Affinity DataIC50: 0.5nMAssay Description:Inhibition of human C-terminal 6His-tagged SYK (356 to 635 residues) expressed in Sf9 insect cells using 5-carboxyfluorescein(FAM)-EEPLYWSFPAKKK-NH2 ...More data for this Ligand-Target Pair
Affinity DataIC50: 0.800nMAssay Description:Inhibition of human C-terminal 6His-tagged SYK (356 to 635 residues) expressed in Sf9 insect cells using 5-carboxyfluorescein(FAM)-EEPLYWSFPAKKK-NH2 ...More data for this Ligand-Target Pair
Affinity DataIC50: 0.900nMAssay Description:Inhibition of human C-terminal 6His-tagged SYK (356 to 635 residues) expressed in Sf9 insect cells using 5-carboxyfluorescein(FAM)-EEPLYWSFPAKKK-NH2 ...More data for this Ligand-Target Pair
Affinity DataIC50: 1.10nMAssay Description:Inhibition of human C-terminal 6His-tagged SYK (356 to 635 residues) expressed in Sf9 insect cells using 5-carboxyfluorescein(FAM)-EEPLYWSFPAKKK-NH2 ...More data for this Ligand-Target Pair
Affinity DataIC50: 1.10nMAssay Description:In vitro binding affinity against substance P receptor using [3H]SP as radioligand in guinea pig lung membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 1.70nMAssay Description:In vitro binding affinity against substance P receptor using [3H]SP as radioligand in guinea pig lung membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 1.70nMAssay Description:In vitro binding affinity against substance P receptor using [3H]SP as radioligand in guinea pig lung membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 1.80nMAssay Description:In vitro binding affinity against substance P receptor using [3H]SP as radioligand in guinea pig lung membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 2nMAssay Description:Inhibition of human recombinant full length N-terminal GST-tagged SYK cytoplasmic domain expressed in baculovirus expression system by Z'-LYTE assayMore data for this Ligand-Target Pair
Affinity DataIC50: 2.30nMAssay Description:Inhibition of human C-terminal 6His-tagged SYK (356 to 635 residues) expressed in Sf9 insect cells using 5-carboxyfluorescein(FAM)-EEPLYWSFPAKKK-NH2 ...More data for this Ligand-Target Pair
Affinity DataIC50: 3nMpH: 8.0 T: 2°CAssay Description:To assess the inhibitory activity of novel inhibitors, the PARP enzyme assay was carried out in reaction mixture consisting of activated salmon teste...More data for this Ligand-Target Pair
Affinity DataIC50: 3.10nMAssay Description:Inhibition of human C-terminal 6His-tagged SYK (356 to 635 residues) expressed in Sf9 insect cells using 5-carboxyfluorescein(FAM)-EEPLYWSFPAKKK-NH2 ...More data for this Ligand-Target Pair
Affinity DataIC50: 3.20nMAssay Description:Inhibition of human C-terminal 6His-tagged SYK (356 to 635 residues) expressed in Sf9 insect cells using 5-carboxyfluorescein(FAM)-EEPLYWSFPAKKK-NH2 ...More data for this Ligand-Target Pair
Affinity DataIC50: 3.5nMAssay Description:In vitro binding affinity against substance P receptor using [3H]SP as radioligand in guinea pig lung membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 3.5nMAssay Description:In vitro binding affinity against substance P receptor using [3H]SP as radioligand in guinea pig lung membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 3.5nMAssay Description:In vitro binding affinity against substance P receptor using [3H]SP as radioligand in guinea pig lung membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 4.30nMAssay Description:In vitro binding affinity against substance P receptor using [3H]SP as radioligand in guinea pig lung membraneMore data for this Ligand-Target Pair
TargetReceptor-type tyrosine-protein kinase FLT3(Homo sapiens (Human))
Takeda California
Curated by ChEMBL
Takeda California
Curated by ChEMBL
Affinity DataIC50: 4.60nMAssay Description:Inhibition of human N-terminal 6His-tagged FLT3 (564 to 993 residues) expressed in Sf9 insect cells using 5-carboxyfluorescein(FAM)-KKKKEEIYFFFG-NH2 ...More data for this Ligand-Target Pair
Affinity DataIC50: 4.60nMAssay Description:In vitro binding affinity against substance P receptor using [3H]SP as radioligand in guinea pig lung membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 4.70nMAssay Description:Inhibition of human C-terminal 6His-tagged SYK (356 to 635 residues) expressed in Sf9 insect cells using 5-carboxyfluorescein(FAM)-EEPLYWSFPAKKK-NH2 ...More data for this Ligand-Target Pair
Affinity DataIC50: 4.90nMAssay Description:In vitro binding affinity against substance P receptor using [3H]SP as radioligand in guinea pig lung membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 5nMAssay Description:In vitro binding affinity against substance P receptor using [3H]SP as radioligand in guinea pig lung membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 5.10nMAssay Description:Inhibition of rat VAP-1 expressed in CHO cells using [14C]-benzylamine as substrate preincubated for 30 mins prior to substrate addition measured aft...More data for this Ligand-Target Pair
Affinity DataIC50: 5.40nMAssay Description:In vitro binding affinity against substance P receptor using [3H]SP as radioligand in guinea pig lung membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 5.40nMAssay Description:In vitro binding affinity against substance P receptor using [3H]SP as radioligand in guinea pig lung membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 6nMAssay Description:In vitro inhibitory concentration against human recombinant Poly (ADP-ribose) polymerase 1More data for this Ligand-Target Pair
Affinity DataIC50: 6.40nMAssay Description:In vitro binding affinity against substance P receptor using [3H]SP as radioligand in guinea pig lung membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 7nMAssay Description:In vitro binding affinity against substance P receptor using [3H]SP as radioligand in guinea pig lung membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 7nMT: 2°CAssay Description:To assess the inhibitory activity of novel inhibitors, the PARP enzyme assay was carried out in reaction mixture consisting of activated salmon teste...More data for this Ligand-Target Pair
Affinity DataIC50: 7.40nMAssay Description:In vitro binding affinity against substance P receptor using [3H]SP as radioligand in guinea pig lung membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 7.60nMAssay Description:In vitro binding affinity against substance P receptor using [3H]SP as radioligand in guinea pig lung membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 8nMT: 2°CAssay Description:To assess the inhibitory activity of novel inhibitors, the PARP enzyme assay was carried out in reaction mixture consisting of activated salmon teste...More data for this Ligand-Target Pair
Affinity DataIC50: 8nMT: 2°CAssay Description:To assess the inhibitory activity of novel inhibitors, the PARP enzyme assay was carried out in reaction mixture consisting of activated salmon teste...More data for this Ligand-Target Pair
Affinity DataIC50: 8nMAssay Description:In vitro binding affinity against substance P receptor using [3H]SP as radioligand in guinea pig lung membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 8.30nMAssay Description:In vitro inhibitory concentration against human recombinant Poly (ADP-ribose) polymerase 1More data for this Ligand-Target Pair
Affinity DataIC50: 8.90nMAssay Description:In vitro inhibitory concentration against human recombinant Poly (ADP-ribose) polymerase 1More data for this Ligand-Target Pair
TargetDual specificity mitogen-activated protein kinase kinase 1(Homo sapiens (Human))
Takeda California
Curated by ChEMBL
Takeda California
Curated by ChEMBL
Affinity DataIC50: 8.90nMAssay Description:Inhibition of MEK1-mediated ERK1 phosphorylation using IPTTPITTYFFFK-5FAM-COOH as substrate by fluorescent polarization assayMore data for this Ligand-Target Pair
Affinity DataIC50: 9nMAssay Description:In vitro binding affinity against substance P receptor using [3H]SP as radioligand in guinea pig lung membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 9nMT: 2°CAssay Description:To assess the inhibitory activity of novel inhibitors, the PARP enzyme assay was carried out in reaction mixture consisting of activated salmon teste...More data for this Ligand-Target Pair
Affinity DataIC50: 9nMAssay Description:In vitro binding affinity against substance P receptor using [3H]SP as radioligand in guinea pig lung membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 9.20nMAssay Description:In vitro binding affinity against substance P receptor using [3H]SP as radioligand in guinea pig lung membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:In vitro binding affinity against substance P receptor using [3H]SP as radioligand in guinea pig lung membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 11nMpH: 8.0 T: 2°CAssay Description:To assess the inhibitory activity of novel inhibitors, the PARP enzyme assay was carried out in reaction mixture consisting of activated salmon teste...More data for this Ligand-Target Pair
Affinity DataIC50: 11nMT: 2°CAssay Description:To assess the inhibitory activity of novel inhibitors, the PARP enzyme assay was carried out in reaction mixture consisting of activated salmon teste...More data for this Ligand-Target Pair
Affinity DataIC50: 11nMAssay Description:In vitro binding affinity against substance P receptor using [3H]SP as radioligand in guinea pig lung membraneMore data for this Ligand-Target Pair
TargetDual specificity mitogen-activated protein kinase kinase 1(Homo sapiens (Human))
Takeda California
Curated by ChEMBL
Takeda California
Curated by ChEMBL
Affinity DataIC50: 11nMAssay Description:Inhibition of MEK1-mediated ERK1 phosphorylation using IPTTPITTYFFFK-5FAM-COOH as substrate by fluorescent polarization assayMore data for this Ligand-Target Pair
Affinity DataIC50: 12nMAssay Description:In vitro binding affinity against substance P receptor using [3H]SP as radioligand in guinea pig lung membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 12nMAssay Description:In vitro inhibitory concentration against human recombinant Poly (ADP-ribose) polymerase 1More data for this Ligand-Target Pair
Affinity DataIC50: 12nMAssay Description:In vitro inhibitory concentration against human recombinant Poly (ADP-ribose) polymerase 1More data for this Ligand-Target Pair
Affinity DataIC50: 12nMAssay Description:In vitro inhibitory concentration against human recombinant Poly (ADP-ribose) polymerase 1More data for this Ligand-Target Pair