Affinity DataKi: 0.100nMAssay Description:Compound was tested for the inhibition activity against HIV-1 proteaseMore data for this Ligand-Target Pair
Affinity DataKi: 0.113nMAssay Description:Inhibitory activity against P2 site in HIV protease.More data for this Ligand-Target Pair
Affinity DataKi: 0.151nMAssay Description:Inhibitory activity against P2 site in HIV protease.More data for this Ligand-Target Pair
Affinity DataKi: 0.162nMAssay Description:Inhibitory activity against P2 site in HIV protease.More data for this Ligand-Target Pair
Affinity DataKi: 0.172nMAssay Description:Inhibitory activity against P2 site in HIV protease.More data for this Ligand-Target Pair
Affinity DataKi: 0.452nMAssay Description:Inhibitory activity against P2 site in HIV protease.More data for this Ligand-Target Pair
Affinity DataKi: 0.550nMAssay Description:Inhibitory activity against P2 site in HIV protease.More data for this Ligand-Target Pair
Affinity DataKi: 0.700nMAssay Description:Compound was tested for its inhibitory activity against HIV-1 proteaseMore data for this Ligand-Target Pair
Affinity DataKi: 0.800nMAssay Description:Compound was tested for its inhibitory activity against HIV-1 proteaseMore data for this Ligand-Target Pair
Affinity DataKi: <1nMAssay Description:Compound was tested for the inhibition activity against HIV-1 proteaseMore data for this Ligand-Target Pair
Affinity DataKi: <1nMAssay Description:Compound was tested for the inhibition activity against HIV-1 proteaseMore data for this Ligand-Target Pair
Affinity DataKi: 2.60nMAssay Description:Inhibitory activity against P2 site in HIV protease.More data for this Ligand-Target Pair
Affinity DataKi: 2.90nMAssay Description:Compound was tested for its inhibitory activity against HIV-1 proteaseMore data for this Ligand-Target Pair
Affinity DataKi: 3.10nMAssay Description:Compound was tested for its inhibitory activity against HIV-1 proteaseMore data for this Ligand-Target Pair
Affinity DataKi: 3.60nMAssay Description:Compound was tested for its inhibitory activity against HIV-1 proteaseMore data for this Ligand-Target Pair
Affinity DataKi: 4nMAssay Description:Compound was tested for the inhibition activity against HIV-1 proteaseMore data for this Ligand-Target Pair
Affinity DataKi: 4.60nMAssay Description:Compound was tested for its inhibitory activity against HIV-1 proteaseMore data for this Ligand-Target Pair
Affinity DataKi: 5nMAssay Description:Compound was tested for its inhibitory activity against HIV-1 proteaseMore data for this Ligand-Target Pair
Affinity DataKi: 7nMAssay Description:Compound was tested for its inhibitory activity against HIV-1 proteaseMore data for this Ligand-Target Pair
Affinity DataKi: 10nMAssay Description:Inhibition constant was evaluated for inhibitory activity against the blood coagulant thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 11nMAssay Description:Compound was tested for the inhibition activity against HIV-1 proteaseMore data for this Ligand-Target Pair
Affinity DataKi: 13nMAssay Description:Compound was tested for its inhibitory activity against HIV-1 proteaseMore data for this Ligand-Target Pair
Affinity DataKi: 16nMAssay Description:Compound was tested for the inhibition activity against HIV-1 proteaseMore data for this Ligand-Target Pair
Affinity DataKi: 50nMAssay Description:Inhibition constant was evaluated for inhibitory activity against the blood coagulant thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 70nMAssay Description:Compound was tested for the inhibition activity against HIV-1 proteaseMore data for this Ligand-Target Pair
Affinity DataKi: 75nMAssay Description:Compound was tested for the inhibition activity against HIV-1 proteaseMore data for this Ligand-Target Pair
Affinity DataKi: 80nMAssay Description:Reversible inhibition of human CYP3A4 in liver microsomes by Dixon and Cornish-Bowden plot analysisMore data for this Ligand-Target Pair
Affinity DataKi: 200nMAssay Description:Inhibition constant was evaluated for inhibitory activity against the blood coagulant thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 300nMAssay Description:Compound was tested for the inhibition activity against HIV-1 proteaseMore data for this Ligand-Target Pair
Affinity DataKi: 600nMAssay Description:Inhibition constant was evaluated for inhibitory activity against the blood coagulant thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 3.06E+3nMAssay Description:Inhibition constant was evaluated for inhibitory activity against the blood coagulant thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 1.56E+4nMAssay Description:Inhibition constant was evaluated for inhibitory activity against the blood coagulant thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 3.17E+4nMAssay Description:Inhibition constant was evaluated for inhibitory activity against the blood coagulant thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 9.72E+4nMAssay Description:Inhibition constant was evaluated for inhibitory activity against the blood coagulant thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 1.10E+7nMAssay Description:Compound was tested for the inhibition activity against HIV-1 proteaseMore data for this Ligand-Target Pair
TargetDimer of Protein farnesyltransferase subunit beta(Homo sapiens (Human))
Keimyung University
Curated by ChEMBL
Keimyung University
Curated by ChEMBL
Affinity DataIC50: 0.0800nMAssay Description:Inhibition of farnesyl transferaseMore data for this Ligand-Target Pair
TargetDimer of Protein farnesyltransferase subunit beta(Homo sapiens (Human))
Keimyung University
Curated by ChEMBL
Keimyung University
Curated by ChEMBL
Affinity DataIC50: 0.0900nMAssay Description:Inhibition of farnesyl transferaseMore data for this Ligand-Target Pair
Affinity DataIC50: 0.100nMT: 2°CAssay Description:Compounds of the invention were initially diluted to 10 mM in 100% DMSO (CALBIOCHEM) for storage and made into kinase buffer solution to create a com...More data for this Ligand-Target Pair
Affinity DataIC50: 0.100nMT: 2°CAssay Description:Compounds of the invention were initially diluted to 10 mM in 100% DMSO (CALBIOCHEM) for storage and made into kinase buffer solution to create a com...More data for this Ligand-Target Pair
TargetDimer of Protein farnesyltransferase subunit beta(Homo sapiens (Human))
Keimyung University
Curated by ChEMBL
Keimyung University
Curated by ChEMBL
Affinity DataIC50: 0.160nMAssay Description:Inhibition of farnesyl transferaseMore data for this Ligand-Target Pair
TargetDimer of Protein farnesyltransferase subunit beta(Homo sapiens (Human))
Keimyung University
Curated by ChEMBL
Keimyung University
Curated by ChEMBL
Affinity DataIC50: 0.200nMAssay Description:Inhibition of farnesyl transferaseMore data for this Ligand-Target Pair
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Korea Research Institute Of Chemical Technology
Curated by ChEMBL
Korea Research Institute Of Chemical Technology
Curated by ChEMBL
Affinity DataIC50: 0.200nMAssay Description:Inhibition of recombinant c-Met by time resolved-fluorescence resonance energy transfer analysisMore data for this Ligand-Target Pair
TargetDimer of Protein farnesyltransferase subunit beta(Homo sapiens (Human))
Keimyung University
Curated by ChEMBL
Keimyung University
Curated by ChEMBL
Affinity DataIC50: 0.210nMAssay Description:Inhibition of farnesyl transferaseMore data for this Ligand-Target Pair
TargetDimer of Protein farnesyltransferase subunit beta(Homo sapiens (Human))
Keimyung University
Curated by ChEMBL
Keimyung University
Curated by ChEMBL
Affinity DataIC50: 0.240nMAssay Description:Inhibition of farnesyl transferaseMore data for this Ligand-Target Pair
TargetDimer of Protein farnesyltransferase subunit beta(Homo sapiens (Human))
Keimyung University
Curated by ChEMBL
Keimyung University
Curated by ChEMBL
Affinity DataIC50: 0.350nMAssay Description:Inhibition of farnesyl transferaseMore data for this Ligand-Target Pair
TargetDimer of Protein farnesyltransferase subunit beta(Homo sapiens (Human))
Keimyung University
Curated by ChEMBL
Keimyung University
Curated by ChEMBL
Affinity DataIC50: 0.370nMAssay Description:Inhibition of farnesyl transferaseMore data for this Ligand-Target Pair
TargetDimer of Protein farnesyltransferase subunit beta(Homo sapiens (Human))
Keimyung University
Curated by ChEMBL
Keimyung University
Curated by ChEMBL
Affinity DataIC50: 0.5nMAssay Description:Inhibition of farnesyl transferaseMore data for this Ligand-Target Pair
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
Lgci
Curated by ChEMBL
Lgci
Curated by ChEMBL
Affinity DataIC50: 0.5nMAssay Description:Inhibition of [3H]-FPP incorporation into Ha-ras protein by FarnesyltransferaseMore data for this Ligand-Target Pair
TargetReceptor-type tyrosine-protein kinase FLT3(Homo sapiens (Human))
Korea Research Institute Of Chemical Technology
Curated by ChEMBL
Korea Research Institute Of Chemical Technology
Curated by ChEMBL
Affinity DataIC50: 0.600nMAssay Description:Inhibition of recombinant FLT3 by time resolved-fluorescence resonance energy transfer analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 0.600nMT: 2°CAssay Description:Compounds of the invention were initially diluted to 10 mM in 100% DMSO (CALBIOCHEM) for storage and made into kinase buffer solution to create a com...More data for this Ligand-Target Pair