Affinity DataIC50: 1.10nMAssay Description:Displacement of [3H]WIN-35428 from human DAT expressed in transfected cell membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 2nMAssay Description:Displacement of [3H]WIN-35428 from human DAT expressed in transfected cell membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 2.5nMAssay Description:Displacement of [3H]-citalopram from human SERT expressed in HEK293 cell membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 3nMAssay Description:Displacement of [3H]-citalopram from human SERT expressed in HEK293 cell membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 3.30nMAssay Description:Displacement of [3H]WIN-35428 from human DAT expressed in transfected cell membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 4.70nMAssay Description:Displacement of [3H]-citalopram from human SERT expressed in HEK293 cell membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 8nMAssay Description:Displacement of [3H]WIN-35428 from human DAT expressed in transfected cell membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 11nMAssay Description:Displacement of [3H]WIN-35428 from human DAT expressed in transfected cell membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 12nMAssay Description:Displacement of [3H]WIN-35428 from human DAT expressed in transfected cell membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 17nMAssay Description:Displacement of [3H]-citalopram from human SERT expressed in HEK293 cell membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 28nMAssay Description:Displacement of [3H]WIN-35428 from human DAT expressed in transfected cell membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 31nMAssay Description:Displacement of [3H]WIN-35428 from human DAT expressed in transfected cell membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 31nMAssay Description:Displacement of [3H]-citalopram from human SERT expressed in HEK293 cell membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 53nMAssay Description:Displacement of [3H]-citalopram from human SERT expressed in HEK293 cell membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 55nMAssay Description:Displacement of [3H]WIN-35428 from human DAT expressed in transfected cell membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 56nMAssay Description:Displacement of [3H]-citalopram from human SERT expressed in HEK293 cell membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 67nMAssay Description:Displacement of [3H]WIN-35428 from human DAT expressed in transfected cell membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 106nMAssay Description:Displacement of [3H]-citalopram from human SERT expressed in HEK293 cell membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 115nMAssay Description:Displacement of [3H]WIN-35428 from human DAT expressed in transfected cell membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 140nMAssay Description:Displacement of [3H]-citalopram from human SERT expressed in HEK293 cell membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 405nMAssay Description:Displacement of [3H]-citalopram from human SERT expressed in HEK293 cell membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 593nMAssay Description:Displacement of [3H]-citalopram from human SERT expressed in HEK293 cell membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 992nMAssay Description:Displacement of [3H]-citalopram from human SERT expressed in HEK293 cell membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 1.54E+3nMAssay Description:Displacement of [3H]WIN-35428 from human DAT expressed in transfected cell membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 2.20E+3nMAssay Description:Displacement of [3H]-citalopram from human SERT expressed in HEK293 cell membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 2.96E+3nMAssay Description:Displacement of [3H]WIN-35428 from human DAT expressed in transfected cell membraneMore data for this Ligand-Target Pair
TargetHTH-type transcriptional regulator ExsA(Pseudomonas aeruginosa)
Paratek Pharmaceuticals
Curated by ChEMBL
Paratek Pharmaceuticals
Curated by ChEMBL
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibition of Pseudomonas aeruginosa 388 ExsA DNA binding activityMore data for this Ligand-Target Pair
TargetHTH-type transcriptional regulator ExsA(Pseudomonas aeruginosa)
Paratek Pharmaceuticals
Curated by ChEMBL
Paratek Pharmaceuticals
Curated by ChEMBL
Affinity DataIC50: 3.50E+3nMAssay Description:Inhibition of Pseudomonas aeruginosa PAO1 ExsA DNA binding activityMore data for this Ligand-Target Pair
TargetHTH-type transcriptional regulator ExsA(Pseudomonas aeruginosa)
Paratek Pharmaceuticals
Curated by ChEMBL
Paratek Pharmaceuticals
Curated by ChEMBL
Affinity DataIC50: 3.70E+3nMAssay Description:Inhibition of Pseudomonas aeruginosa PAO1 ExsA DNA binding activityMore data for this Ligand-Target Pair
TargetHTH-type transcriptional regulator ExsA(Pseudomonas aeruginosa)
Paratek Pharmaceuticals
Curated by ChEMBL
Paratek Pharmaceuticals
Curated by ChEMBL
Affinity DataIC50: 4.60E+3nMAssay Description:Inhibition of Pseudomonas aeruginosa PAO1 ExsA DNA binding activityMore data for this Ligand-Target Pair
TargetHTH-type transcriptional regulator ExsA(Pseudomonas aeruginosa)
Paratek Pharmaceuticals
Curated by ChEMBL
Paratek Pharmaceuticals
Curated by ChEMBL
Affinity DataIC50: 6.70E+3nMAssay Description:Inhibition of Pseudomonas aeruginosa PAO1 ExsA DNA binding activityMore data for this Ligand-Target Pair
TargetHTH-type transcriptional regulator ExsA(Pseudomonas aeruginosa)
Paratek Pharmaceuticals
Curated by ChEMBL
Paratek Pharmaceuticals
Curated by ChEMBL
Affinity DataIC50: 6.90E+3nMAssay Description:Inhibition of Pseudomonas aeruginosa PAO1 ExsA DNA binding activityMore data for this Ligand-Target Pair
TargetHTH-type transcriptional regulator ExsA(Pseudomonas aeruginosa)
Paratek Pharmaceuticals
Curated by ChEMBL
Paratek Pharmaceuticals
Curated by ChEMBL
Affinity DataIC50: 7.30E+3nMAssay Description:Inhibition of Pseudomonas aeruginosa PAO1 ExsA DNA binding activityMore data for this Ligand-Target Pair
TargetHTH-type transcriptional regulator ExsA(Pseudomonas aeruginosa)
Paratek Pharmaceuticals
Curated by ChEMBL
Paratek Pharmaceuticals
Curated by ChEMBL
Affinity DataIC50: 7.50E+3nMAssay Description:Inhibition of Pseudomonas aeruginosa 388 ExsA DNA binding activityMore data for this Ligand-Target Pair
TargetHTH-type transcriptional regulator ExsA(Pseudomonas aeruginosa)
Paratek Pharmaceuticals
Curated by ChEMBL
Paratek Pharmaceuticals
Curated by ChEMBL
Affinity DataIC50: 1.04E+4nMAssay Description:Inhibition of Pseudomonas aeruginosa PAO1 ExsA DNA binding activityMore data for this Ligand-Target Pair
TargetHTH-type transcriptional regulator ExsA(Pseudomonas aeruginosa)
Paratek Pharmaceuticals
Curated by ChEMBL
Paratek Pharmaceuticals
Curated by ChEMBL
Affinity DataIC50: 1.30E+4nMAssay Description:Inhibition of Pseudomonas aeruginosa 388 ExsA DNA binding activityMore data for this Ligand-Target Pair
TargetHTH-type transcriptional regulator ExsA(Pseudomonas aeruginosa)
Paratek Pharmaceuticals
Curated by ChEMBL
Paratek Pharmaceuticals
Curated by ChEMBL
Affinity DataIC50: 3.12E+4nMAssay Description:Inhibition of Pseudomonas aeruginosa PAO1 ExsA DNA binding activityMore data for this Ligand-Target Pair
TargetHTH-type transcriptional regulator ExsA(Pseudomonas aeruginosa)
Paratek Pharmaceuticals
Curated by ChEMBL
Paratek Pharmaceuticals
Curated by ChEMBL
Affinity DataIC50: >4.75E+4nMAssay Description:Inhibition of Pseudomonas aeruginosa PAO1 ExsA DNA binding activityMore data for this Ligand-Target Pair
TargetHTH-type transcriptional regulator ExsA(Pseudomonas aeruginosa)
Paratek Pharmaceuticals
Curated by ChEMBL
Paratek Pharmaceuticals
Curated by ChEMBL
Affinity DataIC50: >4.90E+4nMAssay Description:Inhibition of Pseudomonas aeruginosa PAO1 ExsA DNA binding activityMore data for this Ligand-Target Pair
TargetHTH-type transcriptional regulator ExsA(Pseudomonas aeruginosa)
Paratek Pharmaceuticals
Curated by ChEMBL
Paratek Pharmaceuticals
Curated by ChEMBL
Affinity DataIC50: >5.10E+4nMAssay Description:Inhibition of Pseudomonas aeruginosa PAO1 ExsA DNA binding activityMore data for this Ligand-Target Pair
TargetHTH-type transcriptional regulator ExsA(Pseudomonas aeruginosa)
Paratek Pharmaceuticals
Curated by ChEMBL
Paratek Pharmaceuticals
Curated by ChEMBL
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of Pseudomonas aeruginosa PAO1 ExsA DNA binding activityMore data for this Ligand-Target Pair
TargetHTH-type transcriptional regulator ExsA(Pseudomonas aeruginosa)
Paratek Pharmaceuticals
Curated by ChEMBL
Paratek Pharmaceuticals
Curated by ChEMBL
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of Pseudomonas aeruginosa PAO1 ExsA DNA binding activityMore data for this Ligand-Target Pair