(=O)NCc1ccccc1)[C@H]1c2ccccc2-c2c1c1[nH]c3ccccc3c1c1CNC(=O)c21
C[C@H](OC(=O)NCc1ccccc1)[C@H]1c2ccccc2-c2c1c1[nH]c3ccccc3c1c1CNC(=O)c21
C[C@@H](OC(=O)Nc1ccccc1)[C@H]1c2ccccc2-c2c1c1[nH]c3ccccc3c1c1CNC(=O)c21
C[C@H](OC(=O)Nc1ccccc1)[C@H]1c2ccccc2-c2c1c1[nH]c3ccccc3c1c1CNC(=O)c21
CCOC(=O)CNC(=O)O[C@H](C)[C@H]1c2ccccc2-c2c1c1[nH]c3ccccc3c1c1CNC(=O)c21
CCOC(=O)CNC(=O)O[C@@H](C)[C@H]1c2ccccc2-c2c1c1[nH]c3ccccc3c1c1CNC(=O)c21
C[C@@H](OC(=O)NCCCCl)[C@H]1c2ccccc2-c2c1c1[nH]c3ccccc3c1c1CNC(=O)c21
C[C@H](OC(=O)NCCCCl)[C@H]1c2ccccc2-c2c1c1[nH]c3ccccc3c1c1CNC(=O)c21
C[C@@H](OC(=O)NCC=C)[C@H]1c2ccccc2-c2c3C(=O)NCc3c3c([nH]c4ccccc34)c12
C[C@H](OC(=O)NCC=C)[C@H]1c2ccccc2-c2c3C(=O)NCc3c3c([nH]c4ccccc34)c12
CCNC(=O)O[C@H](C)[C@H]1c2ccccc2-c2c1c1[nH]c3ccccc3c1c1CNC(=O)c21
CN1C(=O)N(Cc2cnc(N)nc12)c1cc(NC(=O)c2cccc(c2)C(F)(F)F)ccc1C
COCC(=O)NC\C=C\c1ccc2ncnc(Nc3ccc(Oc4ccc(C)nc4)c(C)c3)c2c1
CCOc1cc2c(cc1NC(=O)/C=C/CN(C)C)c(c(cn2)C#N)Nc3ccc(c(c3)Cl)F
c1cc(c(c(c1)F)C(=O)n2c(nc(n2)Nc3ccc(cc3)S(=O)(=O)N)N)F
CC[C@H](CO)Nc1nc(NCc2ccccc2)c2ncn(C(C)C)c2n1 |r|
Oc1ccc(cc1)-c1nc(c([nH]1)-c1ccc(F)cc1)-c1ccncc1
NC(=O)c1ccc(cc1)-c1nc(c([nH]1)-c1ccc2OCOc2c1)-c1ccccn1
CCCc1cc(nc2sc(C(N)=O)c(N)c12)N1CCCC(O)C1
CCCc1cc(nc2sc(C(N)=O)c(N)c12)N1CCC(O)CC1
CCCc1cc(nc2sc(C(N)=O)c(N)c12)N1CCNCC1
CCCc1cc(nc2sc(C(N)=O)c(N)c12)N1CCC(N)CC1
CC(C)CC(=O)Nc1[nH]nc2c1CN(C(=O)C1CCN(C)CC1)C2(C)C
CC(C)(C)C(=O)N1Cc2c(NC(=O)c3cc(F)cc(F)c3)[nH]nc2C1(C)C
[H][C@@]12CN(C[C@]1([H])[C@H]2c1cc(nn1C(C)C)-c1cnc(N)c(OC(F)(F)F)c1)C1COC1 |r|
[H][C@@]12CN(C[C@]1([H])[C@H]2c1cc(nn1CC1CC1)-c1cnc(N)c(c1)C(F)(F)F)C1COC1 |r|
O=C1NCCc2[nH]c(cc12)-c1ccncc1
C[C@H](Nc1ncc(Cl)c(Nc2cc(C)n[nH]2)n1)c1ncc(F)cn1 |r|
CN(C[C@@H]1COCCO1)S(=O)(=O)Nc1ccc2ccc3ncc(cc3c(=O)c2c1)-c1cnn(C)c1 |r|
CC(C)Cn1c2ccc(Nc3ncccn3)cc2c2c3CNC(=O)c3c3-c4cn(C)nc4CCc3c12
CSc1ccccc1Nc2c3c(c(ncn3)NCC4CC4)nc(n2)N5CCNCC5
FC(F)(F)c1cccc(NC(=O)Nc2cccc(Nc3ccc4\C(=C\c5ccc[nH]5)C(=O)Nc4c3)c2)c1
CN1CCN(CC1)c1cc(cc(c1)C(F)(F)F)C(=O)Nc1cccc(Nc2ccc3\C(=C\c4[nH]c(C)c(C(O)=O)c4C)C(=O)Nc3c2)c1
Cc1cn(cn1)-c1cc(cc(c1)C(F)(F)F)C(=O)Nc1cccc(Nc2ccc3\C(=C\c4ccc[nH]4)C(=O)Nc3c2)c1
CCN(CC)CCNC(=O)c1c[nH]c(\C=C2/C(=O)Nc3cc(Nc4cccc(NC(=O)c5cc(cc(c5)C(F)(F)F)N5CCN(C)CC5)c4)ccc23)c1
Cc1cn(cn1)-c1cc(cc(c1)C(F)(F)F)C(=O)Nc1cccc(Nc2ccc3\C(=C\c4cccn4C)C(=O)Nc3c2)c1
OCCN1CCN(CC1)c1cc(cc(c1)C(F)(F)F)C(=O)Nc1cccc(Nc2ccc3\C(=C\c4ccc[nH]4)C(=O)Nc3c2)c1
OC1CCN(CC1)c1cc(cc(c1)C(F)(F)F)C(=O)Nc1cccc(Nc2ccc3\C(=C\c4ccc[nH]4)C(=O)Nc3c2)c1
CN1CCN(CC1)c1ccc(cc1C(F)(F)F)C(=O)Nc1cccc(Nc2ccc3\C(=C\c4ccc[nH]4)C(=O)Nc3c2)c1
CN1CCN(CC1)c1cc(cc(c1)C(F)(F)F)C(=O)Nc1cccc(Nc2ccc3\C(=C\c4ccc[nH]4)C(=O)Nc3c2)c1
CN1CCN(CC1)c1cc(C)cc(c1)C(=O)Nc1cccc(Nc2ccc3\C(=C\c4ccc[nH]4)C(=O)Nc3c2)c1
Cc1ccc(NC(=O)Nc2cc(ccc2F)C(F)(F)F)cc1Nc1ccc2\C(=C\c3ccc[nH]3)C(=O)Nc2c1
Cc1ccc(NC(=O)Nc2cccc(c2)C(F)(F)F)cc1Nc1ccc2\C(=C\c3ccc[nH]3)C(=O)Nc2c1
FC(F)(F)c1cccc(c1)C(=O)Nc1cccc(Nc2ccc3\C(=C\c4ccc[nH]4)C(=O)Nc3c2)c1
O=C(Nc1cccc(Nc2ccc3\C(=C\c4ccc[nH]4)C(=O)Nc3c2)c1)c1ccccc1
Nc1ncnn2ccc(C(=O)Nc3ccc(NC(=O)Nc4cccc(F)c4)cc3)c12
CC(=O)Nc1cc(N)cc(c1)-c1cnc2[nH]cc(-c3ccncc3)c2c1
COc1ccc(N)cc1-c1cnc2[nH]cc(-c3ccncc3)c2c1
Nc1ccc(NS(=O)(=O)c2ccccc2)c(c1)-c1cnc2[nH]cc(-c3ccncc3)c2c1
COc1ccc(cc1OC)-c1c[nH]c2ncc(cc12)-c1cncc(NS(=O)(=O)c2ccccc2)c1
COc1ccc(cc1OC)-c1c[nH]c2ncc(cc12)-c1cccc(NS(=O)(=O)c2ccccc2)c1
COc1ccc(cc1OC)-c1c[nH]c2ncc(cc12)-c1cncc(N)c1
COc1ccc(cc1OC)-c1c[nH]c2ncc(cc12)-c1cccc(N)c1
Nc1cccc(c1)-c1cnc2[nH]cc(-c3ccncc3)c2c1
Nc1cccc(c1)-c1cnc2[nH]cc(-c3cccnc3)c2c1
Nc1cccc(c1)-c1cnc2[nH]cc(-c3ccccc3)c2c1
Nc1cccc(c1)-c1cnc2[nH]cc(-c3cccc(c3)C#N)c2c1
Nc1cccc(c1)-c1c[nH]c2ncc(cc12)-c1cccc(c1)C#N
Nc1cncc(c1)-c1cnc2[nH]cc(-c3ccncc3)c2c1
CNc1cccc(c1)-c1cnc2[nH]cc(-c3ccncc3)c2c1
CN(C)c1cccc(c1)-c1cnc2[nH]cc(-c3ccncc3)c2c1
COc1cccc(c1)-c1cnc2[nH]cc(-c3ccncc3)c2c1
CC(=O)Nc1cccc(c1)-c1cnc2[nH]cc(-c3ccncc3)c2c1
Nc1ccc(cc1)-c1cnc2[nH]cc(-c3ccncc3)c2c1
COc1ccc(cc1N)-c1cnc2[nH]cc(-c3ccncc3)c2c1
Nc1cc(ccc1Cl)-c1cnc2[nH]cc(-c3ccncc3)c2c1
Cc1ccc(cc1N)-c1cnc2[nH]cc(-c3ccncc3)c2c1
Nc1cc(ccc1C(=O)N1CCOCC1)-c1cnc2[nH]cc(-c3ccncc3)c2c1
CN(C)CCOc1ccc(cc1N)-c1cnc2[nH]cc(-c3ccncc3)c2c1
COc1cc(N)cc(c1)-c1cnc2[nH]cc(-c3ccncc3)c2c1
Nc1cc(cc(c1)-c1cnc2[nH]cc(-c3ccncc3)c2c1)C(=O)N1CCOCC1
CN(C)CCOc1cc(N)cc(c1)-c1cnc2[nH]cc(-c3ccncc3)c2c1
Nc1cc(OCCN2CCOCC2)cc(c1)-c1cnc2[nH]cc(-c3ccncc3)c2c1
CS(=O)(=O)Nc1cc(N)cc(c1)-c1cnc2[nH]cc(-c3ccncc3)c2c1
Nc1cc(NS(=O)(=O)c2ccccc2)cc(c1)-c1cnc2[nH]cc(-c3ccncc3)c2c1
Cc1ccc(cc1)S(=O)(=O)Nc1cc(N)cc(c1)-c1cnc2[nH]cc(-c3ccncc3)c2c1
Nc1cc(NS(=O)(=O)c2ccc(F)cc2F)cc(c1)-c1cnc2[nH]cc(-c3ccncc3)c2c1
Nc1cc(NS(=O)(=O)c2cccc(c2)C(F)(F)F)cc(c1)-c1cnc2[nH]cc(-c3ccncc3)c2c1
CS(=O)(=O)CCN1CCC(CC1)c1ccc(NC(=O)c2ncc([nH]2)C#N)c(c1)C1=CCCCC1 |t:31|
O=C(Nc1ccc(cc1C1=CCCCC1)C1CCN(CCN2CCOCC2)CC1)c1ncc([nH]1)C#N |t:10|
Cn1cc(-c2ccc3N(CCc3c2)C(=O)Cc2cccc(c2)C(F)(F)F)c2c(N)ncnc12
Cn1cc(NC(=O)c2cnn3ccc(N)nc23)c(n1)-c1cc(Cl)ccc1Cl
NCCCC[C@@H]1NC(=O)c2cc(ccc2NCc2ccc(cc2NC(=O)[C@H](CO)NC1=O)C(N)=O)[N+]([O-])=O
CC(C)(C)Nc1c(Nc2ccnc(Nc3ccc(cc3)-c3ccncc3)n2)c(=O)c1=O
CNCc1cc(F)c(c(OC)c1)-c1cc2c(n[nH]c2cn1)-c1cnn(C)c1
CNCc1cc(F)c(c(F)c1)-c1cc2c(n[nH]c2cn1)-c1cnn(C)c1
CNCc1cc(F)c(-c2cc3c(n[nH]c3cn2)-c2cnn(C)c2)c(c1)C(F)(F)F
CNCc1cc(C)c(c(F)c1)-c1cc2c(n[nH]c2cn1)-c1cnn(C)c1
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1cc(F)ccc1N1CC[C@@H](N)C1 |r|
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1ccc2n(C)ncc2c1N1CC[C@@H](N)C1 |r|
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1cc(F)c2n(C)ncc2c1N1CC[C@@H](N)C1 |r|
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1cc(F)c2nn(C)cc2c1N1CC[C@@H](N)C1 |r|
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1cc2cnn(C)c2cc1N1CC[C@@H](N)C1 |r|
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1ccc2n(C)cnc2c1N1CC[C@@H](N)C1 |r|
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1ccc2sc(C)nc2c1N1CC[C@@H](N)C1 |r|
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1cc(F)c2n(C)ncc2c1N1CCC(N)CC1
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1cc(F)c2n(C)ncc2c1N1CCNCC1
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1cc(F)c2n(C)ncc2c1N1CCNC[C@H]1C |r|
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1cc(F)c2n(C)ncc2c1N1C[C@@H]2C[C@H]1CN2 |r|
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1cc(F)c2n(C)ncc2c1N1C[C@@H]2CC[C@H]1CN2 |r|
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1cc(F)c2n(C)ncc2c1N1C[C@@H](N)C[C@H]1C |r|
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1cc(F)c2n(C)ncc2c1N1C[C@@H](N)C[C@H]1CO |r|
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1cc(F)c2n(C)ncc2c1N1CCC[C@H]1CO |r|
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1cc(F)c2n(C)ncc2c1N1C[C@@H](O)C[C@H]1CN |r|
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1cc(F)c2n(C)ncc2c1N1C[C@H](N)C[C@H]1CO |r|
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1cc(F)c2n(C)ncc2c1N1CC[C@@H](O)[C@@H]1CN |r|
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1cc(F)c2n(C)ncc2c1N1CC[C@H](N)[C@@H]1CO |r|
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1cc(F)ccc1N1C[C@@H](N)C[C@H]1CO |r|
[H][C@@]12CN(c3ccccc3NC(=O)c3ccnc(n3)-c3c(F)cccc3OC)[C@@]([H])(CN1)C2 |r|
[H][C@]12CN(c3cc(c(F)cc3NC(=O)c3ccnc(n3)-c3c(F)cccc3OC)-c3cccnc3)[C@]([H])(CN1)C2 |r|
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1cc(F)c(cc1N1C[C@@H]2C[C@H]1CN2)-c1cccnc1C |r|
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1ccc(cc1N1C[C@@H]2C[C@H]1CN2)-c1cccnc1C |r|
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1ccc(cc1N1C[C@@H](N)C[C@H]1CO)-c1cccnc1C |r|
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1ccc(cc1N1C[C@@H](N)C[C@H]1CO)-c1cnccc1C#N |r|
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1ccc(cc1N1C[C@@H](N)C[C@H]1CO)-c1ncccc1C#N |r|
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1ccc(cc1N1C[C@@H](N)C[C@H]1CO)-c1c(cnn1C)C#N |r|
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1ccc(cc1N1C[C@@H](N)C[C@H]1CO)-c1c(C)nn(C)c1C#N |r|
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1cc(F)ccc1N1C[C@H]2C[C@@H]1CN2 |r|
CO[C@]1(CO)C[C@H]2O[C@]1(C)n1c3ccccc3c3c4CNC(=O)c4c4c5ccccc5n2c4c13
C[C@@]1(O)C[C@H]2O[C@]1(C)n1c3ccccc3c3c4CNC(=O)c4c4c5ccccc5n2c4c13
C[C@]1(O)C[C@H]2O[C@]1(C)n1c3ccccc3c3c4CNC(=O)c4c4c5ccccc5n2c4c13
C[C@]12O[C@H](C[C@@]1(O)C(N)=O)n1c3ccccc3c3c4C(=O)NCc4c4c5ccccc5n2c4c13
COc1cc(NC(=O)Nc2cnc(Nc3ccc(cc3)N3CCOCC3)nc2Oc2ccc(C)cc2OC)cc(OC)c1
Cn1cnc(c1)-c1cnc(OC2CCN(CC2)C(=O)Cc2ccc(OC(F)(F)F)cc2)c(c1)C(N)=O
CNC(=O)c1cc(c(nc1)N)O[C@H]2CN(CC2(F)F)C(=O)Cc3ccc(cc3)OC(F)(F)F
CC(C)(COc1ccc(c(c1)O[C@H]2CCN(C[C@H]2F)C(=O)Cc3ccc(cc3)OC(F)(F)F)C(=O)N)O
Cn1cc(cn1)-c1ccc(OC2CCN(CC2)C(=O)Nc2ccc(OC(F)(F)F)cc2)c(c1)C(N)=O
Cn1cc(cn1)-c1ccc(OC2CCN(CC2)C(=O)Cc2ccc(OC(F)(F)F)cc2)c(c1)C(N)=O
Cn1cc(cn1)-c1ccc(OC2CCN(CC2)C(=O)Cc2ccc(OC(F)(F)F)cc2)c(n1)C(N)=O
C[C@H](C(=O)N1CCC(CC1)Oc1ccc(cc1C(N)=O)-c1cn(C)cn1)c1ccc(OC(F)(F)F)cc1 |r|
C[C@@H](C(=O)N1CCC(CC1)Oc1ccc(cc1C(N)=O)-c1cn(C)cn1)c1ccc(OC(F)(F)F)cc1 |r|
Cn1cnc(c1)-c1ccc(OC2CCN(CC2)C(=O)Cc2ccc(OC(F)(F)F)c(F)c2)c(c1)C(N)=O
Cn1cnc(c1)-c1cnc(O[C@H]2CCN(C[C@@H]2F)C(=O)Cc2ccc(OC(F)(F)F)cc2)c(c1)C(N)=O |r|
Cn1cnc(c1)-c1cnc(O[C@H]2CCN(C[C@H]2F)C(=O)Cc2ccc(OC(F)(F)F)cc2)c(c1)C(N)=O |r|
Cn1cnc(c1)-c1ccc(OC2CCN(CC2(F)F)C(=O)Cc2ccc(OC(F)(F)F)cc2)c(c1)C(N)=O
CC(C)(CO)Oc1ccc(C(N)=O)c(O[C@@H]2CCN(C[C@@H]2F)C(=O)Cc2ccc(OC(F)(F)F)cc2)c1 |r|
Cn1cnc(c1)-c1cnc(N)c(O[C@@H]2CN(C[C@H]2F)C(=O)Cc2ccc(OC(F)(F)F)cc2)c1 |r|
Cn1cnc(c1)-c1cnc(N)c(O[C@@H]2CN(CC2(F)F)C(=O)Cc2ccc(OC(F)(F)F)cc2)c1 |r|
Cn1cc(cn1)-c1ccc(O[C@@H]2CCN(C2)C(=O)Cc2ccc(OC(F)(F)F)cc2)c(n1)C(N)=O |r|
Cn1cnc(c1)-c1cnc(O[C@@H]2CCN(C[C@@H]2F)C(=O)Cc2ccc(OC(F)(F)F)cc2)c(c1)C(N)=O |r|
Cn1cc(cn1)-c1ccc(O[C@H]2CCN(C2)C(=O)Cc2ccc(OC(F)(F)F)cc2)c(n1)C(N)=O |r|
Cn1cnc(c1)-c1ccc(OC2CCN(CC2)C(=O)Cc2ccc(OC3CC3)c(F)c2)c(c1)C(N)=O
CC(C)(O)COc1ccc(C(N)=O)c(O[C@H]2CCN(C[C@@H]2F)C(=O)Cc2ccc(OC(F)(F)F)cc2)c1 |r|
Cn1cnc(c1)-c1ccc(OC2CCN(CC2)C(=O)Cc2ccc(OC(F)(F)F)cc2)c(c1)C(N)=O
CCNC(=O)c1cnc(N)c(O[C@H]2CN(CC2(F)F)C(=O)Cc2ccc(OC(F)(F)F)cc2)c1 |r|
Cn1cnc(c1)-c1cnc(O[C@@H]2CCN(C[C@H]2F)C(=O)Cc2ccc(OC(F)(F)F)cc2)c(c1)C(N)=O |r|
CC(C)(O)COc1ccc(C(N)=O)c(O[C@@H]2CCN(C[C@H]2F)C(=O)Cc2ccc(OC(F)(F)F)cc2)c1 |r|
CC(C)(O)COc1ccc(C(N)=O)c(O[C@@H]2CCN(C[C@@H]2F)C(=O)Cc2ccc(OC(F)(F)F)cc2)c1 |r|
Cn1cnc(c1)-c1cnc(N)c(O[C@H]2CN(C[C@@H]2F)C(=O)Cc2ccc(OC(F)(F)F)cc2)c1 |r|
Cn1cnc(c1)-c1cnc(N)c(O[C@H]2CN(CC2(F)F)C(=O)Cc2ccc(OC(F)(F)F)cc2)c1 |r|
c1cc(c(cc1Cl)CNc2ncc(c(n2)NC3CCCC3)C(=O)NCCCN4CCOC4=O)Cl
Clc1ccc(Cl)c(CNc2ncc(C(=O)NCCCN3CCCC3=O)c(NC3CCCC3)n2)c1
c1ccc(cc1)C(=O)Nc2ccc(cc2)Nc3ccnc4c3-c5ccccc5C(=O)N4
CN1CCN(Cc2ccc(cc2)-c2cnc3[nH]cc(-c4ccc5[nH]ccc5c4)c3c2)CC1
CN(C)c1ccc(Oc2cc(O)cc(O)c2-c2cc(no2)C(=O)NC2CCN(CC2)C2CCC3(CC2)OCCO3)cc1
CC(C)Nc1ccc(Oc2cc(O)cc(O)c2-c2cc(no2)C(=O)NC2CCN(C)CC2)cc1
CN(C)c1ccc(Oc2cc(O)cc(O)c2-c2cc(no2)C(=O)NC2CCN(C)CC2)cc1
CN1CCC(CC1)NC(=O)c2cc(on2)c3c(cc(cc3Oc4ccc(cc4)[N+](=O)[O-])O)O
C[C@H](Nc1nc(Nc2cn(C)cn2)c2cc[nH]c2n1)c1ncc(F)cn1 |r|
C[C@@H](Oc1cc(cnc1N)-c1sc(nc1C)[C@](C)(O)CO)c1cc(F)ccc1-n1nccn1 |r|
CC(C)c1ccc(cc1C#Cc2cnc3n2ccnc3)C(=O)Nc4cc(cc(c4)C(F)(F)F)CN5CCN(CC5)C
CN1CCN(CC1)c1cc(Nc2cc(C)[nH]n2)nc(Sc2ccccc2)n1
CN1CCN(CC1)c1cc(Nc2cc(C)[nH]n2)nc(SCc2ccc(F)cc2)n1
CN1CCN(CC1)c1cc(Nc2cc([nH]n2)C2CCCC2)nc(Sc2ccccc2)n1
CN1CCN(CC1)c1cc(Nc2cc([nH]n2)-c2cccc(F)c2)nc(Sc2ccccc2)n1
CN1CCN(CC1)c1cc(Nc2cc(C)[nH]n2)nc(Sc2ccc(NC(=O)C3CC3)cc2)n1
CN1CCN(CC1)c1cc(Nc2cc(C)[nH]n2)nc(SCc2ccc(C)cc2)n1
COc1cc2c3cnc4[nH]ccc4c3n(CC3CCCCC3)c(=O)c2cc1OC
CCn1cc(-c2ccc3N(CCc3c2)C(=O)Cc2cccc(OC(F)(F)F)c2)c2c(N)ncnc12
CCC[C@H](C)Nc1ncc2c(cn([C@H]3CC[C@H](O)CC3)c2n1)-c1ccc(CN2CCCN(C)CC2)cc1 |r,wU:13.12,wD:16.16,3.3,(17.07,-10.92,;18.4,-10.15,;19.74,-10.92,;21.07,-10.15,;21.07,-8.61,;22.4,-10.92,;23.74,-10.15,;23.74,-8.61,;25.07,-7.84,;26.4,-8.6,;27.88,-8.12,;28.79,-9.38,;27.88,-10.63,;28.63,-11.97,;30.16,-12,;30.91,-13.35,;30.11,-14.67,;30.85,-16.02,;28.57,-14.64,;27.83,-13.29,;26.4,-10.15,;25.07,-10.92,;28.59,-6.76,;30.13,-6.7,;30.84,-5.34,;30.02,-4.03,;30.73,-2.67,;32.27,-2.6,;33,-3.97,;34.51,-4.24,;35.67,-3.22,;35.61,-1.69,;36.96,-.95,;34.36,-.79,;32.87,-1.2,;28.47,-4.1,;27.77,-5.47,)|
CC(C)c1ccc(NC(=O)Nc2cccc(Oc3cncc(n3)-c3ccsc3)c2)cc1
CC(C)(C)c1cccc(NC(=O)Nc2cccc(Oc3cncc(Cl)n3)c2)c1
Cn1cc(cn1)-c1cncc(Oc2cccc(NC(=O)Nc3cccc(c3)C(F)(F)F)c2)n1
Cn1cc(cn1)-c1cncc(Oc2cccc(NC(=O)Nc3cc(on3)C(C)(C)C)c2)n1
CC(C)(C)c1cc(NC(=O)Nc2cccc(Oc3cncc(n3)-c3ccc(cc3)S(C)(=O)=O)c2)no1
Cn1nc(cc1NC(=O)Nc1cccc(Oc2cncc(n2)-c2ccc(cc2)S(C)(=O)=O)c1)C(C)(C)C
Cn1cc(cn1)-c1cncc(n1)-c1ccc(NC(=O)Nc2cc(nn2C)C(C)(C)C)cc1
COc1ccc(cc1)-c1cncc(Oc2cccc(NC(=O)Nc3ccc(cc3)C(C)C)c2)n1
CC(C)(C)c1cc(NC(=O)Nc2cccc(Oc3cncc(Cl)n3)c2)no1
CC(C)c1ccc(NC(=O)Nc2cccc(Oc3cncc(n3)-c3ccc(cc3)S(C)(=O)=O)c2)cc1
CS(=O)(=O)c1ccc(cc1)-c1cncc(Oc2cccc(NC(=O)Nc3cccc(c3)C(F)(F)F)c2)n1
COc1ccc(cc1)-c1cncc(Oc2cccc(NC(=O)Nc3cc(on3)C(C)(C)C)c2)n1
FC(F)(F)c1cccc(NC(=O)Nc2cccc(Oc3cncc(Cl)n3)c2)c1
CC(C)(C)c1cc(NC(=O)Nc2cccc(Oc3cncc(n3)-c3ccsc3)c2)no1
CC(C)(C)c1cc(NC(=O)Nc2cccc(Oc3cncc(n3)-c3ccc(F)cc3)c2)no1
FC(F)(F)c1cccc(NC(=O)Nc2cccc(Oc3cncc(n3)-c3ccsc3)c2)c1
Cn1cc(cn1)-c1cncc(n1)-c1ccc(NC(=O)Nc2cc(no2)C(C)(C)C)cc1
COc1ccc(cc1)-c1cncc(Oc2cccc(NC(=O)Nc3cccc(c3)C(F)(F)F)c2)n1
OC(=O)C1CN(Cc2ccc(OCc3ccc(Cl)c(Cl)c3)cc2)C1
CC(C)n1c(C)nc2c(F)cc(cc12)-c1nc(Nc2ccc3CN(CCN(C)C)CCc3n2)ncc1F
CSc1cccc(NC(=O)Nc2nnc(SCc3cc(=O)n4cc(C)ccc4n3)s2)c1
Fc1ccc(NC(=O)Nc2nnc(SCc3cc(=O)n4cc(Cl)ccc4n3)s2)cc1
CCc1ccc(NC(=O)Nc2nnc(SCc3nc4ccccc4[nH]c3=O)s2)cc1
Cc1ccc(NC(=O)Nc2nnc(SCc3cc(=O)n4cccc(C)c4n3)s2)c(Cl)c1
CCn1c(CCc2ccc(NC(=O)Nc3cccc(OC)c3)cc2)nc2ccccc12
CCn1c(CCc2ccc(NC(=O)Nc3ccc(C)cc3)cc2)nc2ccccc12
COc1cc(NC(=O)Nc2ccc(CCc3nc4ccccc4[nH]3)cc2)cc(OC)c1OC
Brc1cccc(NC(=O)Nc2ccc(CCc3nc4ccccc4[nH]3)cc2)c1
COc1ccccc1NC(=O)Nc1nnc(SCc2cc(=O)n3cccc(C)c3n2)s1
Cc1ccc(NC(=O)Nc2nnc(SCc3cc(=O)n4cc(C)ccc4n3)s2)c(Cl)c1
COc1ccc(OC)c(NC(=O)Nc2nnc(SCc3cc(=O)n4cc(C)ccc4n3)s2)c1
Cc1cccn2c1nc(CSc1nnc(NC(=O)Nc3ccccc3)s1)cc2=O
Fc1ccc(NC(=O)Nc2nnc(SCc3nc4ccccc4[nH]c3=O)s2)cc1Cl
Cn1c(CCc2ccc(NC(=O)Nc3cccc(Br)c3)cc2)nc2ccccc12
Cc1ccc2nc(CSc3nnc(NC(=O)Nc4cccc(C)c4C)s3)cc(=O)n2c1
CCn1c(CCc2ccc(NC(=O)Nc3cc(OC)c(OC)c(OC)c3)cc2)nc2ccccc12
Cc1cc(C)cc(NC(=O)Nc2ccc(CCc3nc4ccccc4n3C)cc2)c1
CCn1c(CCc2ccc(NC(=O)Nc3cc(C)ccc3OC)cc2)nc2ccccc12
CSc1cccc(NC(=O)Nc2ccc(CCc3nc4ccccc4[nH]3)cc2)c1
Cc1ccn2c(c1)nc(CSc1nnc(NC(=O)Nc3ccc(C)c(Cl)c3)s1)cc2=O
CC1=CN2C(=NC(=CC2=O)CSc3nnc(s3)NC(=O)Nc4cccc(c4)C(F)(F)F)C=C1
CCc1ccc(NC(=O)Nc2nnc(SCc3cc(=O)n4cc(C)ccc4n3)s2)cc1
Cc1ccc2nc(CSc3nnc(NC(=O)Nc4ccc(C)c(F)c4)s3)cc(=O)n2c1
CCn1c(CCc2ccc(NC(=O)Nc3ccccc3F)cc2)nc2ccccc12
Cc1ccc(NC(=O)Nc2ccc(CCc3nc4ccccc4n3-c3ccccc3)cc2)cc1
Cn1c(CCc2ccc(NC(=O)Nc3ccc(F)c(Cl)c3)cc2)nc2ccccc12
CCn1c(CCc2ccc(NC(=O)Nc3cc(Cl)c(OC)cc3OC)cc2)nc2ccccc12
O=C(Nc1nnc(SCc2nc3ccccc3[nH]c2=O)s1)Nc1ccccc1
Cn1c(CCc2ccc(NC(=O)Nc3ccccc3F)cc2)nc2ccccc12
CCOc1ccccc1NC(=O)Nc1ccc(CCc2nc3ccccc3n2CC)cc1
Cc1ccc2nc(CSc3nnc(NC(=O)Nc4ccccc4F)s3)cc(=O)n2c1
COC(=O)c1ccccc1NC(=O)Nc1nnc(SCc2cc(=O)n3ccc(C)cc3n2)s1
Cc1ccc(NC(=O)Nc2ccc(CCc3nc4ccccc4[nH]3)cc2)cc1F
Cc1cccc(NC(=O)Nc2ccc(CCc3nc4ccccc4[nH]3)cc2)c1
CCn1c(CCc2ccc(NC(=O)Nc3cccc(Cl)c3)cc2)nc2ccccc12
Cc1ccc2nc(CSc3nnc(NC(=O)Nc4ccccc4C(F)(F)F)s3)cc(=O)n2c1
Cc1cccn2c1nc(CSc1nnc(NC(=O)Nc3cccc(c3)C(F)(F)F)s1)cc2=O
Cc1ccc(NC(=O)Nc2ccc(CCc3nc4ccccc4[nH]3)cc2)cc1Cl
Cc1cccc(NC(=O)Nc2nnc(SCc3cc(=O)n4cccc(C)c4n3)s2)c1
CSc1cccc(NC(=O)Nc2nnc(SCc3cc(=O)n4cccc(C)c4n3)s2)c1
Cc1ccc(NC(=O)Nc2ccc(CCc3nc4ccccc4n3C)cc2)cc1Cl
CCn1c(CCc2ccc(NC(=O)Nc3ccc(C)cc3C)cc2)nc2ccccc12
Cn1c(CCc2ccc(NC(=O)Nc3cccc(c3)C(F)(F)F)cc2)nc2ccccc12
Cc1ccc(NC(=O)Nc2nnc(SCc3cc(=O)n4cc(Cl)ccc4n3)s2)cc1C
FC(F)(F)c1cccc(NC(=O)Nc2nnc(SCc3nc4ccccc4[nH]c3=O)s2)c1
Brc1ccc(NC(=O)Nc2ccc(CCc3nc4ccccc4[nH]3)cc2)cc1
CSc1cccc(NC(=O)Nc2ccc(CCc3nc4ccccc4n3C)cc2)c1
CCOc1ccccc1NC(=O)Nc1ccc(CCc2nc3ccccc3n2C)cc1
CCn1c(CCc2ccc(NC(=O)Nc3cc(OC)cc(OC)c3)cc2)nc2ccccc12
COc1ccc(NC(=O)Nc2nnc(SCc3cc(=O)n4ccc(C)cc4n3)s2)cc1OC
COc1cc(NC(=O)Nc2nnc(SCc3cc(=O)n4ccc(C)cc4n3)s2)cc(OC)c1
COc1ccc(C)cc1NC(=O)Nc1nnc(SCc2cc(=O)n3cccc(C)c3n2)s1
COc1ccc(NC(=O)Nc2ccc(CCc3nc4ccccc4[nH]3)cc2)c(OC)c1
Cn1c(CCc2ccc(NC(=O)Nc3ccccc3C(F)(F)F)cc2)nc2ccccc12
Cc1cccn2c1nc(CSc1nnc(NC(=O)Nc3ccc(F)cc3F)s1)cc2=O
COc1ccc(OC)c(NC(=O)Nc2nnc(SCc3cc(=O)n4cccc(C)c4n3)s2)c1
CCOC(=O)c1ccccc1NC(=O)Nc1nnc(SCc2cc(=O)n3cccc(C)c3n2)s1
Cc1ccc(NC(=O)Nc2ccc(CCc3nc4ccccc4n3C)cc2)c(C)c1
Cn1c(CCc2ccc(NC(=O)Nc3ccccc3Cl)cc2)nc2ccccc12
CCn1c(CCc2ccc(NC(=O)Nc3cccc(c3)C(C)=O)cc2)nc2ccccc12
Clc1cccc(NC(=O)Nc2nnc(SCc3nc4ccccc4[nH]c3=O)s2)c1
COc1ccc(OC)c(NC(=O)Nc2ccc(CCc3nc4ccccc4[nH]3)cc2)c1
FC(F)(F)c1cccc(NC(=O)Nc2ccc(CCc3nc4ccccc4[nH]3)cc2)c1
CCOC(=O)c1ccccc1NC(=O)Nc1nnc(SCc2cc(=O)n3ccc(C)cc3n2)s1
Cc1cccn2c1nc(CSc1nnc(NC(=O)Nc3ccccc3F)s1)cc2=O
COc1cc(NC(=O)Nc2ccc(CCc3nc4ccccc4n3C)cc2)cc(OC)c1
COc1ccc(Cl)cc1NC(=O)Nc1ccc(CCc2nc3ccccc3n2C)cc1
Cc1ccc(NC(=O)Nc2nnc(SCc3cc(=O)n4cccc(C)c4n3)s2)cc1
Cc1ccc(C)c(NC(=O)Nc2nnc(SCc3cc(=O)n4ccccc4n3)s2)c1
Cc1ccc(C)c(NC(=O)Nc2ccc(CCc3nc4ccccc4n3C)cc2)c1
COc1ccc(NC(=O)Nc2nnc(SCc3cc(=O)n4cccc(C)c4n3)s2)cc1OC
Cc1ccc(C)c(NC(=O)Nc2nnc(SCc3cc(=O)n4cccc(C)c4n3)s2)c1
CCOc1ccccc1NC(=O)Nc1nnc(SCc2cc(=O)n3cccc(C)c3n2)s1
COc1cc(OC)c(NC(=O)Nc2ccc(CCc3nc4ccccc4n3C)cc2)cc1Cl
COC(=O)c1ccccc1NC(=O)Nc1nnc(SCc2cc(=O)n3cccc(C)c3n2)s1
Cc1ccc(NC(=O)Nc2nnc(SCc3cc(=O)n4cc(C)ccc4n3)s2)cc1
COc1ccc(OC)c(NC(=O)Nc2nnc(SCc3cc(=O)n4ccc(C)cc4n3)s2)c1
CCn1c(CCc2ccc(NC(=O)Nc3cc(Cl)ccc3OC)cc2)nc2ccccc12
Cc1ccc(Cl)cc1NC(=O)Nc1nnc(SCc2cc(=O)n3cccc(C)c3n2)s1
Cc1ccc(NC(=O)Nc2nnc(SCc3cc(=O)n4cc(Cl)ccc4n3)s2)cc1F
Cc1ccn2c(c1)nc(CSc1nnc(NC(=O)Nc3ccccc3C(F)(F)F)s1)cc2=O
CCn1c(CCc2ccc(NC(=O)Nc3ccc(C)c(C)c3)cc2)nc2ccccc12
Cc1ccc(NC(=O)Nc2nnc(SCc3nc4ccccc4[nH]c3=O)s2)cc1
Cc1ccn2c(c1)nc(CSc1nnc(NC(=O)Nc3cccc(c3)C(F)(F)F)s1)cc2=O
COc1ccc(NC(=O)Nc2ccc(CCc3nc4ccccc4n3C)cc2)c(OC)c1
CCn1c(CCc2ccc(NC(=O)Nc3cccc(C)c3)cc2)nc2ccccc12
CCn1c(CCc2ccc(NC(=O)Nc3cc(OC)ccc3OC)cc2)nc2ccccc12
Cc1cccc(NC(=O)Nc2nnc(SCc3cc(=O)n4cc(C)ccc4n3)s2)c1
COc1ccccc1NC(=O)Nc1nnc(SCc2cc(=O)n3ccc(C)cc3n2)s1
COc1ccc(C)cc1NC(=O)Nc1ccc(CCc2nc3ccccc3[nH]2)cc1
CCn1c(CCc2ccc(NC(=O)Nc3cc(C)cc(C)c3)cc2)nc2ccccc12
Cc1ccc(NC(=O)Nc2nnc(SCc3cc(=O)n4cccc(C)c4n3)s2)cc1Cl
COc1ccccc1NC(=O)Nc1nnc(SCc2cc(=O)n3cc(C)ccc3n2)s1
Fc1ccc(NC(=O)Nc2nnc(SCc3cc(=O)n4ccccc4n3)s2)cc1
Cc1ccc(C)c(NC(=O)Nc2nnc(SCc3cc(=O)n4cc(C)ccc4n3)s2)c1
COc1cccc(NC(=O)Nc2ccc(CCc3nc4ccccc4[nH]3)cc2)c1
COc1ccc(Cl)cc1NC(=O)Nc1ccc(CCc2nc3ccccc3[nH]2)cc1
COc1ccc(OC)c(NC(=O)Nc2ccc(CCc3nc4ccccc4n3C)cc2)c1
CCn1c(CCc2ccc(NC(=O)Nc3cccc(SC)c3)cc2)nc2ccccc12
Cc1cccc(NC(=O)Nc2nnc(SCc3cc(=O)n4cccc(C)c4n3)s2)c1C
CCOc1ccccc1NC(=O)Nc1ccc(CCc2nc3ccccc3n2-c2ccccc2)cc1
Cc1cccn2c1nc(CSc1nnc(NC(=O)Nc3cccc(F)c3)s1)cc2=O
Cc1ccc(NC(=O)Nc2nnc(SCc3cc(=O)n4cccc(C)c4n3)s2)cc1C
Cc1cccn2c1nc(CSc1nnc(NC(=O)Nc3ccc(F)cc3)s1)cc2=O
COc1cccc(NC(=O)Nc2nnc(SCc3cc(=O)n4cccc(C)c4n3)s2)c1
COc1cccc(NC(=O)Nc2nnc(SCc3cc(=O)n4cc(C)ccc4n3)s2)c1
Cc1ccc(NC(=O)Nc2ccc(CCc3nc4ccccc4[nH]3)cc2)cc1C
Cc1ccccc1NC(=O)Nc1nnc(SCc2cc(=O)n3ccccc3n2)s1
Cc1ccc(NC(=O)Nc2ccc(CCc3nc4ccccc4[nH]3)cc2)cc1
CCn1c(CCc2ccc(NC(=O)Nc3ccc4OCOc4c3)cc2)nc2ccccc12
Cc1ccn2c(c1)nc(CSc1nnc(NC(=O)Nc3ccccc3F)s1)cc2=O
Cc1ccc(C)c(NC(=O)Nc2ccc(CCc3nc4ccccc4[nH]3)cc2)c1
Cc1cccn2c1nc(CSc1nnc(NC(=O)Nc3cccc(Cl)c3)s1)cc2=O
Cc1cc(C)cc(NC(=O)Nc2nnc(SCc3cc(=O)n4cccc(C)c4n3)s2)c1
CCc1ccc(NC(=O)Nc2nnc(SCc3cc(=O)n4cccc(C)c4n3)s2)cc1
CCn1c(CCc2ccc(NC(=O)Nc3ccccc3Cl)cc2)nc2ccccc12
Cc1ccc2nc(CSc3nnc(NC(=O)Nc4ccccc4C)s3)cc(=O)n2c1
Cn1c(CCc2ccc(NC(=O)Nc3cccc(Cl)c3)cc2)nc2ccccc12
Clc1cccc(NC(=O)Nc2ccc(CCc3nc4ccccc4[nH]3)cc2)c1
Cc1ccn2c(c1)nc(CSc1nnc(NC(=O)Nc3ccc(C)c(F)c3)s1)cc2=O
CC(=O)Nc1cccc(n1)-c1ccc(Cl)c(c1)C(=O)Nc1cc(nn1-c1ccccc1)C(N)=O
COc1cc(Cl)c(cc1-c1ccccn1)C(=O)Nc1cc(nn1-c1ccccc1)C(N)=O
CC(C)(O)CNC(=O)c1cc(NC(=O)c2cc(c(Cl)cc2Cl)-c2ccccn2)n(n1)-c1ccccc1
CN(C)C(=O)c1cc(NC(=O)c2cc(ccc2Cl)-c2ccccn2)n(n1)-c1ccccc1
NC(=O)c1cc(NC(=O)c2cc(ccc2Cl)-c2cccc(N)n2)n(n1)-c1ccccc1
Cc1cc(NC(=O)c2ccc(Cl)cc2Cl)n(n1)-c1ccccc1
CC(C)(O)CNC(=O)c1cc(NC(=O)c2cc(c(Cl)cc2Cl)-c2ncccc2F)n(n1)-c1ccccc1
NCCNC(=O)c1cc(NC(=O)c2cc(c(Cl)cc2Cl)-c2ccccn2)n(n1)-c1ccccc1
OCCNC(=O)c1cc(NC(=O)c2cc(c(Cl)cc2Cl)-c2ncccc2F)n(n1)-c1ccccc1
OCCNC(=O)c1cc(NC(=O)c2cc(c(Cl)cc2Cl)-c2ccccn2)n(n1)-c1ccccc1
NC(=O)c1cc(NC(=O)c2cc(c(OC(F)F)cc2Cl)-c2ccccn2)n(n1)-c1ccccc1
Cc1cc(Cl)c(cc1-c1ccccn1)C(=O)Nc1cc(nn1-c1ccccc1)C(N)=O
NC(=O)c1cc(NC(=O)c2cc(c(Cl)cc2Cl)-c2cccc(N)n2)n(n1)-c1ccccc1
NC(=O)c1cc(NC(=O)c2cc(ccc2Cl)-c2nc(N)ccc2Cl)n(n1)-c1ccccc1
NC(=O)c1cc(NC(=O)c2cc(ccc2Cl)-c2cccc(n2)C(F)F)n(n1)-c1ccccc1
NC(=O)c1cc(NC(=O)c2cc(ccc2Cl)-c2cccc(n2)C(N)=O)n(n1)-c1ccccc1
NC(=O)c1cc(NC(=O)c2cc(-c3ccccn3)c(cc2Cl)C2CC2)n(n1)-c1ccccc1
NC(=O)c1cc(NC(=O)c2cc(c(Cl)cc2Cl)-c2ccccn2)n(n1)-c1ccccc1
NC(=O)c1cc(NC(=O)c2cc(ccc2Cl)-c2ncccc2F)n(n1)-c1ccccc1
CC(C)(O)CNC(=O)c1cc(NC(=O)c2cc(c(F)cc2Cl)-c2ncccc2F)n(n1)-c1ccccc1
OCCNC(=O)c1cc(NC(=O)c2cc(-c3ccccn3)c(cc2Cl)C(F)(F)F)n(n1)-c1ccccc1
NC(=O)c1cc(NC(=O)c2cc(c(F)cc2Cl)-c2ncccc2F)n(n1)-c1ccccc1
Clc1cc(Cl)c(cc1C(=O)Nc1cc(nn1-c1ccccc1)C(=O)NC1COC1)-c1ccccn1
NC(=O)c1cc(NC(=O)c2cc(c(F)cc2Cl)-c2ccccn2)n(n1)-c1ccccc1
NC(=O)c1cc(NC(=O)c2cc(ccc2Cl)-c2ncccc2Cl)n(n1)-c1ccccc1
COc1cccc(c1)-n1c(=O)[nH]c(=O)n(-c2ccc(Oc3ccccc3)cc2)c1=O
COCCOc1cc(ccc1Oc1ccccc1)-n1c(=O)[nH]c(=O)n(-c2ccc(Cl)cc2)c1=O
COCCOc1cc(ccc1Oc1ccccc1)-n1c(=O)[nH]c(=O)n(-c2cccc(C)c2)c1=O
COCCOc1cc(ccc1Oc1ccccc1)-n1c(=O)[nH]c(=O)n(-c2ccc(C)cc2)c1=O
Cn1c(=O)[nH]c(=O)n(-c2ccc(Oc3ccccc3)c(OCC3COC3)c2)c1=O
CCOc1cc(ccc1Oc1ccccc1)-n1c(=O)[nH]c(=O)n(-c2ccccc2)c1=O
COc1cc(ccc1Oc1ccccc1)-n1c(=O)[nH]c(=O)n(-c2ccccc2)c1=O
O=c1[nH]c(=O)n(-c2ccc(Oc3ccccc3)cc2)c(=O)n1-c1ccccc1
Brc1cc(ccc1Oc1ccccc1)-n1c(=O)[nH]c(=O)n(-c2ccccc2)c1=O
O=c1[nH]c(=O)n(-c2ccc(Oc3ccccc3)c(OCC3COC3)c2)c(=O)n1-c1ccccc1
O=c1[nH]c(=O)n(-c2ccc(Oc3ccccc3)c(OC3CCOC3)c2)c(=O)n1-c1ccccc1
COc1cc(Oc2ccccc2)ccc1-n1c(=O)[nH]c(=O)n(-c2ccccc2)c1=O |(72.02,-7.51,;73.36,-8.28,;73.36,-9.82,;72.02,-10.6,;72.03,-12.14,;70.69,-12.91,;69.36,-12.15,;69.36,-10.61,;68.02,-9.84,;66.69,-10.61,;66.7,-12.16,;68.03,-12.92,;73.37,-12.91,;74.7,-12.13,;74.69,-10.6,;76.02,-9.82,;77.36,-10.59,;77.36,-12.13,;78.69,-9.82,;78.69,-8.28,;80.02,-7.52,;77.36,-7.5,;77.36,-5.96,;78.69,-5.19,;78.69,-3.65,;77.36,-2.88,;76.02,-3.66,;76.03,-5.2,;76.02,-8.28,;74.69,-7.52,)|
Cc1cc(ccc1Oc1ccccc1)-n1c(=O)[nH]c(=O)n(-c2ccccc2)c1=O
COCCOc1cc(ccc1Oc1ccccc1)-n1c(=O)[nH]c(=O)n(-c2cccc(Cl)c2)c1=O
CC(C)Oc1cc(ccc1Oc1ccccc1)-n1c(=O)[nH]c(=O)n(-c2ccccc2)c1=O
[H][C@]12C[C@H]([C@@H](OC)[C@](C)(O1)n1c3ccccc3c3c4CNC(=O)c4c4c5ccccc5n2c4c13)N(C)CCOCCOCCOCCNC(=O)CCC1=[N+]2C(C=C1)=Cc1c(C)cc(C)n1[B-]2(F)F |r,c:63,65,t:60|
[H][C@]12C[C@@H](NCCOCCOCCOCCNC(=O)CCC3=[N+]4C(C=C3)=Cc3c(C)cc(C)n3[B-]4(F)F)[C@@H](OC)[C@](C)(O1)n1c3ccccc3c3c4CNC(=O)c4c4c5ccccc5n2c4c13 |r,c:24,26,t:21|
O=C(Cc1ccc(cc1)-c1ccccc1)Nc1cc([nH]n1)C1CCC1
O=C1c2ccccc2-n2c1nc1ccccc1c2=O
O\N=C1/c2ccccc2-n2c1nc1ccccc1c2=O
Cc1ccc(NC(=O)c2ccc(cc2F)C(F)(F)F)c(n1)-c1ccc(F)cc1
C[C@]1(CCCN1c1nc(Nc2cc([nH]n2)C2CC2)c2cccn2n1)C(=O)Nc1ccc(F)nc1 |r|
COCCNCc1ccc(nc1)-c1cc2nccc(Oc3ccc(NC(=O)C4(CC4)C(=O)Nc4ccc(F)cc4)cc3F)c2s1
Cc1ncc(NC(=O)NC2c3ccccc3-c3ccccc23)c(n1)-c1ccccc1
COc1ccc(cc1)-c1cc2cccc(O)c2c(=O)o1
COC[C@@H](C)Nc1cc(NC(=O)N2CCCc3cc(CN4CCCCOC4=O)c(C=O)nc23)ncc1C#N |r|
CN(CCc1ccc(cc1)-c1ccccc1)Cc1cn(C)c2ccc(cc12)C(=O)Nc1ccc(F)cc1
c1ccc2c(c1)C(=O)c3c(cc(c(c3C2=O)N)N4CCN(CC4)C5CCCCC5)Nc6ccc(cc6)C(=O)O
O=C(NC1c2ccccc2-c2ccccc12)Nc1cccnc1-c1ccccc1
Cn1ccc(n1)-c1cc(ccc1C(F)(F)F)C(=O)Nc1c(nc2ccc(CO)cn12)-c1ccccc1
O[C@H]1CCN(C1)C(=O)c1cnc2ccc(cn12)N1CCCC1c1cc(F)ccc1F |r|
COCCN1C[C@@H](NC(=O)Nc2cc3cc(OC)c(OC)cc3nc2-c2ccccc2)[C@@H](C1)c1ccccc1 |r|
CC(C)c1cc(C(=O)c2cccc(NC(=O)Nc3ccc4ccccc4c3)c2)c2c(N)ncnn12
COCC[C@@H]1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnn(C)c2)[C@@H](N1)c1cnc(Cl)c(F)c1 |r|
COCC[C@@H]1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2cnc3n(C)nc(N=S(C)(C)=O)c3c2)[C@@H](N1)c1ccc(F)c(F)c1 |r|
[H][C@@]12CCc3ccccc3[C@@]1([H])[C@@H](CN2CCOC)NC(=O)Nc1c(C)c(nn1-c1ccccc1)-c1cnn(C)c1 |r|
[H][C@@]12COc3ccccc3[C@]1([H])[C@H](CN2CC(F)(F)F)NC(=O)Nc1c(C)c(OCC2CCN(C)CC2)nn1-c1ccccc1 |r|
CC(C)c1nnc(s1)-c1cnn2ccc(nc12)N1CCCC1c1cc(F)ccc1F
CC(C)(C)c1nnc(o1)-c1cnn2ccc(nc12)N1CCCC1c1cc(F)ccc1F
CC(C)c1cc(C(=O)c2cccc(NC(=O)Nc3ccc(Cl)cc3Cl)c2)c2c(N)ncnn12
CC(C)c1cc(C(=O)c2cccc(NC(=O)Nc3ccc(OCc4ccccc4)cc3)c2)c2c(N)ncnn12
CN(C)CCCc1cc(C(=O)c2cccc(NC(=O)Nc3ccc(Cl)cc3Cl)c2)c2c(N)ncnn12
CCN1CCN(Cc2ccc(NC(=O)Nc3nc4ccc(Oc5ccnc(c5)C(=O)NC)cc4s3)cc2C(F)(F)F)CC1
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)C(C)(C)C)[C@@H](C1)c1ccc(F)c(F)c1 |r|
CC(C)c1cc(C(=O)c2cccc(NC(=O)Nc3ccccc3)c2)c2c(N)ncnn12
COCCN1C[C@@H](NC(=O)Nc2cc3ccccc3nc2-c2ccccc2)[C@@H](C1)c1ccccc1 |r|
COCCN1C[C@@H](NC(=O)Nc2cc3CCCCc3nc2-c2ccccc2)[C@@H](C1)c1ccccc1 |r|
Fc1ccc(NC(=O)c2cnc3ccc(cn23)N2CCCC2c2cc(F)ccc2F)cc1
Nc1nn2cc(cnc2c1C(=O)Nc1ccc(F)cc1)N1CCC[C@@H]1c1cc(F)ccc1F |r|
CC(C)N1Cc2cc(OCCCNC(=O)c3cnn4ccc1nc34)c(F)cc2F
O=C(NC1c2ccccc2-c2ccccc12)Nc1c(nc2ccccn12)-c1ccccc1
Cc1nc(c(NC(=O)Nc2cnc3ccccn23)s1)-c1ccccc1
Nc1nc(c(F)cc1F)-c1ccc(Cl)c(c1)C(=O)Nc1cc(nn1-c1ccccc1)C(=O)NCCCO
C[C@]1(O)CC[C@@H](CC1)NC(=O)c1cc(NC(=O)c2cc(ccc2Cl)-c2nc(N)c(F)cc2F)n(n1)-c1ccccc1 |r,wU:5.8,wD:1.1,(22.7,-36.18,;21.37,-36.96,;21.37,-35.42,;19.85,-37.13,;19.22,-38.54,;20.13,-39.78,;21.66,-39.61,;22.28,-38.21,;19.51,-41.19,;17.98,-41.35,;17.07,-40.11,;17.36,-42.76,;15.85,-43.09,;15.7,-44.62,;14.37,-45.4,;13.03,-44.63,;13.02,-43.09,;11.7,-45.41,;10.36,-44.64,;9.03,-45.41,;9.03,-46.96,;10.37,-47.73,;11.7,-46.96,;13.04,-47.72,;7.71,-44.64,;7.71,-43.1,;6.37,-42.33,;6.38,-40.79,;5.04,-43.1,;3.7,-42.33,;5.04,-44.65,;6.38,-45.41,;6.38,-46.95,;17.1,-45.24,;18.13,-44.09,;17.43,-46.74,;16.29,-47.78,;16.61,-49.28,;18.08,-49.75,;19.22,-48.71,;18.89,-47.21,)|
OC1CN(C1)C(=O)c1cnc2ccc(cn12)N1CCCC1c1cc(F)ccc1F
NC(=O)c1c(N)nn2cc(cnc12)N1CCC[C@@H]1c1cc(F)ccc1F |r|
O=C(NC1c2ccccc2-c2ccccc12)Nc1c(nc2sccn12)-c1ccccc1
COCCN1C[C@@H](NC(=O)Nc2c(C)c(nn2-c2ccccc2)-c2ccnc(C)n2)[C@@H](C1)c1cccc(F)c1 |r|
Nc1cc(CNC(=O)c2cc(NC(=O)c3cc(c(Cl)cc3Cl)-c3cccc(F)n3)n(n2)-c2ccccc2)ccn1
Nc1cc(CNC(=O)c2cc(NC(=O)c3cc(c(F)cc3Cl)-c3cccc(F)n3)n(n2)-c2ccccc2)ccn1
[H][C@]12[C@@H](C[C@@H](CCOC)N1CC(F)(F)c1ccccc21)NC(=O)Nc1c(C)c(nn1-c1ccccc1)-c1cnn(C)c1 |r|
CC(C)c1nnc(o1)-c1cnn2ccc(nc12)N1CCCC1c1cc(F)ccc1F
Cn1ccc(n1)-c1cc(ccc1C(F)(F)F)C(=O)Nc1c(nc2ccc(cn12)C(C)(C)O)-c1ccccc1
CC(C)N1Cc2cc(O[C@@H](C)CNC(=O)c3cnn4cc1cnc34)cc(F)c2Cl |r|
CC(C)(O)c1ccc2nc(c(NC(=O)c3cc(-c4ncccn4)c(cc3F)C(F)(F)F)n2c1)-c1ccccc1
COc1ccc(cn1)-c1n[nH]c2ccc(NCc3ccccc3NS(C)(=O)=O)cc12
CS(=O)(=O)c1ccccc1CNc1ccc2[nH]nc(-c3ccc(nc3)N3CCNCC3)c2c1
CS(=O)(=O)Nc1ccccc1CNc1ccc2[nH]nc(-c3ccc(NC4CCNCC4)nc3)c2c1
CS(=O)(=O)c1ccc(F)cc1CNc1ccc2[nH]nc(-c3ccc(nc3)N3CCNCC3)c2c1
COc1cncc(c1)-c1n[nH]c2ccc(NCc3ccccc3NS(C)(=O)=O)cc12
C(Nc1ccc2[nH]nc(-c3ccc(nc3)N3CCNCC3)c2c1)c1ccccc1
C(Oc1ccc2[nH]nc(-c3ccc(nc3)N3CCNCC3)c2c1)c1ccccc1
CN(Cc1ccccc1)c1ccc2[nH]nc(-c3ccc(nc3)N3CCNCC3)c2c1
CC(C)(Nc1ccc2[nH]nc(-c3ccc(nc3)N3CCNCC3)c2c1)c1ccccc1
CS(=O)(=O)c1ccc(F)cc1CNc1ccc2[nH]nc(-c3cccnc3)c2c1
Cn1cc(cn1)-c1n[nH]c2ccc(NCc3cc(F)ccc3S(C)(=O)=O)cc12
CS(=O)(=O)Nc1ccccc1CNc1ccc2[nH]nc(-c3ccc(nc3)N3CCNCC3)c2c1
C(Cc1ccc2[nH]nc(-c3ccc(nc3)N3CCNCC3)c2c1)c1ccccc1
CS(=O)(=O)c1ccc(F)cc1CNc1ccc2[nH]nc(-c3ccccn3)c2c1
Cn1ccc(n1)-c1n[nH]c2ccc(NCc3cc(F)ccc3S(C)(=O)=O)cc12
CS(=O)(=O)Nc1ccccc1CNc1ccc2[nH]nc(-c3ccc(OC4CCNCC4)nc3)c2c1
CS(=O)(=O)Nc1cccc(CNc2ccc3[nH]nc(-c4ccc(nc4)N4CCNCC4)c3c2)c1
COc1cccc(n1)-c1n[nH]c2ccc(NCc3ccccc3NS(C)(=O)=O)cc12
CS(=O)(=O)Nc1ccc(CNc2ccc3[nH]nc(-c4ccc(nc4)N4CCNCC4)c3c2)cc1
CN1CCC(CC1)Nc1ccc(cc1)C(=O)Nc1cc(n[nH]1)-c1ccc2OCOc2c1
CCc1c(cccc1C(=O)Nc1cc(CN2CCN(C)CC2)cc(c1)C(F)(F)F)C#Cc1cnc2cnccn12
CN1CCN(Cc2cc(NC(=O)c3cc(ccc3C)C#Cc3cnc4cnccn34)cc(c2)C(F)(F)F)CC1
CN1CCN(Cc2cc(NC(=O)c3cccc(C#Cc4cnc5cnccn45)c3C)cc(c2)C(F)(F)F)CC1
CN1CCN(Cc2cc(NC(=O)c3cccc(c3)C#Cc3cnc4cnccn34)cc(c2)C(F)(F)F)CC1
COc1c(cccc1C(=O)Nc1cc(CN2CCN(C)CC2)cc(c1)C(F)(F)F)C#Cc1cnc2cnccn12
CC(C)c1c(cccc1C(=O)Nc1cc(CN2CCN(C)CC2)cc(c1)C(F)(F)F)C#Cc1cnc2cnccn12
CN1CCN(Cc2cc(NC(=O)c3cccc(C#Cc4cnc5cnc(cn45)-c4ccc(N)cc4)c3C)cc(c2)C(F)(F)F)CC1
CN1CCN(Cc2cc(C)cc(NC(=O)c3cccc(C#Cc4cnc5cnc(cn45)-c4ccc(N)cc4)c3C)c2)CC1
CCc1cc(CN2CCN(C)CC2)cc(NC(=O)c2cccc(C#Cc3cnc4cnc(cn34)-c3ccc(N)cc3)c2C)c1
CN1CCN(Cc2cc(NC(=O)c3cccc(C#Cc4cnc5cnc(cn45)-c4ccc(N)cc4)c3C)cc(c2)-c2ccccc2)CC1
CN1CCN(Cc2cc(NC(=O)c3ccc(C)c(c3)C#Cc3cnc4cnccn34)cc(c2)C(F)(F)F)CC1
CC(C)c1cc(CN2CCN(C)CC2)cc(NC(=O)c2cccc(C#Cc3cnc4cnc(cn34)-c3ccc(N)cc3)c2C)c1
CN1CCN(Cc2cc(NC(=O)c3cc(C)cc(c3)C#Cc3cnc4cnccn34)cc(c2)C(F)(F)F)CC1
CN1CCN(Cc2cc(NC(=O)c3cccc(C#Cc4cnc5cnccn45)c3Cl)cc(c2)C(F)(F)F)CC1
CN1CCN(Cc2cc(NC(=O)c3cccc(C#Cc4cnc5cnc(cn45)-c4ccncc4)c3C)cc(c2)C(F)(F)F)CC1
CN1CCN(Cc2cc(NC(=O)c3cccc(C#Cc4cnc5cnc(cn45)-c4ccc(N)cc4)c3C)cc(c2)C(C)(C)C)CC1
CN1CCN(Cc2cc(NC(=O)c3cccc(C#Cc4cnc5cnc(cn45)-c4ccccc4)c3C)cc(c2)C(F)(F)F)CC1
CCCc1c(cccc1C(=O)Nc1cc(CN2CCN(C)CC2)cc(c1)C(F)(F)F)C#Cc1cnc2cnccn12
CC(C)(C)c1cc(NC(=O)Cc2ccc(cc2)-n2cnc3cc(ccc23)-c2ccc(cc2)S(C)(=O)=O)no1
Cn1cc(-c2ccc(F)cc2)c(=O)c2c(Nc3ccc(Oc4ccnc(NC(=O)C5CC5)c4)c(F)c3)nccc12
CN(C)c1ccc(cc1)C(=O)Nc1cccc(NC(=O)COc2ccc3c(c2)occc3=O)c1
CCN1CCN(CC1)c1cc(Nc2ncc(s2)-c2ccncc2)nc(C)n1
CCS(=O)(=O)c1cn(-c2cc(C)[nH]n2)c2nc(N[C@@H](C)c3ccc(F)cn3)ccc12 |r|
C[C@@H](Oc1ccc2c(cn(-c3cc(C)n[nH]3)c2n1)C(=O)N1CCO[C@H](C)C1)c1ccc(F)cn1 |r|
C[C@H](Nc1ccc2ncc(-c3cc(C)n[nH]3)n2n1)c1ccc(F)cc1F |r|
C[C@H](Nc1ccc2ccn(-c3cc(C)n[nH]3)c2n1)c1ccc(F)cc1F |r|
C[C@H](Nc1ccc2c(cn(-c3cc(C)[nH]n3)c2n1)S(C)(=O)=O)c1ccc(F)cc1F |r|
C[C@H](Nc1ccc2c(cn(-c3cc(C)[nH]n3)c2n1)S(=O)(=O)C1COC1)c1ccc(F)cn1 |r|
C[C@H](Nc1ccc2c(cn(-c3cc(C)n[nH]3)c2n1)C(=O)N(C)C)c1ccc(F)cn1 |r|
C[C@H](Nc1ccc2c(cn(-c3cc(C)n[nH]3)c2n1)C(=O)N1CCN(C)CC1)c1ccc(F)cn1 |r|
C[C@H](Nc1ccc2c(cn(-c3cc(C)n[nH]3)c2n1)C1=CCOCC1)c1ccc(F)cn1 |r,t:21|
CC(Oc1ccc2c(cn(-c3cc(C)n[nH]3)c2n1)C(=O)N1CCOCC1)c1ccc(F)cn1
COCc1cn(-c2cc(C)n[nH]2)c2nc(OC(C)c3ccc(F)cn3)ccc12
C[C@H](Nc1ccc2c(cn(-c3cc(C)[nH]n3)c2n1)S(C)(=O)=O)c1ccc(F)cn1 |r|
C[C@H](Nc1ccc2c(cn(-c3cc(C)n[nH]3)c2n1)C(=O)N1CCOCC1)c1ccc(F)cn1 |r|
C[C@H](Oc1ccc2c(cn(-c3cc(C)[nH]n3)c2n1)C(=O)N1CCO[C@@H](C)C1)c1ccc(F)cn1 |r|
CC(C)S(=O)(=O)c1cn(-c2cc(C)[nH]n2)c2nc(N[C@@H](C)c3ccc(F)cn3)ccc12 |r|
O=C(CSc1ncnc2n(ncc12)-c1ccccc1)Nc1cc(nn1-c1ccccc1)C1CC1
O=C(COC(=O)c1ccc2ncsc2c1)Nc1ccc2ccccc2c1
Clc1ccc(C#N)c(NC(=O)COC(=O)CCCc2c[nH]c3ccccc23)c1
FC(F)(F)Oc1ccc(NC(=O)COC(=O)c2ccc3ncsc3c2)cc1
Cc1cc(cc(n1)C#Cc2ccc3c(c2)oc4c3C(=O)c5ccc(cc5C4(C)C)NS(=O)(=O)C)C(=O)NC(C)(C)C
COc1ccc(NC(=O)COC(=O)c2n[nH]c3ccccc23)cc1OC
CC(C)(C)c1cc(NC(=O)CSc2nnnn2-c2ccccc2)n(n1)-c1ccccc1
CC(C)(C)c1cc(NC(=O)COC(=O)c2ccc(cc2)-n2cnnn2)n(n1)-c1ccccc1
CC(C)(C)c1cc(NC(=O)CSc2nnc(-c3cccnc3)n2C2CC2)n(n1)-c1ccccc1
Cc1ccc(cc1)-c1cc(NC(=O)CSc2n[nH]c(N)n2)n(n1)-c1ccccc1
O=C(CSc1nnnn1Cc1ccco1)Nc1cc(nn1-c1ccccc1)-c1ccccc1
CC(C)(C)c1cc(NC(=O)COC(=O)c2ccc(cc2)C#N)n(n1)-c1ccccc1
CC(C)(C)c1ccc(NC(=O)COC(=O)c2ccc3ncsc3c2)cc1
O=C(COC(=O)c1ccc(cc1)-n1cnnn1)Nc1ccc2ccccc2c1
CC(C)(C)c1cc(NC(=O)COC(=O)c2ccc3C(=O)N4CCCC4Nc3c2)n(n1)-c1ccccc1
NC(=O)c1c(NC(=O)COC(=O)CCCc2c[nH]c3ccccc23)sc2CCCc12
NC(=O)c1c(NC(=O)COC(=O)CCC(=O)c2ccc(Cl)cc2)sc2CCCc12
COc1cc(CCC(=O)OCC(=O)Nc2cc(nn2-c2ccccc2)C(C)(C)C)cc(OC)c1OC
CC(C)(C)c1cc(NC(=O)COC(=O)c2ccccc2O)n(n1)-c1ccccc1
CC(C)(C)c1cc(NC(=O)COC(=O)CC2Sc3ccccc3NC2=O)n(n1)-c1ccccc1
CCOc1ccccc1-n1nnnc1SCC(=O)Nc1cc(nn1-c1ccccc1)C(C)(C)C
Cc1cc(NC(=O)CSc2nnnn2-c2ccc(O)cc2)n(n1)-c1ccc(C)cc1
OCc1ccc(cc1)C(=O)OCC(=O)Nc1cccc(c1)C(F)(F)F
FC(F)(F)c1ccc(NC(=O)COC(=O)c2ccc3ncsc3c2)cc1
COc1ccc(cc1)-n1nnnc1SCC(=O)Nc1cc(nn1-c1ccccc1)C(C)(C)C
Cc1cc(NC(=O)CSc2nccn2Cc2ccccc2)n(n1)-c1ccccc1
CC(C)(C)c1cc(NC(=O)COC(=O)c2cnc(Cl)c(Cl)c2)n(n1)-c1ccccc1
CCC(C)c1ccc(NC(=O)COC(=O)c2ccc3ncsc3c2)cc1
Cc1cc(C)cc(c1)-c1cc(NC(=O)CSc2nnc(o2)C2CC2)n(n1)-c1ccccc1
CC(=O)Nc1ccc(cc1)C(=O)OCC(=O)Nc1cc(nn1-c1ccccc1)C(C)(C)C
FC(F)(F)c1ccc(N2CCOCC2)c(NC(=O)COC(=O)Cc2cccc3ccccc23)c1
CCCN([C@@H]1Cc2ccc(cc2C1)C(=O)Nc1cc(cc(c1)C(F)(F)F)-n1cnc(C)c1)c1cncnc1 |r|
Cc1cn(cn1)-c1cc(NC(=O)c2ccc3C[C@@H](Cc3c2)Nc2cncnc2)cc(c1)C(F)(F)F |r|
CCN([C@@H]1Cc2ccc(cc2C1)C(=O)Nc1cc(cc(c1)C(F)(F)F)-n1cnc(C)c1)c1cncnc1 |r|
CCc1cc(NC(=O)c2ccc3C[C@H](Cc3c2)N(C)c2cncnc2)cc(c1)-n1cnc(C)c1 |r|
CC(C)c1cc(NC(=O)c2ccc3C[C@H](Cc3c2)N(C)c2cncnc2)cc(c1)-n1cnc(C)c1 |r|
CN([C@@H]1Cc2ccc(cc2C1)C(=O)Nc1cc(cc(c1)C12CC3CC(CC(C3)C1)C2)-n1cnc(C)c1)c1cncnc1 |r,TLB:18:20:23:27.25.26,THB:25:24:21:27.26.28,25:26:23.24.29:21,28:26:23:29.20.21,28:20:23:27.25.26|
C[C@H]1CN(Cc2cc(ccc12)C(=O)Nc1cc(cc(c1)C(F)(F)F)-n1cnc(C)c1)c1cncnc1 |r|
Cc1cn(cn1)-c1cc(NC(=O)c2ccc3CN(Cc4cncnc4)Cc3c2)cc(c1)C(F)(F)F
Cc1cn(cn1)-c1cc(NC(=O)c2ccc3CC(C)(Cc3c2)Nc2cncnc2)cc(c1)C(F)(F)F
CN([C@@H]1Cc2ccc(cc2C1)C(=O)Nc1cc(cc(c1)C(F)(F)F)-n1cnc(C)c1)c1cncnc1 |r|
Cc1cn(cn1)-c1cc(NC(=O)c2ccc3C[C@H](Cc3c2)Nc2cncnc2)cc(c1)C(F)(F)F |r|
CN([C@@H]1Cc2ccc(cc2C1)C(=O)Nc1cc(cc(c1)-n1cnc(C)c1)C1CCCCC1)c1cncnc1 |r|
CN([C@@H]1Cc2ccc(cc2C1)C(=O)Nc1cc(C)cc(c1)-n1cnc(C)c1)c1cncnc1 |r|
CN([C@@H]1Cc2ccc(cc2C1)C(=O)Nc1cc(cc(c1)C(C)(C)C)-n1cnc(C)c1)c1cncnc1 |r|
Cc1cn(cn1)-c1cc(NC(=O)c2ccc3CN(Cc3c2)c2cncnc2)cc(c1)C(F)(F)F
COc1cc(ccc1OCc2ccc(cc2)C3CC3)C4CN(C4)C(=O)c5cc(ccn5)COC[C@H](CO)O
CCc1ccc2n(C)c(C)c(C(=O)Nc3ccc(Oc4ncnc5cc(OC)c(OC)cc45)c(F)c3)c(=O)c2c1
Cc1c(cccc1-n1cnc2ccccc2c1=O)-c1ccc(C(O)=N)c2[nH]c3cc(ccc3c12)C(C)(C)O
Cc1sc(cc1-c1cnn2cc(Cl)cnc12)C(=O)N[C@@H]1[C@H](N)CCCC1(F)F |r|
FC(F)(F)CNC(=O)c1cc(cs1)-c1cnn2cc(cnc12)-c1ccc(OCCN2CCCCC2)cc1
Cn1cc(cn1)-c1cnc2c(cnn2c1)-c1csc(c1)C(=O)NCC(F)(F)F
Cn1cc(cn1)-c1cnc2c(cnn2c1)-c1csc(c1)C(=O)N[C@@H]1CCCC[C@@H]1N |r|
COc1ccc(cc1OC)-c1cnn2c(N)c(-c3ccccc3)c(OC3CCN(C)CC3)nc12
COC(=O)Nc1ccc(cc1)-c1c(OC2CCN(C)CC2)nc2c(cnn2c1N)-c1ccc(OC)c(OC)c1
COc1ccc(cc1OC)-c1cnn2c(N)c(-c3nccs3)c(OC3CCN(C)CC3)nc12
[H][C@]1(O)CCN(C1)C(=O)Nc1cnn2ccc(nc12)N1CCC[C@@]1([H])c1cc(F)ccc1F |r|
C[C@H]1CCc2ncc(F)cc2[C@@H]2CCCN2c2ccn3ncc(C(=O)N1)c3n2 |r|
Nc1nc2[nH]c(CN3CCN(CC3)c3cc(Cl)cc(Cl)c3)c(CN3CCN(CC3)c3cc(Cl)cc(Cl)c3)c2c(=O)[nH]1
CCCCCCCC(=O)Nc1nc2[nH]c(CN3CCN(Cc4ccc(F)cc4)CC3)c(CN3CCN(Cc4ccc(F)cc4)CC3)c2c(=O)[nH]1
CCCCCCCC(=O)Nc1nc2[nH]c(CN3CCN(Cc4cccc(F)c4)CC3)c(CN3CCN(Cc4cccc(F)c4)CC3)c2c(=O)[nH]1
CCCCCCCC(=O)Nc1nc2[nH]c(CN3CCN(Cc4ccccc4F)CC3)c(CN3CCN(Cc4ccccc4F)CC3)c2c(=O)[nH]1
CCCCCCCC(=O)Nc1nc2[nH]c(CN3CCN(Cc4ccccc4)CC3)c(CN3CCN(Cc4ccccc4)CC3)c2c(=O)[nH]1
C[C@@H](N(C)c1ccn2ncc(NC(=S)N3CC[C@H](O)C3)c2n1)c1cc(F)ccc1F |r|
C[C@@H](N(C)c1ccn2ncc(Nc3c(N4CC[C@H](O)C4)c(=O)c3=O)c2n1)c1cc(F)ccc1F |r|
C[C@@H](N(C)c1ccn2ncc(NC(=O)N(C)CCN(C)C)c2n1)c1cc(F)ccc1F |r|
C[C@@H](N(C)c1ccn2ncc(NC(=O)N3CCN(C)CC3)c2n1)c1cc(F)ccc1F |r|
CC(C)N(C(C)C)C(=O)Nc1cnn2ccc(nc12)N(C)[C@H](C)c1cc(F)ccc1F |r|
C[C@@H](N(C)c1ccn2ncc(NC(=O)N3CC(O)C3)c2n1)c1cc(F)ccc1F |r|
CCC(CO)NC(=O)Nc1cnn2ccc(nc12)N(C)[C@H](C)c1cc(F)ccc1F |r|
C[C@@H](N(C)c1ccn2ncc(NC(=O)N3CCCC(CO)C3)c2n1)c1cc(F)ccc1F |r|
C[C@@H](N(C)c1ccn2ncc(NC(=O)Nc3ccc(O)cc3)c2n1)c1cc(F)ccc1F |r|
C[C@@H](N(C)c1ccn2ncc(NC(=O)N3CC[C@H](O)C3)c2n1)c1cc(F)ccc1F |r|
C[C@@H](Nc1ccn2ncc(NC(=S)N3CC[C@H](O)C3)c2n1)c1cc(F)ccc1F |r|
C[C@@H](Nc1ccn2ncc(Nc3c(N4CC[C@H](O)C4)c(=O)c3=O)c2n1)c1cc(F)ccc1F |r|
C[C@@H](Nc1ccn2ncc(NC(=O)N(C)CCN(C)C)c2n1)c1cc(F)ccc1F |r|
C[C@@H](Nc1ccn2ncc(NC(=O)N3CCN(C)CC3)c2n1)c1cc(F)ccc1F |r|
CC(C)N(C(C)C)C(=O)Nc1cnn2ccc(N[C@H](C)c3cc(F)ccc3F)nc12 |r|
C[C@@H](Nc1ccn2ncc(NC(=O)N3CC(O)C3)c2n1)c1cc(F)ccc1F |r|
CCC(CO)NC(=O)Nc1cnn2ccc(N[C@H](C)c3cc(F)ccc3F)nc12 |r|
C[C@@H](Nc1ccn2ncc(NC(=O)N3CCCC(CO)C3)c2n1)c1cc(F)ccc1F |r|
C[C@@H](Nc1ccn2ncc(NC(=O)Nc3ccc(O)cc3)c2n1)c1cc(F)ccc1F |r|
C[C@@H](Nc1ccn2ncc(NC(=O)N3CC[C@H](O)C3)c2n1)c1cc(F)ccc1F |r|
CC(C)n1cc(c2c1ncnc2N)C(=O)c3ccnc(c3)NC(=O)Nc4ccc(cc4F)F
CC(C)n1cc(C(=O)c2ccnc(NC(=O)Cc3ccc(F)cc3F)c2)c2c(N)ncnc12
CC(C)n1cc(c2c1ncnc2N)C(=O)c3cc(cnc3)NC(=O)Cc4ccc(cc4)Cl
CC(C)n1cc(C(=O)c2cncc(NC(=O)Cc3ccc(cc3)C#N)c2)c2c(N)ncnc12
CC(C)(CO)n1cc(C(=O)c2cncc(NC(=O)Cc3ccc(Cl)cc3)c2)c2cnc(N)nc12
CC(C)(CO)n1cc(c2c1nc(nc2)N)C(=O)c3cc(cnc3)NC(=O)Cc4ccc(cn4)Cl
CC(C)(C)c1cc(NC(=O)Nc2ccc3oc(cc3c2)C(=O)c2cc3cc(O)ccc3[nH]2)no1
CN1CCC(CNC2=NC(=O)\C(S2)=C\c2csc(n2)-c2ccc(OC(F)(F)F)cc2)CC1 |t:7|
OC1CCN(CC1)c1cc(ccn1)-c1cccc(n1)-c1cnc2ccc(nn12)N1CCC[C@@H]1c1cccc(F)c1 |r|
Fc1cccc(c1)[C@H]1CCCN1c1ccc2ncc(-c3cccc(n3)N3CCN(CC3)C(=O)CCCCCNc3cccc4C(=O)N(C5CCC(=O)NC5=O)C(=O)c34)n2n1 |r|
Fc1cccc(c1)[C@H]1CCCN1c1ccc2ncc(-c3cccc(n3)N3CCN(CC3)C(=O)CCOCCNc3cccc4C(=O)N(C5CCC(=O)NC5=O)C(=O)c34)n2n1 |r|
CN1C(=O)CCC(N2C(=O)c3cccc(NCCCCCC(=O)N4CCN(CC4)c4cccc(n4)-c4cnc5ccc(nn45)N4CCC[C@@H]4c4cccc(F)c4)c3C2=O)C1=O |r|
CN1C(=O)CCC(N2C(=O)c3cccc(NCCOCCC(=O)N4CCN(CC4)c4cccc(n4)-c4cnc5ccc(nn45)N4CCC[C@@H]4c4cccc(F)c4)c3C2=O)C1=O |r|
COc1cccc2nc(Nc3cccc(NC(=O)c4ccc(N5CCN(C)CC5)c(c4)C(F)(F)F)c3)ccc12
CCN1CCN(CC1)c1cc(cc(c1)C(F)(F)F)C(=O)Nc1cccc(Nc2ccc3c(OC)cccc3n2)c1
Cc1nc2nc(nn2c(C)c1CC(=O)Nc1cccc(c1)C(F)(F)F)-c1cccnc1
NC(=O)c1ccc(cc1)-c1nnn(CC(=O)Nc2cc(ccc2-n2cncn2)C(F)(F)F)n1
COc1ccc(cc1NC(=O)Nc2ccc3c(c2)sc(n3)NC(=O)c4ccccc4)Cl
O=C(Nc1ccc(cc1N1CCOCC1)N1CCOCC1)c1cnn(n1)-c1ccccc1
COc1ccc(cc1)-n1ncc2c1ncn(CC(=O)Nc1cc(ccc1Cl)C(F)(F)F)c2=O
c1ccc(cc1)Oc2cccc(c2)C(=O)Nc3ccc(cc3N4CCOCC4)N5CCOCC5
CN1CCN(CCCOc2cccc3nc(Nc4ccc(Cl)c(c4)C(F)(F)F)ccc23)CC1
Nc1ncnc2n(CC3CCN(CC3)C(=O)C=C)cc(-c3ccc4OCOc4c3)c12
CNS(=O)(=O)c1ccc2NC(=O)\C(=C/c3cn(C)c4ccc(OC)cc34)c2c1
CN(C)S(=O)(=O)c1ccc2NC(=O)\C(=C/c3cn(C)c4ccc(O)cc34)c2c1
COc1ccc2[nH]cc(\C=C3/C(=O)Nc4ccccc34)c2c1
Cn1cc(\C=C2/C(=O)Nc3ccc(cc23)S(N)(=O)=O)c2ccccc12
COc1ccc2n(C)cc(\C=C3/C(=O)Nc4ccc(cc34)S(N)(=O)=O)c2c1
NS(=O)(=O)c1ccc2NC(=O)\C(=C/c3c[nH]c4ccccc34)c2c1
O=C1Nc2ccccc2\C1=C/c1c[nH]c2ccccc12
Cn1cc(\C=C2/C(=O)Nc3ccccc23)c2ccccc12
COc1ccc2[nH]cc(\C=C3/C(=O)Nc4ccc(cc34)S(N)(=O)=O)c2c1
COc1ccc2n(C)cc(\C=C3/C(=O)Nc4ccc(cc34)S(=O)(=O)N(C)C)c2c1
NS(=O)(=O)c1ccc2NC(=O)\C(=C/c3c[nH]c4ccc(O)cc34)c2c1
Cc1[nH]c2ccccc2c1\C=C1/C(=O)Nc2ccccc12
Clc1[nH]c2ccccc2c1\C=C1\C(=O)Nc2ccccc12
NS(=O)(=O)c1ccc(N\C=C2/C(=O)Nc3ccccc23)cc1
O=C1Nc2ccc3ncsc3c2\C1=C\Nc1ccc(cc1)S(=O)(=O)Nc1ccccn1
Cc1ccc(NC(=O)c2ccc(C)c(c2)C(F)(F)F)cc1C#Cc1nn([C@H]2CC[C@H](O)CC2)c2ncnc(N)c12 |r,wU:26.27,wD:29.31,(-5.46,5.4,;-3.98,5.8,;-3.58,7.29,;-2.09,7.69,;-1,6.6,;.49,7,;1.57,5.91,;1.18,4.42,;3.06,6.31,;3.46,7.79,;4.95,8.19,;6.04,7.1,;7.53,7.5,;5.64,5.62,;4.15,5.22,;6.73,4.53,;8.22,4.93,;6.33,3.04,;7.82,3.44,;-1.4,5.11,;-2.89,4.71,;-3.29,3.22,;-3.68,1.74,;-4.08,.25,;-3.18,-1,;-4.08,-2.24,;-3.68,-3.73,;-2.2,-4.13,;-1.8,-5.62,;-2.89,-6.7,;-2.49,-8.19,;-4.38,-6.31,;-4.77,-4.82,;-5.55,-1.77,;-6.88,-2.54,;-8.22,-1.77,;-8.22,-.23,;-6.88,.54,;-6.88,2.08,;-5.55,-.23,)|
CC(C)(C)c1cc(NC(=O)Nc2ccc(Nc3ncnc4NCCCOc34)cc2)no1
Fc1ccc2NC(=O)C(=C3/Nc4ccccc4/C/3=NOCCN3CCNCC3)c2c1
Fc1cc(F)cc(Cc2ccc3[nH]nc(\C=C\c4ccccn4)c3c2)c1
Fc1cc(F)cc(c1)-c1ccc2[nH]nc(\C=C\c3ccccn3)c2c1
Fc1cc(F)cc(Sc2ccc3[nH]nc(\C=C\c4ccccn4)c3c2)c1
Fc1cc(F)cc(Oc2ccc3[nH]nc(\C=C\c4ccccn4)c3c2)c1
Fc1cc(F)cc(Nc2ccc3[nH]nc(\C=C\c4ccccn4)c3c2)c1
CN(c1ccc2[nH]nc(\C=C\c3ccccn3)c2c1)c1cc(F)cc(F)c1
Fc1cc(F)cc(CCc2ccc3[nH]nc(\C=C\c4ccccn4)c3c2)c1
Fc1cc(F)cc(c1)C#Cc1ccc2[nH]nc(\C=C\c3ccccn3)c2c1
Fc1cc(F)cc(NC(=O)c2ccc3[nH]nc(\C=C\c4ccccn4)c3c2)c1
Fc1cc(F)cc(c1)C(=O)Nc1ccc2[nH]nc(\C=C\c3ccccn3)c2c1
Fc1cc(F)cc(COc2ccc3[nH]nc(\C=C\c4ccccn4)c3c2)c1
Fc1cc(F)cc(OCc2ccc3[nH]nc(\C=C\c4ccccn4)c3c2)c1
Fc1cc(F)cc(CNc2ccc3[nH]nc(\C=C\c4ccccn4)c3c2)c1
Fc1cc(F)cc(NCc2ccc3[nH]nc(\C=C\c4ccccn4)c3c2)c1
CN(Cc1cc(F)cc(F)c1)c1ccc2[nH]nc(\C=C\c3ccccn3)c2c1
CN(Cc1ccc2[nH]nc(\C=C\c3ccccn3)c2c1)c1cc(F)cc(F)c1
C(Nc1ccc2[nH]nc(\C=C\c3ccccn3)c2c1)c1ccccc1
Fc1ccccc1CNc1ccc2[nH]nc(\C=C\c3ccccn3)c2c1
Fc1cccc(CNc2ccc3[nH]nc(\C=C\c4ccccn4)c3c2)c1
Fc1ccc(CNc2ccc3[nH]nc(\C=C\c4ccccn4)c3c2)cc1
Fc1cc(Cl)cc(CNc2ccc3[nH]nc(\C=C\c4ccccn4)c3c2)c1
Fc1cc(Br)cc(CNc2ccc3[nH]nc(\C=C\c4ccccn4)c3c2)c1
Cc1cc(F)cc(CNc2ccc3[nH]nc(\C=C\c4ccccn4)c3c2)c1
COc1cc(F)cc(CNc2ccc3[nH]nc(\C=C\c4ccccn4)c3c2)c1
Fc1cc(CNc2ccc3[nH]nc(\C=C\c4ccccn4)c3c2)cc(c1)C(F)(F)F
Fc1cc(CNc2ccc3[nH]nc(\C=C\c4ccccn4)c3c2)cc(c1)C#N
C[C@H](Nc1ccc2[nH]nc(\C=C\c3ccccn3)c2c1)c1cc(F)cc(F)c1 |r|
C[C@@H](Nc1ccc2[nH]nc(\C=C\c3ccccn3)c2c1)c1cc(F)cc(F)c1 |r|
CN1CCN(CC(=O)Nc2nc(C)c(s2)-c2ccc3c(\C=C\c4ccccn4)n[nH]c3c2)CC1
COc1cc(OC)c(F)c(N2Cc3cnc4[nH]c(cc4c3N(C)C2=O)-c2cnn(C)c2)c1F
COc1cc(OC)c(F)c(N2Cc3cnc4[nH]ccc4c3N(C)C2=O)c1F
CCc1cc(Nc2nc(NCc3ccc(Cl)cc3OC)nc3cccc(OC)c23)n[nH]1
Fc1cc(F)cc(Nc2ncc(Cl)c(n2)N2CCC[C@H]2C(=O)Nc2ccc(N3CCOCC3)c(c2)C(=O)N2CCSCC2)c1 |r|
CN1CCN(CC1)C(=O)c1cc(NC(=O)[C@@H]2CCCN2c2nc(Nc3cc(F)cc(F)c3)ncc2Cl)ccc1N1CCOCC1 |r|
CN(C)C(=O)c1cc(NC(=O)[C@@H]2CCCN2c2nc(Nc3cc(F)cc(F)c3)ncc2Cl)ccc1N1CCN(C)CC1 |r|
CN1CCN(CC1)c1ccc(NC(=O)[C@@H]2CCCN2c2nc(Nc3cc(F)cc(F)c3)ncc2Cl)cc1C(=O)N1CCSCC1 |r|
O[C@H]1CCCC[C@@H]1NC(=O)Cc1ccc(Nc2ncnc3ccsc23)cc1 |r|
O[C@H]1CCCC[C@H]1NC(=O)Cc1ccc(Nc2ncnc3ccsc23)cc1 |r|
FC(F)(F)c1cccc(NC(=O)Cc2ccc(Nc3ncnc4ccsc34)cc2)c1
O=C(Cc1ccc(Nc2ncnc3ccsc23)cc1)Nc1cccc(c1)C#C
Cn1nc(cc1NC(=O)Cc1ccc(Nc2ncnc3ccsc23)cc1)C(C)(C)C
CC(C)(C)c1cc(NC(=O)Cc2ccc(Nc3ncnc4ccsc34)cc2)no1
Cn1cc(cn1)-c1cc2ncnc(Nc3ccc(CC(=O)Nc4cccc(c4)C(F)(F)F)cc3)c2s1
Cn1cc(cn1)-c1cc2ncnc(Nc3ccc(CC(=O)Nc4cccc(c4)C#C)cc3)c2s1
Cn1cc(cn1)-c1cc2ncnc(Nc3ccc(CC(=O)Nc4cc(nn4C)C(C)(C)C)cc3)c2s1
Cn1cc(cn1)-c1cc2ncnc(Nc3ccc(CC(=O)Nc4nc(cs4)C(C)(C)C)cc3)c2s1
Cn1cc(cn1)-c1cc2ncnc(Nc3ccc(CC(=O)Nc4cc(nn4CCN4CCOCC4)C(C)(C)C)cc3)c2s1
Cn1cc(cn1)-c1cc2ncnc(Nc3ccc(CC(=O)Nc4ccc5OCCOc5c4)cc3)c2s1
Cn1cc(cn1)-c1cc2ncnc(Nc3ccc(CC(=O)Nc4ccc(cc4)C(C)(C)C)cc3)c2s1
Cn1cc(cn1)-c1cc2ncnc(Nc3ccc(CC(=O)Nc4ccc(F)c(Cl)c4)cc3)c2s1
Cn1cc(cn1)-c1cc2ncnc(Nc3ccc(CC(=O)NCc4cccc(F)c4)cc3)c2s1
Cn1cc(cn1)-c1cc2ncnc(Nc3ccc(CC(=O)Nc4cccnc4)cc3)c2s1
Cn1cc(cn1)-c1cc2ncnc(Nc3ccc(NC(=O)Nc4cc(nn4C)C(C)(C)C)cc3)c2s1
CS(=O)(=O)c1ccc(cc1)-c1cc2ncnc(Nc3ccc(CC(=O)Nc4ccc(F)c(Cl)c4)cc3)c2s1
COc1cc(cc(OC)c1OC)-c1cc2ncnc(Nc3ccc(CC(=O)Nc4ccc(F)c(Cl)c4)cc3)c2s1
Fc1ccc(NC(=O)Cc2ccc(Nc3ncnc4cc(sc34)-c3ccc(OCCN4CCCC4)cc3)cc2)cc1Cl
CNC(=O)c1ccc(Nc2ncc(c(NCc3ccccc3Cl)n2)C(F)(F)F)cc1
CNC(=O)c1ccc(Nc2ncc(c(Nc3ccccc3OC)n2)C(F)(F)F)cc1
CNC(=O)c1ccc(cc1)Nc2ncc(c(n2)NCc3c(nccn3)N(C)S(=O)(=O)C)C(F)(F)F
Nc1ncnc2n(cc(-c3cccc(O)c3)c12)[C@@H]1C[C@H](CO)C1 |r,wU:17.19,19.22,(11.65,-9.07,;11.66,-10.61,;12.99,-11.37,;13,-12.92,;11.66,-13.69,;10.32,-12.92,;8.86,-13.4,;7.95,-12.16,;8.85,-10.91,;8.37,-9.46,;6.87,-9.15,;6.38,-7.69,;7.41,-6.53,;8.92,-6.85,;9.95,-5.7,;9.4,-8.31,;10.32,-11.38,;8.4,-14.88,;7.03,-15.58,;7.73,-16.95,;7.26,-18.42,;8.3,-19.56,;9.1,-16.25,)|
Nc1ncnc2n(cc(-c3cccc(O)c3)c12)C1CCCC1
CC(=O)N1CCN(CC1)[C@H]1C[C@H](C1)n1cc(-c2cc(O)ccc2F)c2c(N)ncnc12 |r,wU:11.14,9.9,(5.38,-23.19,;6.89,-22.87,;7.92,-24.01,;7.36,-21.4,;6.33,-20.26,;6.8,-18.8,;8.31,-18.48,;9.35,-19.61,;8.87,-21.08,;8.78,-17.01,;8.08,-15.64,;9.45,-14.94,;10.15,-16.31,;9.91,-13.47,;9,-12.23,;9.9,-10.98,;9.42,-9.52,;10.45,-8.37,;9.97,-6.91,;11,-5.76,;8.46,-6.59,;7.43,-7.75,;7.92,-9.21,;6.9,-10.36,;11.37,-11.45,;12.7,-10.67,;12.7,-9.13,;14.04,-11.43,;14.05,-12.98,;12.71,-13.76,;11.37,-12.99,)|
CCC[C@H](C)Nc1ncc2c(cn([C@H]3CC[C@H](O)CC3)c2n1)C1CCN(CC1)C(=O)c1cc(C)nc(C)c1 |r,wU:13.12,wD:3.3,16.16,(-8.93,-2.23,;-7.59,-1.46,;-6.26,-2.23,;-4.93,-1.46,;-4.93,.08,;-3.59,-2.23,;-2.26,-1.46,;-2.26,.08,;-.93,.85,;.41,.08,;1.87,.56,;2.78,-.69,;1.87,-1.94,;2.35,-3.4,;3.85,-3.72,;4.33,-5.19,;3.3,-6.33,;3.78,-7.79,;1.79,-6.01,;1.32,-4.55,;.41,-1.46,;-.93,-2.23,;2.35,2.02,;3.85,2.34,;4.33,3.81,;3.3,4.95,;1.79,4.63,;1.32,3.16,;3.78,6.41,;3.04,7.77,;5.26,6.02,;6.35,7.1,;7.84,6.71,;8.93,7.79,;8.24,5.22,;7.15,4.13,;7.55,2.64,;5.66,4.53,)|
CC1(C)N(Cc2ccccc2)Cc2c(NC(=O)c3ccccc3)n[nH]c12
Cc1cccc(CN2Cc3c(NC(=O)c4ccccc4)n[nH]c3C2(C)C)c1
COc1cccc(CN2Cc3c(NC(=O)c4ccccc4)n[nH]c3C2(C)C)c1
CC1(C)N(Cc2cccc(c2)C#N)Cc2c(NC(=O)c3ccccc3)n[nH]c12
CC1(C)N(Cc2cccc(I)c2)Cc2c(NC(=O)c3ccccc3)n[nH]c12
CC1(C)N(Cc2cccc(Br)c2)Cc2c(NC(=O)c3ccccc3)n[nH]c12
CC1(C)N(Cc2cccc(Cl)c2)Cc2c(NC(=O)c3ccccc3)n[nH]c12
CC1(C)N(Cc2cccc(F)c2)Cc2c(NC(=O)c3ccccc3)n[nH]c12
CC1(C)N(Cc2cccc(c2)[N+]([O-])=O)Cc2c(NC(=O)c3ccccc3)n[nH]c12
O[C@@H]1CCN(C1)C(=O)Nc1cnn2ccc(nc12)N1CCC[C@H]1c1cc(F)ccc1F |r|
CC1(C)N(Cc2ccccc2F)Cc2c(NC(=O)c3ccccc3)n[nH]c12
CC1(C)N(Cc2ccc(F)cc2)Cc2c(NC(=O)c3ccccc3)n[nH]c12
CC1(C)N(Cc2cc(F)cc(F)c2)Cc2c(NC(=O)c3ccccc3)n[nH]c12
CC1(C)N(Cc2cccc(F)c2F)Cc2c(NC(=O)c3ccccc3)n[nH]c12
CC1(C)N(Cc2cc(F)ccc2F)Cc2c(NC(=O)c3ccccc3)n[nH]c12
CC1(C)N(Cc2ccc(F)c(F)c2)Cc2c(NC(=O)c3ccccc3)n[nH]c12
CC1(C)N(Cc2ccc(F)cc2F)Cc2c(NC(=O)c3ccccc3)n[nH]c12
CC1(C)N(Cc2c(F)cccc2F)Cc2c(NC(=O)c3ccccc3)n[nH]c12
Cc1ccc(CN2Cc3c(NC(=O)c4ccccc4)n[nH]c3C2(C)C)cc1F
Cc1ccc(F)c(CN2Cc3c(NC(=O)c4ccccc4)n[nH]c3C2(C)C)c1
CC1(C)N(Cc2cc(cc(c2)C(F)(F)F)C(F)(F)F)Cc2c(NC(=O)c3ccccc3)n[nH]c12
CC1(C)N(Cc2cc(F)cc(c2)C(F)(F)F)Cc2c(NC(=O)c3ccccc3)n[nH]c12
CC1(C)N(Cc2cc(F)c(F)c(F)c2)Cc2c(NC(=O)c3ccccc3)n[nH]c12
CC1(C)N(Cc2cccc(F)c2F)Cc2c(NC(=O)c3ccc4ccccc4c3)n[nH]c12
CC1(C)N(Cc2cc(F)cc(F)c2)Cc2c(NC(=O)c3ccc4ccccc4c3)n[nH]c12
CC1(C)N(Cc2cc(F)cc(F)c2)Cc2c(NC(=O)c3ccc4ncccc4c3)n[nH]c12
CC1(C)N(Cc2cccc(F)c2F)Cc2c(NC(=O)c3ccc(F)cc3)n[nH]c12
CC1(C)N(Cc2cc(F)cc(F)c2)Cc2c(NC(=O)c3ccc(F)cc3)n[nH]c12
CC1(C)N(Cc2cccc(F)c2F)Cc2c(NC(=O)c3ccc(Br)cc3)n[nH]c12
CC1(C)N(Cc2cc(F)cc(F)c2)Cc2c(NC(=O)c3ccc(Br)cc3)n[nH]c12
CC1(C)N(Cc2cccc(F)c2F)Cc2c(NC(=O)c3ccc(cc3)N3CCOCC3)n[nH]c12
CC1(C)N(Cc2cc(F)cc(F)c2)Cc2c(NC(=O)c3ccc(cc3)N3CCOCC3)n[nH]c12
CN(C)c1ccc(cc1)C(=O)Nc1n[nH]c2c1CN(Cc1cc(F)cc(F)c1)C2(C)C
CN1CCN(CC1)c1ccc(cc1)C(=O)Nc1n[nH]c2c1CN(Cc1cccc(F)c1F)C2(C)C
CN1CCN(CC1)c1ccc(cc1)C(=O)Nc1n[nH]c2c1CN(Cc1cc(F)cc(F)c1)C2(C)C
CC1(C)N(Cc2cc(F)cc(F)c2)Cc2c(NC(=O)c3ccc(cc3)N3CC[N+](C)(Cc4cc(F)cc(F)c4)CC3)n[nH]c12
CC1(C)N(Cc2cccc(F)c2F)Cc2c(NC(=O)c3cccc(c3)N3CCOCC3)n[nH]c12
CC1(C)N(Cc2cc(F)cc(F)c2)Cc2c(NC(=O)c3cccc(c3)N3CCOCC3)n[nH]c12
CN(C)c1cccc(c1)C(=O)Nc1n[nH]c2c1CN(Cc1cccc(F)c1F)C2(C)C
CN(C)c1cccc(c1)C(=O)Nc1n[nH]c2c1CN(Cc1cc(F)cc(F)c1)C2(C)C
CN1CCN(CC1)c1cccc(c1)C(=O)Nc1n[nH]c2c1CN(Cc1cccc(F)c1F)C2(C)C
CN1CCN(CC1)c1cccc(c1)C(=O)Nc1n[nH]c2c1CN(Cc1cc(F)cc(F)c1)C2(C)C
CN(C)c1ccc(cc1)C(=O)Nc1n[nH]c2c1CN(Cc1cccc(F)c1F)C2(C)C
COCc1ccc(OC(F)(F)F)c(CNC(=O)Nc2c(nc3c(C)nccn23)-c2ccccc2)c1
C[C@H]1CNCc2cnn3ccc(nc23)N(C)Cc2cc(F)ccc2O1 |r|
CN1Cc2cc(F)ccc2OCCN(Cc2cnn3ccc1nc23)S(C)(=O)=O
CCS(=O)(=O)N1CCOc2ccc(F)cc2CN(C)c2ccn3ncc(C1)c3n2
CN1Cc2cc(F)ccc2OCCN(Cc2cnn3ccc1nc23)S(=O)(=O)CCl
CN1Cc2cc(F)ccc2OCCN(Cc2cnn3ccc1nc23)C(C)=O
C[C@H]1CN(Cc2cnn3ccc(nc23)N(C)Cc2cc(F)ccc2O1)S(C)(=O)=O |r|
CCS(=O)(=O)N1C[C@H](C)Oc2ccc(F)cc2CN(C)c2ccn3ncc(C1)c3n2 |r|
C[C@H]1CN(Cc2cnn3ccc(nc23)N(C)Cc2cc(F)ccc2O1)C(C)=O |r|
CCS(=O)(=O)N1CCCOc2ccc(F)cc2CN(C)c2ccn3ncc(C1)c3n2
Fc1cnc2OCC3(CC3)NC(=O)c3cnn4ccc(nc34)N3CCCC[C@@H]3c2c1 |r|
Fc1cnc2OCC3(CC3)NC(=O)c3cnn4ccc(nc34)N3CCNC[C@@H]3c2c1 |r|
Fc1cnc2OCC3(CC3)NC(=O)c3cnn4ccc(nc34)N3CCOC[C@@H]3c2c1 |r|
C[C@H]1CNS(=O)(=O)c2cnn3ccc(N[C@H](C)c4cc(F)ccc4O1)nc23 |r|
C[C@H]1Nc2ccn3ncc(C(=O)N[C@H](C)C(=O)Nc4ccc(F)cc14)c3n2 |r|
C[C@H]1Nc2ccn3ncc(C(=O)N4CCC(CC4)c4ccc(F)cc14)c3n2 |r,wD:1.0,(25.51,-11.86,;25.1,-13.39,;23.21,-13.56,;21.78,-14.28,;20.43,-13.42,;19,-14.14,;18.92,-15.74,;17.67,-16.75,;18.24,-18.26,;19.85,-18.18,;21.19,-18.94,;21.18,-20.52,;22.51,-18.19,;23.83,-18.95,;25.16,-18.19,;25.16,-16.65,;23.79,-15.86,;22.51,-16.61,;26.48,-15.89,;27.81,-16.65,;29.14,-15.89,;29.13,-14.34,;30.45,-13.58,;27.81,-13.59,;26.48,-14.35,;20.26,-16.62,;21.69,-15.89,)|
C[C@H]1Nc2ccn3ncc(C(=O)N4CCN(CC4)c4ccc(F)cc14)c3n2 |r|
C[C@@H]1COc2ncc(F)cc2C23CC2CCN3c2ccn3ncc(C(=O)N1)c3n2 |r|
Cn1cc(cn1)-c1cnn2ccc(nc12)N1CCC[C@@H]1c1cc(F)ccc1F |r|
Cn1cc(cn1)-c1cnn2ccc(nc12)N1CCC[C@@H]1c1cc(F)ccc1OCC(F)F |r|
C[C@@H](Nc1ccn2ncc(-c3cnn(C)c3)c2n1)c1cc(F)ccc1OCC(F)F |r|
C[C@@H](Nc1ccn2ncc(-c3cnn(CCO)c3)c2n1)c1cc(F)ccc1OCC(F)F |r|
CC1(C)Oc2c(Nc3ccc(NC(=O)Nc4ccc(Cl)c(c4)C(F)(F)F)cc3)ncnc2NC1=O
CC1(C)Oc2c(Nc3ccc(NC(=O)Nc4cccc(c4)C(F)(F)F)cc3)ncnc2NC1=O
CC1(C)Oc2c(Nc3ccc(NC(=O)Nc4cc(cc(c4)C(F)(F)F)C(F)(F)F)cc3)ncnc2NC1=O
CC(C)(C)c1cc(NC(=O)Nc2ccc(Nc3ncnc4NC(=O)C(C)(C)Oc34)cc2)no1
CC(C)(C)c1cc(NC(=O)Nc2ccc(Nc3ncnc4NC(=O)C(C)(C)Oc34)cc2)on1
CC(C)(C)c1cc(NC(=O)Nc2ccc(Nc3ncnc4NC(=O)C(C)(C)Oc34)cc2)n(n1)C(C)(C)C
CC(C)(C)c1cc(NC(=O)Nc2ccc(Nc3ncnc4NC(=O)C(C)(C)Oc34)cc2)n(n1)C1CCCCC1
CC(C)(C)c1cc(NC(=O)Nc2ccc(Nc3ncnc4NC(=O)C(C)(C)Oc34)cc2)n(n1)-c1ccccc1
CC(C)(C)c1cc(NC(=O)Nc2cccc(Nc3ncnc4NC(=O)C(C)(C)Oc34)c2)n(n1)-c1ccccc1
CC(C)(C)c1cc(NC(=O)Nc2ccc(Nc3ncnc4NC(=O)C(C)(C)Oc34)c3ccccc23)n(n1)-c1ccccc1
CC(C)(C)c1cc(NC(=O)Nc2ccc(Nc3ncnc4NC(=O)C(C)(C)Oc34)cc2F)n(n1)-c1ccccc1
CSc1cc(Nc2ncnc3NC(=O)C(C)(C)Oc23)ccc1NC(=O)Nc1cc(nn1-c1ccccc1)C(C)(C)C
CC(C)(C)c1cc(NC(=O)Nc2ccc(Nc3ncnc4NC(=O)C(C)(C)Oc34)cc2C(F)(F)F)n(n1)-c1ccccc1
Cc1cc(Nc2ncnc3NC(=O)C(C)(C)Oc23)ccc1NC(=O)Nc1cc(nn1-c1ccccc1)C(C)(C)C
Cc1cc(NC(=O)Nc2cc(nn2-c2ccccc2)C(C)(C)C)ccc1Nc1ncnc2NC(=O)C(C)(C)Oc12
COc1cc(Nc2ncnc3NC(=O)C(C)(C)Oc23)ccc1NC(=O)Nc1cc(nn1-c1ccccc1)C(C)(C)C
COc1cc(NC(=O)Nc2cc(nn2-c2ccccc2)C(C)(C)C)ccc1Nc1ncnc2NC(=O)C(C)(C)Oc12
Cc1cc(NC(=O)Nc2cc(nn2-c2ccc(F)cc2)C(C)(C)C)ccc1Nc1ncnc2NC(=O)C(C)(C)Oc12
Cc1cc(NC(=O)Nc2cc(nn2-c2cccc(F)c2)C(C)(C)C)ccc1Nc1ncnc2NC(=O)C(C)(C)Oc12
Cc1cc(NC(=O)Nc2cc(nn2-c2ccccc2F)C(C)(C)C)ccc1Nc1ncnc2NC(=O)C(C)(C)Oc12
Cc1ccc(cc1)-n1nc(cc1NC(=O)Nc1ccc(Nc2ncnc3NC(=O)C(C)(C)Oc23)c(C)c1)C(C)(C)C
Cc1cc(NC(=O)Nc2cc(nn2-c2ccc(cc2)C(F)(F)F)C(C)(C)C)ccc1Nc1ncnc2NC(=O)C(C)(C)Oc12
Cc1cc(NC(=O)Nc2cc(nn2-c2ccc(OC(F)(F)F)cc2)C(C)(C)C)ccc1Nc1ncnc2NC(=O)C(C)(C)Oc12
Cc1cc(NC(=O)Nc2cc(nn2-c2ccc(Cl)cc2)C(C)(C)C)ccc1Nc1ncnc2NC(=O)C(C)(C)Oc12
Cc1cc(NC(=O)Nc2cc(nn2-c2ccc3ccccc3c2)C(C)(C)C)ccc1Nc1ncnc2NC(=O)C(C)(C)Oc12
Cc1cc(NC(=O)Nc2cc(nn2-c2cccnc2)C(C)(C)C)ccc1Nc1ncnc2NC(=O)C(C)(C)Oc12
Cc1cc(NC(=O)Nc2cc(nn2-c2ccc(F)c(F)c2)C(C)(C)C)ccc1Nc1ncnc2NC(=O)C(C)(C)Oc12
Cc1cc(NC(=O)Nc2cc(nn2-c2c(F)c(F)c(F)c(F)c2F)C(C)(C)C)ccc1Nc1ncnc2NC(=O)C(C)(C)Oc12 |(-6.52,.89,;-5.13,.12,;-3.8,.88,;-2.45,.08,;-1.13,.85,;.24,.12,;.21,-1.47,;1.53,.94,;2.92,.16,;3.1,-1.37,;4.62,-1.66,;5.35,-.31,;4.31,.83,;4.6,2.35,;6.04,2.86,;7.26,1.84,;6.33,4.38,;7.84,4.88,;5.19,5.39,;5.48,6.91,;3.75,4.88,;2.53,5.9,;3.46,3.36,;1.94,2.86,;5.29,-3.05,;6.82,-3.16,;4.53,-4.38,;6.06,-4.38,;-2.46,-1.44,;-3.79,-2.2,;-5.15,-1.48,;-6.48,-2.24,;-6.48,-3.76,;-7.84,-4.55,;-7.84,-6.07,;-6.52,-6.85,;-5.15,-6.13,;-3.83,-6.91,;-2.48,-6.12,;-1.16,-6.89,;-2.47,-4.6,;-1.93,-3.14,;-.92,-4.88,;-3.79,-3.82,;-5.16,-4.54,)|
Cc1cc(NC(=O)Nc2cc(nn2-c2ccccc2)-c2ccccc2)ccc1Nc1ncnc2NC(=O)C(C)(C)Oc12
Cc1cc(NC(=O)Nc2cc(nn2-c2ccccc2)C2CC2)ccc1Nc1ncnc2NC(=O)C(C)(C)Oc12
Cc1ccc(NC(=O)Nc2ccc(Nc3ncnc4NC(=O)C(C)(C)Oc34)cc2)cc1
CC1(C)Oc2c(Nc3ccc(NC(=O)Nc4cccc(F)c4)cc3)ncnc2NC1=O
CC1(C)Oc2c(Nc3ccc(NC(=O)Nc4ccc(F)c(F)c4)cc3)ncnc2NC1=O
CC1(C)Oc2c(Nc3ccc(NC(=O)Nc4ccc(cc4)C#N)cc3)ncnc2NC1=O
CC1(C)Oc2c(Nc3ccc(NC(=O)NC4CCCCC4)cc3)ncnc2NC1=O
[H][C@]12C[C@]3([H])C[C@]([H])(C1)CC(C2)(C3)NC(=O)Nc1ccc(Nc2ncnc3NC(=O)C(C)(C)Oc23)cc1 |r,TLB:8:1:12:6.5.9,8:6:12:2.1.11,THB:2:3:9:1.8.11,2:1:12.3.5:9|
CC(C)(C)NC(=O)Nc1ccc(Nc2ncnc3NC(=O)C(C)(C)Oc23)cc1
CC1(C)Oc2c(Nc3ccc(NC(=O)NCC=C)cc3)ncnc2NC1=O
CCNC(=O)Nc1ccc(Nc2ncnc3NC(=O)C(C)(C)Oc23)cc1
Cn1nc(cc1NC(=O)Nc1ccc(Nc2ncnc3NC(=O)C(C)(C)Oc23)cc1)C(C)(C)C
CC(C)n1nc(cc1NC(=O)Nc1ccc(Nc2ncnc3NC(=O)C(C)(C)Oc23)cc1)C(C)(C)C
CN(C)C(=O)c1ccc(Nc2ncc(c(N[C@@H]3CC[C@H](N)CC3)n2)C(F)(F)F)cc1 |r,wU:16.15,19.19,(85.12,-20.14,;83.79,-20.91,;83.79,-22.45,;82.45,-20.15,;82.45,-18.61,;81.12,-20.92,;81.12,-22.46,;79.79,-23.23,;78.46,-22.46,;77.13,-23.24,;75.79,-22.47,;74.46,-23.24,;73.12,-22.47,;73.12,-20.92,;74.45,-20.15,;74.45,-18.61,;75.78,-17.84,;77.11,-18.61,;78.44,-17.84,;78.44,-16.3,;79.78,-15.53,;77.11,-15.53,;75.77,-16.3,;75.79,-20.92,;71.79,-20.15,;71.79,-18.61,;70.46,-20.93,;70.45,-19.38,;78.45,-20.93,;79.78,-20.15,)|
Cn1ccc2cc(Nc3ncc(c(N[C@@H]4CC[C@H](N)CC4)n3)C(F)(F)F)ccc2c1=O |r,wU:14.13,17.17,(14.79,-47.72,;13.46,-48.49,;13.46,-50.03,;12.13,-50.8,;10.79,-50.04,;9.46,-50.81,;8.13,-50.04,;6.8,-50.81,;5.46,-50.05,;4.13,-50.82,;2.79,-50.05,;2.79,-48.5,;4.12,-47.73,;4.12,-46.19,;5.45,-45.42,;6.78,-46.19,;8.11,-45.42,;8.11,-43.88,;9.45,-43.11,;6.78,-43.11,;5.44,-43.88,;5.46,-48.5,;1.46,-47.73,;1.46,-46.19,;.13,-48.5,;.12,-46.96,;8.12,-48.51,;9.45,-47.73,;10.79,-48.5,;12.12,-47.72,;12.12,-46.18,)|
CN1Cc2nn(C)c(C#N)c2-c2cnc3[nH]cc(-c4cn(CCCC1=O)nc4C(F)(F)F)c3c2
NS(=O)(=O)c1ccc(CNc2nc(Nc3cccc(CN4CCOCC4)c3)ncc2Br)cc1
NS(=O)(=O)c1ccc(CNc2nc(Nc3cccc(CN4CCOCC4)c3)ncc2C2CC2)cc1
NS(=O)(=O)c1ccc(CNc2nc(Nc3cccc(NC(=O)N4CCCC4)c3)ncc2Br)cc1
NS(=O)(=O)c1ccc(CNc2nc(Nc3cccc(NC(=O)N4CCCC4)c3)ncc2C2CC2)cc1
CN1CCN(CC1)c1cc(Nc2cc(C)n[nH]2)nc(Nc2ccc(CC(=O)Nc3cccc(F)c3)cc2)n1
Cc1nc2cnc3cc(F)c(cc3c2n1[C@H]1CCN(C[C@@H]1F)C(=O)CO)-c1ccc(Oc2ncccn2)cc1Cl |r|
CN(C)CCCOc1ccc2c(NCCc3cnc(NC(=O)Nc4cccc(Cl)c4)s3)ncnc2c1
CCOc1cc2ncnc(NCCc3ccc(NC(=O)Nc4cccc(Cl)c4)cc3)c2cc1F
CCOc1cc2ncnc(Nc3ccc(NC(=O)Nc4cccc(Cl)c4)cc3)c2cc1F
Fc1cc2ncnc(NCCc3ccc(NC(=O)Nc4cccc(Cl)c4)cc3)c2cc1F
CCOc1cc2c(NCCc3ccc(NC(=O)Nc4cccc(Cl)c4)cc3)ncnc2cc1F
CCOc1cc2ncnc(NCCc3ccc(NC(=O)Nc4ccccc4)cc3)c2cc1F
CCOc1cc2ncnc(NCCc3ccc(NC(=O)Nc4cccc(F)c4)cc3)c2cc1F
CCOc1cc2ncnc(NCCc3ccc(NC(=O)Nc4cccc(c4)C(F)(F)F)cc3)c2cc1F
CCOc1cc2ncnc(NCCc3ccc(NC(=O)Nc4ccc(F)c(Cl)c4)cc3)c2cc1F
CCOc1cc2ncnc(NCCc3ccc(NC(=O)Nc4ccc(Cl)c(c4)C(F)(F)F)cc3)c2cc1F
CCOc1cc2ncnc(NCCc3ccc(NC(=O)Nc4cc(Cl)ccc4OC)cc3)c2cc1F
CCOc1cc2ncnc(NCCc3ccc(NC(=O)Nc4cc(ccc4OC)C(F)(F)F)cc3)c2cc1F
COc1cc2nccc(Oc3ccc(NC(=O)C4(CC4)C(=O)Nc4ccc(F)cc4)cc3)c2cc1OC
COc1cc2c(ccnc2cc1OCCCN3CCOCC3)Oc4ccc(cc4F)NC(=O)C5(CC5)C(=O)Nc6ccc(cc6)F
CNC(=O)c1ccc(cc1C(F)(F)F)-c1ccc(=O)n(CCc2ccc3ncc(cc3c2)-c2cnn(c2)C2CCOCC2)n1
c1cc2c3cc1CCN4C(=O)C=CC(=N4)c5ccc(c(c5)C(F)(F)F)C(=O)NCCCCn6cc(cn6)-c(c3)cn2
CNC(=O)c1cccc(c1)-c1cnc2cc(-c3cnn(C)c3)c(OC)nn12
CNC(=O)c1cccc(c1)-c1cnc2cc(-c3cnn(C)c3)c(O[C@H]3CCOC3)nn12 |r|
CNC(=O)c1cncc(c1)-c1cnc2cc(-c3cnn(C)c3)c(OC3CCOC3)nn12
CNC(=O)c1ccc(F)c(c1)-c1cnc2cc(-c3cnn(C)c3)c(OC)nn12
CNC(=O)c1cc(C)cc(c1)-c1cnc2cc(-c3cnn(c3)C(C)C)c(O[C@H]3CCOC3)nn12 |r|
CNC(=O)c1cc(C)c(F)c(c1)-c1cnc2cc(-c3cnn(C)c3)c(O[C@H]3CCOC3)nn12 |r|
CNC(=O)c1cc(C(F)F)c(F)c(c1)-c1cnc2cc(-c3cnn(C)c3)c(O[C@H]3CCOC3)nn12 |r|
CNC(=O)c1cc(F)c(F)c(c1)-c1cnc2cc(-c3cnn(C)c3)c(O[C@H]3CCOC3)nn12 |r|
CO[C@H](C(=O)N1Cc2[nH]nc(NC(=O)c3ccc(cc3)N3CCN(C)CC3)c2C1)c1ccccc1 |r|
CN1CCC(CC1)Nc1ccc(cc1)C(=O)Nc1cc(n[nH]1)-c1ccc2OCCc2c1
CN1CCC(CC1)Nc1ccc(cc1)C(=O)Nc1cc(n[nH]1)-c1ccc2OCCOc2c1
COc1ccc(cc1OC)-c1cc(NC(=O)c2ccc(NC3CCN(C)CC3)cc2)[nH]n1
CN1CCC(CC1)Nc1ccc(cc1)C(=O)Nc1cc(n[nH]1)-c1ccc2OC(F)(F)Oc2c1
CN1CCC(CC1)Nc1ccc(cc1)C(=O)Nc1cc(n[nH]1)-c1cc2ccccc2s1
CN1CCC(CC1)Nc1ccc(cc1)C(=O)Nc1cc([nH]n1)-c1ccc2ncn(Cc3ccccc3)c2c1
C[C@@H](Nc1ccn2ncc(-c3cn[nH]c3)c2n1)c1cc(F)ccc1F |r|
CCn1cc(cn1)-c1cnn2ccc(N[C@H](C)c3cc(F)ccc3F)nc12 |r|
C[C@@H](Nc1ccn2ncc(-c3cnn(c3)C(F)F)c2n1)c1cc(F)ccc1F |r|
C[C@@H](Nc1ccn2ncc(-c3cnn(CCC#N)c3)c2n1)c1cc(F)ccc1F |r|
C[C@@H](Nc1ccn2ncc(-c3cnn(CCO)c3)c2n1)c1cc(F)ccc1F |r|
C[C@@H](Nc1ccn2ncc(-c3cnn(c3)S(C)(=O)=O)c2n1)c1cc(F)ccc1F |r|
C[C@@H](Nc1ccn2ncc(-c3cnn(c3)C3CC3)c2n1)c1cc(F)ccc1F |r|
C[C@@H](Nc1ccn2ncc(-c3cnn(c3)C3CCC3)c2n1)c1cc(F)ccc1F |r|
C[C@@H](Nc1ccn2ncc(-c3cnn(c3)C3CCCC3)c2n1)c1cc(F)ccc1F |r|
C[C@@H](Nc1ccn2ncc(-c3cnn(c3)C3CCOC3)c2n1)c1cc(F)ccc1F |r|
C[C@@H](Nc1ccn2ncc(-c3cnn(c3)C3CCOCC3)c2n1)c1cc(F)ccc1F |r|
COCCn1cc(cn1)-c1cnn2ccc(N[C@H](C)c3cc(F)ccc3F)nc12 |r|
C[C@@H](Nc1ccn2ncc(-c3cnn(CC(C)(C)O)c3)c2n1)c1cc(F)ccc1F |r|
C[C@@H](Nc1ccn2ncc(-c3cnn(c3)C3COC3)c2n1)c1cc(F)ccc1F |r|
CC1(C)c2oc3cc(ccc3c2C(=O)c2ccc(OCCN3CCOCC3)cc12)C#Cc1cc(OCC2CC2)ccn1
CC1(C)c2oc3cc(ccc3c2C(=O)c2ccc(OCCN3CCOCC3)cc12)C#Cc1cncc(OCC2CC2)c1
CC1(COc2ccnc(c2)C#Cc2ccc3c4c(oc3c2)C(C)(C)c2cc(OCCN3CCOCC3)ccc2C4=O)CC1
CC1(C)c2oc3cc(ccc3c2C(=O)c2ccc(OCCN3CCOCC3)cc12)C#Cc1cc(OCC2CCC2)ccn1
CC1(C)c2oc3cc(ccc3c2C(=O)c2ccc(OCCN3CCOCC3)cc12)C#Cc1cc(OCCC2CC2)ccn1
CC1(C)c2oc3cc(ccc3c2C(=O)c2ccc(OCCN3CCOCC3)cc12)C#Cc1cc(OCC(F)(F)F)ccn1
CC1(C)c2oc3cc(ccc3c2C(=O)c2ccc(OCCN3CCOCC3)cc12)C#Cc1cc(OCC2(CO)CC2)ccn1
COCCOc1ccnc(c1)C#Cc1ccc2c3c(oc2c1)C(C)(C)c1cc(OCCN2CCOCC2)ccc1C3=O
CC1(C)c2oc3cc(ccc3c2C(=O)c2ccc(OCCN3CCOCC3)cc12)C#Cc1cc(ccn1)C(=O)NC1CC1
CC1(C)c2oc3cc(ccc3c2C(=O)c2ccc(OCCN3C4CCC3COC4)cc12)C#Cc1cc(OCC2CC2)ccn1
CC1(C)c2oc3cc(ccc3c2C(=O)c2ccc(OCCN3CCCOCC3)cc12)C#Cc1cc(OCC2CC2)ccn1
CC1(C)c2oc3cc(ccc3c2C(=O)c2ccc(OCCN3CC4(COC4)C3)cc12)C#Cc1cc(OCC2CC2)ccn1
CC1(C)c2oc3cc(ccc3c2C(=O)c2ccc(OCCN3CCNC(=O)C3)cc12)C#Cc1cc(OCC2CC2)ccn1
CC1(C)NC(=O)N(CCOc2ccc3C(=O)c4c(oc5cc(ccc45)C#Cc4cc(OCC5CC5)ccn4)C(C)(C)c3c2)C1=O
CC1(C)c2oc3cc(ccc3c2C(=O)c2ccc(cc12)N1CCOCC1)C#Cc1cc(OCC2CC2)ccn1
CC1(C)c2oc3cc(ccc3c2C(=O)c2ccc(cc12)N1CC2(COC2)C1)C#Cc1cc(OCC2CC2)ccn1
CC1(C)c2oc3cc(ccc3c2C(=O)c2ccc(cc12)N1CCNC(=O)C1)C#Cc1cc(OCC2CC2)ccn1
CC1(C)c2oc3cc(ccc3c2C(=O)c2ccc(NS(C)(=O)=O)cc12)C#Cc1cc(OCC2CC2)ccn1
CC1(C)c2oc3cc(ccc3c2C(=O)c2ccc(NS(C)(=O)=O)cc12)C#Cc1cc(OCC(F)(F)F)ccn1
CC1(C)c2oc3cc(ccc3c2C(=O)c2ccc(NS(C)(=O)=O)cc12)C#Cc1cc(ccn1)C(=O)NC1CC1
CC(C)(C)NC(=O)c1ccnc(c1)C#Cc1ccc2c3c(oc2c1)C(C)(C)c1cc(NS(C)(=O)=O)ccc1C3=O
Cc1cnc(cc1C(=O)NC(C)(C)C)C#Cc1ccc2c3c(oc2c1)C(C)(C)c1cc(NS(C)(=O)=O)ccc1C3=O
Cc1c(ccnc1C#Cc1ccc2c3c(oc2c1)C(C)(C)c1cc(NS(C)(=O)=O)ccc1C3=O)C(=O)NC(C)(C)C
CCc1cc(cc(n1)C#Cc1ccc2c3c(oc2c1)C(C)(C)c1cc(NS(C)(=O)=O)ccc1C3=O)C(=O)NC(C)(C)C
CCCc1cc(cc(n1)C#Cc1ccc2c3c(oc2c1)C(C)(C)c1cc(NS(C)(=O)=O)ccc1C3=O)C(=O)NC(C)(C)C
CC(C)(C)NC(=O)c1cc(nc(c1)C(F)(F)F)C#Cc1ccc2c3c(oc2c1)C(C)(C)c1cc(NS(C)(=O)=O)ccc1C3=O
CC(C)(C)NC(=O)c1cc(Cl)nc(c1)C#Cc1ccc2c3c(oc2c1)C(C)(C)c1cc(NS(C)(=O)=O)ccc1C3=O
CC(C)(C)NC(=O)c1cc(nc(c1)C#Cc1ccc2c3c(oc2c1)C(C)(C)c1cc(NS(C)(=O)=O)ccc1C3=O)C#N
CN1CCN(C1=O)c1cnn2ccc(nc12)N1CCC[C@@H]1c1cc(F)ccc1F |r|
Fc1ccc(cc1)-c1cnn2ccc(nc12)N1CCC[C@@H]1c1cc(F)ccc1F |r|
Cc1ccc(cn1)-c1cnn2ccc(nc12)N1CCC[C@@H]1c1cc(F)ccc1F |r|
Fc1ccc(F)c(c1)[C@H]1CCCN1c1ccn2ncc(-c3cn[nH]c3)c2n1 |r|
Cn1cc(-c2cnn3ccc(nc23)N2CCC[C@@H]2c2cc(F)ccc2F)c(n1)C(F)(F)F |r|
FC(F)n1cc(cn1)-c1cnn2ccc(nc12)N1CCC[C@@H]1c1cc(F)ccc1F |r|
Fc1ccc(F)c(c1)[C@H]1CCCN1c1ccn2ncc(-c3cnn(c3)C3COC3)c2n1 |r|
FCCOc1ccc(F)cc1[C@H]1CCCN1c1ccn2ncc(-c3cn[nH]c3)c2n1 |r|
FC(F)COc1ccc(F)cc1[C@H]1CCCN1c1ccn2ncc(-c3cn[nH]c3)c2n1 |r|
Fc1ccc(OCC(F)(F)F)c(c1)[C@H]1CCCN1c1ccn2ncc(-c3cn[nH]c3)c2n1 |r|
CC(C)(C)c1cc(\C=C(/C#N)C(N)=S)cc(c1O)C(C)(C)C
CC(=O)Nc1ccc(cc1)-n1cnc2cc(ccc12)-c1ccc(OCCN2CCCCC2)cc1
Cc1ccc(cc1C#Cc2cnc3n2nccc3)C(=O)Nc4ccc(c(c4)C(F)(F)F)CN5CCN(CC5)C
CNC(=O)c1cc(Oc2ccc(NC(=O)Nc3cc(nn3-c3ccc4ncccc4c3)C(C)(C)C)c(F)c2)ccn1
Cc1cc(Nc2nc(NCc3ccc(F)cc3)nc3ccccc23)n[nH]1
Cc1cc(Nc2nc(NCc3ccc(Cl)cc3)nc3ccccc23)n[nH]1
Cc1cc(Nc2nc(NCc3ccc(Br)cc3)nc3ccccc23)n[nH]1
Cc1cc(Nc2nc(NCc3ccc(cc3)C#N)nc3ccccc23)n[nH]1
Cc1cc(Nc2nc(NCc3ccc(C)cc3)nc3ccccc23)n[nH]1
Cc1cc(Nc2nc(NCc3ccc(cc3)C(F)(F)F)nc3ccccc23)n[nH]1
Cc1cc(Nc2nc(NCc3ccc(OC(F)(F)F)cc3)nc3ccccc23)n[nH]1
Cc1cc(Nc2nc(NCc3ccccc3F)nc3ccccc23)n[nH]1
Cc1cc(Nc2nc(NCc3ccc(F)cc3F)nc3ccccc23)n[nH]1
Cc1cc(Nc2nc(NCc3cc(F)ccc3F)nc3ccccc23)n[nH]1
Cc1cc(Nc2nc(NCc3c(F)cccc3F)nc3ccccc23)n[nH]1
Cc1cc(Nc2nc(NCc3ccc(F)c(F)c3)nc3ccccc23)n[nH]1
Cc1cc(Nc2nc(NCc3cc(F)cc(F)c3)nc3ccccc23)n[nH]1
Cc1cc(Nc2nc(NCc3cc(F)c(F)c(F)c3)nc3ccccc23)n[nH]1
Cc1cc(Nc2nc(nc3ccc(Cl)cc23)N2CCOCC2)n[nH]1
Fc1ccc(CNc2nc(Nc3cc([nH]n3)C3CC3)c3ccccc3n2)cc1
Fc1ccc(CNc2nc(Nc3cc([nH]n3)C3CC3)c3ccccc3n2)c(F)c1
CCc1cc(Nc2nc(NCc3ccc(F)cc3)nc3ccccc23)n[nH]1
CCc1cc(Nc2nc(NCc3ccc(F)cc3F)nc3ccccc23)n[nH]1
Fc1ccc(CNc2nc(Nc3cc([nH]n3)-c3ccccc3)c3ccccc3n2)cc1
Fc1ccc(CNc2nc(Nc3cc([nH]n3)-c3ccccc3)c3ccccc3n2)c(F)c1
Cc1cc(Nc2nc(NCc3ccc(F)cc3F)nc3ccc(F)cc23)n[nH]1
Fc1ccc(CNc2nc(Nc3cc([nH]n3)C3CC3)c3cc(F)ccc3n2)c(F)c1
Cc1cc(Nc2nc(NCc3ccc(F)cc3F)nc3ccc(Cl)cc23)n[nH]1
Fc1ccc(CNc2nc(Nc3cc([nH]n3)C3CC3)c3cc(Cl)ccc3n2)c(F)c1
Fc1ccc(CNc2nc(Nc3cc([nH]n3)C3CC3)c3cc(Br)ccc3n2)c(F)c1
Cc1cc(Nc2nc(NCc3ccc(F)cc3F)nc3ccc(C)cc23)n[nH]1
Cc1ccc2nc(NCc3ccc(F)cc3F)nc(Nc3cc([nH]n3)C3CC3)c2c1
Cc1cc(Nc2nc(NCc3ccc(F)cc3F)nc3ccc(cc23)C(F)(F)F)n[nH]1
Cc1cc(Nc2nc(NCc3ccc(F)cc3F)nc3cc(F)ccc23)n[nH]1
Cc1cc(Nc2nc(NCc3ccc(F)cc3F)nc3cc(Cl)ccc23)n[nH]1
Fc1ccc(CNc2nc(Nc3cc([nH]n3)C3CC3)c3ccc(Cl)cc3n2)c(F)c1
Cc1cc(Nc2nc(NCc3ccc(F)cc3F)nc3cc(Br)ccc23)n[nH]1
Fc1ccc(CNc2nc(Nc3cc([nH]n3)C3CC3)c3ccc(Br)cc3n2)c(F)c1
Cc1cc(Nc2nc(NCc3ccc(F)cc3F)nc3cc(C)ccc23)n[nH]1
Cc1ccc2c(Nc3cc([nH]n3)C3CC3)nc(NCc3ccc(F)cc3F)nc2c1
Cc1cc(Nc2nc(NCc3ccc(F)cc3F)nc3cc(ccc23)C(F)(F)F)n[nH]1
Fc1ccc(CNc2nc(Nc3cc([nH]n3)C3CC3)c3ccc(cc3n2)C(F)(F)F)c(F)c1
CN(C)c1ccc(Nc2ncc(Cl)c(NCc3cccc(F)c3)n2)cc1
CC(C)OCc1ccc(Nc2ncc(Cl)c(NCc3cccc(F)c3)n2)cc1
Fc1cccc(CNc2nc(Nc3ccc(cc3)N3CCOCC3=O)ncc2Cl)c1
NS(=O)(=O)c1ccc(Nc2ncc(Cl)c(NCc3cccc(F)c3)n2)cc1
Fc1cccc(CNc2nc(Nc3ccc(cc3)N3CCOCC3)ncc2Cl)c1
CN1CCN(CC1)c1ccc(Nc2ncc(Cl)c(NCc3cccc(F)c3)n2)cc1
CCN1CCN(CC1)c1ccc(Nc2ncc(Cl)c(NCc3cccc(F)c3)n2)cc1
NC(=O)c1ccc(Nc2ncc(Cl)c(NCc3cccc(F)c3)n2)cc1
CCOCc1ccc(Nc2ncc(Cl)c(NCc3cccc(F)c3)n2)cc1
OCc1ccc(Nc2ncc(Cl)c(NCc3cccc(F)c3)n2)cc1
NS(=O)(=O)c1cccc(Nc2ncc(Cl)c(NCc3cccc(F)c3)n2)c1
Fc1cccc(CNc2nc(Nc3cccc(c3)N3CCOCC3)ncc2Cl)c1
CN1CCN(CC1)c1cccc(Nc2ncc(Cl)c(NCc3cccc(F)c3)n2)c1
CN1CCN(CC1)C(=O)c1ccc(Nc2ncc(Cl)c(NCc3cccc(F)c3)n2)cc1
Fc1cccc(CNc2nc(Nc3ccc(cc3)C(=O)N3CCOCC3)ncc2Cl)c1
CN1CCN(CC1)C(=O)c1cccc(Nc2ncc(Cl)c(NCc3cccc(F)c3)n2)c1
Fc1cccc(CNc2nc(Nc3cccc(c3)C(=O)N3CCOCC3)ncc2Cl)c1
Fc1cccc(CNc2nc(Nc3cccc(c3)C(=O)N3CCCCC3)ncc2Cl)c1
CCN1CCN(CC1)C(=O)c1cccc(Nc2ncc(Cl)c(NCc3cccc(F)c3)n2)c1
CC(C)N1CCN(CC1)C(=O)c1cccc(Nc2ncc(Cl)c(NCc3cccc(F)c3)n2)c1
Fc1cccc(CNc2nc(Nc3cccc(c3)C(=O)N3CCNC(=O)C3)ncc2Cl)c1
CN1CCCN(CC1)C(=O)c1cccc(Nc2ncc(Cl)c(NCc3cccc(F)c3)n2)c1
Fc1cccc(CNc2nc(Nc3cccc(c3)C(=O)N3CCCNCC3)ncc2Cl)c1
CN(C)C1CCN(CC1)C(=O)c1cccc(Nc2ncc(Cl)c(NCc3cccc(F)c3)n2)c1
CNC1CCN(CC1)C(=O)c1cccc(Nc2ncc(Cl)c(NCc3cccc(F)c3)n2)c1
NC1CCN(CC1)C(=O)c1cccc(Nc2ncc(Cl)c(NCc3cccc(F)c3)n2)c1
CN1CCC(CC1)NC(=O)c1cccc(Nc2ncc(Cl)c(NCc3cccc(F)c3)n2)c1
Fc1cccc(CNc2nc(Nc3cccc(c3)C(=O)NC3CCNCC3)ncc2Cl)c1
C[C@@H]1CCCN(C1)C(=O)c1cccc(Nc2ncc(Cl)c(NCc3cccc(F)c3)n2)c1 |r|
C[C@H]1CCCN(C1)C(=O)c1cccc(Nc2ncc(Cl)c(NCc3cccc(F)c3)n2)c1 |r|
Fc1cccc(CNc2nc(Nc3cccc(c3)C(=O)N[C@H]3CCCNC3)ncc2Cl)c1 |r|
Fc1cccc(CNc2nc(Nc3cccc(c3)C(=O)N[C@@H]3CCCNC3)ncc2Cl)c1 |r|
Fc1cccc(CNc2nc(Nc3cccc(c3)C(=O)N[C@@H]3CCCNC3)ncc2C(F)(F)F)c1 |r|
Fc1cccc(CNc2nc(Nc3cccc(c3)C(=O)N[C@H]3CCCNC3)ncc2C(F)(F)F)c1 |r|
Fc1cccc(CNc2nc(Nc3cccc(c3)C(=O)NC3CCCNC3)ncc2C(F)(F)F)c1
Fc1ccc(CNc2nc(Nc3cccc(c3)C(=O)N[C@@H]3CCCNC3)ncc2C(F)(F)F)cc1 |r|
Fc1ccc(CNc2nc(Nc3cccc(c3)C(=O)N[C@H]3CCCNC3)ncc2C(F)(F)F)cc1 |r|
Fc1ccc(CNc2nc(Nc3cccc(c3)C(=O)NC3CCCNC3)ncc2C(F)(F)F)cc1
Fc1ccccc1CNc1nc(Nc2cccc(c2)C(=O)NC2CCCNC2)ncc1Cl
Fc1ccc(CNc2nc(Nc3cccc(c3)C(=O)NC3CCCNC3)ncc2Cl)cc1
Fc1cccc(CNc2nc(Nc3cccc(c3)C(=O)NC3CCCNC3)ncc2Cl)c1F
Fc1ccc(CNc2nc(Nc3cccc(c3)C(=O)NC3CCCNC3)ncc2Cl)c(F)c1
Fc1ccc(F)c(CNc2nc(Nc3cccc(c3)C(=O)NC3CCCNC3)ncc2Cl)c1
Fc1cccc(F)c1CNc1nc(Nc2cccc(c2)C(=O)NC2CCCNC2)ncc1Cl
Fc1ccc(CNc2nc(Nc3cccc(c3)C(=O)NC3CCCNC3)ncc2Cl)cc1F
Fc1cc(F)cc(CNc2nc(Nc3cccc(c3)C(=O)NC3CCCNC3)ncc2Cl)c1
Fc1cc(CNc2nc(Nc3cccc(c3)C(=O)NC3CCCNC3)ncc2Cl)cc(F)c1F
Fc1cccc(c1)C1CCCN1c1nc(Nc2cccc(c2)C(=O)NC2CCCNC2)ncc1Cl
Fc1ccc(cc1)C1CCCN1c1nc(Nc2cccc(c2)C(=O)NC2CCCNC2)ncc1Cl
Fc1cc(F)cc(c1)C1CCCN1c1nc(Nc2cccc(c2)C(=O)NC2CCCNC2)ncc1Cl
Fc1cc(cc(F)c1F)C1CCCN1c1nc(Nc2cccc(c2)C(=O)NC2CCCNC2)ncc1Cl
Fc1cccc(CNc2nc(Nc3cccc(c3)C(=O)NC3CCCNC3)ncc2F)c1
Fc1cccc(CNc2nc(Nc3cccc(c3)C(=O)NC3CCCNC3)ncc2Br)c1
Cc1cnc(Nc2cccc(c2)C(=O)NC2CCCNC2)nc1NCc1cccc(F)c1
[O-][N+](=O)c1cnc(Nc2cccc(c2)C(=O)NC2CCCNC2)nc1NCc1cccc(F)c1
Fc1cccc(CNc2nc(Nc3cccc(c3)C(=O)NC3CCCNC3)nc3ccsc23)c1
Fc1cccc(CNc2nc(Nc3cccc(c3)C(=O)NC3CCCNC3)nc3sccc23)c1
Cn1ccc2c(NCc3cccc(F)c3)nc(Nc3cccc(c3)C(=O)NC3CCCNC3)nc12
Fc1cccc(CNc2nc(Nc3cccc(c3)C(=O)NC3CCCNC3)nc3[nH]ccc23)c1
Fc1cccc(CNc2nc(Nc3cccc(c3)C(=O)NC3CCCNC3)nc3cc[nH]c23)c1
Fc1ccc2CN3CCOc4cn5ncc(C(=O)NCCOc2c1)c5nc34
Fc1ccc2CN3CCCOC4=Cn5ncc(c5NC34)C(=O)NCCOc2c1 |t:11|
C[C@H]1COc2cn3ncc4C(=O)NCCOc5cc(F)ccc5CN1c2nc34 |r|
C[C@H]1CN2Cc3ccc(F)cc3OCCNC(=O)c3cnn4cc(O1)c2nc34 |r|
C[C@@H]1CN2Cc3ccc(F)cc3OCCNC(=O)c3cnn4cc(O1)c2nc34 |r|
C[C@@H]1COc2cn3ncc4C(=O)NCCOc5cc(F)ccc5CN1c2nc34 |r|
CC1(C)COc2cc(F)ccc2CN2CCOc3cn4ncc(C(=O)N1)c4nc23
C[C@@H]1COc2cn3ncc4C(=O)NC(C)(C)COc5cc(F)ccc5CN1c2nc34 |r|
CC1(C)COc2cc(F)ccc2CN2CCCOC3=Cn4ncc(c4NC23)C(=O)N1 |t:19|
C[C@@H]1COc2cn3ncc4C(=O)NC[C@H](C)Oc5cc(F)ccc5CN1c2nc34 |r|
C[C@@H]1COc2cn3ncc4C(=O)NC[C@@H](C)Oc5cc(F)ccc5CN1c2nc34 |r|
C[C@@H]1COc2cn3ncc4C(=O)NC[C@H](C)Oc5ccccc5CN1c2nc34 |r|
C[C@@H]1COc2cn3ncc4C(=O)NC[C@H](C)Oc5cc(Cl)ccc5CN1c2nc34 |r|
CN1Cc2ccc(F)cc2OCCNC(=O)c2cnn3cc(F)c1nc23
CN1Cc2ccc(F)cc2OCC(C)(C)NC(=O)c2cnn3cc(F)c1nc23
COC(=O)c1ccc2c(C(Nc3ccc(cc3)N(C)C(=O)CN3CCN(C)CC3)c3ccccc3)c(O)[nH]c2c1
Cc1c(cccc1C(=O)Nc1cc(Cl)cc(c1)C(F)(F)F)C#Cc1cnc2ccc(nn12)N1CCC[C@H](N)C1 |r|
Cc1c2cc(NC(=O)CCCCCN[C@H]3CCCN(C3)c3ccc4ncc(C#C2)n4n3)cc1C(=O)Nc1cc(Cl)cc(c1)C(F)(F)F |r|
Cc1c2cc(NC(=O)CCCCCCN[C@H]3CCCN(C3)c3ccc4ncc(C#C2)n4n3)cc1C(=O)Nc1cc(Cl)cc(c1)C(F)(F)F |r|
Cc1c2cc(NC(=O)CCCCCCCN[C@H]3CCCN(C3)c3ccc4ncc(C#C2)n4n3)cc1C(=O)Nc1cc(Cl)cc(c1)C(F)(F)F |r|
Cc1c2cc(NOCCCCC(=O)N[C@H]3CCCN(C3)c3ccc4ncc(C#C2)n4n3)cc1C(=O)Nc1cc(Cl)cc(c1)C(F)(F)F |r|
CN1CCNC(=O)CCCCOc2cc(C#Cc3cnc4ccc1nn34)c(C)c(c2)C(=O)Nc1cc(Cl)cc(c1)C(F)(F)F
CN1CCNC(=O)CCCCOc2cc(C#Cc3cnc4ccc1nn34)c(C)c(c2)C(=O)Nc1cc(cc(c1)C(F)(F)F)-n1cnc(C)c1
CN1CCN(Cc2cc(NC(=O)c3cc4OCCCCC(=O)NCCN(C)c5ccc6ncc(C#Cc(c4)c3C)n6n5)cc(c2)C(F)(F)F)CC1
FCCNC(=O)c1cnc2ccc(nn12)N1C[C@@H](F)C[C@@H]1c1cccc(F)c1 |r|
C[C@@H]1CCN(C[C@@H]1n1ccc2cnc3[nH]ccc3c12)C(=O)CC#N |r|
[H][C@@]12C[C@](O)(CO)[C@](C)(O1)n1c3ccccc3c3c4CNC(=O)c4c4c5ccccc5n2c4c13
CN1CCC(CC1)n1cc(Nc2nc(OC3(C)CC3)c3nc(ccc3n2)-c2cncnc2)cn1
CN1CCC(CC1)n1cc(Nc2nc(OC3(C)CC3)c3nc(c(F)cc3n2)-c2cnc(C)nc2)cn1
CC(C)Nc1nc(Nc2cnn(c2)C2CC3(C2)CN(C)C3)nc2cc(F)c(nc12)-c1cnc(C)nc1
CC(=O)N1CCC(CC1)n1cc(Nc2nc(OC3CCOCC3)c3nc(C)ccc3n2)cn1
CC(C)C[C@@H](NC(=O)C1(CCCCC1)C(F)(F)F)C(=O)Nc1nnc(Cc2ccc(cc2)C#N)s1 |r|
O=C(Nc1cc(ccn1)C(=O)Nc1cnccc1-c1ccccc1)C1CC1
Fc1ccc(cc1)-c1ccncc1NC(=O)c1ccnc(NC(=O)C2CC2)c1
Clc1ccc(cc1)-c1ccncc1NC(=O)c1ccnc(NC(=O)C2CC2)c1
O=C1Nc2ccccc2\C1=C\Nc1ccc(cc1)-n1nccn1
Fc1cccc(Cc2cnc3[nH]nc(Nc4cccc(c4)C(=O)N4CCOCC4)c3c2)c1
O=C(N1CCOCC1)c1cccc(Nc2n[nH]c3ncc(Cc4ccccc4)cc23)c1
Clc1cccc(Cc2cnc3[nH]nc(Nc4cccc(c4)C(=O)N4CCOCC4)c3c2)c1
Brc1cccc(Cc2cnc3[nH]nc(Nc4cccc(c4)C(=O)N4CCOCC4)c3c2)c1
[O-][N+](=O)c1cccc(Cc2cnc3[nH]nc(Nc4cccc(c4)C(=O)N4CCOCC4)c3c2)c1
FC(F)(F)c1cccc(Cc2cnc3[nH]nc(Nc4cccc(c4)C(=O)N4CCOCC4)c3c2)c1
Fc1ccccc1Cc1cnc2[nH]nc(Nc3cccc(c3)C(=O)N3CCOCC3)c2c1
Fc1ccc(Cc2cnc3[nH]nc(Nc4cccc(c4)C(=O)N4CCOCC4)c3c2)cc1
Fc1cccc(Cc2cnc3[nH]nc(Nc4cccc(c4)C(=O)N4CCOCC4)c3c2)c1F
Fc1ccc(Cc2cnc3[nH]nc(Nc4cccc(c4)C(=O)N4CCOCC4)c3c2)c(F)c1
Fc1ccc(F)c(Cc2cnc3[nH]nc(Nc4cccc(c4)C(=O)N4CCOCC4)c3c2)c1
Fc1cccc(F)c1Cc1cnc2[nH]nc(Nc3cccc(c3)C(=O)N3CCOCC3)c2c1
Fc1ccc(Cc2cnc3[nH]nc(Nc4cccc(c4)C(=O)N4CCOCC4)c3c2)cc1F
Fc1cc(F)cc(Cc2cnc3[nH]nc(Nc4cccc(c4)C(=O)N4CCOCC4)c3c2)c1
Fc1cc(Cc2cnc3[nH]nc(Nc4cccc(c4)C(=O)N4CCOCC4)c3c2)cc(F)c1F
CN1CCN(CC1)C(=O)c1cccc(Nc2n[nH]c3ncc(Cc4cc(F)ccc4F)cc23)c1
OC1CCN(CC1)C(=O)c1cccc(Nc2n[nH]c3ncc(Cc4cc(F)ccc4F)cc23)c1
OC1CCCN(C1)C(=O)c1cccc(Nc2n[nH]c3ncc(Cc4cc(F)ccc4F)cc23)c1
Fc1ccc(F)c(Cc2cnc3[nH]nc(Nc4cccc(c4)C(=O)N4CCNCC4)c3c2)c1
NC1CCN(CC1)C(=O)c1cccc(Nc2n[nH]c3ncc(Cc4cc(F)ccc4F)cc23)c1
Fc1ccc(F)c(Cc2cnc3[nH]nc(Nc4cccc(c4)C(=O)NC4CCNCC4)c3c2)c1
Fc1ccc(F)c(Cc2cnc3[nH]nc(Nc4ccc(cc4)C(=O)N4CCOCC4)c3c2)c1
CN1CCN(CC1)C(=O)c1ccc(Nc2n[nH]c3ncc(Cc4cc(F)ccc4F)cc23)cc1
OC1CCN(CC1)C(=O)c1ccc(Nc2n[nH]c3ncc(Cc4cc(F)ccc4F)cc23)cc1
OC1CCCN(C1)C(=O)c1ccc(Nc2n[nH]c3ncc(Cc4cc(F)ccc4F)cc23)cc1
Fc1ccc(F)c(Cc2cnc3[nH]nc(Nc4ccc(cc4)C(=O)N4CCNCC4)c3c2)c1
NC1CCN(CC1)C(=O)c1ccc(Nc2n[nH]c3ncc(Cc4cc(F)ccc4F)cc23)cc1
Fc1ccc(F)c(Cc2cnc3[nH]nc(Nc4ccc(cc4)C(=O)NC4CCNCC4)c3c2)c1
CN1CCN(CC1)C(=O)c1cccc(c1)-c1n[nH]c2ncc(Cc3cc(F)ccc3F)cc12
OC1CCN(CC1)C(=O)c1cccc(c1)-c1n[nH]c2ncc(Cc3cc(F)ccc3F)cc12
OC1CCCN(C1)C(=O)c1cccc(c1)-c1n[nH]c2ncc(Cc3cc(F)ccc3F)cc12
Fc1ccc(F)c(Cc2cnc3[nH]nc(-c4cccc(c4)C(=O)N4CCNCC4)c3c2)c1
CN1CCN(CC1)C(=O)c1ccc(cc1)-c1n[nH]c2ncc(Cc3cc(F)ccc3F)cc12
OC1CCN(CC1)C(=O)c1ccc(cc1)-c1n[nH]c2ncc(Cc3cc(F)ccc3F)cc12
OC1CCCN(C1)C(=O)c1ccc(cc1)-c1n[nH]c2ncc(Cc3cc(F)ccc3F)cc12
Fc1ccc(F)c(Cc2cnc3[nH]nc(-c4ccc(cc4)C(=O)N4CCNCC4)c3c2)c1
O[C@@H]1CCCN(C1)C(=O)c1cccc(c1)-c1n[nH]c2ncc(Cc3cc(F)ccc3F)cc12 |r|
O[C@H]1CCCN(C1)C(=O)c1cccc(c1)-c1n[nH]c2ncc(Cc3cc(F)ccc3F)cc12 |r|
CC(C)(O)Cn1cc(cn1)-c1cnc2Nc3ccc(C#N)c(CCCCOc4ccccc4[C@@H](CO)Nc1n2)c3 |r|
COc1c(Nc2cc(C)[nH]n2)nc(Sc2ccc(cc2F)S(=O)(=O)Cc2cccc(c2F)[N+]([O-])=O)nc1N1CCOCC1
CC(C)Nc1cc(F)cc(c1)-c1n[nH]c2ncc(cc12)-c1cccc(c1)S(C)(=O)=O
CC(=O)Nc1cc(F)cc(c1)-c1n[nH]c2ncc(cc12)-c1cccc(c1)S(C)(=O)=O
CS(=O)(=O)c1cccc(c1)-c1cnc2[nH]nc(-c3cc(F)cc(NC(=O)Nc4ccccc4)c3)c2c1
CS(=O)(=O)c1cccc(c1)-c1cnc2[nH]nc(-c3cc(F)cc(NC(=O)Nc4cccnc4)c3)c2c1
CS(=O)(=O)c1cccc(c1)-c1cnc2[nH]nc(-c3cc(F)cc(NC(=O)Nc4cncnc4)c3)c2c1
Fc1cc(NC(=O)Nc2cncnc2)cc(c1)-c1n[nH]c2ncc(cc12)-c1ccc(CN2CCOCC2)cc1
CN1CCN(Cc2ccc(cc2)-c2cnc3[nH]nc(-c4cc(F)cc(NC(=O)Nc5cncnc5)c4)c3c2)CC1
Cc1ncc(c(NC(=O)NC2c3ccccc3-c3ccccc23)n1)-c1ccccc1
CCOc1nn(c(NC(=O)N[C@H]2CN(CCOC)C[C@@H]2c2ccc(F)c(F)c2)c1C)-c1ccccc1 |r|
CC(=O)NCc1ncc(NC(=O)c2ccc(c(c2)-c2cn(C)cn2)C(F)(F)F)c(n1)-c1ccccc1
Cn1ccc(n1)-c1cc(ccc1C(F)(F)F)C(=O)Nc1cc(cnc1-c1ccccc1)C(O)=O
Cn1ccc(n1)-c1cc(ccc1C(F)(F)F)C(=O)Nc1cc(OP(O)(O)=O)cnc1-c1ccccc1
Cn1ccc(n1)-c1cc(ccc1C(F)(F)F)C(=O)Nc1cc(O)cnc1-c1ccccc1
OCCN1CCN(Cc2cn(nn2)-c2cccc(NC(=O)c3cc(F)cc(F)c3)c2)CC1
OC[C@@H]1CCCN1Cc1cn(nn1)-c1cccc(NC(=O)c2cc(F)cc(F)c2)c1 |r|
OCCN1CCN(CC1)c1nc(cs1)-c1cccc(NC(=O)c2cc(F)cc(F)c2)c1
CN1CCN(CC1)c1ccc(NCc2cn(nn2)-c2cccc(CNc3cc(F)cc(F)c3)c2)cc1C(=O)N1CCOCC1
Fc1cc(F)cc(c1)C(=O)c1ccc2NC(=O)\C(=C/c3ccc[nH]3)c2c1
Fc1cc(F)cc(Cc2ccc3NC(=O)\C(=C/c4ccc[nH]4)c3c2)c1
Fc1cc(F)cc(c1)C(=O)Nc1ccc2NC(=O)\C(=C/c3ccc[nH]3)c2c1
Fc1cc(F)cc(CNc2ccc3NC(=O)\C(=C/c4ccc[nH]4)c3c2)c1
Fc1cc(F)cc(COc2ccc3NC(=O)\C(=C/c4ccc[nH]4)c3c2)c1
O=C1Nc2ccc(NCc3ccccc3)cc2\C1=C\c1ccc[nH]1
Fc1cccc(CNc2ccc3NC(=O)\C(=C/c4ccc[nH]4)c3c2)c1
Clc1cccc(CNc2ccc3NC(=O)\C(=C/c4ccc[nH]4)c3c2)c1
Brc1cccc(CNc2ccc3NC(=O)\C(=C/c4ccc[nH]4)c3c2)c1
Fc1ccccc1CNc1ccc2NC(=O)\C(=C/c3ccc[nH]3)c2c1
Fc1ccc(CNc2ccc3NC(=O)\C(=C/c4ccc[nH]4)c3c2)cc1
Fc1ccc(CNc2ccc3NC(=O)\C(=C/c4ccc[nH]4)c3c2)cc1F
Fc1ccc(CNc2ccc3NC(=O)\C(=C/c4ccc[nH]4)c3c2)c(F)c1
Fc1ccc(F)c(CNc2ccc3NC(=O)\C(=C/c4ccc[nH]4)c3c2)c1
Fc1cccc(CNc2ccc3NC(=O)\C(=C/c4ccc[nH]4)c3c2)c1F
Fc1cccc(F)c1CNc1ccc2NC(=O)\C(=C/c3ccc[nH]3)c2c1
Fc1cc(F)c(F)c(CNc2ccc3NC(=O)\C(=C/c4ccc[nH]4)c3c2)c1
Fc1cc(F)c(F)c(CNc2ccc3NC(=O)\C(=C/c4ccc[nH]4)c3c2)c1F
Fc1cc(Cl)cc(CNc2ccc3NC(=O)\C(=C/c4ccc[nH]4)c3c2)c1
Fc1cc(Br)cc(CNc2ccc3NC(=O)\C(=C/c4ccc[nH]4)c3c2)c1
Cc1cc(F)cc(CNc2ccc3NC(=O)\C(=C/c4ccc[nH]4)c3c2)c1
Fc1cc(CNc2ccc3NC(=O)\C(=C/c4ccc[nH]4)c3c2)cc(c1)C(F)(F)F
COc1cc(F)cc(CNc2ccc3NC(=O)\C(=C/c4ccc[nH]4)c3c2)c1
Fc1ccc(Cl)c(CNc2ccc3NC(=O)\C(=C/c4ccc[nH]4)c3c2)c1
Fc1ccc(Br)c(CNc2ccc3NC(=O)\C(=C/c4ccc[nH]4)c3c2)c1
Cc1ccc(F)cc1CNc1ccc2NC(=O)\C(=C/c3ccc[nH]3)c2c1
Fc1ccc(c(CNc2ccc3NC(=O)\C(=C/c4ccc[nH]4)c3c2)c1)C(F)(F)F
COc1ccc(F)cc1CNc1ccc2NC(=O)\C(=C/c3ccc[nH]3)c2c1
Fc1cc(F)cc(CNc2ccc3NC(=O)\C(=C/c4cccs4)c3c2)c1
Fc1cc(F)cc(CNc2ccc3NC(=O)\C(=C/c4cncs4)c3c2)c1
Cc1cc(C)c(\C=C2/C(=O)Nc3ccc(NCc4cc(F)cc(F)c4)cc23)[nH]1
Fc1cc(F)cc(CNc2ccc3NC(=O)\C(=C/c4ccn[nH]4)c3c2)c1
Fc1cc(F)cc(CNc2ccc3NC(=O)\C(=C/c4cnc[nH]4)c3c2)c1
Fc1cc(F)cc(CNc2ccc3NC(=O)\C(=C/c4ncc[nH]4)c3c2)c1
Cc1nc[nH]c1\C=C1/C(=O)Nc2ccc(NCc3cc(F)cc(F)c3)cc12
Fc1ccc(F)c(CNc2ccc3NC(=O)\C(=C/c4cnc[nH]4)c3c2)c1
COc1ccc(F)cc1CNc1ccc2NC(=O)\C(=C/c3cnc[nH]3)c2c1
CN(C)S(=O)(=O)Nc1cccc(c1)-c1cnn(c1)-c1ccc(cc1)C(F)(F)F
CN1CCCCOc2cc(C#Cc3cnc4ccc(NCCC1=O)nn34)c(C)c(c2)C(=O)Nc1cc(cc(c1)C(F)(F)F)-n1cnc(C)c1
Cc1cn(cn1)-c1cc(NC(=O)c2cc3OCCCCNC(=O)CCNc4ccc5ncc(C#Cc(c3)c2C)n5n4)cc(c1)C(F)(F)F
CN1CCNc2ccc3ncc(C#Cc4cc(OCCCCC1=O)cc(C(=O)Nc1cc(cc(c1)C(F)(F)F)-n1cnc(C)c1)c4C)n3n2
Cc1cn(cn1)-c1cc(NC(=O)c2cc3OCCCCC(=O)NCCNc4ccc5ncc(C#Cc(c3)c2C)n5n4)cc(c1)C(F)(F)F
Cc1cn(cn1)-c1cc(NC(=O)c2cc3OCCCCNC(=O)CNC(=O)c4ccc5ncc(C#Cc(c3)c2C)n5n4)cc(c1)C(F)(F)F
Cc1cn(cn1)-c1cc(NC(=O)c2cc3OCCCCCCCNC(=O)c4ccc5ncc(C#Cc(c3)c2C)n5n4)cc(c1)C(F)(F)F
Cc1cn(cn1)-c1cc(NC(=O)c2cc3OCCCCCCNC(=O)c4ccc5ncc(C#Cc(c3)c2C)n5n4)cc(c1)C(F)(F)F
Cc1cn(cn1)-c1cc(NC(=O)c2cc3OCCCCCNC(=O)c4ccc5ncc(C#Cc(c3)c2C)n5n4)cc(c1)C(F)(F)F
Cc1cn(cn1)-c1cc(NC(=O)c2cc3OCCCCCCCCNC(=O)c4ccc5ncc(C#Cc(c3)c2C)n5n4)cc(c1)C(F)(F)F
Cc1c2cc(OCCCCCCCNC(=O)c3ccc4ncc(C#C2)n4n3)cc1C(=O)Nc1cc(nn1-c1ccc(Cl)cc1)C(C)(C)C
Cc1c(NC(=O)Nc2ccc(Cl)c(c2)C(F)(F)F)cc2OCCCCCCCNC(=O)c3ccc4ncc(C#Cc1c2)n4n3
CN1CCN(Cc2ccc(NC(=O)c3cc4OCCCCCCCNC(=O)c5ccc6ncc(C#Cc(c4)c3C)n6n5)cc2C(F)(F)F)CC1
CN1CCN(Cc2cc(NC(=O)c3cc4OCCCCCCCNC(=O)c5ccc6ncc(C#Cc(c4)c3C)n6n5)cc(c2)C(F)(F)F)CC1
Cc1c2cc(OCCCCCCCNC(=O)c3ccc4ncc(C#C2)n4n3)cc1C(=O)Nc1cc(Cl)cc(c1)C(F)(F)F
Cc1c2cc(OCCCCCCCNC(=O)c3ccc4ncc(C#C2)n4n3)cc1C(=O)Nc1cc(CN2CCOCC2)cc(c1)C(F)(F)F
Cc1c2cc(OCCCCCCCNC(=O)c3ccc4ncc(C#C2)n4n3)cc1C(=O)Nc1cc(cc(c1)C(F)(F)F)N1CCC(CC1)N1CCOCC1
CN1CCCN(Cc2cc(NC(=O)c3cc4OCCCCCCCNC(=O)c5ccc6ncc(C#Cc(c4)c3C)n6n5)cc(c2)C(F)(F)F)CC1
CC(C)c1cc(CN2CCN(C)CC2)cc(NC(=O)c2cc3OCCCCCCCNC(=O)c4ccc5ncc(C#Cc(c3)c2C)n5n4)c1
CN1CCN(Cc2cc(NC(=O)c3cc4OCCCCCCCNC(=O)c5ccc6ncc(C#Cc(c4)c3C)n6n5)cc(c2)C(C)(C)C)CC1
Cc1c2cc(cc1C(=O)Nc3cc(cc(c3)C4CC4)CN5CCN(CC5)C)OCCCCCCCNC(=O)c6ccc7ncc(n7n6)C#C2
C[C@H]1CNC(=O)c2ncn3ccc(N[C@H](C)c4cc(F)ccc4O1)nc23 |r|
Cc1cc(Nc2nc(NCc3ccc4OCCNc4c3)nc3n(ncc23)C2CCOCC2)n[nH]1
CN1CCOc2ccc(CNc3nc(Nc4cc(C)[nH]n4)c4cnn(C5CCOCC5)c4n3)cc12
Cc1cc(Nc2nc(NCc3ccc4OCCCNc4c3)nc3n(ncc23)C2CCOCC2)n[nH]1
Cc1cc(Nc2nc(NCc3ccc(F)c(c3)N3CCSCC3)nc3n(ncc23)C2CCOCC2)n[nH]1
Cc1cc(Nc2nc(NCc3ccc(F)c(c3)N3CCOCC3)nc3n(ncc23)C2CCOCC2)n[nH]1
Cc1cc(Nc2nc(NCc3ccc(F)c(NC4CCOCC4)c3)nc3n(ncc23)C2CCOCC2)n[nH]1
Cc1cc(Nc2nc(NCc3ccc(Cl)c(NC4CCOCC4)c3)nc3n(ncc23)C2CCOCC2)n[nH]1
Cc1cc(Nc2nc(NCc3ccc(F)c(NC4CCOC4)c3)nc3n(ncc23)C2CCOCC2)n[nH]1
Cc1cc(Nc2nc(NCc3ccc(Cl)c(NC4CCOC4)c3)nc3n(ncc23)C2CCOCC2)n[nH]1
COCCN(C)c1cc(CNc2nc(Nc3cc(C)[nH]n3)c3cnn(C4CCOCC4)c3n2)ccc1F
COCCN(C)c1cc(CNc2nc(Nc3cc(C)[nH]n3)c3cnn(C4CCOCC4)c3n2)ccc1Cl
CC(CO)Nc1cc(CNc2nc(Nc3cc(C)[nH]n3)c3cnn(C4CCOCC4)c3n2)ccc1F
CC(CO)Nc1cc(CNc2nc(Nc3cc(C)[nH]n3)c3cnn(C4CCOCC4)c3n2)ccc1Cl
Cc1cc(Nc2nc(NCc3ccc(Cl)c(NC4CCS(=O)(=O)CC4)c3)nc3n(ncc23)C2CCOCC2)n[nH]1
Cc1cc(Nc2nc(NCc3ccc(Cl)c(NC4CCS(=O)(=O)C4)c3)nc3n(ncc23)C2CCOCC2)n[nH]1
Cc1cc(Nc2nc(NCc3ccc(Cl)c(NCCS(C)(=O)=O)c3)nc3n(ncc23)C2CCOCC2)n[nH]1
Cc1cc(Nc2nc(NCc3ccc(Cl)c(c3)C(=O)Nc3ccccc3)nc3n(ncc23)C2CCOCC2)n[nH]1
Cc1cc(Nc2nc(NCc3ccc(F)cc3F)nc3n(ncc23)C2CCOCC2)n[nH]1
Cc1cc(Nc2nc(NCc3ccc(Cl)c(c3)C(=O)Nc3ccccc3F)nc3n(ncc23)C2CCOCC2)n[nH]1
Cc1cc(Nc2nc(NCc3ccc(Cl)c(c3)C(=O)Nc3ccccc3Cl)nc3n(ncc23)C2CCOCC2)n[nH]1
Cc1cc(Nc2nc(NCc3ccc(Cl)c(c3)C(=O)Nc3ccccc3Br)nc3n(ncc23)C2CCOCC2)n[nH]1
Cc1cc(Nc2nc(NCc3ccc(Cl)c(c3)C(=O)Nc3cccc(F)c3)nc3n(ncc23)C2CCOCC2)n[nH]1
Cc1cc(Nc2nc(NCc3ccc(Cl)c(c3)C(=O)Nc3cccc(Cl)c3)nc3n(ncc23)C2CCOCC2)n[nH]1
Cc1cc(Nc2nc(NCc3ccc(Cl)c(c3)C(=O)Nc3cccc(Br)c3)nc3n(ncc23)C2CCOCC2)n[nH]1
Cc1cc(Nc2nc(NCc3ccc(Cl)c(c3)C(=O)Nc3ccc(F)cc3)nc3n(ncc23)C2CCOCC2)n[nH]1
Cc1cc(Nc2nc(NCc3ccc(Cl)c(c3)C(=O)Nc3ccc(Cl)cc3)nc3n(ncc23)C2CCOCC2)n[nH]1
Cc1cc(Nc2nc(NCc3ccc(Cl)c(c3)C(=O)Nc3ccc(Br)cc3)nc3n(ncc23)C2CCOCC2)n[nH]1
Cc1cc(Nc2nc(NCc3ccc(Cl)c(c3)C(=O)Nc3cccc(C)c3)nc3n(ncc23)C2CCOCC2)n[nH]1
Cc1cc(Nc2nc(NCc3ccc(Cl)c(c3)C(=O)Nc3cccc(c3)C#N)nc3n(ncc23)C2CCOCC2)n[nH]1
Cc1cc(Nc2nc(NCc3ccc(Cl)c(c3)C(=O)Nc3cccc(OC(F)(F)F)c3)nc3n(ncc23)C2CCOCC2)n[nH]1
COc1cccc(NC(=O)c2cc(CNc3nc(Nc4cc(C)[nH]n4)c4cnn(C5CCOCC5)c4n3)ccc2Cl)c1
COc1ccc(NC(=O)c2cc(CNc3nc(Nc4cc(C)[nH]n4)c4cnn(C5CCOCC5)c4n3)ccc2Cl)cc1OC
Cc1cc(Nc2nc(NCc3ccc(Cl)c(c3)C(=O)Nc3ccc(F)c(F)c3)nc3n(ncc23)C2CCOCC2)n[nH]1
Cc1cc(Nc2nc(NCc3ccc(Cl)c(c3)C(=O)Nc3cc(F)cc(F)c3)nc3n(ncc23)C2CCOCC2)n[nH]1
Cc1cc(Nc2nc(NCc3ccc(Cl)c(c3)C(=O)Nc3cccc(F)c3F)nc3n(ncc23)C2CCOCC2)n[nH]1
Cc1cc(Nc2nc(NCc3ccc(Cl)c(c3)C(=O)Nc3cc(F)ccc3F)nc3n(ncc23)C2CCOCC2)n[nH]1
Cc1cc(Nc2nc(NCc3ccc(Cl)c(c3)C(=O)Nc3cc(F)c(F)c(F)c3)nc3n(ncc23)C2CCOCC2)n[nH]1
Cc1cc(Nc2nc(NCc3ccc(Cl)c(c3)C(=O)Nc3cc(F)ccc3F)nc3n(ncc23)C2CC(C)(C)OC(C)(C)C2)n[nH]1
Cc1cc(Nc2nc(NCc3ccc(Cl)c(c3)C(=O)Nc3cc(F)ccc3F)nc3n(ncc23)C2CCS(=O)(=O)CC2)n[nH]1
Cc1cc(Nc2nc(NCc3ccc(Cl)c(c3)C(=O)Nc3cc(F)ccc3F)nc3n(ncc23)C2CCN(CC2)S(C)(=O)=O)n[nH]1
CC(=O)N1CCC(CC1)n1ncc2c(Nc3cc(C)[nH]n3)nc(NCc3ccc(Cl)c(c3)C(=O)Nc3cc(F)ccc3F)nc12
Cc1cc(Nc2nc(NCc3ccc(Cl)c(c3)C(=O)Nc3cc(F)ccc3F)nc3[nH]ncc23)n[nH]1
Cc1cc(Nc2nc(NCc3ccc(Cl)c(c3)C(=O)Nc3cc(F)ccc3F)nc3n(C)ncc23)n[nH]1
CC(C)n1ncc2c(Nc3cc(C)[nH]n3)nc(NCc3ccc(Cl)c(c3)C(=O)Nc3cc(F)ccc3F)nc12
CC(C)n1ncc2c(Nc3cc(C)[nH]n3)nc(NC(C)c3ccc(Cl)c(c3)C(=O)Nc3cc(F)ccc3F)nc12
CC(C)n1ncc2c(Nc3cc(C)[nH]n3)nc(NCc3cnc(Cl)c(c3)C(=O)Nc3cc(F)ccc3F)nc12
CC(C)n1ncc2c(Nc3cc(C)[nH]n3)nc(NCc3cc(C(=O)Nc4cc(F)ccc4F)c(Cl)cn3)nc12
CCc1cc(Nc2nc(NCc3ccc(Cl)c(c3)C(=O)Nc3cc(F)ccc3F)nc3n(ncc23)C(C)C)n[nH]1
CC(C)n1ncc2c(Nc3cc([nH]n3)C3CC3)nc(NCc3ccc(Cl)c(c3)C(=O)Nc3cc(F)ccc3F)nc12
CN1CCN(Cc2ccc(NC(=O)[C@@H]3CCN(C3)c3ccc4ncc(-c5cccnc5)n4n3)cc2C(F)(F)F)CC1 |r|
CN1CCN(Cc2ccc(NC(=O)[C@@H]3CCN(C3)c3ccc4nccn4n3)cc2C(F)(F)F)CC1 |r|
CN1CCN(Cc2ccc(NC(=O)[C@@H]3CCN(C3)c3ccc4ncc(-c5cnn(CCO)c5)n4n3)cc2C(F)(F)F)CC1 |r|
CN1CCN(Cc2ccc(NC(=O)[C@@H]3CCN(C3)c3ccc4ncc(-c5cn[nH]c5)n4n3)cc2C(F)(F)F)CC1 |r|
CN1CCN(Cc2ccc(NC(=O)[C@@H]3CCN(C3)c3ccc4ncc(-c5cnn(c5)C5CCOCC5)n4n3)cc2C(F)(F)F)CC1 |r|
CN1CCN(Cc2ccc(NC(=O)[C@@H]3CCN(C3)c3ccc4ncc(-c5ccc(N)nc5)n4n3)cc2C(F)(F)F)CC1 |r|
CN1CCN(Cc2cc(NC(=O)[C@@H]3CCN(C3)c3ccc4ncc(-c5ccccn5)n4n3)cc(c2)C(F)(F)F)CC1 |r|
CN1CCN(Cc2cc(NC(=O)[C@H]3CCN(C3)c3ccc4ncc(-c5ccccn5)n4n3)cc(c2)C(F)(F)F)CC1 |r|
Cc1cn(cn1)-c1cc(NC(=O)[C@@H]2CCN(C2)c2ccc3ncc(-c4ccccn4)n3n2)cc(c1)C(F)(F)F |r|
CN1CCN(Cc2ccc(NC(=O)[C@@H]3CCN(C3)c3ccc4ncc(-c5ccccn5)n4n3)cc2C(F)(F)F)CC1 |r|
FC(F)(F)c1cc(NC(=O)N[C@@H]2CCN(C2)c2ccc3ncc(-c4ccccn4)n3n2)ccc1Cl |r|
Cc1conc1NC(=O)N[C@@H]1CCN(C1)c1ccc2ncc(-c3ccccn3)n2n1 |r|
CC(C)(O)c1cc2nn(CCS(C)(=O)=O)cc2cc1NC(=O)c1cccc(n1)C(F)(F)F
CC(C)(CCn1cc2cc(c(cc2n1)C(C)(C)O)NC(=O)c3cccc(n3)C(F)(F)F)O
CC(C)Oc1c(cn2cc(nc2n1)C34CC(C3)(OC4)C)C(=O)NC5=CC=CN(C5=O)C6CC6
COc1cc(Nc2nccc(-c3cc(C(=O)N[C@@H](C)CN4CCC4)n(C)n3)n2)cc(OC)c1
C1CN(CCO1)c1ccc(Nc2nc(cn3ccnc23)-c2ccc3cn[nH]c3c2)cc1
NC(=O)Nc1n[nH]c2ccc(Cc3cc(F)cc(F)c3)cc12
CNC(=O)Nc1n[nH]c2ccc(Cc3cc(F)cc(F)c3)cc12
CCOC(=O)Nc1n[nH]c2ccc(Cc3cc(F)cc(F)c3)cc12
Fc1cc(F)cc(Cc2ccc3[nH]nc(-c4ccncc4)c3c2)c1
Fc1cc(F)cc(Cc2ccc3[nH]nc(-c4cccnc4)c3c2)c1
Fc1cc(F)cc(Cc2ccc3[nH]nc(-c4ccccn4)c3c2)c1
Fc1cc(F)cc(Cc2ccc3[nH]nc(-c4cn[nH]c4)c3c2)c1
Fc1cc(F)cc(Cc2ccc3[nH]nc(-c4ccn[nH]4)c3c2)c1
Fc1cc(F)cc(Cc2ccc3[nH]nc(-c4ccoc4)c3c2)c1
Cn1cc(-c2n[nH]c3ccc(Cc4cc(F)cc(F)c4)cc23)cn1
O=C(Nc1cccc(Nc2ccc3c(-c4cn[nH]c4)n[nH]c3c2)c1)c1ccccc1
O=C(Nc1cccc(Nc2ccc3c(-c4cn[nH]c4)n[nH]c3c2)c1)c1cccc(F)c1
O=C(Nc1cccc(Nc2ccc3c(-c4cn[nH]c4)n[nH]c3c2)c1)c1cccc(Cl)c1
O=C(Nc1cccc(Nc2ccc3c(-c4cn[nH]c4)n[nH]c3c2)c1)c1cccc(Br)c1
Cc1cccc(C(=O)Nc2cccc(Nc3ccc4c(-c5cn[nH]c5)n[nH]c4c3)c2)c1
O=C(Nc1cccc(Nc2ccc3c(-c4cn[nH]c4)n[nH]c3c2)c1)c1cccc(C(F)(F)F)c1
O=C(Nc1ccccc1)Nc1cccc(Nc2ccc3c(-c4cn[nH]c4)n[nH]c3c2)c1
O=C(Nc1cccc(F)c1)Nc1cccc(Nc2ccc3c(-c4cn[nH]c4)n[nH]c3c2)c1
O=C(Nc1cccc(Cl)c1)Nc1cccc(Nc2ccc3c(-c4cn[nH]c4)n[nH]c3c2)c1
O=C(Nc1cccc(Br)c1)Nc1cccc(Nc2ccc3c(-c4cn[nH]c4)n[nH]c3c2)c1
Cc1cccc(NC(=O)Nc2cccc(Nc3ccc4c(-c5cn[nH]c5)n[nH]c4c3)c2)c1
O=C(Nc1cccc(Nc2ccc3c(-c4cn[nH]c4)n[nH]c3c2)c1)Nc1cccc(C(F)(F)F)c1
CC(C)c1cccc(NC(=O)Nc2cccc(Nc3ccc4c(-c5cn[nH]c5)n[nH]c4c3)c2)c1
CC(C)(C)c1cccc(NC(=O)Nc2cccc(Nc3ccc4c(-c5cn[nH]c5)n[nH]c4c3)c2)c1
CN(C)c1cccc(NC(=O)Nc2cccc(Nc3ccc4c(-c5cn[nH]c5)n[nH]c4c3)c2)c1
O=C(Nc1cccc(Nc2ccc3c(-c4cn[nH]c4)n[nH]c3c2)c1)Nc1cccc(N2CCOCC2)c1
CC(C)(C)c1cc(NC(=O)Nc2cccc(Nc3ccc4c(-c5cn[nH]c5)n[nH]c4c3)c2)on1
CC(C)(C)c1cc(NC(=O)Nc2cccc(Nc3ccc4c(-c5cn[nH]c5)n[nH]c4c3)c2)no1
Cn1nc(C(C)(C)C)cc1NC(=O)Nc1cccc(Nc2ccc3c(-c4cn[nH]c4)n[nH]c3c2)c1
CC(C)n1nc(C(C)(C)C)cc1NC(=O)Nc1cccc(Nc2ccc3c(-c4cn[nH]c4)n[nH]c3c2)c1
CC(C)(C)c1cc(NC(=O)Nc2cccc(Nc3ccc4c(-c5cn[nH]c5)n[nH]c4c3)c2)n(C(C)(C)C)n1
CC(C)(C)c1cc(NC(=O)Nc2cccc(Nc3ccc4c(-c5cn[nH]c5)n[nH]c4c3)c2)n(C2CCCCC2)n1
CC(C)(C)c1cc(NC(=O)Nc2cccc(Nc3ccc4c(-c5cn[nH]c5)n[nH]c4c3)c2)n(-c2ccccc2)n1
CC(C)(C)c1cc(NC(=O)Nc2cccc(Nc3ccc4c(-c5cn[nH]c5)n[nH]c4c3)c2)n(-c2ccc(F)cc2)n1
CC(C)(C)c1cc(NC(=O)Nc2cccc(Nc3ccc4c(-c5cn[nH]c5)n[nH]c4c3)c2)n(-c2ccc(Cl)cc2)n1
CC(C)(C)c1cc(NC(=O)Nc2cccc(Nc3ccc4c(-c5cn[nH]c5)n[nH]c4c3)c2)n(-c2ccc(Br)cc2)n1
CC(C)(C)c1cc(NC(=O)Nc2cccc(Nc3ccc4c(-c5cn[nH]c5)n[nH]c4c3)c2)n(-c2cccc(F)c2)n1
CC(C)(C)c1cc(NC(=O)Nc2cccc(Nc3ccc4c(-c5cn[nH]c5)n[nH]c4c3)c2)n(-c2ccccc2F)n1
CC(C)(C)c1cc(NC(=O)Nc2cccc(Nc3ccc4c(-c5cn[nH]c5)n[nH]c4c3)c2)n(-c2ccc(F)c(F)c2)n1
CC(C)(C)c1cc(NC(=O)Nc2cccc(Nc3ccc4c(-c5cn[nH]c5)n[nH]c4c3)c2)n(-c2cc(F)cc(F)c2)n1
CC(C)(C)c1cc(NC(=O)Nc2cccc(Nc3ccc4c(-c5cn[nH]c5)n[nH]c4c3)c2)n(-c2cc(F)ccc2F)n1
CC(C)(C)c1cc(NC(=O)Nc2cccc(Nc3ccc4c(-c5cn[nH]c5)n[nH]c4c3)c2)n(-c2ccc(F)cc2F)n1
CCN1CCN(c2ccc(NC(=O)c3cc(O[C@H](C)c4c(Cl)ccc(F)c4Cl)c[nH]c3=O)c(OC)c2)CC1
C[C@@H](Nc1c[nH]c(=O)c(C(=O)Nc2ccccc2)c1)c1c(Cl)ccc(F)c1Cl
C[C@@H](Nc1c[nH]c(=O)c(C(=O)Nc2ccc(N3CCOCC3)cc2)c1)c1c(Cl)ccc(F)c1Cl
C[C@@H](Nc1c[nH]c(=O)c(C(=O)Nc2ccc(CN3CCOCC3)cc2)c1)c1c(Cl)ccc(F)c1Cl
C[C@@H](Nc1c[nH]c(=O)c(C(=O)Nc2ccc(OCCN3CCOCC3)cc2)c1)c1c(Cl)ccc(F)c1Cl
C[C@@H](Nc1c[nH]c(=O)c(C(=O)Nc2ccc(CN3CCN(C)CC3)cc2)c1)c1c(Cl)ccc(F)c1Cl
C[C@@H](Nc1c[nH]c(=O)c(C(=O)Nc2ccc(CN3CCN(C)CC3)c(C(F)(F)F)c2)c1)c1c(Cl)ccc(F)c1Cl
CNC(=O)c1ccc(NC(=O)c2cc(N[C@H](C)c3c(Cl)ccc(F)c3Cl)c[nH]c2=O)cc1F
C[C@@H](Nc1c[nH]c(=O)c(C(=O)Nc2cccc(CN3CCCCC3)c2)c1)c1c(Cl)ccc(F)c1Cl
C[C@@H](Nc1c[nH]c(=O)c(C(=O)Nc2cnn(C)c2)c1)c1c(Cl)ccc(F)c1Cl
C[C@@H](Nc1c[nH]c(=O)c(C(=O)Nc2cnn(CCO)c2)c1)c1c(Cl)ccc(F)c1Cl
C[C@@H](Nc1c[nH]c(=O)c(C(=O)Nc2cnn(C3CCNCC3)c2)c1)c1c(Cl)ccc(F)c1Cl
C[C@@H](Nc1c[nH]c(=O)c(C(=O)Nc2ccc(N3CCOCC3)nc2)c1)c1c(Cl)ccc(F)c1Cl
C[C@@H](Nc1c[nH]c(=O)c(C(=O)Nc2ccc(N3CCN(C)CC3)nc2)c1)c1c(Cl)ccc(F)c1Cl
C[C@@H](Nc1c[nH]c(=O)c(C(=O)Nc2ccc(CN3CCN(C)CC3)cc2)c1)c1ccc(F)cc1
C[C@@H](Nc1c[nH]c(=O)c(C(=O)Nc2ccc(CN3CCN(C)CC3)cc2)c1)c1ccccc1F
C[C@@H](Nc1c[nH]c(=O)c(C(=O)Nc2ccc(CN3CCN(C)CC3)cc2)c1)c1cccc(F)c1
C[C@@H](Nc1c[nH]c(=O)c(C(=O)Nc2ccc(CN3CCN(C)CC3)cc2)c1)c1ccc(F)cc1F
C[C@@H](Nc1c[nH]c(=O)c(C(=O)Nc2ccc(CN3CCN(C)CC3)cc2)c1)c1cc(F)ccc1F
C[C@@H](Nc1c[nH]c(=O)c(C(=O)Nc2ccc(CN3CCN(C)CC3)cc2)c1)c1cc(F)cc(F)c1
C[C@@H](Nc1c[nH]c(=O)c(C(=O)Nc2ccc(CN3CCN(C)CC3)cc2)c1)c1ccc(Cl)cc1Cl
C[C@@H](Nc1c[nH]c(=O)c(C(=O)Nc2ccc(CN3CCN(C)CC3)cc2)c1)c1cc(Cl)cc(Cl)c1
Cc1ccc([C@@H](C)Nc2c[nH]c(=O)c(C(=O)Nc3ccc(CN4CCN(C)CC4)cc3)c2)cc1
Cc1cccc([C@@H](C)Nc2c[nH]c(=O)c(C(=O)Nc3ccc(CN4CCN(C)CC4)cc3)c2)c1
Cc1ccc([C@@H](C)Nc2c[nH]c(=O)c(C(=O)Nc3ccc(CN4CCN(C)CC4)cc3)c2)cc1C
CN1CCN(c2ccc(C(=O)Nc3n[nH]c4ccc(-c5cc(F)cc(F)c5)cc34)cc2)CC1
CN1CCN(CC1)c1ccc(cc1)C(=O)Nc1n[nH]c2ccc(Cc3cc(F)cc(F)c3)cc12
CN1CCN(c2ccc(C(=O)Nc3n[nH]c4ccc(Oc5cc(F)cc(F)c5)cc34)cc2)CC1
C[C@@H](Oc1ccc2[nH]nc(NC(=O)c3ccc(N4CCN(C)CC4)cc3)c2c1)c1c(Cl)ccc(F)c1Cl
CN1CCN(c2ccc(-c3ccnc(Nc4n[nH]c5ccc(Cc6cc(F)cc(F)c6)cc45)n3)cc2)CC1
CN1CCN(c2ccc3c(Nc4n[nH]c5ccc(Cc6cc(F)cc(F)c6)cc45)n[nH]c3c2)CC1
CC(C)n1nc(Nc2n[nH]c3ccc(Cc4cc(F)cc(F)c4)cc23)c2ccc(N3CCN(C)CC3)cc21
CN1CCN(c2ccc3c(Nc4n[nH]c5ccc(Cc6cc(F)cc(F)c6)cc45)nn(CCO)c3c2)CC1
COCCn1nc(Nc2n[nH]c3ccc(Cc4cc(F)cc(F)c4)cc23)c2ccc(N3CCN(C)CC3)cc21
COCCCn1nc(Nc2n[nH]c3ccc(Cc4cc(F)cc(F)c4)cc23)c2ccc(N3CCN(C)CC3)cc21
CN1CCN(c2ccc3c(Nc4n[nH]c5ccc(Cc6cc(F)cc(F)c6)cc45)nn(CC(N)=O)c3c2)CC1
COCC(COC)Cn1nc(Nc2n[nH]c3ccc(Cc4cc(F)cc(F)c4)cc23)c2ccc(N3CCN(C)CC3)cc21
CN1CCN(c2ccc3c(Nc4n[nH]c5ccc(Cc6cc(F)cc(F)c6)cc45)nn(C4COC4)c3c2)CC1
CN1CCN(c2ccc3c(Nc4n[nH]c5ccc(Cc6cc(F)cc(F)c6)cc45)nn(CC4CNC4)c3c2)CC1
CN1CCN(c2ccc3c(Nc4n[nH]c5ccc(Cc6cc(F)cc(F)c6)cc45)nn(CC4CN(C(=O)OC(C)(C)C)C4)c3c2)CC1
CN1CCN(c2ccc3c(Nc4n[nH]c5ccc(Cc6cc(F)cc(F)c6)cc45)nn(C4CCOCC4)c3c2)CC1
CN1CCN(c2ccc3c(Nc4n[nH]c5ccc(Cc6cc(F)cc(F)c6)cc45)nn(CC4CCOCC4)c3c2)CC1
CN1CCN(c2ccc3c(Nc4n[nH]c5ccc(Cc6cc(F)cc(F)c6)cc45)nn(CC4CCC(O)CC4)c3c2)CC1
CN1CCN(c2ccc3c(Nc4n[nH]c5ccc(Cc6cc(F)cc(F)c6)cc45)nn(C4CCNCC4)c3c2)CC1
CN1CCN(c2ccc3c(Nc4n[nH]c5ccc(Cc6cc(F)cc(F)c6)cc45)nn(C4CCN(C(=O)OC(C)(C)C)CC4)c3c2)CC1
CN1CCN(c2ccc3c(Nc4n[nH]c5ccc(Cc6cc(F)cc(F)c6)cc45)nn(CC4CCNCC4)c3c2)CC1
CN1CCC(Cn2nc(Nc3n[nH]c4ccc(Cc5cc(F)cc(F)c5)cc34)c3ccc(N4CCN(C)CC4)cc32)CC1
CN1CCN(c2ccc3c(Nc4n[nH]c5ccc(Cc6cc(F)cc(F)c6)cc45)nn(CC4CCN(C(=O)OC(C)(C)C)CC4)c3c2)CC1
CN1CCN(c2ccc3c(Nc4n[nH]c5ccc(Cc6cc(F)cc(F)c6)cc45)nn(Cc4ccccc4)c3c2)CC1
Fc1cc(F)cc(Cc2ccc3[nH]nc(Nc4n[nH]c5ccccc45)c3c2)c1
CN(C)CCN(C)c1ccc2c(Nc3n[nH]c4ccc(Cc5cc(F)cc(F)c5)cc34)n[nH]c2c1
CN(C)C1CCN(c2ccc3c(Nc4n[nH]c5ccc(Cc6cc(F)cc(F)c6)cc45)n[nH]c3c2)C1
Fc1cc(F)cc(Cc2ccc3[nH]nc(Nc4n[nH]c5cc(N6CCCCC6)ccc45)c3c2)c1
Fc1cc(F)cc(Cc2ccc3[nH]nc(Nc4n[nH]c5cc(N6CCOCC6)ccc45)c3c2)c1
C[C@@H]1CN(c2ccc3c(Nc4n[nH]c5ccc(Cc6cc(F)cc(F)c6)cc45)n[nH]c3c2)C[C@H](C)O1
CN1CC=C(c2ccc3c(Nc4n[nH]c5ccc(Cc6cc(F)cc(F)c6)cc45)n[nH]c3c2)CC1
CN(C)C1CCN(c2ccc3c(Nc4n[nH]c5ccc(Cc6cc(F)cc(F)c6)cc45)n[nH]c3c2)CC1
CN1CCCN(c2ccc3c(Nc4n[nH]c5ccc(Cc6cc(F)cc(F)c6)cc45)n[nH]c3c2)CC1
Fc1cc(F)cc(Cc2ccc3[nH]nc(Nc4ncnc5ccccc45)c3c2)c1
CN(C)C1CCN(c2ccc3c(Nc4n[nH]c5ccc(Cc6cc(F)cc(F)c6)cc45)ncnc3c2)C1
Fc1cc(F)cc(Cc2ccc3[nH]nc(Nc4ncnc5cc(N6CCCCC6)ccc45)c3c2)c1
Fc1cc(F)cc(Cc2ccc3[nH]nc(Nc4ncnc5cc(N6CCOCC6)ccc45)c3c2)c1
C[C@@H]1CN(c2ccc3c(Nc4n[nH]c5ccc(Cc6cc(F)cc(F)c6)cc45)ncnc3c2)C[C@H](C)O1
CN1CCN(c2ccc3c(Nc4n[nH]c5ccc(Cc6cc(F)cc(F)c6)cc45)ncnc3c2)CC1
CN1CCCN(c2ccc3c(Nc4n[nH]c5ccc(Cc6cc(F)cc(F)c6)cc45)ncnc3c2)CC1
CN1CCN(CC1)CC(=O)N(C)c2ccc(cc2)N/C(=C\3/c4ccc(cc4NC3=O)C(=O)OC)/c5ccccc5
Cn1cc(-c2ccc3c(c2)ncn3-c2ccc(CC(=O)Nc3cc(C(C)(C)C)on3)cc2)cn1
COc1ccc(F)cc1CNc1ccc2[nH]nc(-c3cn[nH]c3)c2c1
COc1ccc(F)cc1CNc1ccc2[nH]nc(-n3cccn3)c2c1
COc1ccc(F)cc1CNc1ccc2[nH]nc(-n3cc(F)cn3)c2c1
COc1ccc(F)cc1CNc1ccc2[nH]nc(-n3cc(C(F)(F)F)cn3)c2c1
COc1ccc(F)cc1CNc1ccc2[nH]nc(-n3cnc(C(F)(F)F)c3)c2c1
COc1ccc(F)cc1CNc1ccc2[nH]nc(C(N)=O)c2c1
CNC(=O)c1n[nH]c2ccc(NCc3cc(F)ccc3OC)cc12
COc1ccc(F)cc1CNc1ccc2[nH]nc(C(=O)NC3CC3)c2c1
COc1ccc(F)cc1CNc1ccc2[nH]nc(C(=O)NCC(F)F)c2c1
COc1ccc(F)cc1CNc1ccc2[nH]nc(C(=O)N3CCC(F)(F)C3)c2c1
COc1ccc(F)cc1CNc1ccc2[nH]nc(C(=O)N3CCC(O)C3)c2c1
COc1ccc(F)cc1CNc1ccc2[nH]nc(C(=O)NO)c2c1
COc1ccc(F)cc1CNc1ccc2[nH]nc(-c3ccc(F)cc3)c2c1
COc1ccc(F)cc1CNc1ccc2[nH]nc(-c3cccc(F)c3)c2c1
COc1ccc(F)cc1CNc1ccc2[nH]nc(C#N)c2c1
CNC(=O)c1n[nH]c2ccc(NCc3cc(F)ccc3OC(C)C)cc12
CNC(=O)c1n[nH]c2ccc(NCc3cc(F)ccc3OC3CCOC3)cc12
CNC(=O)c1n[nH]c2ccc(NCc3cc(F)ccc3OC3CCOCC3)cc12
CNC(=O)c1n[nH]c2ccc(NCc3cc(F)ccc3OCCO)cc12
CNC(=O)c1n[nH]c2ccc(NCc3cc(F)ccc3OC(F)F)cc12
CNC(=O)c1n[nH]c2ccc(NCc3cc(F)ccc3OCCF)cc12
CNC(=O)c1n[nH]c2ccc(NCc3cc(F)ccc3OCC(F)F)cc12
CNC(=O)c1n[nH]c2ccc(NCc3cc(F)ccc3OCC(F)(F)F)cc12
CNC(=O)c1n[nH]c2ccc(NCc3cc(F)ccc3P(C)(C)=O)cc12
CNC(=O)c1n[nH]c2ccc(NCc3cc(F)ccc3S(C)(=O)=O)cc12
Fc1ccc(OCC(F)F)c(CNc2ccc3[nH]nc(-c4cnoc4)c3c2)c1
N#Cc1n[nH]c2ccc(NCc3cc(F)ccc3OCC(F)F)cc12
Fc1ccc(OCC(F)F)c(CNc2ccc3[nH]nc(-n4ccnn4)c3c2)c1
Fc1ccc(OCC(F)F)c(CNc2ccc3[nH]nc(-n4cncn4)c3c2)c1
C[C@H](Nc1ccc2[nH]nc(-n3cncn3)c2c1)c1cc(F)ccc1OCC(F)F
C[C@@H](Nc1ccc2[nH]nc(-n3cncn3)c2c1)c1cc(F)ccc1OCC(F)F
CC(=O)N[C@H]1CC[C@H](c2ncc(Cl)c(Nc3ccccc3S(=O)(=O)C(C)C)n2)CC1
Cc1ccccc1NS(=O)(=O)c1ccc2c(c1)/C(=C/c1nc3ccccc3[nH]1)C(=O)N2
CCN1CCN(c2ccc(NC(=O)Nc3ccc(-c4cc(C(=O)NC)c5ncccc5n4)cc3)cc2C(F)(F)F)CC1
CCOc1nn(-c2ccccc2)c(NC(=O)NC2CN(CCOC)C[C@H]2c2ccc(F)c(F)c2)c1C
CC(Nc1cc(-c2cnn(C3CCNCC3)c2)cnc1N)c1cc(F)ccc1F
CC(Nc1cc(-c2cnn(CCCO)c2)cnc1N)c1cc(F)ccc1F
CC(Nc1cc(-c2cnn(C3CCN(C)CC3)c2)cnc1N)c1cc(F)ccc1F
Nc1ncc(-c2cnn(C3CCNCC3)c2)cc1NCc1ccccc1
Cc1cc(NC(=O)Nc2cc(C(C)(C)C)nn2-c2ccc(Cl)cc2)ccc1Nc1cccc2c1OC(C)(C)C(=O)N2
Cc1nn2c(-c3ccccc3)ccnc2c1C#N
Cc1ccc(-c2ccnc3c(C#N)c(C)nn23)cc1
Cc1nn2c(-c3ccc(Cl)cc3)ccnc2c1C#N
Cc1nn2c(-c3ccc(Br)cc3)ccnc2c1C#N
COc1ccc(-c2ccnc3c(C#N)c(C)nn23)cc1
Cc1nn2c(-c3ccccc3)ccnc2c1C(N)=O
Cc1ccc(-c2ccnc3c(C(N)=O)c(C)nn23)cc1
Cc1nn2c(-c3ccc(Cl)cc3)ccnc2c1C(N)=O
Cc1nn2c(-c3ccc(Br)cc3)ccnc2c1C(N)=O
COc1ccc(-c2ccnc3c(C(N)=O)c(C)nn23)cc1
Cc1nn2c(-c3ccccc3)ccnc2c1/C(N)=N/O
Cc1ccc(-c2ccnc3c(/C(N)=N/O)c(C)nn23)cc1
Cc1nn2c(-c3ccc(Cl)cc3)ccnc2c1/C(N)=N/O
Cc1nn2c(-c3ccc(Br)cc3)ccnc2c1/C(N)=N/O
COc1ccc(-c2ccnc3c(/C(N)=N/O)c(C)nn23)cc1
Cc1nc(-c2c(C)nn3c(-c4ccccc4)ccnc23)no1
Cc1ccc(-c2ccnc3c(-c4noc(C)n4)c(C)nn23)cc1
Cc1nc(-c2c(C)nn3c(-c4ccc(Cl)cc4)ccnc23)no1
Cc1nc(-c2c(C)nn3c(-c4ccc(Br)cc4)ccnc23)no1
COc1ccc(-c2ccnc3c(-c4noc(C)n4)c(C)nn23)cc1
C[C@@H](C(F)(F)F)N(Cc1ccc(cc1)F)C(=O)CN2C(=O)[C@]3(CCc4c3ccc(c4)NC(=O)NC)OC2=O
Cc1ccc(C(=O)Nc2cccc(C(F)(F)F)c2)cc1Nc1nc(-c2cccnc2)nc2nn(C)cc12
Cc1ccc(C(=O)Nc2cccc(C(F)(F)F)c2)cc1Nc1nc(-c2cccnc2)nc2c1cnn2C
C[C@@]1(O)C[C@@H](C1)c1nc(-c2ccc3ccc(nc3c2)-c2ccccc2)c2c(N)nccn12 |r,wU:1.1,4.6,wD:1.0,(18.42,-37.26,;17.1,-36.49,;16.31,-37.82,;17.79,-35.11,;16.41,-34.42,;15.72,-35.8,;15.93,-32.97,;16.83,-31.71,;15.91,-30.47,;16.38,-29.01,;15.35,-27.88,;15.81,-26.41,;17.32,-26.08,;17.78,-24.62,;19.27,-24.29,;20.31,-25.42,;19.85,-26.89,;18.35,-27.21,;17.89,-28.68,;21.81,-25.09,;22.85,-26.23,;24.35,-25.9,;24.82,-24.43,;23.77,-23.29,;22.27,-23.63,;14.45,-30.96,;13.11,-30.19,;13.11,-28.65,;11.78,-30.96,;11.78,-32.51,;13.12,-33.28,;14.46,-32.5,)|
CC(C)S(=O)(=O)c1ccccc1Nc2ncnc(n2)Nc3ccc(cc3OC)N4CCC(CC4)N5CCN(CC5)C
C[C@H]1CC(=O)Nc2cc(C(=O)NCCC3CC3)ccc2N1C(=O)N1CC2CC2C1
Cc1cn(CCN2CCN(CC2)c2ccccc2-c2cc(cc(c2)C(=O)NCCCN2CCCC2)C#N)c2ccccc12
CCc1cc(Nc2nccc(n2)-c2c(nc3ccccn23)-c2ccc(OC)c(c2)C(=O)Nc2c(F)cccc2F)c(OC)cc1N1CCC(CC1)N1CCN(CC1)S(C)(=O)=O
Cc1nc2ccsc2c(n1)Nc3c4c([nH]n3)C(N(C4)C(=O)N[C@H](CN(C)C)c5ccccc5)(C)C
CCN1CCN(Cc2ccc(Nc3ncc(F)c(n3)-c3cc(F)c4nc(C)n(C(C)C)c4c3)nc2)CC1
O=C(NCC#N)c1ccc(cc1)-c1ccnc(Nc2ccc(cc2)N2CCOCC2)n1
CCc1cccc(CC)c1NC(=O)c1nn(C)c-2c1CCc1cnc(Nc3ccc(cc3OC(F)(F)F)C(=O)NC3CCN(C)CC3)nc-21
O=C1c2ccccc2-c2n[nH]c3cccc1c23
C[C@H]1Oc2cc(cnc2N)-c2c(nn(C)c2C#N)CN(C)C(=O)C2C=CC(F)=CC21
CC[C@@H]1CN(C[C@@H]1c1cnc2cnc3[nH]ccc3n12)C(=O)NCC(F)(F)F |r|
Cc1c[nH]c2nccc(Oc3c(F)cc(Nc4cc(Cl)nc(N)n4)cc3F)c12