Compile Data Set for Download or QSAR
maximum 50k data
Found 2 Enz. Inhib. hit(s) with Target = 'Adenosine receptor A2b' and Ligand = 'BDBM50170137'
TargetAdenosine receptor A2b(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50170137(1-Benzyl-7-methyl-3-propyl-1H,6H-pyrrolo[2,1-f]pur...)
Affinity DataIC50:  400nMAssay Description:Antagonist activity at human cloned adenosine A2B cells expressed in CHO cells assessed as inhibition of NECA-stimulated cAMP productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50170137(1-Benzyl-7-methyl-3-propyl-1H,6H-pyrrolo[2,1-f]pur...)
Affinity DataIC50:  400nMAssay Description:Inhibition of 100 nM NECA-stimulated cAMP production in CHO cells expressing human adenosine A2B receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed