Compile Data Set for Download or QSAR
maximum 50k data
Found 29 with Last Name = 'tanguturi' and Initial = 'p'
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Universit£

Curated by ChEMBL
LigandPNGBDBM50595851(CHEMBL5192735)
Affinity DataKi:  0.920nMAssay Description:Displacement of [3H]-HS665 from KOR in guinea pig brain membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Universit£

Curated by ChEMBL
LigandPNGBDBM50595850(CHEMBL5188021)
Affinity DataKi:  1.10nMAssay Description:Displacement of [3H]-HS665 from KOR in guinea pig brain membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Universit£

Curated by ChEMBL
LigandPNGBDBM50595847(CHEMBL5199097)
Affinity DataKi:  1.30nMAssay Description:Displacement of [3H]-HS665 from KOR in guinea pig brain membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Universit£

Curated by ChEMBL
LigandPNGBDBM50399881(CHEMBL2180639)
Affinity DataKi:  1.90nMAssay Description:Displacement of [3H]-HS665 from KOR in guinea pig brain membranesMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Universit£

Curated by ChEMBL
LigandPNGBDBM50595846(CHEMBL5183917)
Affinity DataKi:  2.30nMAssay Description:Displacement of [3H]-HS665 from KOR in guinea pig brain membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Universit£

Curated by ChEMBL
LigandPNGBDBM50595852(CHEMBL5194818)
Affinity DataKi:  3nMAssay Description:Displacement of [3H]-HS665 from KOR in guinea pig brain membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Universit£

Curated by ChEMBL
LigandPNGBDBM50595849(CHEMBL5169404)
Affinity DataKi:  3.10nMAssay Description:Displacement of [3H]-HS665 from KOR in guinea pig brain membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Universit£

Curated by ChEMBL
LigandPNGBDBM50595853(CHEMBL5177451)
Affinity DataKi:  3.60nMAssay Description:Displacement of [3H]-HS665 from KOR in guinea pig brain membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Universit£

Curated by ChEMBL
LigandPNGBDBM50595848(CHEMBL5179970)
Affinity DataKi:  4.40nMAssay Description:Displacement of [3H]-HS665 from KOR in guinea pig brain membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetOxytocin receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50406324(CHEMBL5275543)
Affinity DataEC50:  0.730nMAssay Description:Biological activity against Oxytocin receptor in ratMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetOxytocin receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50406325(CHEMBL5279634)
Affinity DataEC50:  160nMAssay Description:Antagonism against Tachykinin receptor 2 in rat vas deferens(RVD)More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetOxytocin receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50406326(CHEMBL5280014)
Affinity DataEC50:  0.280nMAssay Description:Antagonism against Tachykinin receptor 2 in rat vas deferens(RVD)More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetOxytocin receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50205990(CHEMBL395429 | OXYTOCIN)
Affinity DataEC50:  2.30nMAssay Description:Biological activity against Oxytocin receptor in ratMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetOxytocin receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50406327(CHEMBL5281925)
Affinity DataEC50:  3.80E+3nMAssay Description:Antagonism against Tachykinin receptor 2 in rat vas deferens(RVD)More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetOxytocin receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50406328(CHEMBL5266871)
Affinity DataEC50:  7.00E+3nMAssay Description:Antagonism against Tachykinin receptor 2 in rat vas deferens(RVD)More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetOxytocin receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50406329(CHEMBL5273426)
Affinity DataEC50:  0.540nMAssay Description:Antagonism against Tachykinin receptor 2 in rat vas deferens(RVD)More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetOxytocin receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50406330(CHEMBL5271164)
Affinity DataEC50:  220nMAssay Description:Antagonism against Tachykinin receptor 2 in rat vas deferens(RVD)More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetOxytocin receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50406331(CHEMBL5286119)
Affinity DataEC50:  0.0600nMAssay Description:Biological activity against Oxytocin receptor in ratMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetVasopressin V1a receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50044777(Arginine Vasopressin | Beta-Hypophamine | CHEBI:34...)
Affinity DataEC50:  32nMAssay Description:Biological activity against Oxytocin receptor in ratMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Universit£

Curated by ChEMBL
LigandPNGBDBM50595853(CHEMBL5177451)
Affinity DataEC50:  7.90nMAssay Description:Agonist activity at KOR in guinea pig brain membranes assessed as stimulation of [35S]GTPgammaS binding measured after 1 hr by liquid scintillation c...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Universit£

Curated by ChEMBL
LigandPNGBDBM50595852(CHEMBL5194818)
Affinity DataEC50:  1.86E+3nMAssay Description:Agonist activity at KOR in guinea pig brain membranes assessed as stimulation of [35S]GTPgammaS binding measured after 1 hr by liquid scintillation c...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Universit£

Curated by ChEMBL
LigandPNGBDBM50595851(CHEMBL5192735)
Affinity DataEC50:  955nMAssay Description:Agonist activity at KOR in guinea pig brain membranes assessed as stimulation of [35S]GTPgammaS binding measured after 1 hr by liquid scintillation c...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetVasopressin V1b receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50044777(Arginine Vasopressin | Beta-Hypophamine | CHEBI:34...)
Affinity DataEC50:  11nMAssay Description:Antagonism against Tachykinin receptor 2 in rat vas deferens(RVD)More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Universit£

Curated by ChEMBL
LigandPNGBDBM50595849(CHEMBL5169404)
Affinity DataEC50:  5.10nMAssay Description:Agonist activity at KOR in guinea pig brain membranes assessed as stimulation of [35S]GTPgammaS binding measured after 1 hr by liquid scintillation c...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Universit£

Curated by ChEMBL
LigandPNGBDBM50595848(CHEMBL5179970)
Affinity DataEC50:  1.35E+3nMAssay Description:Agonist activity at KOR in guinea pig brain membranes assessed as stimulation of [35S]GTPgammaS binding measured after 1 hr by liquid scintillation c...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Universit£

Curated by ChEMBL
LigandPNGBDBM50595847(CHEMBL5199097)
Affinity DataEC50:  22nMAssay Description:Agonist activity at KOR in guinea pig brain membranes assessed as stimulation of [35S]GTPgammaS binding measured after 1 hr by liquid scintillation c...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Universit£

Curated by ChEMBL
LigandPNGBDBM50595846(CHEMBL5183917)
Affinity DataEC50:  26nMAssay Description:Agonist activity at KOR in guinea pig brain membranes assessed as stimulation of [35S]GTPgammaS binding measured after 1 hr by liquid scintillation c...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Universit£

Curated by ChEMBL
LigandPNGBDBM21130(N-methyl-2-phenyl-N-[(5R,7S,8S)-7-(pyrrolidin-1-yl...)
Affinity DataEC50:  1.45E+3nMAssay Description:Agonist activity at KOR in guinea pig brain membranes assessed as stimulation of [35S]GTPgammaS binding measured after 1 hr by liquid scintillation c...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Universit£

Curated by ChEMBL
LigandPNGBDBM50595850(CHEMBL5188021)
Affinity DataEC50:  9.55E+3nMAssay Description:Agonist activity at KOR in guinea pig brain membranes assessed as stimulation of [35S]GTPgammaS binding measured after 1 hr by liquid scintillation c...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed