Affinity DataKi: 2.66nMAssay Description:Displacement of [3H]-CP55940 from human recombinant cannabinoid CB2 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 174nMAssay Description:Displacement of [3H]CCK8 from rat pancreas CCK1 receptor at by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 275nMAssay Description:Displacement of [3H]CCK8 from rat pancreas CCK1 receptor at by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 347nMAssay Description:Displacement of [3H]CCK8 from rat pancreas CCK1 receptor at by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 387nMAssay Description:Displacement of [3H]-CP55940 from human recombinant cannabinoid CB2 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 467nMAssay Description:Displacement of [3H]CCK8 from rat pancreas CCK1 receptor at by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 468nMAssay Description:Displacement of [3H]CCK8 from rat pancreas CCK1 receptor at by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 537nMAssay Description:Displacement of [3H]CCK8 from rat pancreas CCK1 receptor at by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 676nMAssay Description:Displacement of [3H]CCK8 from rat pancreas CCK1 receptor at by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 1.02E+3nMAssay Description:Displacement of [3H]CCK8 from rat pancreas CCK1 receptor at by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 1.02E+3nMAssay Description:Displacement of [3H]CCK8 from rat pancreas CCK1 receptor at by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 1.07E+3nMAssay Description:Displacement of [3H]CCK8 from rat pancreas CCK1 receptor at by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 1.45E+3nMAssay Description:Displacement of [3H]CCK8 from rat pancreas CCK1 receptor at by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 1.48E+3nMAssay Description:Displacement of [3H]CCK8 from rat pancreas CCK1 receptor at by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 1.58E+3nMAssay Description:Displacement of [3H]CCK8 from rat pancreas CCK1 receptor at by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 1.58E+3nMAssay Description:Displacement of [3H]CCK8 from rat pancreas CCK1 receptor at by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 1.58E+3nMAssay Description:Displacement of [3H]CCK8 from rat pancreas CCK1 receptor at by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 1.66E+3nMAssay Description:Displacement of [3H]CCK8 from rat pancreas CCK1 receptor at by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 2.04E+3nMAssay Description:Displacement of [3H]CCK8 from rat pancreas CCK1 receptor at by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 2.23E+3nMAssay Description:Displacement of [3H]CCK8 from rat pancreas CCK1 receptor at by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 2.24E+3nMAssay Description:Displacement of [3H]CCK8 from rat pancreas CCK1 receptor at by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 2.57E+3nMAssay Description:Displacement of [3H]CCK8 from rat pancreas CCK1 receptor at by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 2.57E+3nMAssay Description:Displacement of [3H]CCK8 from rat pancreas CCK1 receptor at by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 2.69E+3nMAssay Description:Displacement of [3H]CCK8 from rat pancreas CCK1 receptor at by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 3.09E+3nMAssay Description:Displacement of [3H]CCK8 from rat pancreas CCK1 receptor at by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 3.24E+3nMAssay Description:Displacement of [3H]CCK8 from rat pancreas CCK1 receptor at by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 3.31E+3nMAssay Description:Displacement of [3H]CCK8 from rat pancreas CCK1 receptor at by liquid scintillation countingMore data for this Ligand-Target Pair
TargetEnoyl-[acyl-carrier-protein] reductase [NADH](Francisella tularensis subsp. tularensis (strain S...)
Naval Research Laboratories
Curated by ChEMBL
Naval Research Laboratories
Curated by ChEMBL
Affinity DataKi: 3.40E+3nMAssay Description:Competitive inhibition of C-terminal His6-tagged Francisella tularensis SCHU S4 FabI expressed in Escherichia coli BL21 (DE3) using CrCoA as substrat...More data for this Ligand-Target Pair
Affinity DataKi: 4.07E+3nMAssay Description:Displacement of [3H]CCK8 from rat pancreas CCK1 receptor at by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 5.13E+3nMAssay Description:Displacement of [3H]CCK8 from rat pancreas CCK1 receptor at by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 5.13E+3nMAssay Description:Displacement of [3H]CCK8 from rat pancreas CCK1 receptor at by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 6.61E+3nMAssay Description:Displacement of [3H]CCK8 from rat pancreas CCK1 receptor at by liquid scintillation countingMore data for this Ligand-Target Pair
TargetEnoyl-[acyl-carrier-protein] reductase [NADH](Francisella tularensis subsp. tularensis (strain S...)
