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Found 30 with Last Name = 'dutta' and Initial = 'd'
TargetSigma intracellular receptor 2(Homo sapiens (Human))
University Of Kansas

Curated by ChEMBL
LigandPNGBDBM50606398(ML-246 | Metarrestin | Ml-246)
Affinity DataKi:  244nMAssay Description:Binding affinity to sigma2 receptor (unknown origin) by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
University Of Kansas

Curated by ChEMBL
LigandPNGBDBM50606398(ML-246 | Metarrestin | Ml-246)
Affinity DataKi:  1.22E+3nMAssay Description:Binding affinity to alpha2C receptor (unknown origin) by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
University Of Kansas

Curated by ChEMBL
LigandPNGBDBM50606398(ML-246 | Metarrestin | Ml-246)
Affinity DataKi:  3.26E+3nMAssay Description:Binding affinity to alpha1D receptor (unknown origin) by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
University Of Kansas

Curated by ChEMBL
LigandPNGBDBM50606398(ML-246 | Metarrestin | Ml-246)
Affinity DataKi:  3.41E+3nMAssay Description:Binding affinity to DAT receptor (unknown origin) by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetHistamine H1 receptor(Homo sapiens (Human))
University Of Kansas

Curated by ChEMBL
LigandPNGBDBM50606398(ML-246 | Metarrestin | Ml-246)
Affinity DataKi:  3.56E+3nMAssay Description:Binding affinity to H1 receptor (unknown origin) by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetLow molecular weight protein-tyrosine phosphatase A(Mycobacterium tuberculosis)
Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50331863(6-(4-Hydroxy-benzyl)-9-(phenyl-phenylamino-methyl)...)
Affinity DataKi:  8.00E+3nMAssay Description:Inhibition of Mycobacterium tuberculosis recombinant protein tyrosine phosphatase A by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLow molecular weight protein-tyrosine phosphatase A(Mycobacterium tuberculosis)
Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50345500(6-oxo-1,2,9,10-tetradehydro-3,4,5,6-tetrahydro-5-b...)
Affinity DataKi:  2.25E+4nMAssay Description:Non-competitive inhibition of Mycobacterium tuberculosis PTPA using p-nitrophenyl phosphate as substrate by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLow molecular weight protein-tyrosine phosphatase A(Mycobacterium tuberculosis)
Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50331859(4,9-Dioxo-3-(phenyl-phenylamino-methyl)-[1,5]diazo...)
Affinity DataKi:  3.63E+4nMAssay Description:Inhibition of Mycobacterium tuberculosis recombinant protein tyrosine phosphatase A by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLow molecular weight protein-tyrosine phosphatase A(Mycobacterium tuberculosis)
Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50331860(9-(Phenyl-phenylamino-methyl)-[1,4,7]triazecane-2,...)
Affinity DataKi:  8.55E+4nMAssay Description:Inhibition of Mycobacterium tuberculosis recombinant protein tyrosine phosphatase A by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLow molecular weight protein-tyrosine phosphatase A(Mycobacterium tuberculosis)
Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50345501(CHEMBL1784317 | rac-6-oxo-1,2,3,4,5,6,7,8,9,10-dec...)
Affinity DataKi:  1.01E+5nMAssay Description:Non-competitive inhibition of Mycobacterium tuberculosis PTPA using p-nitrophenyl phosphate as substrate by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLow molecular weight protein-tyrosine phosphatase A(Mycobacterium tuberculosis)
Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50331858(6-(Phenyl-phenylamino-methyl)-[1,4]diazepane-2,5-d...)
Affinity DataKi:  1.40E+5nMAssay Description:Inhibition of Mycobacterium tuberculosis recombinant protein tyrosine phosphatase A by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLow molecular weight protein-tyrosine phosphatase A(Mycobacterium tuberculosis)
Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50331864(3,6,9-Trimethyl-12-(phenyl-phenylamino-methyl)-1,4...)
Affinity DataKi:  1.99E+5nMAssay Description:Inhibition of Mycobacterium tuberculosis recombinant protein tyrosine phosphatase A by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLow molecular weight protein-tyrosine phosphatase A(Mycobacterium tuberculosis)
Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50331861(9-(Furan-2-yl-phenylamino-methyl)-[1,4,7]triazecan...)
Affinity DataKi:  2.15E+5nMAssay Description:Inhibition of Mycobacterium tuberculosis recombinant protein tyrosine phosphatase A by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLow molecular weight protein-tyrosine phosphatase A(Mycobacterium tuberculosis)
Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50331862(3,6-Dimethyl-9-(phenyl-phenylamino-methyl)-[1,4,7]...)
Affinity DataKi:  2.20E+5nMAssay Description:Inhibition of Mycobacterium tuberculosis recombinant protein tyrosine phosphatase A by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
University Of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50206892(CHEMBL3948489)
Affinity DataIC50:  730nMAssay Description:Inhibition of acetylcholinesterase (unknown origin) assessed as reduction in formation of 5-thio-2-nitrobenzoate from acetylthiocholine iodide preinc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
University Of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50206895(CHEMBL3983017)
Affinity DataIC50:  830nMAssay Description:Inhibition of acetylcholinesterase (unknown origin) assessed as reduction in formation of 5-thio-2-nitrobenzoate from acetylthiocholine iodide preinc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
University Of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50206890(CHEMBL3910830)
Affinity DataIC50:  980nMAssay Description:Inhibition of acetylcholinesterase (unknown origin) assessed as reduction in formation of 5-thio-2-nitrobenzoate from acetylthiocholine iodide preinc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
University Of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50206891(CHEMBL3921785)
Affinity DataIC50:  1.01E+3nMAssay Description:Inhibition of acetylcholinesterase (unknown origin) assessed as reduction in formation of 5-thio-2-nitrobenzoate from acetylthiocholine iodide preinc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
University Of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50206897(CHEMBL3945423)
Affinity DataIC50:  1.09E+3nMAssay Description:Inhibition of acetylcholinesterase (unknown origin) assessed as reduction in formation of 5-thio-2-nitrobenzoate from acetylthiocholine iodide preinc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
University Of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM10404((1S,12S,14R)-9-methoxy-4-methyl-11-oxa-4-azatetrac...)
Affinity DataIC50:  1.30E+3nMAssay Description:Inhibition of acetylcholinesterase (unknown origin) assessed as reduction in formation of 5-thio-2-nitrobenzoate from acetylthiocholine iodide preinc...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Homo sapiens (Human))
University Of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50206885(CHEMBL3930722)
Affinity DataIC50:  1.35E+3nMAssay Description:Inhibition of acetylcholinesterase (unknown origin) assessed as reduction in formation of 5-thio-2-nitrobenzoate from acetylthiocholine iodide preinc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
University Of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50206896(CHEMBL3958208)
Affinity DataIC50:  1.48E+3nMAssay Description:Inhibition of acetylcholinesterase (unknown origin) assessed as reduction in formation of 5-thio-2-nitrobenzoate from acetylthiocholine iodide preinc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
University Of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50206889(CHEMBL3928840)
Affinity DataIC50:  1.59E+3nMAssay Description:Inhibition of acetylcholinesterase (unknown origin) assessed as reduction in formation of 5-thio-2-nitrobenzoate from acetylthiocholine iodide preinc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
University Of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50206893(CHEMBL3901794)
Affinity DataIC50:  1.80E+3nMAssay Description:Inhibition of acetylcholinesterase (unknown origin) assessed as reduction in formation of 5-thio-2-nitrobenzoate from acetylthiocholine iodide preinc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
University Of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50206886(CHEMBL3955393)
Affinity DataIC50:  1.93E+3nMAssay Description:Inhibition of acetylcholinesterase (unknown origin) assessed as reduction in formation of 5-thio-2-nitrobenzoate from acetylthiocholine iodide preinc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
University Of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50206894(CHEMBL3972865)
Affinity DataIC50:  2.27E+3nMAssay Description:Inhibition of acetylcholinesterase (unknown origin) assessed as reduction in formation of 5-thio-2-nitrobenzoate from acetylthiocholine iodide preinc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
University Of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50206887(CHEMBL3976003)
Affinity DataIC50:  3.18E+3nMAssay Description:Inhibition of acetylcholinesterase (unknown origin) assessed as reduction in formation of 5-thio-2-nitrobenzoate from acetylthiocholine iodide preinc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
University Of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50206888(CHEMBL3984034)
Affinity DataIC50:  3.22E+3nMAssay Description:Inhibition of acetylcholinesterase (unknown origin) assessed as reduction in formation of 5-thio-2-nitrobenzoate from acetylthiocholine iodide preinc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLow molecular weight protein-tyrosine phosphatase A(Mycobacterium tuberculosis)
Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50345500(6-oxo-1,2,9,10-tetradehydro-3,4,5,6-tetrahydro-5-b...)
Affinity DataIC50:  1.10E+5nMAssay Description:Non-competitive inhibition of Mycobacterium tuberculosis PTPA using p-nitrophenyl phosphate as substrate by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLow molecular weight protein-tyrosine phosphatase A(Mycobacterium tuberculosis)
Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50345501(CHEMBL1784317 | rac-6-oxo-1,2,3,4,5,6,7,8,9,10-dec...)
Affinity DataIC50:  2.36E+5nMAssay Description:Non-competitive inhibition of Mycobacterium tuberculosis PTPA using p-nitrophenyl phosphate as substrate by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed