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Found 93 with Last Name = 'park' and Initial = 'oh'
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50170264(CHEMBL361931 | N-{4-[3-(4-tert-Butyl-benzyl)-thiou...)
Affinity DataIC50:  8.40nMAssay Description:Inhibitory effect on capsaicin (0.5 uM)-induced calcium uptake in rat DRG neurons upon incubation at RT for 10 minutesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rattus norvegicus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM20321(3-[(4-tert-butylphenyl)methyl]-1-[(3-fluoro-4-meth...)
Affinity DataIC50:  37nMAssay Description:Inhibition of [Ca2+] uptake in dorsal root ganglion (DRG) neurons from neonatal Sprague-Dawley ratMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM20321(3-[(4-tert-butylphenyl)methyl]-1-[(3-fluoro-4-meth...)
Affinity DataIC50:  37nMAssay Description:Inhibitory effect on capsaicin (0.5 uM)-induced calcium uptake in rat DRG neurons upon incubation at RT for 10 minutesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50172566(CHEMBL196291 | N-{4-[3-(4-tert-Butyl-benzyl)-thiou...)
Affinity DataIC50:  41nMAssay Description:Inhibitory effect on capsaicin (0.5 uM)-induced calcium uptake in rat DRG neurons upon incubation at RT for 10 minutesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50172563(1-(1H-Benzotriazol-5-ylmethyl)-3-(4-tert-butyl-ben...)
Affinity DataIC50:  50nMAssay Description:Inhibitory effect on capsaicin (0.5 uM)-induced calcium uptake in rat DRG neurons upon incubation at RT for 10 minutesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM20321(3-[(4-tert-butylphenyl)methyl]-1-[(3-fluoro-4-meth...)
Affinity DataIC50:  54nMAssay Description:Concentration required to inhibit [3H]-RTX radioligand binding towards transient receptor potential cation channel (subfamily V, member 1) expressed ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50170263(CHEMBL189418 | N-{4-[3-(4-tert-Butyl-benzyl)-thiou...)
Affinity DataIC50:  71nMAssay Description:Inhibitory effect on capsaicin (0.5 uM)-induced calcium uptake in rat DRG neurons upon incubation at RT for 10 minutesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50172578(CHEMBL196085 | N-{2-Bromo-4-[3-(4-tert-butyl-benzy...)
Affinity DataIC50:  80nMAssay Description:Inhibitory effect on capsaicin (0.5 uM)-induced calcium uptake in rat DRG neurons upon incubation at RT for 10 minutesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rattus norvegicus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM20315(3-[(4-tert-butylphenyl)methyl]-1-[(4-methanesulfon...)
Affinity DataIC50:  110nMAssay Description:Inhibition of [Ca2+] uptake in dorsal root ganglion (DRG) neurons from neonatal Sprague-Dawley ratMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM20315(3-[(4-tert-butylphenyl)methyl]-1-[(4-methanesulfon...)
Affinity DataIC50:  110nMAssay Description:Inhibitory effect on capsaicin (0.5 uM)-induced calcium uptake in rat DRG neurons upon incubation at RT for 10 minutesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50172590(CHEMBL196255 | N-{4-[3-(3,5-Di-tert-butyl-benzyl)-...)
Affinity DataIC50:  200nMAssay Description:Inhibitory effect on capsaicin (0.5 uM)-induced calcium uptake in rat DRG neurons upon incubation at RT for 10 minutesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50172587(CHEMBL197770 | N-{4-[3-(4-tert-Butyl-benzyl)-ureid...)
Affinity DataIC50:  240nMAssay Description:Inhibitory effect on capsaicin (0.5 uM)-induced calcium uptake in rat DRG neurons upon incubation at RT for 10 minutesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50172567(CHEMBL197222 | N-{4-[3-(4-tert-Butyl-benzyl)-ureid...)
Affinity DataIC50:  240nMAssay Description:Inhibitory effect on capsaicin (0.5 uM)-induced calcium uptake in rat DRG neurons upon incubation at RT for 10 minutesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50172598(CHEMBL197781 | N-(4-[({4-tert-Butylbenzyl}aminocar...)
Affinity DataIC50:  300nMAssay Description:Inhibitory effect on capsaicin (0.5 uM)-induced calcium uptake in rat DRG neurons upon incubation at RT for 10 minutesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50172595(CHEMBL196229 | N-{4-[3-(4-Chloro-benzyl)-thioureid...)
Affinity DataIC50:  340nMAssay Description:Inhibitory effect on capsaicin (0.5 uM)-induced calcium uptake in rat DRG neurons upon incubation at RT for 10 minutesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50172581(CHEMBL194592 | N-(4-{3-[2-(4-tert-Butyl-phenyl)-et...)
Affinity DataIC50:  370nMAssay Description:Inhibitory effect on capsaicin (0.5 uM)-induced calcium uptake in rat DRG neurons upon incubation at RT for 10 minutesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50172560(CHEMBL382920 | N-{2-Fluoro-4-[3-(4-propyl-benzyl)-...)
Affinity DataIC50:  460nMAssay Description:Inhibitory effect on capsaicin (0.5 uM)-induced calcium uptake in rat DRG neurons upon incubation at RT for 10 minutesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50172582(CHEMBL198139 | N-{4-[3-(4-Butyl-benzyl)-thioureido...)
Affinity DataIC50:  470nMAssay Description:Inhibitory effect on capsaicin (0.5 uM)-induced calcium uptake in rat DRG neurons upon incubation at RT for 10 minutesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50172565(CHEMBL198300 | N-{2-Fluoro-4-[3-(4-isopropyl-benzy...)
Affinity DataIC50:  520nMAssay Description:Inhibitory effect on capsaicin (0.5 uM)-induced calcium uptake in rat DRG neurons upon incubation at RT for 10 minutesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50172593(CHEMBL196281 | N-{4-[3-(4-Bromo-benzyl)-thioureido...)
Affinity DataIC50:  570nMAssay Description:Inhibitory effect on capsaicin (0.5 uM)-induced calcium uptake in rat DRG neurons upon incubation at RT for 10 minutesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rattus norvegicus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM20284(CHEMBL391997 | CPZ | Capsazepine | N-[2-(4-chlorop...)
Affinity DataIC50:  590nMAssay Description:Inhibition of [Ca2+] uptake in dorsal root ganglion (DRG) neurons from neonatal Sprague-Dawley ratMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50172562(CHEMBL197350 | N-{2-Fluoro-4-[3-(4-iodo-benzyl)-th...)
Affinity DataIC50:  630nMAssay Description:Inhibitory effect on capsaicin (0.5 uM)-induced calcium uptake in rat DRG neurons upon incubation at RT for 10 minutesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50172586(CHEMBL198457 | N-{2-Fluoro-4-[3-(2-methyl-benzyl)-...)
Affinity DataIC50:  670nMAssay Description:Inhibitory effect on capsaicin (0.5 uM)-induced calcium uptake in rat DRG neurons upon incubation at RT for 10 minutesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50172575(5-[3-(4-tert-Butyl-benzyl)-thioureidomethyl]-2-met...)
Affinity DataIC50:  720nMAssay Description:Inhibitory effect on capsaicin (0.5 uM)-induced calcium uptake in rat DRG neurons upon incubation at RT for 10 minutesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50172596(CHEMBL198994 | N-{4-[4-(tert-butyl)benzylamino(1-c...)
Affinity DataIC50:  730nMAssay Description:Inhibitory effect on capsaicin (0.5 uM)-induced calcium uptake in rat DRG neurons upon incubation at RT for 10 minutesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50172585(1-(1H-Benzoimidazol-5-ylmethyl)-3-(4-tert-butyl-be...)
Affinity DataIC50:  790nMAssay Description:Inhibitory effect on capsaicin (0.5 uM)-induced calcium uptake in rat DRG neurons upon incubation at RT for 10 minutesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50172572(CHEMBL196553 | N-{4-[3-(4-Ethyl-benzyl)-thioureido...)
Affinity DataIC50:  1.10E+3nMAssay Description:Inhibitory effect on capsaicin (0.5 uM)-induced calcium uptake in rat DRG neurons upon incubation at RT for 10 minutesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50172601(CHEMBL197558 | N-{4-[(3-Anthracen-9-yl-thioureido)...)
Affinity DataIC50:  1.10E+3nMAssay Description:Inhibitory effect on capsaicin (0.5 uM)-induced calcium uptake in rat DRG neurons upon incubation at RT for 10 minutesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50172600(CHEMBL198508 | N-{2-Fluoro-4-[3-(3-methyl-benzyl)-...)
Affinity DataIC50:  1.30E+3nMAssay Description:Inhibitory effect on capsaicin (0.5 uM)-induced calcium uptake in rat DRG neurons upon incubation at RT for 10 minutesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50172579(CHEMBL196372 | N-{2-Fluoro-4-[3-(4-methyl-benzyl)-...)
Affinity DataIC50:  1.50E+3nMAssay Description:Inhibitory effect on capsaicin (0.5 uM)-induced calcium uptake in rat DRG neurons upon incubation at RT for 10 minutesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50172574(CHEMBL370797 | N-{4-[3-(4-tert-Butyl-benzyl)-thiou...)
Affinity DataIC50:  1.50E+3nMAssay Description:Inhibitory effect on capsaicin (0.5 uM)-induced calcium uptake in rat DRG neurons upon incubation at RT for 10 minutesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50172561(CHEMBL198443 | N-{4-[3-(4-tert-Butyl-phenyl)-thiou...)
Affinity DataIC50:  1.60E+3nMAssay Description:Inhibitory effect on capsaicin (0.5 uM)-induced calcium uptake in rat DRG neurons upon incubation at RT for 10 minutesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50172569(1-(4-tert-Butyl-benzyl)-3-(1H-indol-5-ylmethyl)-th...)
Affinity DataIC50:  1.80E+3nMAssay Description:Inhibitory effect on capsaicin (0.5 uM)-induced calcium uptake in rat DRG neurons upon incubation at RT for 10 minutesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50172564(CHEMBL382921 | N-(4-{3-[3-(4-tert-Butyl-phenyl)-pr...)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibitory effect on capsaicin (0.5 uM)-induced calcium uptake in rat DRG neurons upon incubation at RT for 10 minutesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50172589(CHEMBL197516 | N-[4-(3-Benzhydryl-thioureidomethyl...)
Affinity DataIC50:  2.50E+3nMAssay Description:Inhibitory effect on capsaicin (0.5 uM)-induced calcium uptake in rat DRG neurons upon incubation at RT for 10 minutesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50172594(CHEMBL195919 | N-{2-Fluoro-4-[(3-naphthalen-1-yl-t...)
Affinity DataIC50:  2.60E+3nMAssay Description:Inhibitory effect on capsaicin (0.5 uM)-induced calcium uptake in rat DRG neurons upon incubation at RT for 10 minutesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50172591(CHEMBL194293 | N-{4-[4-(tert-butyl)benzylamino(met...)
Affinity DataIC50:  3.10E+3nMAssay Description:Inhibitory effect on capsaicin (0.5 uM)-induced calcium uptake in rat DRG neurons upon incubation at RT for 10 minutesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50172592(CHEMBL373044 | {4-[3-(4-tert-Butyl-benzyl)-thioure...)
Affinity DataIC50:  3.60E+3nMAssay Description:Inhibitory effect on capsaicin (0.5 uM)-induced calcium uptake in rat DRG neurons upon incubation at RT for 10 minutesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50172599(5-[3-(4-tert-Butyl-benzyl)-ureidomethyl]-2-methane...)
Affinity DataIC50:  3.70E+3nMAssay Description:Inhibitory effect on capsaicin (0.5 uM)-induced calcium uptake in rat DRG neurons upon incubation at RT for 10 minutesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50172573(CHEMBL193908 | N-{4-[3-(4-tert-Butyl-benzyl)-thiou...)
Affinity DataIC50:  5.90E+3nMAssay Description:Inhibitory effect on capsaicin (0.5 uM)-induced calcium uptake in rat DRG neurons upon incubation at RT for 10 minutesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50172576(CHEMBL196423 | N-{4-[4-(tert-butyl)benzylamino(eth...)
Affinity DataIC50:  6.20E+3nMAssay Description:Inhibitory effect on capsaicin (0.5 uM)-induced calcium uptake in rat DRG neurons upon incubation at RT for 10 minutesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50172584(CHEMBL372982 | N-[4-(3-Benzyl-thioureidomethyl)-2-...)
Affinity DataIC50:  9.70E+3nMAssay Description:Inhibitory effect on capsaicin (0.5 uM)-induced calcium uptake in rat DRG neurons upon incubation at RT for 10 minutesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50172580(CHEMBL198455 | N-{4-[3-(4-tert-Butyl-benzyl)-thiou...)
Affinity DataIC50:  1.09E+4nMAssay Description:Inhibitory effect on capsaicin (0.5 uM)-induced calcium uptake in rat DRG neurons upon incubation at RT for 10 minutesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Ovis aries (Sheep))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50097197((E)-6-((1R,4aR,7S)-1,4a,7-Trimethyl-7-vinyl-1,2,3,...)
Affinity DataIC50:  1.32E+4nMAssay Description:Inhibitory activity against Prostaglandin G/H synthase 2 from sheep placental cotyledonsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Homo sapiens (Human))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50097195((1R,4aR,7S)-7-(2-Fluoro-ethyl)-1,4a,7-trimethyl-1,...)
Affinity DataIC50:  1.84E+4nMAssay Description:Inhibitory activity against Prostaglandin G/H synthase 1 from rabbit renal microsomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Homo sapiens (Human))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50097201((1R,4aR,7S)-1,4a,7-Trimethyl-7-vinyl-1,2,3,4,4a,6,...)
Affinity DataIC50:  1.84E+4nMAssay Description:Inhibitory activity against Prostaglandin G/H synthase 1 from rabbit renal microsomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Homo sapiens (Human))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50097210(3-((1S,4aR,7S)-1,4a,7-Trimethyl-7-vinyl-1,2,3,4,4a...)
Affinity DataIC50:  2.11E+4nMAssay Description:Inhibitory activity against Prostaglandin G/H synthase 1 from rabbit renal microsomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rattus norvegicus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50222457(CHEMBL136158)
Affinity DataIC50:  2.43E+4nMAssay Description:Inhibition of [Ca2+] uptake in dorsal root ganglion (DRG) neurons from neonatal Sprague-Dawley ratMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Homo sapiens (Human))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50097199(((1S,4aR,7S)-1,4a,7-Trimethyl-7-vinyl-1,2,3,4,4a,6...)
Affinity DataIC50:  2.81E+4nMAssay Description:Inhibitory activity against Prostaglandin G/H synthase 1 from rabbit renal microsomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50172588(CHEMBL197933 | N-[4-(3-tert-Butyl-thioureidomethyl...)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibitory effect on capsaicin (0.5 uM)-induced calcium uptake in rat DRG neurons upon incubation at RT for 10 minutesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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