Naval Research Laboratories
Curated by ChEMBL
Naval Research Laboratories
Curated by ChEMBL
Affinity DataKi: 7.00E+3nMAssay Description:Competitive inhibition of C-terminal His6-tagged Francisella tularensis SCHU S4 FabI expressed in Escherichia coli BL21 (DE3) using CrCoA as substrat...More data for this Ligand-Target Pair
Affinity DataKi: 8.32E+3nMAssay Description:Displacement of [3H]CCK8 from rat pancreas CCK1 receptor at by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 9.55E+3nMAssay Description:Displacement of [3H]CCK8 from rat pancreas CCK1 receptor at by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]CCK8 from rat pancreas CCK1 receptor at by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]CCK8 from rat pancreas CCK1 receptor at by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 1.74E+4nMAssay Description:Displacement of [3H]CCK8 from rat pancreas CCK1 receptor at by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 2.04E+4nMAssay Description:Displacement of [3H]CCK8 from rat pancreas CCK1 receptor at by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataIC50: 0.130nMAssay Description:Inhibition of MEK U911-activated ERK2 (unknown origin) using ERKtide as substrate preincubated for 20 mins followed by substrate addition in presence...More data for this Ligand-Target Pair
Affinity DataIC50: 0.200nMAssay Description:Inhibition of ERK2 (unknown origin) in the presence of 1 mM ATPMore data for this Ligand-Target Pair
Affinity DataIC50: <0.300nMAssay Description:Inhibition of MEK U911-activated ERK2 (unknown origin) using ERKtide as substrate preincubated for 20 mins followed by substrate addition in presence...More data for this Ligand-Target Pair
Affinity DataIC50: <0.300nMAssay Description:Inhibition of MEK U911-activated ERK2 (unknown origin) using Erktide as substrate preincubated with enzyme for 20 mins prior to substrate addition by...More data for this Ligand-Target Pair
Affinity DataIC50: <0.300nMAssay Description:Inhibition of MEK U911-activated ERK2 (unknown origin) using ERKtide as substrate preincubated for 20 mins followed by substrate addition in presence...More data for this Ligand-Target Pair
Affinity DataIC50: <0.300nMAssay Description:Inhibition of MEK U911-activated ERK2 (unknown origin) using Erktide as substrate preincubated with enzyme for 20 mins prior to substrate addition by...More data for this Ligand-Target Pair
Affinity DataIC50: <0.300nMAssay Description:Inhibition of MEK U911-activated ERK2 (unknown origin) using ERKtide as substrate preincubated for 20 mins followed by substrate addition in presence...More data for this Ligand-Target Pair
Affinity DataIC50: <0.300nMAssay Description:Inhibition of MEK U911-activated ERK2 (unknown origin) using Erktide as substrate preincubated with enzyme for 20 mins prior to substrate addition by...More data for this Ligand-Target Pair
Affinity DataIC50: <0.300nMAssay Description:Inhibition of ERK2 (unknown origin) in the presence of 60 uM ATPMore data for this Ligand-Target Pair
Affinity DataIC50: <0.300nMAssay Description:Inhibition of MEK U911-activated ERK2 (unknown origin) using ERKtide as substrate preincubated for 20 mins followed by substrate addition in presence...More data for this Ligand-Target Pair
Affinity DataIC50: <0.300nMAssay Description:Inhibition of ERK2 (unknown origin) in the presence of 60 uM ATPMore data for this Ligand-Target Pair