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Found 141 with Last Name = 'cerbara' and Initial = 'i'
Target72 kDa type IV collagenase(Homo sapiens (Human))
Colosseum Combinatorial Chemistry Centre For Technology (C4T Scarl)

Curated by ChEMBL
LigandPNGBDBM50026872(CHEMBL1233506 | SC-74020)
Affinity DataIC50: <0.100nMAssay Description:Inhibition of full length MMP2 using Mca-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2 as substrate preincubated for 1 hr prior substrate addition measured after 3...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMatrix metalloproteinase-9(Homo sapiens (Human))
Colosseum Combinatorial Chemistry Centre For Technology (C4T Scarl)

Curated by ChEMBL
LigandPNGBDBM50366175(CHEMBL1957606)
Affinity DataIC50:  0.5nMAssay Description:Inhibition of MMP9 catalytic domain using Mca-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2 as substrate preincubated for 1 hr prior substrate addition measured af...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
Colosseum Combinatorial Chemistry Centre For Technology (C4T Scarl)

Curated by ChEMBL
LigandPNGBDBM50366175(CHEMBL1957606)
Affinity DataIC50:  0.800nMAssay Description:Inhibition of full length MMP2 using Mca-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2 as substrate preincubated for 1 hr prior substrate addition measured after 3...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMatrix metalloproteinase-9(Homo sapiens (Human))
Colosseum Combinatorial Chemistry Centre For Technology (C4T Scarl)

Curated by ChEMBL
LigandPNGBDBM50366203(CHEMBL1957601)
Affinity DataIC50:  2nMAssay Description:Inhibition of MMP9 catalytic domain using Mca-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2 as substrate preincubated for 1 hr prior substrate addition measured af...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Mus musculus (Mouse))
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM19130((2E,4E,6R)-7-[4-(dimethylamino)phenyl]-N-hydroxy-4...)
Affinity DataIC50:  2nMAssay Description:Inhibition of mouse HDAC1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil collagenase(Homo sapiens (Human))
Colosseum Combinatorial Chemistry Centre For Technology (C4T Scarl)

Curated by ChEMBL
LigandPNGBDBM50366175(CHEMBL1957606)
Affinity DataIC50:  4nMAssay Description:Inhibition of MMP8 catalytic domain using Mca-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2 as substrate preincubated for 1 hr prior substrate addition measured af...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMatrix metalloproteinase-9(Homo sapiens (Human))
Colosseum Combinatorial Chemistry Centre For Technology (C4T Scarl)

Curated by ChEMBL
LigandPNGBDBM50366205(CHEMBL1957603)
Affinity DataIC50:  5nMAssay Description:Inhibition of MMP9 catalytic domain using Mca-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2 as substrate preincubated for 1 hr prior substrate addition measured af...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMatrix metalloproteinase-14(Homo sapiens (Human))
Colosseum Combinatorial Chemistry Centre For Technology (C4T Scarl)

Curated by ChEMBL
LigandPNGBDBM50366175(CHEMBL1957606)
Affinity DataIC50:  5nMAssay Description:Inhibition of MMP14 catalytic domain using Mca-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2 as substrate preincubated for 1 hr prior substrate addition measured a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 2b(Zea mays)
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM19130((2E,4E,6R)-7-[4-(dimethylamino)phenyl]-N-hydroxy-4...)
Affinity DataIC50:  7.10nMAssay Description:Inhibition of maize Histone deacetylase 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 2b(Zea mays)
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM19130((2E,4E,6R)-7-[4-(dimethylamino)phenyl]-N-hydroxy-4...)
Affinity DataIC50:  7.20nMAssay Description:Concentration required for inhibition of histone deacetylase HD2 in vitro.Checked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 2b(Zea mays)
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM19130((2E,4E,6R)-7-[4-(dimethylamino)phenyl]-N-hydroxy-4...)
Affinity DataIC50:  7.20nMAssay Description:Inhibition of maize histone deacetylase 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
Colosseum Combinatorial Chemistry Centre For Technology (C4T Scarl)

