Compile Data Set for Download or QSAR
maximum 50k data
Found 71 with Last Name = 'cavanaugh' and Initial = 'ck'
TargetEcdysone receptor(Aedes aegypti)
Rheogene

Curated by ChEMBL
LigandPNGBDBM50128466(CHEMBL291513 | [(2R,4S)-6-Fluoro-4-(4-fluoro-pheny...)
Affinity DataEC50:  3.00E+3nMAssay Description:Effective concentration for ecdysone-dependent transactivation in mammalian cell line expressing Aedes aegypti ecdysone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEcdysone receptor(Aedes aegypti)
Rheogene

Curated by ChEMBL
LigandPNGBDBM50128468((4-Chloro-phenyl)-[(2R,4S)-6-fluoro-4-(4-fluoro-ph...)
Affinity DataEC50:  640nMAssay Description:Effective concentration for ecdysone-dependent transactivation in mammalian cell line expressing Aedes aegypti ecdysone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEcdysone receptor(Aedes aegypti)
Rheogene

Curated by ChEMBL
LigandPNGBDBM50128467(((2R,4S)-2,6-Dimethyl-4-p-tolylamino-3,4-dihydro-2...)
Affinity DataEC50:  3.33E+4nMAssay Description:Effective concentration for ecdysone-dependent transactivation in mammalian cell line expressing Aedes aegypti ecdysone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEcdysone receptor(Aedes aegypti)
Rheogene

Curated by ChEMBL
LigandPNGBDBM50128469(CHEMBL56663 | [(2R,4S)-6-Fluoro-4-(4-fluoro-phenyl...)
Affinity DataEC50:  1.14E+3nMAssay Description:Effective concentration for ecdysone-dependent transactivation in mammalian cell line expressing Aedes aegypti ecdysone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEcdysone receptor(Aedes aegypti)
Rheogene

Curated by ChEMBL
LigandPNGBDBM50128471(CHEMBL59557 | [(2R,4S)-6-Fluoro-4-(4-fluoro-phenyl...)
Affinity DataEC50:  1.10E+4nMAssay Description:Effective concentration for ecdysone-dependent transactivation in mammalian cell line expressing Aedes aegypti ecdysone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEcdysone receptor(Aedes aegypti)
Rheogene

Curated by ChEMBL
LigandPNGBDBM50128470(CHEMBL416140 | [(2R,4S)-6-Fluoro-4-(4-fluoro-pheny...)
Affinity DataEC50:  3.19E+3nMAssay Description:Effective concentration for ecdysone-dependent transactivation in mammalian cell line expressing Aedes aegypti ecdysone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEcdysone receptor(Aedes aegypti)
Rheogene

Curated by ChEMBL
LigandPNGBDBM50128472(CHEMBL294491 | [(2R,4S)-6-Fluoro-4-(4-fluoro-pheny...)
Affinity DataEC50:  1.36E+3nMAssay Description:Effective concentration for ecdysone-dependent transactivation in mammalian cell line expressing Aedes aegypti ecdysone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEcdysone receptor(Aedes aegypti)
Rheogene

Curated by ChEMBL
LigandPNGBDBM50128473(((2R,4S)-2,6-Dimethyl-4-p-tolylamino-3,4-dihydro-2...)
Affinity DataEC50:  3.33E+4nMAssay Description:Effective concentration for ecdysone-dependent transactivation in mammalian cell line expressing Aedes aegypti ecdysone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEcdysone receptor(Aedes aegypti)
Rheogene

Curated by ChEMBL
LigandPNGBDBM50128474((4-Methoxy-phenyl)-((2R,4S)-2-methyl-4-phenylamino...)
Affinity DataEC50:  1.43E+3nMAssay Description:Effective concentration for ecdysone-dependent transactivation in mammalian cell line expressing Aedes aegypti ecdysone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEcdysone receptor(Aedes aegypti)
Rheogene

Curated by ChEMBL
LigandPNGBDBM50128475((3-Fluoro-phenyl)-((2R,4S)-2-methyl-4-phenylamino-...)
Affinity DataEC50:  750nMAssay Description:Effective concentration for ecdysone-dependent transactivation in mammalian cell line expressing Aedes aegypti ecdysone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEcdysone receptor(Aedes aegypti)
Rheogene

Curated by ChEMBL
LigandPNGBDBM50128476(CHEMBL61369 | [(2R,4S)-6-Fluoro-4-(4-fluoro-phenyl...)
Affinity DataEC50:  3.33E+4nMAssay Description:Effective concentration for ecdysone-dependent transactivation in mammalian cell line expressing Aedes aegypti ecdysone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEcdysone receptor(Aedes aegypti)
Rheogene

Curated by ChEMBL
LigandPNGBDBM50128479(CHEMBL57186 | [(2R,4S)-6-Fluoro-4-(4-fluoro-phenyl...)
Affinity DataEC50:  1.73E+3nMAssay Description:Effective concentration for ecdysone-dependent transactivation in mammalian cell line expressing Aedes aegypti ecdysone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEcdysone receptor(Aedes aegypti)
Rheogene

Curated by ChEMBL
LigandPNGBDBM50128478(CHEMBL301460 | [(2R,4S)-6-Fluoro-4-(4-fluoro-pheny...)
Affinity DataEC50:  1.00E+3nMAssay Description:Effective concentration for ecdysone-dependent transactivation in mammalian cell line expressing Aedes aegypti ecdysone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEcdysone receptor(Aedes aegypti)
Rheogene

Curated by ChEMBL
LigandPNGBDBM50128477(((2R,4S)-2-Methyl-4-phenylamino-3,4-dihydro-2H-qui...)
Affinity DataEC50:  1.12E+3nMAssay Description:Effective concentration for ecdysone-dependent transactivation in mammalian cell line expressing Aedes aegypti ecdysone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEcdysone receptor(Aedes aegypti)
Rheogene

Curated by ChEMBL
LigandPNGBDBM50128480(((2R,4S)-2,6-Dimethyl-4-p-tolylamino-3,4-dihydro-2...)
Affinity DataEC50:  4.41E+3nMAssay Description:Effective concentration for ecdysone-dependent transactivation in mammalian cell line expressing Aedes aegypti ecdysone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEcdysone receptor(Aedes aegypti)
Rheogene

Curated by ChEMBL
LigandPNGBDBM50128481(((2R,4S)-2,6-Dimethyl-4-p-tolylamino-3,4-dihydro-2...)
Affinity DataEC50:  5.32E+3nMAssay Description:Effective concentration for ecdysone-dependent transactivation in mammalian cell line expressing Aedes aegypti ecdysone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEcdysone receptor(Aedes aegypti)
Rheogene

Curated by ChEMBL
LigandPNGBDBM50128309(3,5-Dimethyl-benzoic acid N-tert-butyl-N'-(2-ethyl...)
Affinity DataEC50:  440nMAssay Description:Effective concentration for ecdysone-dependent transactivation in mammalian cell line expressing Aedes aegypti ecdysone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEcdysone receptor(Aedes aegypti)
Rheogene

Curated by ChEMBL
LigandPNGBDBM50128484(CHEMBL58731 | [(2R,4S)-6-Fluoro-4-(4-fluoro-phenyl...)
Affinity DataEC50:  990nMAssay Description:Effective concentration for ecdysone-dependent transactivation in mammalian cell line expressing Aedes aegypti ecdysone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEcdysone receptor(Aedes aegypti)
Rheogene

Curated by ChEMBL
LigandPNGBDBM50128483((4-Chloro-phenyl)-((2R,4S)-2-methyl-4-phenylamino-...)
Affinity DataEC50:  980nMAssay Description:Effective concentration for ecdysone-dependent transactivation in mammalian cell line expressing Aedes aegypti ecdysone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEcdysone receptor(Aedes aegypti)
Rheogene

Curated by ChEMBL
LigandPNGBDBM50128482(CHEMBL58694 | [(2R,4S)-6-Fluoro-4-(4-fluoro-phenyl...)
Affinity DataEC50:  920nMAssay Description:Effective concentration for ecdysone-dependent transactivation in mammalian cell line expressing Aedes aegypti ecdysone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEcdysone receptor(Aedes aegypti)
Rheogene

Curated by ChEMBL
LigandPNGBDBM50128485(CHEMBL291343 | [(2R,4S)-6-Fluoro-4-(4-fluoro-pheny...)
Affinity DataEC50:  1.48E+3nMAssay Description:Effective concentration for ecdysone-dependent transactivation in mammalian cell line expressing Aedes aegypti ecdysone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEcdysone receptor(Aedes aegypti)
Rheogene

Curated by ChEMBL
LigandPNGBDBM50128486(((2R,4S)-2-Methyl-4-phenylamino-3,4-dihydro-2H-qui...)
Affinity DataEC50:  1.21E+3nMAssay Description:Effective concentration for ecdysone-dependent transactivation in mammalian cell line expressing Aedes aegypti ecdysone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEcdysone receptor(Aedes aegypti)
Rheogene

Curated by ChEMBL
LigandPNGBDBM50128493(((2R,4S)-2,6-Dimethyl-4-p-tolylamino-3,4-dihydro-2...)
Affinity DataEC50:  3.33E+4nMAssay Description:Effective concentration for ecdysone-dependent transactivation in mammalian cell line expressing Aedes aegypti ecdysone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEcdysone receptor(Aedes aegypti)
Rheogene

Curated by ChEMBL
LigandPNGBDBM50128494((3-Methoxy-phenyl)-((2R,4S)-2-methyl-4-phenylamino...)
Affinity DataEC50:  700nMAssay Description:Effective concentration for ecdysone-dependent transactivation in mammalian cell line expressing Aedes aegypti ecdysone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEcdysone receptor(Aedes aegypti)
Rheogene

Curated by ChEMBL
LigandPNGBDBM50128488(((2R,4S)-2,6-Dimethyl-4-p-tolylamino-3,4-dihydro-2...)
Affinity DataEC50:  3.00E+3nMAssay Description:Effective concentration for ecdysone-dependent transactivation in mammalian cell line expressing Aedes aegypti ecdysone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEcdysone receptor(Aedes aegypti)
Rheogene

Curated by ChEMBL
LigandPNGBDBM50128490(((2R,4S)-2,6-Dimethyl-4-p-tolylamino-3,4-dihydro-2...)
Affinity DataEC50:  5.00E+3nMAssay Description:Effective concentration for ecdysone-dependent transactivation in mammalian cell line expressing Aedes aegypti ecdysone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEcdysone receptor(Aedes aegypti)
Rheogene

Curated by ChEMBL
LigandPNGBDBM50128489(((2R,4S)-2-Methyl-4-phenylamino-3,4-dihydro-2H-qui...)
Affinity DataEC50:  1.18E+3nMAssay Description:Effective concentration for ecdysone-dependent transactivation in mammalian cell line expressing Aedes aegypti ecdysone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEcdysone receptor(Aedes aegypti)
Rheogene

Curated by ChEMBL
LigandPNGBDBM50128487(CHEMBL57114 | [(2R,4S)-6-Fluoro-4-(4-fluoro-phenyl...)
Affinity DataEC50:  870nMAssay Description:Effective concentration for ecdysone-dependent transactivation in mammalian cell line expressing Aedes aegypti ecdysone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEcdysone receptor(Aedes aegypti)
Rheogene

Curated by ChEMBL
LigandPNGBDBM50128491(((2R,4S)-2,6-Dimethyl-4-p-tolylamino-3,4-dihydro-2...)
Affinity DataEC50:  3.33E+4nMAssay Description:Effective concentration for ecdysone-dependent transactivation in mammalian cell line expressing Aedes aegypti ecdysone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEcdysone receptor(Aedes aegypti)
Rheogene

Curated by ChEMBL
LigandPNGBDBM50128492((4-Chloro-phenyl)-((2R,4S)-2,6-dimethyl-4-p-tolyla...)
Affinity DataEC50:  2.15E+3nMAssay Description:Effective concentration for ecdysone-dependent transactivation in mammalian cell line expressing Aedes aegypti ecdysone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEcdysone receptor(Aedes aegypti)
Rheogene

Curated by ChEMBL
LigandPNGBDBM50128495(((2R,4S)-2,6-Dimethyl-4-p-tolylamino-3,4-dihydro-2...)
Affinity DataEC50:  5.40E+3nMAssay Description:Effective concentration for ecdysone-dependent transactivation in mammalian cell line expressing Aedes aegypti ecdysone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEcdysone receptor(Aedes aegypti)
Rheogene

Curated by ChEMBL
LigandPNGBDBM50128497(((2R,4S)-2,6-Dimethyl-4-p-tolylamino-3,4-dihydro-2...)
Affinity DataEC50:  1.84E+3nMAssay Description:Effective concentration for ecdysone-dependent transactivation in mammalian cell line expressing Aedes aegypti ecdysone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEcdysone receptor(Aedes aegypti)
Rheogene

Curated by ChEMBL
LigandPNGBDBM50128496(((2R,4S)-2-Methyl-4-phenylamino-3,4-dihydro-2H-qui...)
Affinity DataEC50:  990nMAssay Description:Effective concentration for ecdysone-dependent transactivation in mammalian cell line expressing Aedes aegypti ecdysone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEcdysone receptor(Aedes aegypti)
Rheogene

Curated by ChEMBL
LigandPNGBDBM50128498(((2R,4S)-2,6-Dimethyl-4-p-tolylamino-3,4-dihydro-2...)
Affinity DataEC50:  8.71E+3nMAssay Description:Effective concentration for ecdysone-dependent transactivation in mammalian cell line expressing Aedes aegypti ecdysone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEcdysone receptor(Choristoneura fumiferana)
Rheogene

Curated by ChEMBL
LigandPNGBDBM50128297(5-Ethyl-2,3-dihydro-benzo[1,4]dioxine-6-carboxylic...)
Affinity DataEC50:  390nMAssay Description:Dose affording 50% of maximum transactivation for ecdysone receptor from Choristoneura fumiferana (CfEcR) and a luciferase reporter gene in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEcdysone receptor(Choristoneura fumiferana)
Rheogene

Curated by ChEMBL
LigandPNGBDBM50128298(CHEMBL299671 | N-[1-(3,5-Dimethyl-benzoyl)-1-ethyl...)
Affinity DataEC50:  6.23E+3nMAssay Description:Dose affording 50% of maximum transactivation for ecdysone receptor from Choristoneura fumiferana (CfEcR) and a luciferase reporter gene in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEcdysone receptor(Bombyx mori)
Rheogene

Curated by ChEMBL
LigandPNGBDBM50128299(4-Methyl-benzo[1,3]dioxole-5-carboxylic acid [1-(3...)
Affinity DataEC50:  3.68E+3nMAssay Description:Dose affording 50% of maximum transactivation for ecdysone receptor from Bombyx mori (BmEcR) and a beta-galactosidase reporter gene in HEK-293 cell-l...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEcdysone receptor(Bombyx mori)
Rheogene

Curated by ChEMBL
LigandPNGBDBM50128300(CHEMBL55869 | N-[1-(3,5-Dimethyl-benzoyl)-cyclohex...)
Affinity DataEC50:  1.41E+3nMAssay Description:Dose affording 50% of maximum transactivation for ecdysone receptor from Bombyx mori (BmEcR) and a beta-galactosidase reporter gene in HEK-293 cell-l...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEcdysone receptor(Choristoneura fumiferana)
Rheogene

Curated by ChEMBL
LigandPNGBDBM50128301(CHEMBL54575 | N-[1-(3,5-Dimethyl-benzoyl)-cyclobut...)
Affinity DataEC50:  1.00E+4nMAssay Description:Dose affording 50% of maximum transactivation for ecdysone receptor from Choristoneura fumiferana (CfEcR) and a luciferase reporter gene in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEcdysone receptor(Bombyx mori)
Rheogene

Curated by ChEMBL
LigandPNGBDBM50128301(CHEMBL54575 | N-[1-(3,5-Dimethyl-benzoyl)-cyclobut...)
Affinity DataEC50:  8.52E+3nMAssay Description:Dose affording 50% of maximum transactivation for ecdysone receptor from Bombyx mori (BmEcR) and a beta-galactosidase reporter gene in HEK-293 cell-l...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEcdysone receptor(Bombyx mori)
Rheogene

