Affinity DataKi: 3.20nMAssay Description:Binding affinity for 5-hydroxytryptamine 1F receptor was determinedMore data for this Ligand-Target Pair
Affinity DataKi: 6.30nMAssay Description:Binding affinity for 5-hydroxytryptamine 1E receptor was determinedMore data for this Ligand-Target Pair
Affinity DataKi: 7.90nMAssay Description:Binding affinity for Dopamine receptor D3 was determinedMore data for this Ligand-Target Pair
Affinity DataKi: 13nMAssay Description:Binding affinity for 5-hydroxytryptamine 1B receptor was determinedMore data for this Ligand-Target Pair
Affinity DataKi: 16nMAssay Description:Binding affinity for Dopamine receptor D2 was determinedMore data for this Ligand-Target Pair
Affinity DataKi: 20nMAssay Description:Binding affinity for 5-hydroxytryptamine 2A receptor was determinedMore data for this Ligand-Target Pair
Affinity DataKi: 25nMAssay Description:Binding affinity for 5-hydroxytryptamine 2B receptor was determinedMore data for this Ligand-Target Pair
Affinity DataKi: 40nMAssay Description:Binding affinity of the compound for C-C chemokine receptor type 2B was determinedMore data for this Ligand-Target Pair
Affinity DataKi: 40nMAssay Description:Inhibition of [125I]-MCP-1 binding to the cloned C-C chemokine receptor type 2B expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 50nMAssay Description:Binding affinity of the compound at C-C chemokine receptor type 2 was determinedMore data for this Ligand-Target Pair
Affinity DataKi: 50nMAssay Description:Inhibition of [125I]MCP-1 binding to the cloned C-C chemokine receptor type 2B expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 50nMAssay Description:Inhibition of [125I]-MCP-1 binding to the cloned C-C chemokine receptor type 2B expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 50nMAssay Description:Antagonist activity against C-C chemokine receptor type 2More data for this Ligand-Target Pair
Affinity DataKi: 63nMAssay Description:Binding affinity for 5-hydroxytryptamine 7 receptor was determinedMore data for this Ligand-Target Pair
Affinity DataKi: 79nMAssay Description:Binding affinity for 5-hydroxytryptamine 2C receptor was determinedMore data for this Ligand-Target Pair
Affinity DataKi: 79nMAssay Description:Inhibition of [125I]-MCP-1 binding to the cloned C-C chemokine receptor type 2B expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 79nMAssay Description:Binding affinity for 5-hydroxytryptamine 6 receptor was determinedMore data for this Ligand-Target Pair
Affinity DataKi: 79nMAssay Description:Antagonist activity against C-C chemokine receptor type 2More data for this Ligand-Target Pair
Affinity DataKi: 79nMAssay Description:Inhibition of [125I]-MCP-1 binding to the cloned C-C chemokine receptor type 2B expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 100nMAssay Description:Binding affinity for 5-hydroxytryptamine 1A receptor was determinedMore data for this Ligand-Target Pair
Affinity DataKi: 126nMAssay Description:Inhibition of [125I]-MCP-1 binding to the cloned C-C chemokine receptor type 2B expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 126nMAssay Description:Inhibition of [125I]-MCP-1 binding to the cloned C-C chemokine receptor type 2B expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 150nMAssay Description:Reversible binding potential for rat ATP-Citrate Lyase as carbon-carbon bond cleavage activity in citrate substrateMore data for this Ligand-Target Pair
Affinity DataKi: 220nMAssay Description:Inhibitory activity against human recombinant ATP-Citrate Lyase (ACL) enzymeMore data for this Ligand-Target Pair
Affinity DataKi: 234nMAssay Description:Antagonist activity against C-C chemokine receptor type 2More data for this Ligand-Target Pair
Affinity DataKi: 251nMAssay Description:Inhibition of [125I]-MCP-1 binding to the cloned C-C chemokine receptor type 2B expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 251nMAssay Description:Inhibition of [125I]MCP-1 binding to the cloned C-C chemokine receptor type 2B expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 300nMAssay Description:Inhibitory activity against human recombinant ATP-Citrate Lyase (ACL) enzymeMore data for this Ligand-Target Pair
Affinity DataKi: 300nMAssay Description:Inhibitory activity against human recombinant ATP-Citrate Lyase (ACL) enzymeMore data for this Ligand-Target Pair
Affinity DataKi: 316nMAssay Description:Inhibition of [125I]MCP-1 binding to the cloned C-C chemokine receptor type 2B expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 350nMAssay Description:Antagonist activity against C-C chemokine receptor type 2More data for this Ligand-Target Pair
Affinity DataKi: 360nMAssay Description:Antagonist activity against C-C chemokine receptor type 2More data for this Ligand-Target Pair
Affinity DataKi: 360nMAssay Description:Antagonist activity against C-C chemokine receptor type 2More data for this Ligand-Target Pair
Affinity DataKi: 370nMAssay Description:Inhibitory activity against human recombinant ATP-Citrate Lyase (ACL) enzymeMore data for this Ligand-Target Pair
Affinity DataKi: 420nMAssay Description:Antagonist activity against C-C chemokine receptor type 2More data for this Ligand-Target Pair
Affinity DataKi: 460nMAssay Description:Antagonist activity against C-C chemokine receptor type 2More data for this Ligand-Target Pair
Affinity DataKi: 501nMAssay Description:Binding affinity for 5-hydroxytryptamine 2B receptor was determinedMore data for this Ligand-Target Pair
Affinity DataKi: 520nMAssay Description:Antagonist activity against C-C chemokine receptor type 2More data for this Ligand-Target Pair
Affinity DataKi: 550nMAssay Description:Inhibitory activity against human recombinant ATP-Citrate Lyase (ACL) enzymeMore data for this Ligand-Target Pair
Affinity DataKi: 550nMAssay Description:Antagonist activity against C-C chemokine receptor type 2More data for this Ligand-Target Pair
Affinity DataKi: 560nMAssay Description:Antagonist activity against C-C chemokine receptor type 2More data for this Ligand-Target Pair
Affinity DataKi: 590nMAssay Description:Antagonist activity against C-C chemokine receptor type 2More data for this Ligand-Target Pair
Affinity DataKi: 620nMAssay Description:Inhibitory activity against human recombinant ATP-Citrate Lyase (ACL) enzymeMore data for this Ligand-Target Pair
Affinity DataKi: 630nMAssay Description:Inhibition of [125I]-MCP-1 binding to the cloned C-C chemokine receptor type 2B expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 631nMAssay Description:Inhibition of [125I]-MCP-1 binding to the cloned C-C chemokine receptor type 2B expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 631nMAssay Description:Inhibition of [125I]MCP-1 binding to the cloned C-C chemokine receptor type 2B expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 660nMAssay Description:Antagonist activity against C-C chemokine receptor type 2More data for this Ligand-Target Pair
Affinity DataKi: 700nMAssay Description:Inhibitory activity was tested agianst rat ATP-Citrate Lyase (ACL) enzymeMore data for this Ligand-Target Pair
Affinity DataKi: 700nMAssay Description:Inhibitory activity was tested agianst rat ATP-Citrate Lyase (ACL) enzymeMore data for this Ligand-Target Pair
Affinity DataKi: 710nMAssay Description:Inhibitory activity against human recombinant ATP-Citrate Lyase (ACL) enzymeMore data for this Ligand-Target Pair