Curated by ChEMBL
LigandPNGBDBM50366173(CHEMBL1957604)
Affinity DataIC50:  9nMAssay Description:Inhibition of full length MMP2 using Mca-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2 as substrate preincubated for 1 hr prior substrate addition measured after 3...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
Colosseum Combinatorial Chemistry Centre For Technology (C4T Scarl)

Curated by ChEMBL
LigandPNGBDBM50366203(CHEMBL1957601)
Affinity DataIC50:  9nMAssay Description:Inhibition of full length MMP2 using Mca-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2 as substrate preincubated for 1 hr prior substrate addition measured after 3...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 2b(Zea mays)
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50134805(6,9-Dibenzyl-12-(6-oxiranyl-6-oxo-hexyl)-decahydro...)
Affinity DataIC50:  10nMAssay Description:Concentration required for inhibition of histone deacetylase HD2 in vitro.Checked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
Colosseum Combinatorial Chemistry Centre For Technology (C4T Scarl)

Curated by ChEMBL
LigandPNGBDBM50366205(CHEMBL1957603)
Affinity DataIC50:  10nMAssay Description:Inhibition of full length MMP2 using Mca-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2 as substrate preincubated for 1 hr prior substrate addition measured after 3...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
Colosseum Combinatorial Chemistry Centre For Technology (C4T Scarl)

Curated by ChEMBL
LigandPNGBDBM50366204(CHEMBL1957602)
Affinity DataIC50:  13nMAssay Description:Inhibition of full length MMP2 using Mca-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2 as substrate preincubated for 1 hr prior substrate addition measured after 3...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMatrix metalloproteinase-9(Homo sapiens (Human))
Colosseum Combinatorial Chemistry Centre For Technology (C4T Scarl)

Curated by ChEMBL
LigandPNGBDBM50366204(CHEMBL1957602)
Affinity DataIC50:  16nMAssay Description:Inhibition of MMP9 catalytic domain using Mca-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2 as substrate preincubated for 1 hr prior substrate addition measured af...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMacrophage metalloelastase(Homo sapiens (Human))
Colosseum Combinatorial Chemistry Centre For Technology (C4T Scarl)

Curated by ChEMBL
LigandPNGBDBM50366175(CHEMBL1957606)
Affinity DataIC50:  19nMAssay Description:Inhibition of MMP12 catalytic domain using Mca-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2 as substrate preincubated for 1 hr prior substrate addition measured a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 2b(Zea mays)
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50139952(CHEMBL268286 | N-Hydroxy-3-[1-methyl-4-(3-phenyl-p...)
Affinity DataIC50:  43nMAssay Description:Concentration required for inhibition of histone deacetylase HD2 in vitro.Checked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 2b(Zea mays)
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50139952(CHEMBL268286 | N-Hydroxy-3-[1-methyl-4-(3-phenyl-p...)
Affinity DataIC50:  43nMAssay Description:Concentration required for inhibition of histone deacetylase HD2 in vitro.Checked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 2b(Zea mays)
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM19149(CHEMBL98 | N-hydroxy-N'-phenyloctanediamide | SAHA...)
Affinity DataIC50:  50nMAssay Description:Concentration required for inhibition of histone deacetylase HD2 in vitro.Checked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 2b(Zea mays)
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50140882((E)-3-(5-Benzoyl-1-methyl-1H-pyrrol-3-yl)-N-hydrox...)
Affinity DataIC50:  50nMAssay Description:Inhibition of maize histone deacetylase 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 2b(Zea mays)
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM19149(CHEMBL98 | N-hydroxy-N'-phenyloctanediamide | SAHA...)
Affinity DataIC50:  50nMAssay Description:Inhibition of maize histone deacetylase 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 2b(Zea mays)
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50140882((E)-3-(5-Benzoyl-1-methyl-1H-pyrrol-3-yl)-N-hydrox...)
Affinity DataIC50:  50nMAssay Description:Inhibition of maize Histone deacetylase 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 2b(Zea mays)
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM19149(CHEMBL98 | N-hydroxy-N'-phenyloctanediamide | SAHA...)
Affinity DataIC50:  50nMAssay Description:Inhibition of maize Histone deacetylase 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
Colosseum Combinatorial Chemistry Centre For Technology (C4T Scarl)