Curated by ChEMBL
LigandPNGBDBM50128302(CHEMBL59044 | N-[1-(3,5-Dimethyl-benzoyl)-cyclohex...)
Affinity DataEC50:  1.81E+3nMAssay Description:Dose affording 50% of maximum transactivation for ecdysone receptor from Bombyx mori (BmEcR) and a beta-galactosidase reporter gene in HEK-293 cell-l...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEcdysone receptor(Choristoneura fumiferana)
Rheogene

Curated by ChEMBL
LigandPNGBDBM50128303(3-Methoxy-N-[1-(2-methoxy-benzoyl)-cyclopentyl]-2-...)
Affinity DataEC50:  6.61E+3nMAssay Description:Dose affording 50% of maximum transactivation for ecdysone receptor from Choristoneura fumiferana (CfEcR) and a luciferase reporter gene in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEcdysone receptor(Choristoneura fumiferana)
Rheogene

Curated by ChEMBL
LigandPNGBDBM50128304(CHEMBL52252 | N-[4-(3,5-Dimethyl-benzoyl)-tetrahyd...)
Affinity DataEC50:  1.80E+3nMAssay Description:Dose affording 50% of maximum transactivation for ecdysone receptor from Choristoneura fumiferana (CfEcR) and a luciferase reporter gene in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEcdysone receptor(Choristoneura fumiferana)
Rheogene

Curated by ChEMBL
LigandPNGBDBM50128305(3-methoxy-2-methylbenzoic acid 2-(3,5-dimethylbenz...)
Affinity DataEC50:  280nMAssay Description:Dose affording 50% of maximum transactivation for ecdysone receptor from Choristoneura fumiferana (CfEcR) and a luciferase reporter gene in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEcdysone receptor(Bombyx mori)
Rheogene

Curated by ChEMBL
LigandPNGBDBM50128305(3-methoxy-2-methylbenzoic acid 2-(3,5-dimethylbenz...)
Affinity DataEC50:  100nMAssay Description:Dose affording 50% of maximum transactivation for ecdysone receptor from Bombyx mori (BmEcR) and a beta-galactosidase reporter gene in HEK-293 cell-l...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEcdysone receptor(Bombyx mori)
Rheogene

Curated by ChEMBL
LigandPNGBDBM50128306(3-Methoxy-N-[1-(2-methoxy-benzoyl)-cycloheptyl]-2-...)
Affinity DataEC50:  1.94E+3nMAssay Description:Dose affording 50% of maximum transactivation for ecdysone receptor from Bombyx mori (BmEcR) and a beta-galactosidase reporter gene in HEK-293 cell-l...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEcdysone receptor(Bombyx mori)
Rheogene

Curated by ChEMBL
LigandPNGBDBM50128297(5-Ethyl-2,3-dihydro-benzo[1,4]dioxine-6-carboxylic...)
Affinity DataEC50:  740nMAssay Description:Dose affording 50% of maximum transactivation for ecdysone receptor from Bombyx mori (BmEcR) and a beta-galactosidase reporter gene in HEK-293 cell-l...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEcdysone receptor(Choristoneura fumiferana)
Rheogene

Curated by ChEMBL
LigandPNGBDBM50128302(CHEMBL59044 | N-[1-(3,5-Dimethyl-benzoyl)-cyclohex...)
Affinity DataEC50:  1.25E+3nMAssay Description:Dose affording 50% of maximum transactivation for ecdysone receptor from Choristoneura fumiferana (CfEcR) and a luciferase reporter gene in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEcdysone receptor(Bombyx mori)
Rheogene

Curated by ChEMBL
LigandPNGBDBM50128307(CHEMBL56411 | N-[4-(3,5-Dimethyl-benzoyl)-tetrahyd...)
Affinity DataEC50:  1.00E+4nMAssay Description:Dose affording 50% of maximum transactivation for ecdysone receptor from Bombyx mori (BmEcR) and a beta-galactosidase reporter gene in HEK-293 cell-l...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEcdysone receptor(Bombyx mori)
Rheogene

Curated by ChEMBL
LigandPNGBDBM50128298(CHEMBL299671 | N-[1-(3,5-Dimethyl-benzoyl)-1-ethyl...)
Affinity DataEC50:  4.53E+3nMAssay Description:Dose affording 50% of maximum transactivation for ecdysone receptor from Bombyx mori (BmEcR) and a beta-galactosidase reporter gene in HEK-293 cell-l...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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