Curated by ChEMBL
LigandPNGBDBM50366174(CHEMBL1957605)
Affinity DataIC50:  53nMAssay Description:Inhibition of full length MMP2 using Mca-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2 as substrate preincubated for 1 hr prior substrate addition measured after 3...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 2b(Zea mays)
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50139949(CHEMBL13200 | N-Hydroxy-3-[1-methyl-4-(6-phenyl-he...)
Affinity DataIC50:  71nMAssay Description:Concentration required for inhibition of histone deacetylase HD2 in vitro.Checked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 2b(Zea mays)
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50139949(CHEMBL13200 | N-Hydroxy-3-[1-methyl-4-(6-phenyl-he...)
Affinity DataIC50:  71nMAssay Description:Inhibitory concentration against histone deacetylase HD2 enzyme.Checked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 2b(Zea mays)
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50135752((2E)-N-hydroxy-3-[1-methyl-4-(phenylacetyl)-1H-pyr...)
Affinity DataIC50:  100nMAssay Description:Inhibitory concentration against histone deacetylase HD2 enzyme.Checked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 2b(Zea mays)
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50139935(CHEMBL12927 | N-Hydroxy-3-[1-methyl-4-(1-phenyl-cy...)
Affinity DataIC50:  100nMAssay Description:Concentration required for inhibition of histone deacetylase HD2 in vitro.Checked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil collagenase(Homo sapiens (Human))
Colosseum Combinatorial Chemistry Centre For Technology (C4T Scarl)

Curated by ChEMBL
LigandPNGBDBM50366174(CHEMBL1957605)
Affinity DataIC50:  100nMAssay Description:Inhibition of MMP8 catalytic domain using Mca-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2 as substrate preincubated for 1 hr prior substrate addition measured af...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 2b(Zea mays)
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50135752((2E)-N-hydroxy-3-[1-methyl-4-(phenylacetyl)-1H-pyr...)
Affinity DataIC50:  100nMAssay Description:Inhibitory concentration against histone deacetylase HD2 enzyme.Checked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 2b(Zea mays)
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50139935(CHEMBL12927 | N-Hydroxy-3-[1-methyl-4-(1-phenyl-cy...)
Affinity DataIC50:  101nMAssay Description:Concentration required for inhibition of histone deacetylase HD2 in vitro.Checked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 2b(Zea mays)
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50139942((5S,8S,11S)-5,8-Dimethyl-11-(6-oxiranyl-6-oxo-hexy...)
Affinity DataIC50:  110nMAssay Description:Concentration required for inhibition of histone deacetylase HD2 in vitro.Checked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 2b(Zea mays)
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50139937(CHEMBL274906 | N-Hydroxy-3-[1-methyl-4-(5-phenyl-p...)
Affinity DataIC50:  110nMAssay Description:Concentration required for inhibition of histone deacetylase HD2 in vitro.Checked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 2b(Zea mays)
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50139937(CHEMBL274906 | N-Hydroxy-3-[1-methyl-4-(5-phenyl-p...)
Affinity DataIC50:  110nMAssay Description:Inhibitory concentration against histone deacetylase HD2 enzyme.Checked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Mus musculus (Mouse))
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM19149(CHEMBL98 | N-hydroxy-N'-phenyloctanediamide | SAHA...)
Affinity DataIC50:  112nMAssay Description:Inhibition of mouse HDAC1More data for this Ligand-Target Pair
TargetHistone deacetylase 2b(Zea mays)
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50139945(CHEMBL273731 | N-Hydroxy-3-[1-methyl-4-(naphthalen...)
Affinity DataIC50:  115nMAssay Description:Concentration required for inhibition of histone deacetylase HD2 in vitro.Checked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 2b(Zea mays)
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50139945(CHEMBL273731 | N-Hydroxy-3-[1-methyl-4-(naphthalen...)
Affinity DataIC50:  115nMAssay Description:Concentration required for inhibition of histone deacetylase HD2 in vitro.Checked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 2b(Zea mays)
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50139947(CHEMBL265077 | N-Hydroxy-3-[1-methyl-4-(4-phenyl-b...)
Affinity DataIC50:  129nMAssay Description:Inhibitory concentration against histone deacetylase HD2 enzyme.Checked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 2b(Zea mays)
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50139947(CHEMBL265077 | N-Hydroxy-3-[1-methyl-4-(4-phenyl-b...)
Affinity DataIC50:  130nMAssay Description:Concentration required for inhibition of histone deacetylase HD2 in vitro.Checked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 2b(Zea mays)
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50139944(CHEMBL12890 | N-Hydroxy-3-[1-methyl-4-(naphthalene...)
Affinity DataIC50:  144nMAssay Description:Concentration required for inhibition of histone deacetylase HD2 in vitro.Checked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 2b(Zea mays)
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50139944(CHEMBL12890 | N-Hydroxy-3-[1-methyl-4-(naphthalene...)
Affinity DataIC50:  145nMAssay Description:Inhibitory concentration against histone deacetylase HD2 enzyme.Checked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMatrix metalloproteinase-14(Homo sapiens (Human))
Colosseum Combinatorial Chemistry Centre For Technology (C4T Scarl)

Curated by ChEMBL
LigandPNGBDBM50366173(CHEMBL1957604)
Affinity DataIC50:  160nMAssay Description:Inhibition of MMP14 catalytic domain using Mca-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2 as substrate preincubated for 1 hr prior substrate addition measured a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-1(Homo sapiens (Human))
Colosseum Combinatorial Chemistry Centre For Technology (C4T Scarl)

Curated by ChEMBL
LigandPNGBDBM50366204(CHEMBL1957602)
Affinity DataIC50:  160nMAssay Description:Inhibition of MMP3 catalytic domain using Mca-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2 as substrate preincubated for 1 hr prior substrate addition measured af...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 2b(Zea mays)
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50139930(CHEMBL269230 | N,N'-Dihydroxy-2-(1-methyl-4-phenyl...)
Affinity DataIC50:  200nMAssay Description:Inhibitory concentration against histone deacetylase HD2 enzyme.Checked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
Colosseum Combinatorial Chemistry Centre For Technology (C4T Scarl)

Curated by ChEMBL
LigandPNGBDBM50366200(CHEMBL1957598)
Affinity DataIC50:  200nMAssay Description:Inhibition of full length MMP2 using Mca-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2 as substrate preincubated for 1 hr prior substrate addition measured after 3...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 2b(Zea mays)
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50139930(CHEMBL269230 | N,N'-Dihydroxy-2-(1-methyl-4-phenyl...)
Affinity DataIC50:  200nMAssay Description:Concentration required for inhibition of histone deacetylase HD2 in vitro.Checked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 2b(Zea mays)
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50139951(CHEMBL273454 | N-Hydroxy-3-[1-methyl-4-(8-phenyl-o...)
Affinity DataIC50:  209nMAssay Description:Inhibitory concentration against histone deacetylase HD2 enzyme.Checked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 2b(Zea mays)
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50139951(CHEMBL273454 | N-Hydroxy-3-[1-methyl-4-(8-phenyl-o...)
Affinity DataIC50:  209nMAssay Description:Inhibitory concentration against histone deacetylase HD2 enzyme.Checked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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